Configure Receptors:

1200015E14Rik 17Beta-HSD Type 3 5-HT Transporter 5-HT-S1 5-HT-S1A 5-HT1 5-HT1 like 5-HT1A 5-HT1B 5-HT1C 5-HT1D 5-HT1Dalpha 5-HT1Db 5-HT1DBeta 5-HT1E 5-HT1F 5-HT2 5-HT2A 5-HT2B 5-HT2C 5-HT2c VGI 5-HT3 5-HT4 5-HT5 5-HT5a 5-HT5B 5-HT6 5-HT7 5-Lipoxygenase Acetylcholinesterase Acetylcholinesterase, AChE Activated p21cdc42Hs kinase Activator Protein AP-1 ADENOSINE ADENOSINE A1 ADENOSINE A1 high ADENOSINE A1 low ADENOSINE A2 ADENOSINE A2a ADENOSINE A2B ADENOSINE A3 Adenosine A4 Adenosine Deaminase ADA Adenosine Kinase, AK Adenosine transporter Adenylate cyclase Adenylate cyclase Forskolin Adrenaline Adrenaline 1 Adrenaline 2 Adrenaline alpha1 Adrenaline alpha2 Adrenaline beta1 Adrenergic Alpha adrenergic Alpha1 adrenergic Alpha1A adrenergic Alpha1B adrenergic Alpha1C adrenergic Alpha1D adrenergic Alpha2 adrenergic Alpha2A adrenergic Alpha2B adrenergic Alpha2C adrenergic Alpha2D adrenergic Beta adrenergic Beta1 adrenergic Beta1,2 adrenergic Beta2 adrenergic Beta3 Akt aldose reductase all-trans-retinoic acid, atRA Alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid Anandamid membrane transporter, AMT Anaplastic lymphoma kinase (Ki-1) androgen Androgen Receptor ANF Angiotensin ANGIOTENSIN AT1 Angiotensin AT2 Angiotensin II AT1 Angiotensin II AT1A Angiotensin II AT1B Angiotensin II AT2 Angiotensin II, central Angiotensin IV Angiotensin-converting enzyme, ACE AP2 associated kinase 1 Arg-vasopressin V1 ATPase (Na+, K+) atrial natriuretic peptide, ANP Aurora kinase C B lymphoid tyrosine kinase B1 B1 BRADYKININ B2 BRADYKININ Benzodiazepine central Benzodiazepine peripheral beta-amyloid BHE BHSK BHSP Bile Salt Export Pump, BSEP BMP2 inducible kinase BMX non-receptor tyrosine kinase Bombesin Bombesin 1 Bombesin 2 Bombesin 3 Bombesin 4 Bruton agammaglobulinemia tyrosine kinase butyrylcholinesterase, BuChE C-src tyrosine kinase calcineurin Calcitonin Gene-Related Peptide Calcitonin Gene-related Peptide (CGRP) Calcitonin Gene-Related Peptide 1 Calcium channel Calcium channel (DHP) Calcium channel (Type L) Calcium channel (Type N) Calcium channel (Type T,L) Calcium channel (VER) Calcium channel diltiazem Calcium channel verapamil binding site Calcium/calmodulin-dependent protein kinase (CaM kinase) II alpha Calcium/calmodulin-dependent protein kinase (CaM kinase) II beta Calcium/calmodulin-dependent protein kinase (CaM kinase) II delta Calcium/calmodulin-dependent protein kinase (CaM kinase) II gamma Calcium/calmodulin-dependent protein kinase I Calcium/calmodulin-dependent protein kinase ID Calcium/calmodulin-dependent protein kinase IG Calcium/calmodulin-dependent protein kinase kinase 1, alpha Calcium/calmodulin-dependent protein kinase kinase 2, beta calmodulin kinase calpain calpain-1 CANNABINOID CB1 CANNABINOID CB2 Carbonic Anhydrase Isozymes, CA I Carbonic Anhydrase Isozymes, CA II Carbonic Anhydrase Isozymes, CA IX Carboxypeptidase CPG2 Casein kinase 1 Delta Casein kinase 1, epsilon Casein kinase 1, gamma 1 Casein kinase 1, gamma 2 casein kinase-1 casein kinase-2 caspase-2 caspase-3 caspase-6 caspase-7 caspase-8 Cathepsin D CCK A CCK B CCR5 CDC-like kinase 1 CDC-like kinase 2 CDC-like kinase 3 CDC-like kinase 4 CDK1 CDK2 CDK4 CDK5 activator-binding protein C53 CGRP CGRP1 Chemoattractant receptor-homologous, CRTH2 Chemokine CXCR1 Chemokine CXCR2 Chemokine CXCR3 Chemokine CXCR4 Chemokine receptor 5 Chemokine US28 Chloride channel, TBOB Chloride ionophore Cholecystokinin Cholecystokinin 1 Cholecystokinin 2 Cholecystokinin A Cholecystokinin B Cholecystokinin central Cholecystokinin peripheral Choline Acetyltransferase Choline Uptake Cholinergic, muscarinic Cholinergic, muscarinic M1 Cholinergic, muscarinic M2 Cholinergic, muscarinic M3 Cholinergic, muscarinic M4 Cholinergic, muscarinic M5 Cholinergic, nicotinic Cholinergic, Nicotinic Alpha1Beta1DeltaGamma Cholinergic, Nicotinic Alpha1Beta2 Cholinergic, Nicotinic Alpha2Beta2 Cholinergic, Nicotinic Alpha2Beta4 Cholinergic, Nicotinic Alpha3Beta2 Cholinergic, Nicotinic Alpha3Beta4 Cholinergic, Nicotinic Alpha3Beta4x Cholinergic, Nicotinic Alpha4Beta2 Cholinergic, Nicotinic Alpha4Beta4 Cholinergic, Nicotinic Alpha6 Cholinergic, Nicotinic Alpha6Beta2 Cholinergic, Nicotinic Alpha6Beta3Beta4Alpha5 Cholinergic, Nicotinic Alpha6Beta4 Cholinergic, Nicotinic Alpha7 Cholinergic, Nicotinic Alpha7/5-HT3 Cholinergic, Nicotinic Muscle Corticotropin-Releasing Factor COX-1 COX-2 CRF CRF-R1 CRF-R2 Alpha CRF-R2 Beta CRF1 CRF2 Beta Cyclin G associated kinase Cyclin-dependent kinase 2 Death-associated kinase 3 Death-associated protein kinase 2 Deoxyuridine triphosphatase Dihyrofolate Reductase, DHFR Dipeptidyl peptidase DPP II Dipeptidyl peptidase DPP IV DOPAMINE DOPAMINE D1 Dopamine D1 high Dopamine D1 low Dopamine D1A Dopamine D1B DOPAMINE D2 DOPAMINE D2 Long DOPAMINE D2 Short DOPAMINE D2/D4 Dopamine D2A Dopamine D2B DOPAMINE D3 Dopamine D3A DOPAMINE D4 DOPAMINE D5 Dopamine Transporter Dopamine Uptake Dopamine, cocaine site Dopamine1-like Dopamine2-like DRI Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A dUTPase EGF EGF-R Eledoisin ENDOTHELIN ENDOTHELIN A ENDOTHELIN B EPH receptor A2 EPH receptor A3 EPH receptor A4 EPH receptor A5 EPH receptor A6 EPH receptor A7 EPH receptor A8 EPH receptor B1 EPH receptor B2 EPH receptor B4 Epidermal growth factor receptor estrogen estrogen alpha estrogen beta Estrogen receptor alpha Estrogen receptor beta Excitatory Amino Acid EAAT1 Excitatory Amino Acid EAAT2 Excitatory Amino Acid EAAT3 Export Pump, ABCC2 extracellular-regulated protein kinase, ERK Fatty Acid Amide Hydrolic, FAAH Fer (fps/fes related) tyrosine kinase (phosphoprotein NCP94) FGF FGF-R2 FGFR-1, (cyto) FGFR-1, (FL) Fibroblast growth factor receptor 1 Fibroblast growth factor receptor 2 Fibroblast growth factor receptor 3 FKBP12 Fms-related tyrosine kinase 3 Fms-related tyrosine kinase 4 Follicle-Stimulating Hormone, FSH Formyl peptide Receptor FYN oncogene related to SRC, FGR, YES Fyn-related kinase GABA GABA A GABA A alpha1 GABA A Alpha1Beta1Gamma2 GABA A Alpha1Beta2 GABA A Alpha1Beta2Gamma2 GABA A Alpha1Beta3Gamma2 GABA A alpha2 GABA A Alpha2Beta1Gamma2 GABA A Alpha2Beta2Gamma2 GABA A Alpha2Beta3Gamma2 GABA A alpha3 GABA A Alpha3Beta1Gamma2 GABA A Alpha3Beta2Gamma2 GABA A Alpha3Beta3Gamma2 GABA A Alpha4Beta2Gamma2 GABA A Alpha4Beta3Gamma2 GABA A Alpha4Gamma2 GABA A alpha5 GABA A Alpha5Beta1Gamma2 GABA A Alpha5Beta2Gamma2 GABA A Alpha5Beta3Gamma2 GABA A Alpha5m10Beta2Gamma2 GABA A Alpha5m8Beta2Gamma2 GABA A Alpha5m9Beta2Gamma2 GABA A alpha6 GABA A Alpha6Beta1Gamma2 GABA A Alpha6Beta2Gamma2 GABA A Alpha6Beta3Gamma2 GABA A anti-Alpha1 GABA A anti-Alpha3 GABA A Benzodiazepine GABA A Benzodiazepine brain GABA A Benzodiazepine liver GABA A Benzodiazepine omega1 GABA A Benzodiazepine omega2 GABA A Benzodiazepine omega5 GABA A Benzodiazepine Type I GABA A Benzodiazepine Type II GABA A Benzodiazepine Type IIL GABA A Benzodiazepine Type IIM GABA A Beta2Gamma2 GABA B GABA B rho 1 GABA C GABA receptor alpha-1 subunit GABA receptor alpha-2 subunit GABA receptor alpha-3 subunit GABA receptor alpha-5 subunit GABA uptake GABA, Chloride, TBOB GABA-PICROTOXIN GALANIN Galanin R1 Galanin R2 Galanin R3 Gamma hydroxybutyric, GHB Gardner-Rasheed feline sarcoma viral (v-fgr) oncogene homolog Gastrin-Releasing peptide glucagon Glucocorticoid Glucocorticoid receptor GLUK5 GluR1 -40 mV GluR1 -80 mV Glutamate AMPA 1 Glutamate AMPA 2 Glutamate AMPA 3 Glutamate AMPA 4 Glutamate AMPA 5 Glutamate AMPA 6 Glutamate Chloride Glutamate delta 2 Glutamate, GluR1 Glutamate-AMPA Glutamate-AMPA, GluR3 Glutamate-KA Glutamate-Kainate Glutamate-Kainate 2 Glutamate-Kainate 4 Glutamate-Kainate 5 Glutamate-Kainate 7 Glutamate-Kainate EAA1 Glutamate-Kainate, GluR5 Glutamate-Kainate, GluR6 Glutamate-NMDA Glutamate-NMDA-Channel Glutamate-NMDA-Glycine Glutamate-NMDA-MK801 Glutamate-NMDA-Polyamine Glutamic acid decarboxylase Glutamine synthetase Glutaminyl cyclase Glycine Glycine, non-strychnine Glycine, strychnine Glycine-1-transporter Glycine-2-transporter Glycogen Synthase Kinase 3 Glycogen synthase kinase 3 Gonadotropin-Releasing Hormone, GnRH-R GPR103 GPR109B GPR7 GR Alkaline Fosfatase Grb2-SH2 Growth Hormone GSK-3 Hemopoietic cell kinase Heptyrosine aminotransferase, HepTAT HER1 HER2 HERG HISTAMINE H1 HISTAMINE H2 Histamine H2-Gs alpha S HISTAMINE H3 Histamine H3L HISTAMINE H4 IGF-IR IKK Imidazoline I1 Imidazoline I2 imipramine Inositol Triphosphate Inositol Trisphosphate 1 Inositol Trisphosphate 4 Inositol Trisphosphate 5 Insulin insulin kinase-beta Insulin receptor Interleukin Interleukin 1-Alpha Interleukin 1-beta Itk JAK3 Janus kinase 1 (a protein tyrosine kinase) Janus kinase 2 (a protein tyrosine kinase) KDR KHEYLRF-NH2 (AF2) Kinase insert domain receptor (a type III receptor tyrosine kinase) Kinase insert domain(KDR) Lck Leukotriene 2 Leukotriene b1 Leukotriene B4 Leukotriene B4 R1 Leukotriene B4 R2 Leukotriene Cysteinyl 1 Leukotriene Cysteinyl 2 Leukotriene D4 Leukotriene D4 Alpha Leukotriene D4 Beta LIM domain kinase 1 Liver X, LXR alpha Liver X, LXR beta Luteinizing Hormone-Releasing Hormone LHRH Lymphocyte-specific protein tyrosine kinase Lysophosphatidic Acid 1 Lysophosphatidic Acid 2 Lysophosphatidic Acid 3 m-AChR M1 M2 M3 M4 M5 malonyl-CoA decarboxylase, MCD MAO A MAO B MAP kinase MAP kinase interacting serine/threonine kinase 2 Map Kinase P38 Alpha MAP Kinase P38 Beta MAP Kinase P38 Delta MAP Kinase P38 Gamma MAP/microtubule affinity-regulating kinase 2 Matrix Metalloproteinase, MMP-1 Matrix Metalloproteinase, MMP-13 Matrix Metalloproteinase, MMP-2 Matrix Metalloproteinase, MMP-3 Matrix Metalloproteinase, MMP-8 Matrix Metalloproteinase, MMP-9 Matrix Metalloproteinase, MPP-2 Matrix Metalloproteinase, MPP-9 MEK Melanin Concentrating Hormone 1 Melanin Concentrating Hormone 2 Melanocortin MC1 Melanocortin MC3 Melanocortin MC4 Melanocortin MC5 Melatonin Melatonin 1A Melatonin 1B Melatonin 1C Met Met proto-oncogene (hepatocyte growth factor receptor) metabotropic glutamate 1 metabotropic glutamate 1/2 metabotropic glutamate 1/5-D metabotropic glutamate 1/DA Metabotropic Glutamate 1a metabotropic glutamate 1b metabotropic glutamate 1c metabotropic glutamate 2 metabotropic glutamate 2/1 metabotropic glutamate 2/3 metabotropic glutamate 3 metabotropic glutamate 3/1a metabotropic glutamate 3/1c metabotropic glutamate 4 metabotropic glutamate 4/1-F metabotropic glutamate 4a metabotropic glutamate 5 metabotropic glutamate 5/1-C metabotropic glutamate 5/1-F metabotropic glutamate 5a metabotropic glutamate 5b metabotropic glutamate 6 metabotropic glutamate 7 metabotropic glutamate 8 Methionine Aminopeptidase, ecMetAP mineralocorticoid Mineralocorticoid receptor Mitegen-Activated Protein Kinase Kinase Mitogen-activated protein kinase 10 Mitogen-activated protein kinase 11 Mitogen-activated protein kinase 12 Mitogen-activated protein kinase 8 Mitogen-activated protein kinase 9 Mitogen-activated protein kinase kinase kinase 4 Mitogen-activated protein kinase kinase kinase 5 Mitogen-activated protein kinase kinase kinase kinase 5 Mixed Lineage Kinase-7, MLK-7K MK2 Monoamine Oxidase A Monoamine Oxidase B Motilin Multidrug Resistance Transporter MDR 1 Myosin light chain kinase 2, skeletal muscle n-AChR N-Methyl-D-Aspartate NET Neurokinin NK1 Neurokinin NK2 Neurokinin NK3 Neuromedin B Neuronal acetylcholine receptor protein alpha-3 subunit Neuronal acetylcholine receptor protein alpha-4 subunit Neuronal acetylcholine receptor protein alpha-7 subunit Neuropeptide Y Neuropeptide Y1 Neuropeptide Y2 Neurotensin Neurotensin 1 Neurotensin 2 Neurotrophic tyrosine kinase, receptor, type 1 Neurotrophic tyrosine kinase, receptor, type 2 NGF Nicotinic Alpha-Bungarotoxin nicotinic central Nicotinic neuronal, alpha-BGTX-insensitive NIH 3T3 NIMA (never in mitosis gene a)- related kinase 9 NIMA (never in mitosis gene a)-related kinase 2 NIMA (never in mitosis gene a)-related kinase 6 Nischarin Nitric-oxide synthase, NOS (constitutive ) Nitric-oxide synthase, NOS (inducible) Nitrogen oxide synthase - neuronal NMB NMDA NMDA PCP SITE Nociceptin receptor Nociceptin/Orphanin FQ, NOP receptor Non-receptor tyrosine kinase Tyk2 Noradrenaline Uptake Norepinephrine transporter Norepinephrine transporter Norepinephrine Uptake NOS NOS neuronal NPFF NPFF2 NPY-Y1 NPY-Y2 NPY-Y4 NPY-Y5 NR2B NR2B Channel Blocker NRI NT OPIATE Delta Opiate Delta 1 OPIATE Kappa Opiate Kappa 1 OPIATE Kappa 3 OPIATE Mu OPIATE Mu 2 Opiate non-selective OPIATE ORL-1 OPIATE Sigma OPIOID Delta OPIOID Kappa OPIOID Kappa 3 OPIOID Mu OPIOID Mu 2 OPIOID Sigma Organic Anion Transporter OATP1B3 ouabain Oxytocin P21 (CDKN1A)-activated kinase 3 P21 (CDKN1A)-activated kinase 6 P21(CDKN1A)-activated kinase 4 P21(CDKN1A)-activated kinase 7 P21/Cdc42/Rac1-activated kinase 1 (STE20 homolog, yeast) P38 mitogen activated protein kinase p3TP-Lux PACAP PACAP-27 PACAP-38 PAF Platelet activating factor papain PAR2 PARATHYROID HT1 PARATHYROID HT2 PBR PCTAIRE protein kinase 1 PDGF PDGF-Rbeta PGD2 phencyclidine Phenylethanolamine-N-methyl transferase, PNMT Phenylethanolamine-N-methyl transferase, PNMT-3 Phorbol ester Phosphatidylcholine specific phospholipase C, PC-PLC Phosphodiesterase 1 Phosphodiesterase 3 Phosphodiesterase 4 Phosphodiesterase 5 Phosphoinositide specific phospholipase C, PI-PLC Phosphorylase kinase, gamma 1 (muscle) Phosphorylase kinase, gamma 2 (testis) Pim-1 oncogene Pim-2 oncogene PKA PKC alpha PKC beta PKC gamma PKC-alpha PKC-beta2 Plasmepsin I Plasmepsin II Platelet-derived growth factor receptor, alpha polypeptid Platelet-derived growth factor receptor, beta polypeptide Polyamine Transporter Potassium (voltage dependent) Potassium Channel Potassium channel (ATP modulatory) Potassium Channel (Ca2+ dependent) Potassium channel, Apamin Potassium Channel, Ca2+ Act., VI Potassium Channel, Ca2+ Act., VS PPAR-delta Pregnane X receptor progesterone Progesterone receptor Prolactin Releasing Peptide Receptor Prostaglandin D Prostaglandin D2 Prostaglandin E1 Prostaglandin E2 Prostaglandin E3 Prostaglandin E4 Prostaglandin EP1 Prostaglandin EP2 Prostaglandin EP3 Prostaglandin EP4 Prostaglandin F Prostaglandin H2 Prostaglandin I Prostaglandin I2 Prostaglandin Transporter ProstaglandinF2Alpha Proteasome Protein Kinase Protein kinase C Protein Kinase C- alpha Protein Kinase C- delta Protein Kinase D-GST Protein Kinase G Protein kinase, AMP-activated, alpha 1 catalytic subunit Protein kinase, cAMP-dependent, catalytic, alpha Protein kinase, membrane associated tyrosine/threonine 1 Protein-tyrosine kinase Tie2 Proteinase-Activated Receptor 2 PrRP PTK2 protein tyrosine kinase 2 PTK6 protein tyrosine kinase 6 Purinergic, P2X Purinergic, P2X1 Purinergic, P2X2 Purinergic, P2X3 Purinergic, P2X4 Purinergic, P2X7 Purinergic, P2Y PurinergicP2X2/3 Raf Receptor-interacting serine-threonine kinase 2 Ret proto-oncogene Rho Kinase Ribosomal protein S6 kinase, 90kDa, polypeptide 2 Ribosomal protein S6 kinase, 90kDa, polypeptide 3 Ribosomal protein S6 kinase, 90kDa, polypeptide 5 S643b Serine/threonine kinase 10 Serine/threonine kinase 16 Serine/threonine kinase 17a (apoptosis-inducing) Serine/threonine kinase 17b (apoptosis-inducing) Serine/threonine kinase 18 Serine/threonine kinase 3 mouse Serine/threonine kinase 36 (fused homolog, Drosophila) Serine/threonine kinase 38 like Serine/threonine kinase 4 Serine/threonine kinase 6 Serotonin Serum/glucocorticoid regulated kinase Sigma Sigma 2 receptor Sigma opioid receptor Sigma-1 Sigma-2 Signal transducer and activator of transcription 3,Stat3 SLC-1 Small conductance calcium-activated potassium channel protein 3 Sodium (Site 1) Sodium (Site 2) Sodium Channel SOMATOSTATIN SOMATOSTATIN SST1 SOMATOSTATIN SST2 SOMATOSTATIN SST3 SOMATOSTATIN SST4 SOMATOSTATIN SST5 sphingosine-1-phosphate 1 S1P1 sphingosine-1-phosphate 3 S1P3 sphingosine-1-phosphate 4 S1P4 sphingosine-1-phosphate 5 S1P5 Spleen tyrosine kinase Src Kinase STE20-like kinase (yeast) Substance K Substance P Syk Synaptic vesicular amine transporter TA1 tachykinin TBPS TEK tyrosine kinase, endothelial (venous malformations, multiple cutaneous and mucosal) Testosterone TG 1019 Thrombin Thrombin FIIa Thrombin FXa Thrombin trypsin Thromboxane Thromboxane A2 Thromboxane Alpha Thromboxane B2 Thromboxane Beta Thromboxane prostanoid Thymidylate Synthase thyroid alpha thyroid beta Thyrotropin-releasing Hormone thyrotropin-releasing hormone R1 thyrotropin-releasing hormone R2 thyrotropin-releasing hormone R3 TNF-alpha TRAF2 and NCK interacting kinase Transforming Growth Factor Beta RIIK Transforming Growth Factor Beta RIK TRH Tripeptidyl Peptidase TPP II TSPO TTK protein kinase Tumor Necrosis Factor alpha TXA2/PGH2 Tyrosine kinase receptor ron Urotensin-II V-abl Abelson murine leukemia viral oncogene homolog V-abl Abelson murine leukemia viral oncogene homolog 1 V-abl Abelson murine leukemia viral oncogene homolog 1 (E255K) V-abl Abelson murine leukemia viral oncogene homolog 1 (H396P) V-abl Abelson murine leukemia viral oncogene homolog 1 (M351T) V-abl Abelson murine leukemia viral oncogene homolog 1 (Q252H) V-abl Abelson murine leukemia viral oncogene homolog 1 (T3151) V-abl Abelson murine leukemia viral oncogene homolog 1 (Y253F) V-abl Abelson murine leukemia viral oncogene homolog 2 V-erb-b2 erythroblastic leukemia viral oncogene homolog 2 V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog (avian) V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian) V-yes-1 Yamaguchi sarcoma viral oncogene homolog 1 V-yes-1 Yamaguchi sarcoma viral related oncogene homolog V1 Vanilloid receptor Vanilloid VR1 VASOPRESSIN V1 VASOPRESSIN V1A VASOPRESSIN V1B VASOPRESSIN V2 Vasopressin V3 VEGF-R2 VIP VIP 1 VIP 2 Vitamin D, VDR VMAT1 VMAT2 Y1 Y2 Y4 Y5 Zacopride site-R Zeta-chain (TCR) associated protein kinase 70kDa

Receptor List:

Configure Compounds:

1-(5-Chloropyridin-2-yl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(Aminomethyl)dibenzo[b,e]bicyclo[2.2.2]octadiene Hydrochloride 9-Aminomethyl-10,10-dimethyl-9,10-dihydroanthracene Oxalate 9-Aminomethyl-9,10-dihydro-9,10-methanoanthracene Hydrochloride 9-Methyl-9-aminomethyl-9,10-dihydroanthracene Oxalate α-Methylalanyl-L-proline butylamide hydrochloride hemihydrate ((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methanamine ((RS)-alpha-M4CPG) (+)(R)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+)(R)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+)-(1R,3'R)-Quinuclidin-3'-yl 1-(3-Thienyl)1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monooxalate (+)-(1S,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (+)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (+)-(3'R)-Quinuclidin-3'-yl 1-Benzyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (+)-(R)-4-Methyl-1-[2-(4-chlorophenoxy)-1-methyl-ethyl]piperidine hydrochloride (+)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-2-methyl-propyl]piperidine hydrochloride (+)-(S)-4-Methyl-1-[2-(4-chlorophenoxy)-propyl]piperidine hydrochloride (+)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-1-methyl-propyl]piperidine hydrochloride (+)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-butyl]piperidine hydrochloride (+)-1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (+)-1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (+)-1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine (+)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide (+)-1-[(1R)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride (+)-1-[(1S)-1-(3-Chlorophenyl)-2-(dimethylamino)ethyl]cyclohexanol (+)-1-[(1S)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride (+)-1-[(1S,2R,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (+)-1-[(1S,2S,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (+)-1-{(1R)-2-(4-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride (+)-1-{(1S)-2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride (+)-1-{(1S,2R,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (+)-1-{(1S,2S,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (+)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (+)-3-(4-Chlorophenyl)-N'-[(4-cyanophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (+)-3-(4-Chlorophenyl)-N'-[(4-iodophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (+)-6-chloro-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (+)-6-fluorodinapsoline hydrobromide (+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazo... (+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazo... (+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole (+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole (+)-8-hydroxy-2-(di-n-propylamino)tetralin (+)-alpha-Methylphenylethylamine (+)-Methyl(1S,2R,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (+)-t-ADA (+)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine (+)-trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione (+)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine (+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol (+-)-MCPG (+/-) BMY-14802 (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid (+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]... (+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol (+/-)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+/-)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+/-)-11-chlorodinapsoline hydrobromide (+/-)-11-nitrodinapsoline hydrobromide (+/-)-2,3-Dimethyldinapsoline hydrobromide (+/-)-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (+/-)-2-methyldinapsoline hydrobromide (+/-)-2-propyldinapsoline hydrobromide (+/-)-3-Ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxylic Acid (+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide (+/-)-3-Fluoromethyl-7-(N-2,2,2-trifluoroethylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-3,3,3-trifluoropropylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-3-methoxypropylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-ethylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-propylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-thiomorpholinoaminosulfonyl)-THIQ (+/-)-3-Methyl-1,2,3,4-tetrahydroisoquinoline (+/-)-3-methyldinapsoline hydrobromide (+/-)-3-n-butyldinapsoline hydrobromide (+/-)-3-perfluorobutyldinapsoline hydrobromide (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(1-cyclopropylethyl)pyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(1-methylcyclopropyl)pyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(cyclopropylmethyl)pyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-tert-butylpyrimidin-2-amine (+/-)-7,7'-dimethyldinapsoline hydrobromide (+/-)-7-Bromo-9,10-dihydro-9-(4-ethylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Bromo-9,10-dihydro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Bromo-9,10-dihydro-9-[4-(2'-hydroxy)ethylpiperazin-1-yl]pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9,10-dihydro-9-(4-ethylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9,10-dihydro-9-(4-methylhexahydro-1H-1,4-diazepin-1-yl)pyrrolo-[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9,10-dihydro-9-[4-(2'-hydroxy)ethylpiperazin-1-yl]pyrrolo-[2,1-b][1,3]benzothiazepine (+/-)-7-chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-ethyldinapsoline hydrobromide (+/-)-7-methoxycarbonylmethyldinapsoline (+/-)-7-methyldinapsoline hydrobromide (+/-)-8-hydroxy-2-(di-n-propylamino)tetralin (+/-)-9,10-Dihydro-7-fluoro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-9,10-Dihydro-7-fluoro-9-[4-(2'-hydroxy)ethylpiperazin-1-yl]pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-9,10-Dihydro-9-(4-ethylpiperazin-1-yl)-7-fluoropyrrolo[2,1-b][1,3]benzothiazepine (+/-)-AP5 (+/-)-BMY-1402 (+/-)-cis-1-Phenyl-3-(trimethylammoniumyl)-1,2,3,4-tetrahydronaphthalene Iodide (+/-)-Methyl 5-[({trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazin-1-yl}carbonyl)amino]pyridine-2-carboxylat... (+/-)-N-(4-(2-(Dimethylamino)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide monohydrochloride (+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride (+/-)-o-chloro-trans-H2-PAT (+/-)-o-methyl-trans-H2-PAT (+/-)-p-chloro-trans-H2-PAT (+/-)-p-fluoro-trans-H2-PAT (+/-)-p-methyl-trans-H2-PAT (+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahydrobenzo[a]phenanthridine (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(1-oxidopyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(2-methylpyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(4-methylpyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(5-methylpyridin-3-yl)piperazine-1-carboxamide hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(6-methylpyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-2-ylpiperazine-1-carboxamide Hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-3-ylpiperazine-1-carboxamide Hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-4-ylpiperazine-1-carboxamide Hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-2-ylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-4-ylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-5-ylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(methylthio)pyridin-3-yl]piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(2-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(4-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide Hydrochlorid... (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(5-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(6-hydroxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(6-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-ACPD (+/-)-trans-N-(2-Hydroxycyclopropyl)palmitamide (+/-)-trans-N-(6-Acetylpyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-N-(6-Aminopyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-N-(6-Chloropyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-N-(6-Cyanopyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+_)-erythro-2-(1-Methylpiperidin-2-yl)-Chroman (+_)-erythro-5-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)-erythro-6-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)-erythro-7-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)-erythro-7-Hydroxy-2-(1-methylpyrrolidin-2-yl)chroman (+_)-erythro-8-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-2-(1-Methylpiperidin-2-yl)-Chroman (+_)threo-5-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-6-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-7-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-7-Hydroxy-2-(1-methylpyrrolidin-2-yl)chroman (+_)threo-8-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (-)(S)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (-)(S)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (-)-(1S,3'R)-Quinuclidin-3'-yl 1-(3-Thienyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Mono-(-)-tartrate (-)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (-)-(2S,5R)-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]piperazine-1-carboxamide (-)-(3'R)-Quinuclidin-3'-yl 1-Benzyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (-)-(R)-4-Methyl-1-[2-(4-chlorophenoxy)-propyl]piperidine hydrochloride (-)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-1-methyl-propyl]piperidine hydrochloride (-)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-butyl]piperidine hydrochloride (-)-(S)-4-Methyl-1-[2-(4-chlorophenoxy)-1-methyl-ethyl]piperidine hydrochloride (-)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-2-methyl-propyl]piperidine hydrochloride (-)-1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (-)-1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (-)-1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine (-)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide (-)-1-[(1R)-1-(3-Chlorophenyl)-2-(dimethylamino)ethyl]cyclohexanol (-)-1-[(1R)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride (-)-1-[(1R,2R,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (-)-1-[(1R,2S,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo-[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (-)-1-[(1S)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride (-)-1-{(1R)-2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride (-)-1-{(1R,2R,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (-)-1-{(1R,2S,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (-)-1-{(1S)-2-(4-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride (-)-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (-)-2-aminoadipic acid (-)-3-(4-Chlorophenyl)-N'-[(4-cyanophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (-)-3-(4-Chlorophenyl)-N'-[(4-iodophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide (-)-3-{(Cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)-1-methylpropyl]amino}-8-fluorochromane-5-carboxamide (-)-3-{Cyclobutyl[3-(5,7-difluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide (-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane- (-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-propylpyrimidin-2-amine (-)-6-fluorodinapsoline hydrobromide (-)-7,9-difluoro-5-(6-methyl-7-oxa-bicyclo[4.1.0]hept-2-yl)-2,2,4-trimethyl 2,5-dihydro-(1H)-6-oxa-1-aza-chrysen (-)-8-hydroxy-2-(di-n-propylamino)tetralin (-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol (-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)-Indolactam V (-)-Indolactam V (low PS) (-)-Methyl(1R,2S,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (-)-NANM (-)-Octylindolactam V (-)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine (-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone (-)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine (-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol (-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (1'RS)-(2S)-2-Amino-4-[(1'-aminoethyl)(hydroxy)phosphinyl]butyric Acid (1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-ylcarbamoyl)(phenyl)methyl acetate (1,2,3,4-Tetrahydro-acridin-9-yl)-[8-(1,2,3,4-tetrahydro-acridin-9-ylsulfanyl)-octyl]-amine (1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-carbamic acid benzyl ester (1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-yl)methanol (1-Benzenesulfonyl-5-fluoro-2-methyl-1H-indol-3-yl)-acetic acid (1-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (14-dimethylaminomethyl-6H,13H-pyrazino[1,2-a;4,5-a']diindol-7-ylmethyl)-dimethyl-amine (14S)-14-Hydroxydihydromorphinone (15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide (15R)-8-cyano-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxami... (15S)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide (15S)-8-cyano-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxami... (1H-Benzimidazol-2-yl)-thiazol-2-yl-amin (1H-Indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (1H-Indol-2-yl)-(4-phenethyl-piperazin-1-yl)-methanone (1H-Indol-2-yl)-(piperazin-1-yl)-methanone (1R)-benzo[b]thiophen-3-yl((4aR)-1-(4-fluorophenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl)methanol (1R,13S,14R)-24-(cyclopropylmethyl)-13,20-dihydroxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa... (1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 (1R,2R,3R,4R,5S,7R,9S,10R)-1-Benzoyloxy-9-cinnamoyloxy-2,3-diacetoxy-dihydro-beta-agarofuran (1R,2R,3R,4R,5S,7R,9S,10R)-1-Benzoyloxy-9-cinnamoyloxy-2,3-dihydroxy-dihydro-beta-agarofuran (1R,2R,3R,4R,5S,7R,9S,10R)-2-Acetoxy-1-benzoyloxy-9-cinnamoyloxy-3-hydroxy-dihydro-beta-agarofuran (1R,2R,3R,4R,5S,7R,9S,10R)-3-Acetoxy-1-benzoyloxy-9-cinnamoyloxy-2-hydroxy-dihydro-beta-agarofuran (1R,2R,3S,4S,5S,6R,7R,9S,10S)-1-Benzoyloxy-4-hydroxy-2,3,6,9,15-pentaacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1R,2R,4S)-2-(6-chloro-5-(3-methoxyphenyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane (1R,2R,4S)-2-(6-chloro-5-(4-fluorophenyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane (1R,2R,4S)-2-(6-chloro-5-phenylpyridin-3-yl)-7-azabicyclo[2.2.1]heptane (1R,2R,5S )-6-benzyl-2-benzyloxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane (1R,2R,5S )-6-benzyl-2-methoxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane (1R,2R,5S )-6-benzyl-8-(2-phenylethyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol (1R,2R,5S )-6-benzyl-8-methyl-6,8-diazabicyclo[3.2.2]nonan-2-ol (1R,2R,5S)-methyl 8-(2-(3,4-dichlorophenyl)acetyl)-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (1R,2S)-2-(tert-butylamino)-1-phenylpropan-1-ol (1R,2S)-N-Arachidonoylcyclopropanolamide (1R,2S)-N-Oleoylcyclopropanolamide (1R,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1R,2S,4R,5S,6R,7R,8S,9R,10S)-8,9-Dibenzoyloxy-1,2,6,15-tetraacetoxy-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-1,2,6,9,15-pentaacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-1,9-Dibenzoyloxy-2,6,15-triacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-9-Benzoyloxy-1,2,6,15-tetraacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-9-Benzoyloxy-1-hydroxy-2,6,15-triacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4S,5S) Acetic Acid 4-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonooxy-bicyclo[3.1.0]hex-1-ylmethyl Ester (1R,2S,4S,5S) Acetic Acid 4-(2-chloro-6-methylamino-purin-9-yl)-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl Ester (1R,2S,4S,5S) Phosphoric Acid mono-[4-(2-chloro-6-methylamino-purin-9-yl)-1-hydroxymethyl-bicyclo-[3.1.0] hex-2-yl] Ester (1R,2S,4S,5S) Phosphoric Acid mono-[4-(2-chloro-6-methylamino-purin-9-yl)-2-hydroxy-bicyclo[3.1.0]hex-1-ylmethyl] Ester (1R,2S,4S,5S,6R,7R,8S,9R,10R)-6-Acetoxy-4,8-dihydroxy-1,2,9-tribenzoyloxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,8S,9R,10S)-2,6-Diacetoxy-4-hydroxy,1,8,9-tribenzoyloxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,8S,9R,10S)-8,9-Dibenzoyloxy-4,15-dihydroxy-1,2,6-triacetoxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,8S,9R,10S)-8,9-Dibenzoyloxy-4-hydroxy-1,2,6,15-tetraacetoxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,9S,10S)-2,15-Diacetoxy-1,9-dibenzoyloxy-4,6-dihydroxy-8-oxo-dihydro-beta-agarofuran (1R,2S,5S )-6-Benzyl-8-(2-phenylethyl)-6,8-diazabidiazabicyclo (1R,2S,5S )-6-Benzyl-8-methyl-6,8-diazabicyclo-[3.2.2]nonan-2-ol (1R,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (1R,3'S)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (1R,3S)-1-(Aminomethyl)-3,4-dihydro-5,6-dihydroxy-3-phenyl-1H-2-benzopyran Hydrochloride (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid (1R,4R)-2-(2,5-diazabicyclo[2.2.1]hept-2-yl)-thieno[3,2-b]pyridine (1R,4R)-2-(3-methyl-(1,2,4)-thiadiazol-5-yl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(3-pyridinylmethyl)-2,5-diazabicyclo[2.2.1]-heptane (1R,4R)-2-(5,6-dichloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1R,4R)-2-(5-bromo-6-chloropyridine-3-sulfonyl)-2,5-diazabicyclo[2.2.1]heptane (1R,4R)-2-(5-trifluoromethyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-chloro-5-methoxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-chloro-5-methyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-chloropyridine-3-carbonyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1R,4R)-3-(2,5-diazabicyclo[2.2.1]hept-2-yl)-thieno[3,2-b]pyridine (1R,5S )-6-benzyl-8-methyl-6,8-diazabicyclo[3.2.2]-nonane-2-one dimethyl acetal (1R,9R,10S)-4-carbamoyl-17-(cyclopropylmethyl)-3,10-dihydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptad... (1R,9R,10S,13R)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-... (1R,9R,10S,13S)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-... (1R,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-15-(prop-2-en-1-yl)-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5... (1R,9R,18S,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^{1,32}.0^{2,7}.... (1RS,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate (1RS,3'R)-Quinuclidin-3'-yl 1-Phenylisoindoline-2-carboxylate (1S)-1-((4aR)-1-(4-fluorophenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl)but-3-en-1-ol (1S,11S,13S,17R,18R,20R,27S,29R,30R,31S,35E)-14,26-bis(cyclohex-2-en-1-yl)-35-(2-hydroxyethylidene)-19-phenyl-21-oxa-8,14,19,... (1S,11S,13S,17R,18R,20R,27S,29R,30R,31S,35E)-14,26-bis[(3,4-dimethoxyphenyl)methyl]-35-(2-hydroxyethylidene)-19-phenyl-21-oxa... (1S,11S,13S,17R,18R,20R,27S,29R,30R,31S,35E)-35-(2-hydroxyethylidene)-14,26-dimethyl-19-phenyl-21-oxa-8,14,19,26-tetraazadeca... (1S,11S,13S,18R,20R,27S,29R,30R,31S,35E)-35-(2-hydroxyethylidene)-14,26-bis[(4-nitrophenyl)methyl]-19-phenyl-21-oxa-8,14,19,2... (1S,2R)-1-(3-methyl-1H-indol-1-yl)-3-(methylamino)-1-phenylpropan-2-ol (1S,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1S,2R,6S,14R,15S,16R)-3-(cyclopropylmethyl)-16-[(2R)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-3-azahexacyclo[13.2... (1S,2S)-1-[(R)-2-[4-(2,4-Dimethylphenyl)piperazyl]-ethyl]-2-methyl-2-phenylcyclopropane (1S,2S)-1-[(S)-2-[4-(2,4-Dimethylphenyl)piperazyl]-ethyl]-2-methyl-2-phenylcyclopropane (1S,2S)-1-[4-(2,4-Dimethylphenyl)piperazyl]methyl-2-methyl-2-phenylcyclopropane (1S,2S)-N-Arachidonoylcyclopropanolamide (1S,2S)-N-Oleoylcyclopropanolamide (1S,2S,13R,21R)-22-(cyclopropylmethyl)-2-hydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{1... (1S,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1S,2S,5R)-methyl 8-(2-(3,4-dichlorophenyl)acetyl)-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (1S,2S,5R,6S)-2-[(2'S)-(2'-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylicAcid (1S,2S,7S,8R,12S,20R,24R,32R)-9,33-bis(cyclopropylmethyl)-2,7-dihydroxy-19,25-dioxa-9,22,33-triazaundecacyclo[24.9.1.1^{8,14}... (1S,3'S)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (1S,3R)-1-aminocyclopentane-1,3-dicarboxylic (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid (1S,4S)-2-(2-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(2-quinolinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(2-thiazolyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-methylisothiazol-5-yl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(3-nitrophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-pyridazinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-quinolinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(4-chloro-1-phthalazinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(4-nitrophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(4-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(5-aminocarbonyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(5-aminomethyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(5-cyano-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(5-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(5-pyrimidinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-1,3-pyrimidin-4-yl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-3-pyridinyl)-5,5-dimethyl-2,5-diazabicyclo-[2.2.1]heptanium iodide (1S,4S)-2-(6-chloro-3-pyridinyl)-5-ethyl-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-3-pyridinyl)-5-methyl-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(6-chloro-5-hydroxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(6-chloro-5-methyl-3-pyridazinyl)-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(6-chloropyridin-3-yl)-2,5-diazabicyclo[2.2.1]-heptanone (1S,4S)-2-(6-fluoro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-methyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-nitro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(phenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-[5-hydroxy-3-pyridinyl]-2,5-diazabicyclo[2.2.1]-heptane (1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,... (1S,5R,13R,14S,17S)-4-(cyclobutylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(1... (1S,5R,13R,14S,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,... (1S,5R,13R,17R)-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxa... (1S,5R,13R,17S)-10-carbamoyl-4-(cyclopropylmethyl)-17-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.... (1S,5R,13R,17S)-17-hydroxy-14-oxo-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13S,14S,17R)-14-hydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)... (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-... (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octad... (1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide (1S,9R,10S)-17-(cyclobutylmethyl)-10-hydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-triene-4-carboxamide (1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxa... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis(cyclohex-2-en-1-yl)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundeca... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis(naphthalen-2-ylmethyl)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaund... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(2E)-but-2-en-1-yl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundeca... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(3,4-dimethoxyphenyl)methyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetra... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(4-bromophenyl)methyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaund... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(4-nitrophenyl)methyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaund... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[2-(acetyloxy)ethyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundeca... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-dibenzyl-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-dimethyl-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-15,31-bis(prop-2-en-1-yl)-10,26-dioxa-8,15,24,31-tetraazaundecacycl... (2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(4,4-difluoropiperidin-1-yl)methanone (2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2,2-diphenyl-[1,3]dioxolo[4,5-c]pyridin-6-yl)-piperidin-1-ylmethanone (2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2-(2,4-dichlorophenyl)-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2-(2,4-dichlorophenyl)-6-fluoro-2-(2-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2-(2,4-dichlorophenyl)-6-fluoro-2-(4-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2-(2-chloro-4-fluorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3,4-dichlorophenoxy)-5-(4-(4-fluoropiperidin-1-yl)but-1-ynyl)phenyl)-N-methylmethanamine (2-(3,4-dichlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3,4-dichlorophenoxy)-5-(4-thiomorpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3-chlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3-fluorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(4-chloro-3-(trifluoromethyl)phenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(4-chlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(Methylamino)-4-phenylthiazol-5-yl)(phenyl)methanone (2-Aminoethyl)benzene (2-Bromo-5-(4-(((2,4-difluorobenzyl)(2-methyl-3-((methylsulfonyl)amino)phenyl)amino)methyl)phenoxy)phenoxy)acetic Acid (2-Chloro-5-{4-[((2,4-difluorobenzyl){2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic Acid (2-chloroethyl)(2-(methylsulfonyloxyethyl)amino)aminobenzyl-L-glutamic acid (23R, 25R)-DLAM-03I (23R, 25R)-DLAM-2P (23R, 25R)-DLAM-3P (23R, 25R)-DLAM-4P (23R, 25R)-DLAM-MPM (23R, 25S)-DLAM-03I (23R, 25S)-DLAM-2P (23R, 25S)-DLAM-3P (23R, 25S)-DLAM-4P (23R, 25S)-DLAM-MPM (23R,25R)-DLAM-1P (23R,25S)-DLAM-1P (23S, 25R)-DLAM-03I (23S, 25R)-DLAM-2P (23S, 25R)-DLAM-3P (23S, 25R)-DLAM-4P (23S, 25R)-DLAM-MPM (23S, 25S)-DLAM-03I (23S, 25S)-DLAM-1P (23S, 25S)-DLAM-2P (23S, 25S)-DLAM-3P (23S, 25S)-DLAM-4P (23S, 25S)-DLAM-MPM (23S,25R)-DLAM-1P (2E)-3-[6-(Acetylamino)-3-pyridinyl]-N-{2-[2,4-dichloro-3-({[2-methoxy-1-(2-methoxyethyl)-1H-benzimidazol-4-yl]oxy}methyl)met... (2E)-N-{2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(2-pyridinylmethoxy)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl}-3-{6-[(4-py... (2R,2'R))-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2R,2'R)-2-(1-methyl-2-pyrrolidinyl)-1,4-benzodioxane hydrochloride (2R,2'S)-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)-piperidine (2RS,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroquinoline-2-carboxylate (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-bromo-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-chloro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (2S)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}pyrrolidine-2-carboxamide (2S)-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)amino]-2-benzyl-3-oxopropanoyl}amino)p... (2S)-2-Amino-4-[(1'-aminoethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(2'-Aminoethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(2'-Carboxyethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(aminomethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(hydroxymethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]-3-phenylpropanoic acid bis(tetraflurobor... (2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]-3-phenylpropanoic acid bis(tetrafluorobor... (2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]propanoic acid bis(tetrafluoroborate) (2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]propanoic acid bis(tetrafluoroborate) (2S)-2-{[4-(6-Bromoquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-2-{[4-(6-Chloroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-2-{[4-(6-Fluoroquinolin-2-yl)-1,4-diazepan-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline (2S)-2-{[4-(6-Fluoroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-6-allyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol (2S)-8-Methyl-2-({4-[6-(trifluoromethoxy)quinolin-2-yl]piperazin-1-yl}methyl)-2,3-dihydro-[1,4]dioxino[2,3-f]quinoline (2S)-8-Methyl-2-[(4-quinolin-2-yl-1,4-diazepan-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]-quinoline (2S)-8-Methyl-2-[(4-quinolin-2-ylpiperazin-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-8-Methyl-2-{[(2R)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline (2S)-8-Methyl-2-{[(2S)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline (2S)-8-Methyl-2-{[4-(6-nitroquinolin-2-yl)piperazin-1-yl]-methyl}-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-Aminobutyryl-(2S)-azetidine carboxamide trifluoroacetate hydrate (2S)-Aminobutyryl-(2S)-indoline carboxylic acid ethylamide hydrogen oxalate hydrate (2S)-Aminobutyryl-(2S)-indoline carboxylic acid methylamide hydrogen oxalate hydrate (2S)-Aminobutyryl-(2S)-indoline carboxylic acid propylamide hydrogen oxalate hydrate (2S)-Aminobutyryl-(4S)-fluoro-L-proline n-Butylamide Trifluoroacetate (2S)-Aminobutyryl-(R)-pipecolinic acid amide trifluoroacetate (2S)-Aminobutyryl-(S)-nipecotamide hydrogen oxalate (2S)-Aminobutyryl-4-cis-benzyl-L-proline n-butylamide Hydrogen Oxalate (2S)-Aminobutyryl-4-thia-L-prolinamide trifluoroacetate hemihydrate (2S)-Aminobutyryl-L-pipecolinic acid n-butylamide trifluoroacetate (2S)-Aminobutyryl-L-prolinamide trifluoroacetate hemihydrate (2S)-Aminobutyryl-L-proline (R)-sec-butylamide hydrogen oxalate (2S)-Aminobutyryl-L-proline 3-methylthiopropylamide hydrogen oxalate hemihydrate (2S)-Aminobutyryl-L-proline isobutylamide trifluoroacetate (2S)-Aminobutyryl-L-proline n-butylamide hydrogen oxalate (2S)-Aminobutyryl-L-proline n-pentylamide hydrogen oxalate (2S)-Aminobutyryl-L-proline n-propylamide trifluoroacetate (2S)-Aminobutyryl-L-proline-(2S)-methylbutylamide hydrogen oxalate hemihydrate (2S, 1'S, 2'S)-2-(carboxycyclopropyl)glycine (2S,2'R-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2S,2'S)-2-(1-methyl-2-pyrrolidinyl)-1,4-benzodioxane hydrochloride (2S,2'S-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2S,3S,4R,5S)-5-(6-(cyclopentylamino)-9H-purin-8-yl)-3,4-dihydroxy-N-(1-(4-(N-(1-phenethylpiperidin-4-yl)propionamido)phenyl)... (2S,3S,4S,5R,6S)-6-(5-((R)-2-(5,6-diethyl-2,3-dihydro-1H-inden-2-ylamino)-1-hydroxyethyl)-2-oxo-1,2-dihydroquinolin-8-yloxy)-... (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamid... (2S,5R)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(piperidin-1-ylsulfonyl)piperidine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid (2S,6S,2R)-2-[6-(2-(1-Naphthalene)-sulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-(2-Naphthalene)-sulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-(2-Thiophen)-carboxyl-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-(2-Thiophene)-sulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Acetyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Anisoyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Benzoyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Benzylsulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Butylsulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Butyryloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Isobutyryloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Isopropylsulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Chloro-benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Fluoro-benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Nitro-benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Toluenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Propionyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Toluyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-bromo-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-chloro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (3'R)-Quinuclidin-3'-yl 1-(2-Thienyl)1,2,3,4-tetrahydroisoquinoline-2-carboxylate (3'R)-Quinuclidin-3'-yl 1-Cyclohexyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate (3'R,4RS)-Quinuclidin-3'-yl 4-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate (3,5-Dinitropyridin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (3-((2-(4,6-dimorpholino-1,3,5-triazin-2-yl)hydrazono)methyl)-1H-indol-1-yl)(p-tolyl)methanone (3-Amino-1(R,S)-ethylpropyl)methylphosphinic acid (3-Amino-1(R,S)-hydroxypropyl)methylphosphinic acid (3-Amino-2(R)-hydroxypropyl)methylphosphinic acid (3-Amino-2(R,S)-hydroxypropyl)(cyclohexylmethyl)phosphinic Acid Hydrochloride (3-Amino-2(R,S)-hydroxypropyl)(diethoxymethyl)phosphinic Acid (3-Amino-2(R,S)-hydroxypropyl)(difluoromethyl)phosphinic acid (3-Amino-2(R,S)-hydroxypropyl)benzylphosphinic Acid Hydrochloride (3-Amino-2(R,S)-hydroxypropyl)n-butylphosphinic Acid Hydrochloride (3-Amino-2(S)-hydroxypropyl)(1,1-diethoxymethyl)phosphinic Acid (3-Amino-2(S)-hydroxypropyl)methylphosphinic acid (3-Aminopropyl)(1(R,S)-hydroxybenzyl)phosphinic acid (3-Aminopropyl)(1,1-difluoro-n-butyl)phosphinic acid hydrochloride (3-Aminopropyl)(2-cyclohexylethyl)phosphinic acid hydrochloride (3-Aminopropyl)(2-phenylethyl)phosphinic acid (3-Aminopropyl)(2-pyridylmethyl)phosphinic acid (3-Aminopropyl)(3-N-phthalimido-2-(R,S)-hydroxypropyl)phosphinic Acid (3-Aminopropyl)(3-oxobutyl)phosphinic Acid (3-Aminopropyl)(cyclohexylmethyl)phosphinic acid (3-Aminopropyl)(hydroxymethyl)phosphinic acid (3-Aminopropyl)benzylphosphinic acid (3-Aminopropyl)isobutylphosphinic acid (3-Aminopropyl)methylphosphinic acid (3-Aminopropyl)phenylphosphinic acid (3-Aminopropyl)tert-butylphosphinic acid (3-Aminopropyl)[(R,S)-tetrahydrofuran-2-yl]phosphinic acid (3-Aminopropyl)[(R,S)-tetrahydropyran-2-yl]phosphinic acid (3-Aminopropyl)[(tetrahydropyran-2(R,S)-yl)ethyl]phosphinic acid (3-Aminopropyl)[[(R,S)-tetrahydropyran-2-yl]methyl]phosphinic acid (3-Ph-Pr6)His7,DAla11,DPro13,Psi13-14,Phe14-Bn(6-14) (3aR,5R,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3R)-(-)-3-((Cyclopropylmethyl){[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}amino)-8-fluorochromane-5-carboxamide (3R)-(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide (3R)-(-)-8-Fluoro-3-[{[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}(propyl)amino]chromane-5-carboxamide (3R)-(-)-8-Fluoro-3-{[(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl]amino}chromane-5-carboxamide (3R)-(-)-8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)-amino}-N-methylchromane-5-carboxamide (3R)-(-)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine (3R)-1,1-Dibutyl-3-(4,5-diphenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Dibutyl-3-(4-phenyl-1,3-thiazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline Hydrochloride (3R)-1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-1,2,3,4-tetrahydro[1]benzothieno[2,3-c]pyridine (3R)-1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Diethyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Dihexyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Dipentyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(2-Nitrophenyl)-3-(4-phenyl-1H-imidazol-2-y1)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(4-Dimethylaminophenyl)-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(4-Methoxyphenyl)-3-(4-phenyl-1H-imidazol-2-y1)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(n-Pentyl)-3-(4-Phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-Cyclohexyl-1-methyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-Cyclohexyl-3-(4-Phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline Fumarate (3R)-3-((3-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-8-azabicyclo[3.2.1]octan-8-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[... (3R)-3-(4-Phenyl-1H-imidazol-2-yl)-1-(4-pyridinyl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-3-(4-Phenyl-1H-imidazol-2-yl)spiro[Beta-carboline-1,2'-adamantyl] Dihydrochloride (3R)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide (3R)-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-3,4-dihydro-2H-chromen- (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dion... (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6a... (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-di... (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6... (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2... (3R,4S)-3-(benzofuran-2-ylmethyl)-4-(4-methoxyphenyl)-1-phenylazetidin-2-one (3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin-3-yl)propyl)azetidin-2-one (3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-N-isobutylpiperidine-3-carboxamide (3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-N-isobutylpiperidine-3-sulfonamide (3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-N-isopentylpiperidine-3-sulfonamide (3R,6S)-1-(4-chlorophenyl)-N-cyclobutyl-6-(2,4-dichlorophenyl)piperidine-3-carboxamide (3R,6S)-1-(4-chlorophenyl)-N-cyclohexyl-6-(2,4-dichlorophenyl)piperidine-3-carboxamide (3R,6S)-1-(4-chlorophenyl)-N-cyclohexyl-6-(2,4-dichlorophenyl)piperidine-3-sulfonamide (3R,6S)-N-(4-chlorobenzyl)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidine-3-carboxamide (3S)-(+)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine (3S)-1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (3S)-3-((2-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)ethylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (3S)-3-((2-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)ethylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one... (3S)-3-((3-( 6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-o... (3S)-3-({[2-({4-[amino(imino)methyl]benzyl}oxy)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}carbonyl}amino)-3-phenylpro... (3S)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide (3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-one (3S,4S)-5-(4-Bromobenzyloxy)-3-hydroxy-4-(2-thiophen-2-ylacetylamino)pentanoic Acid [(S)-1-((S)-1-Carbamoyl-3-methylbutylcarb... (3S,4S)-5-(4-Bromobenzyloxy)-4-(3,3-diphenylpropionylamino)-3-hydroxypentanoic Acid [(S)-1-((S)-1-Carbamoyl-3-methylbutylcarb... (3S,4S)-5-(4-Bromobenzyloxy)-4-diphenylacetylamino-3-hydroxypentanoic Acid [(S)-1-((S)-1-Carbamoyl-3-methylbutylcarbamoyl)eth... (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6a... (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine... (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',... (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione (4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxybenzofuran-2-yl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methan... (4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol (4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)(1-methyl-1H-pyrrol-2-yl)meth... (4-(Benzylamino)piperidin-1-yl)-(naphthalen-2-yl)methadone (4-(furan-2-yl)-2-(2-(thiophen-2-yl)ethylamino)thiazol-5-yl)(phenyl)methanone (4-(Methylsulfonyl)phenyl)(4-phenyl-2-(phenylamino)-thiazol-5-yl)methanone (4-benzhydrylpiperazin-1-yl)(cyclohexyl)methanone (4-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (4-Chlorophenyl)(2-(methylamino)-4-phenylthiazol-5-yl)methanone (4-Ethyl-piperazin-1-yl)-(1H-indol-2-yl)-methanone (4-Ethynyl-cyclohex-3-enyl)-dipropyl-amine (4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol (4-Methoxyphenyl)(2-(methylamino)-4-phenylthiazol-5-yl)methanone (4-Methoxyphenyl)(4-phenyl-2-(phenylamino)thiazol-5-yl)methanone (4-Nitrobenzyl)-6-thioguanosine (4-Phenyl-2-(phenylamino)thiazol-5-yl)(p-toluyl)methanone (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)imidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)imidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)imidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-imidazo[1,2-a]pyridine (4-{2-[4-(2,2-Dimethyl-[1,3]dioxan-5-ylmethoxy)phenyl]vinyl}phenyl)dimethylamine (4-{4-[(Benzyl{2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic Acid (4aR,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol (4aS,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol (4bS,7R,8aR)-4b-benzyl-7-hydroxy-7-(prop-1-ynyl)-N-(pyridin-4-ylmethyl)-4b,5,6,7,8,8a,9,10-octahydrophenanthrene-2-carboxamid... (4R)-3,4-Dihydrosalvinorin C (4R)-3,4-Dihydrosalvinorin E (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid (4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-10-(3-guanidinopropyl)-16-(4... (5,7- Dichloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5,7-Difluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5,7-Dimethyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-(4-(((2,4-Difluorobenzyl)(2-methyl-3-((methylsulfonyl)amino)phenyl)amino)methyl)phenoxy)-2-fluorophenoxy)acetic Acid (5-(4-(4-cyclopropylpiperazin-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-cyclopropylpiperazin-1-yl)butyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-fluoropiperidin-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-isopropyl-1,4-diazepan-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-isopropylpiperazin-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-isopropylpiperazin-1-yl)butyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-bromo-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-Bromopyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (5-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine (5-Fluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Hydroxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Methoxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate (5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate (5aR,6S)-1-(4-Fluorophenyl)-6-((S)-1-methoxy-1-(thiophen-2-yl)-ethyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinol... (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione (5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid (5R,2'R)-5-(1-methyl-2-pyrrolidinyl)oxazolidinone (5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid (5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5R,2'S)-5[1'-methylpyrrolidin-2'-yl]-1,3-oxazolidin-2-one (5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5S,2'S)-5-(1-methyl-2-pyrrolidinyl)oxazolidinone (5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (6-(4-((phenethylamino)methyl)phenoxy)pyridin-3-yl)(piperidin-1-yl)methanone (6-(methylsulfonyl)-1-pentyl-1H-indol-3-yl)(naphthalen-2-yl)methanone (6-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (6-bromo-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone (6-chloro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone (6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone (6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (6-fluoro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-ylmethanone (6-fluoro-2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (6-methyl-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone (6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one (6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride (6S,10bR)-6-(4-methoxyphenyl)-9-(3-(piperidin-1-yl)propoxy)-1,2,3,5,6,10b-hexahydropyrrolo[2,1-a]isoquinoline (6S,7S)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride (7-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (8R,9S,13S,14S,17S)-17-(2-(2-(2-hydroxyphenyl)-1H-indol-3-yl)ethynyl)-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclo... (8R,9S,13S,14S,17S)-17-(2-(2-(2-methoxyphenyl)-1H-indol-3-yl)ethynyl)-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclo... (9S,10R,11S,13S,14S,17R)-11,17-dihydroxy-17-(2-hydroxyacetyl)-10,13-dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-1H-c... (anthracen-9-ylmethyl)-3,3-triamine (anthracen-9-ylmethyl)-4,4-triamine (±)-7-Chloro-1-hydroxymethyl-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (±)-7-Chloro-1-methoxymethyl-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (±)-7-Chloro-9-[4-[2-(imidazolidin-2-on-1-yl)ethyl]piperazin-1-yl]-9,10-dihydro pyrrolo[2,1-b][1,3]benzothiazepine (±)-alpha-Methylbenzeneethanamine (C33H41N3O5Cl2·0.7F3CCO2H) C, H, N (C34H40N3O6Cl) C, H, N (C34H42N3O5Cl·2F3CCO2H) C, H, N (C34H46Cl2N6O8•1.5H2O), C, H, N (C34H46Cl2N6O8•3H2O), C, H, N (C34H46Cl2N6O8•H2O), C, H, N (C35H40N3O7Cl) C, H, N (C35H41N4O6Cl·1.3H2O) C, H, N (C35H48Cl2N6O8), C, H, N (C35H48Cl2N6O8•2.5H2O), C, H, N (C35H48Cl2N6O8•H2O), C, H, N (C37H52Cl2N6O8), C, H, N (C37H52Cl2N6O8•1.5H2O), C, H, N (C37H52Cl2N6O8•2.5H2O), C, H, N (C38H36N3O8Cl) C, H, N (C38H54Cl2N6O10•H2O), C, H, N (C40H41N3O8·0.5H2O) C, H, N (C41H49N3O7·0.9F3CCO2H) C, H, N (C42H51N3O7) C, H, N (C42H62Cl2N6O8•0.5H2O), C, H, N (C42H62Cl2N6O8•1.5H2O), C, H, N (C43H49N3O9·0.8H2O) C, H, N (C46H45N3O10) C, H, N (D-Ala(2),MePhe(4),Gly-ol(5))enkephalin (D-T6-D-W8,9)galol (E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-propenone (E)-3-Aminopropen-2-yl)methylphosphinic acid (E)-3-[2-(2-Methyl-4-thiazolyl)vinyl]pyridine (E)-9-(2-(cinnamyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione (E)-CH2OCOC(CH3)3 (E)-N-(Adamant-1-yl)-6-[2-(4-methoxyphenyl)vinyl]-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (E/Z)-11-(2-butenyloxy)-N-propylnoraporphine (N-acetyl 2-benzyltryptamine) (R)(+)-BrAPB (R)-(+)-3-Fluoromethyl-7-(N-2,2,2-trifluoroethylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-3,3,3-trifluoropropylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-3-methoxypropylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-ethylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-propylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-thiomorpholinoaminosulfonyl)-THIQ (R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride (R)-(-)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid (R)-(-)-7-chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (R)-(-)-9,10-Dihydro-7-fluoro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (R)-(-)-N-butyl-2-methoxy-11-hydroxynoraporphine (R)-(-)-N-ethyl-2-methoxy-11-hydroxynoraporphine (R)-(1-benzyl-4-(4-methoxybenzyl)piperazin-2-yl)methanol (R)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; iodide (R)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(tetrahydro-2H-pyran-4-y... (R)-1-(10,11-dihydro-dibenzo[b,f]azepin-5-yl)-3-methylamino-propan-2-ol (R)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol (R)-1-(2-(1-(3,4-Dichloro-benzene sulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine (R)-1-(2-(1-(3-bromo-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine (R)-1-(2-(1-(3-methoxy-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl-4-methyl piperidine (R)-1-(2-(2-ethoxyphenyl)-1-phenylethyl)piperazine (R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine (R)-1-(4-Fluorophenyl)-2-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)propan-2... (R)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol (R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine (R)-1-Cyclohexyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol (R)-1-Cyclopropyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol (R)-10-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-10-Methyl-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-11-(2-methylallyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-11-(3-methylbut-2-enyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-11-(allyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-11-Amino-2-methoxyaporphine (R)-11-Ethyl-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-2,11-Diaminoaporphine (R)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (R)-2-((1-methylpyrrolidin-2-yl)methyl)-1H-pyrrolo[2,3-b]pyridine (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-4-methylpentan-2-ol (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-4-phenylbutan-2-ol (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)hexan-2-ol (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)pent-4-en-2-ol (R)-2-((R)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine (R)-2-((R)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine (R)-2-((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)-1-methylpyrrolidine hydrochloride (R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid (R)-2-(2-phenyl-2-(piperazin-1-yl)ethyl)phenol (R)-2-(4-hydroxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-2-(4-Hydroxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol (R)-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid (R)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid (R)-2-Methoxyaporphin-11-yl pentanoate (R)-3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate (R)-3-((4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)piperidin-1-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)... (R)-3-((4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (R)-3-(1H-indol-4-yl)-N-methyl-3-(thiophen-2-yl)propan-1-amine hydrochloride (R)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride (R)-3-(3,4-dichlorophenyl)-N-methyl-3-(naphthalen-1-yl)propan-1-amine hydrochloride (R)-3-Carboxy-4-hydroxyphenylglycine (R)-3-Hydroxyphenylglycine (R)-4-(1H-indol-4-yl)-N-methyl-4-(thiophen-2-yl)butan-1-amine hydrochloride (R)-4-(3,4-dichlorophenyl)-4-(1H-indol-4-yl)-N-methylbutan-1-amine hydrochloride (R)-4-(3,4-dichlorophenyl)-N-methyl-4-(naphthalen-1-yl)butan-1-amine hydrochloride (R)-4-(3-(2-amino-4-(4-fluorophenyl)thiazol-5-yl)pyrrolidin-1-yl)-1-(4-fluorophenyl)butan-1-one (R)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline (R)-4-(4-Methylpentanoyl)-8-(4-methylpentylidene)-1-thia-4-azaspiro[4.5]decane-3-carboxylic Acid (R)-4-Carboxyphenylglycine (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) (R)-4-Methylhomoibotenic acid (R)-4-Oxo-1-pentyl-N-(1-phenylethyl)-7-(pyrrolidin-1-yl)-1,4-dihydroquinoline-3-carboxamide (R)-5,6,6a,7-Tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-5-(2-Azetidnylmethoxy)-2-Chloropyridine (R)-5-2-Azetidnylmethoxy)-2-Chloropyridine (R)-5a,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene (R)-6,10-Dimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-6-(1-methyl-pyrrolidin-2-yl)-quinoline (R)-6-bromo-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-6-chloro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-6-Chloro-3-(1-phenylethyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide (R)-6-fluoro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-6-Methyl-2-phenyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol (R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-7-Ethoxy-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide (R)-7-Fluoro-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide (R)-7-Methyl-1,6,6a,7,8,9-hexahydro-1,7-diaza-benzo[cd]pyren-2-one (R)-7-Methyl-6a,7,8,9-tetrahydro-2H,6H-2,7-diaza-benzo[cd]pyren-1-one (R)-7-Methyl-6a,7,8,9-tetrahydro-6H-1-oxa-7-aza-benzo[cd]pyren-2-one (R)-7-Methyl-6a,7,8,9-tetrahydro-6H-2-oxa-7-aza-benzo[cd]pyren-1-one (R)-7-[8-(2-Oxo-1,2,3,4-tetrahydro-quinolin-7-ylmethyl)-3-aza-bicyclo[3.2.1]oct-3-ylmethyl]-7,8-dihydro-3H-1,6,9-trioxa-3-aza... (R)-8-(3-Methylbutylidene)-4-(5-methylhexanoyl)-1-thia-4-azaspiro[4.5]decane-3-carboxylic Acid (R)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide (R)-ABT-089 [2-Methyl-3-(2-(S)-pyrrolidinylmethoxy)pyridine] (R)-ACPA (R)-AMPA (R)-AP5 (R)-aspartic acid (R)-Bu-HIBO (R)-Chlopheniramine (R)-chlorpheniramine (R)-CPPene (R)-Demethyl-ACPA (R)-Epinephrine (R)-Hexbutinol (R)-HIBO (R)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-benzo[d]imidazol-2-amine (R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(1H-indol-3-yl)-2-oxoacetamide (R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide (R)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide (R)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea (R)-N-methyl-3-(naphthalen-1-yl)-3-(thiophen-2-yl)propan-1-amine hydrochloride (R)-N-methyl-4-(naphthalen-1-yl)-4-(thiophen-2-yl)butan-1-amine hydrochloride (R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide (R)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexa-hydropyrazino[1,2-a]quinolin-3-yl)butyl]amide (R)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}am... (R)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide (R)-SIB-1508Y (R)-Trihexyphenidyl (R)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone (R,S)-4-Carboxy-3-hydroxyphenylglycine (R,S)-alpha-Methyl-4-carboxyphenylglycine (R/S)-2-(1H-indol-3-yl)-N-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-2-oxoacetamide (R/S)-2-(5-nitro-1H-indol-3-yl)-N-(5-nitro-2,3-dihydro-1H-inden-1-yl)-2-oxoacetamide (R/S)-N-(5-fluoro-2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide (R/S)-N-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide (RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine (RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine (RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine (RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine (RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine (RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine (RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine (RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine (RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate (RS) PPG (RS)-2-Amino-3-(3-hydroxy-4-pentyl-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-(3-hydroxy-4-phenylethyl-5-isoxazolyl)-propionic Acid (RS)-2-amino-3-(3-hydroxy-5-isoxazolyl)propionic acid (RS)-2-Amino-3-(4-heptyl-3-hydroxy-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-[3-hydroxy-4-(2-phenolyl)-5-isoxazolyl]-propionic Acid (RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate (RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate (RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate (RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate (RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate (RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate (RS)-2-amino-5-(3-hydoxy-5-methylisoxazol-4-yl)pentanoic acid (RS)-2-amino-5-(3-hydroxy-5-methylisoxazol-4-yl)pentanoic acid (RS)-3-sec-Butyl-2-chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]-pyridin-6(7H)-one (RS)-3-sec-Butyl-2-chloro-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one (RS)-3-sec-Butyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one (RS)-3-sec-Butyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one (RS)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) (RS)-HIBO (RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine (S)-(+)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid (S)-(+)-Amphetamine (S)-(+)-Br-HIBO (S)-(+)-Bu-HIBO (S)-(-)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride (S)-(2)-Me-Tet-AMPA (S)-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(2-methoxypyrrolidin-1-yl)methanone (S)-1,1,1-Trifluoro-2-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)propan-2-ol (S)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; iodide (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[,5-b]isoquinolin-6-yl)-1-(thiazol-2-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(3-methylthiophen-2-yl)-... (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(5-methylthiophen-2-yl)-... (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-2-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-3-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-4-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-2-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-3-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-m-tolylethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-o-tolylethanol (S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-phenylethanol (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)-2-methylpropan-2-ol (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol (S)-1-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-N-(5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl)pyrrolidine-2-carboxami... (S)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine (S)-1-(4-Chlorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol (S)-1-(4-Fluorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]-isoquinolin-6-yl)ethanol (S)-1-(5-Chlorothiophen-2-yl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-... (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-2-methyl-propan-2-ol (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol (S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol (S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-amide (S)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine (S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide (S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide (S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-oxopyrrolidine-2-carboxamide (S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide (S)-1-acetyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide (S)-1-acetyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)pyrrolidine-2-carboxamide (S)-1-benzoyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide (S)-1-benzoyl-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide (S)-1-benzoyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-5-oxopyrrolidine-2-carboxamide (S)-1-benzoyl-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide (S)-1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-1-thiophen-3-yl-ethanol (S)-1-{2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-isochroman-6-carboxylic acid methylamide (S)-2,3-dichloro-N-(2-cyclopropylethyl)-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-(2H-pyran-4-yl)-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-(pentan-3-yl)-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-(pyrrolidin-3-yl)-N-(2,2,2-trifluoroethyl)benzamide (S)-2,3-dichloro-N-cyclopentyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-ethyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-neopentyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-phenyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-propyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-Dihydro-1H-indole-2-carboxylic Acid {(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbam... (S)-2,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2-((1-methylpyrrolidin-2-yl)methyl)-1H-pyrrolo[2,3-b]pyridine (S)-2-((4-(1H-Indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)-methyl)-8-methyl-2,3-dihydro-[1,4]dioxino-[2,3-f]quinoline (S)-2-((R)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)-1-methylpyrrolidine hydrochloride (S)-2-((S)-(2,3-dichlorophenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-chloro-4-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-methoxy-4-(trifluoromethyl)phenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-bromo-2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(2-fluorophenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(3-fluorophenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(4-fluorophenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(m-tolyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(o-tolyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(p-tolyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-1-yl)propano... (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-2-yl)propano... (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-phenylpropanoic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-4-phenylbutanoic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanedioic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)succinic acid (S)-2-((S)-2-Aminopropanoylamino)-4-methylpentanoic Acid Amide (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-isobutylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-methylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenethylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-4-phenylbutanoic acid (S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionyl}-amino)-3-phenyl-propionic... (S)-2-(methylamino)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-3-phenylpropanamide (S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(N-ethyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (S)-2-amino-3-(1H-indol-3-yl)-N-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-2-amino-3-(1H-indol-3-yl)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-2-amino-3-(1H-indol-3-yl)-N-(3-oxo-3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl)propanamide (S)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid (S)-2-amino-3-(naphthalen-2-yl)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-2-amino-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-3-phenylpropanamide (S)-2-amino-N1,N5-bis(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)pentanediamide (S)-2-Aminoadipic acid (S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine (S)-2-chloro-3-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2-chloro-4-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2-chloro-5-((1-methylpyrrolidin-2-yl)methoxy)-3-(2-(pyridin-4-yl)vinyl)pyridine (S)-2-chloro-N-isobutyl-N-(pyrrolidin-3-yl)-3-(trifluoromethyl)benzamide (S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-3-biphenyl-4-yl-propionic ac... (S)-3,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3,5-DHPG (S)-3,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3,5-dihydroxyphenylglycine; (S)-3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate (S)-3-(1H-indol-3-yl)-2-(methylamino)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-3-(1H-indol-4-yl)-N-methyl-3-(thiophen-2-yl)propan-1-amine hydrochloride (S)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride (S)-3-(3,4-dichlorophenyl)-N-methyl-3-(naphthalen-1-yl)propan-1-amine hydrochloride (S)-3-(3-Methanesulfonyl-phenyl)-1-propyl-piperidine (S)-3-(4-chlorophenyl)-N-(4-chlorophenylsulfonyl)-N'-methyl-4-phenyl-4,5-dihydropyrazole-1-carboxamidine (S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-propionic acid (S)-3-bromo-1,2,9,10-tetramethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (S)-3-bromo-1,9,10-trimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-2-ol (S)-3-Carboxy-4-hydroxyphenylglycine (S)-3-chloro-2-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3-chloro-N-isobutyl-2-methyl-N-(pyrrolidin-3-yl)benzamide (S)-3-chloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid (S)-3-cyclohexyl-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)propanoic acid (S)-3-fluoro-N-isobutyl-2-methyl-N-(pyrrolidin-3-yl)benzamide (S)-3-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)-2-(trifluoromethyl)benzamide (S)-3-hydroxyphenylglycine (S)-3-Hydroxyphenylglycine (S)-3-iodo-1,2,9,10-tetramethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (S)-3-iodo-1,9,10-trimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-2-ol (S)-3-methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole (S)-4-(1-(3,4-dimethylphenyl)hexyl)-1H-indene hydrochloride (S)-4-(1H-indol-4-yl)-N-methyl-4-(thiophen-2-yl)butan-1-amine hydrochloride (S)-4-(3,4-dichlorophenyl)-N-methyl-4-(naphthalen-1-yl)butan-1-amine hydrochloride (S)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline (S)-4-carboxy-3-hydroxyphenylglycine (S)-4-carboxy-phenylglycine (S)-4-Carboxyphenylglycine (S)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) (S)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine(10) (S)-4-Methylhomoibotenic acid (S)-4C3HPG (S)-4CPG (S)-5-((R)-1-methylpyrrolidin-2-yl)oxazolidin-2-one (S)-5-(5-methoxypyridin-3-yl)-N-methylpent-4-en-2-amine (S)-5-allyl-10-ethynyl-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-5-allyl-9-(ethynyloxy)-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-5-allyl-9-cyanato-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-5-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanoic acid (S)-6-(1-methylpyrrolidin-2-yl)-quinoline (S)-6-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)hexanoic acid (S)-6-chloro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (S)-6-Chloro-3-(1-phenylethyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide (S)-6-fluoro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (S)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline (S)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide (S)-9-methoxy-2,2,4-trimethyl-5-phenyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-ABT-089 [2-Methyl-3-(2-(S)-pyrrolidinylmethoxy)pyridine] (S)-ACPA (S)-alpha-Phenylethylamine (S)-AMPA (S)-AP5 (S)-aspartic acid (S)-ATPA (S)-Chlopheniramine (S)-Demethyl-ACPA (S)-Glu (S)-Hexbutinol (S)-HIBO (S)-N-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)benzamide (S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)benzamide (S)-N-(2,3-dichlorobenzyl)-N-(pyrrolidin-3-yl)isobutyramide (S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide (S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclopentanecarbonyl)pyrrolidine-2-carboxamide (S)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (S)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide (S)-N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide (S)-N-(4-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)butyl)-2-naphthamide (S)-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide (S)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea (S)-N-isobutyl-2-isopropyl-N-(pyrrolidin-3-yl)benzamide (S)-N-methyl-3-(naphthalen-1-yl)-3-(thiophen-2-yl)propan-1-amine hydrochloride (S)-N-methyl-4-(naphthalen-1-yl)-4-(thiophen-2-yl)butan-1-amine hydrochloride (S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-2-yl)methyl)amino]benzenepropaneamide bis(trifluoroa... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-3-yl)methyl)amino]benzenepropaneamide bis(trifluoroa... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-4-yl)methyl)amino]benzenepropaneamide bis(trifluoroa... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-2-phenylethyl) amino]benzenepropaneamide bis-(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-dimethylbutyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-phenylprop- 2-enyl)amino]benzenepropaneamide bis(trifluoroace... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-phenylpropyl)amino]benzenepropaneamide bis-(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-cyclohexylmethyl)amino]benzenepropaneamide bis(trifluoroacetate... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxobutyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxoethyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxohexyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxophenylmethyl)amino]benzenepropaneamide bis-(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxopropyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)-butyl]amide (S)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}am... (S)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide (S)-SIB-1508Y (S)-tert-butyl 1,5-dioxo-1,5-bis(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethylamino)pentan-2-ylcarbamate (S)-tert-butyl 3-(1H-indol-3-yl)-1-oxo-1-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethylamino)propan-2-ylcarbamate (S)-tert-butyl 3-(1H-indol-3-yl)-1-oxo-1-(3-oxo-3-(1,2,3,4-tetrahydroacridin-9-ylamino)propylamino)propan-2-ylcarbamate (S)-Thio-ATPA (S)-Trihexyphenidyl (S)-UH-301 (S)-Zopiclone (S)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone (S)ACPA (S,S)-1-cyclopentyl-2-(5-fluoro-2-methoxy-phenyl)-1-morpholin-2-yl-ethanol (S,S)-2-(6-aminopyridin-3-yl)-2,5-diazabicyclo[2.2.1]-heptane (Z)-3-Aminopropen-2-yl)methylphosphinic acid (Z)-5-(2'-(3'-((E)-1''-hydroxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,... (Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,... (Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H... (Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quino... (Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline (Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline (Z)-CH2OCOC(CH3)3 (Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride ([Dmt1]DALDA) + 1 mM GTP +-(1H-Indol-2-yl)-(3-methyl-piperazin-1-yl)-methanone ,14-endoetheno – 7 a (1-(R)-hydroxy-1 methylbutyl)-tetrahydro-nororipavine 1 1'-(o-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1'-(p-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1'-Acetyle-(3R)-(4-Phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydrospiro[Beta-carboline-1,4'-piperidine] 1'-benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4'-piperidine] 1, 10-diamiodecane 1, 12-DB-3-4-3 1, 2-Benzenediol, 4-(2-amino-1-hydroxyethyl)- 1, HENECA 1,1-Dibutyl-6-chloro(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline 1,1-Dibutyl-6-chloro-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline 1,1-dimethyl-2-quinolin-6-yl-pyrrolidinium iodide 1,1-dimethyl-4-phenylpiperazinium iodide 1,2,3,11b-Tetrahydro[1]benzothiopyrano[4,3,2-de]isoquinolin-8,9-diol 1,2,3,4,10,14b-hexahydro-2-methyl-6-triflouromethanesulfonoxydibenzo[c,f]pyrazino[1,2-a]azepin, (+/-) 1,2,3,4,10,14b-Hexahydro-6-hydroxy-2-methyldibenzo[c,f]pyrazino[1,2-a]azepin, (+/-) 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+) 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+/-) 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(-) 1,2,3,4,5,6-Hexahydro-2-benzazocine 1,2,3,4-Tetrahydroisoquinoline 1,2,3,4-Tetrahydroisoquinoline, THIQ 1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1,2,3,7,8,9-Hexadropyrano[2,3-g], 1-(1-indolinyl)-2-propylamines 1,2,3.4-Tetrahydro[2,7]naphthyrldine oxalate 1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol 1,3,7-n-tripropylxantine 1,3,7-Trimethy1-8-(3-aminostyryl)xanthine 1,3,7-trimethyl 1,3,7-Trimethyl-8-(2,3-dimethoxystyryl)xanthine 1,3,7-Trimethyl-8-(2-methoxystyryl)xanthine 1,3,7-Trimethyl-8-(3,4-dimethoxystyryl)xanthine 1,3,7-Trimethyl-8-(3,5-dimethoxystyryl)xanthine 1,3,7-Trimethyl-8-(3-aminostyryl)xanthine 1,3,7-Trimethyl-8-(3-nitrostyryl)xanthine 1,3,7-Trimethyl-8-(4-methoxystyryl)xanthine 1,3,7-Trimethyl-8-[2-(3-aminophenyl)ethyl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-(benzyloxy)styryl]-xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-(benzyloxy)styryl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-[(4-amino-trans-butenyl)oxy]styryl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-[(4-aminobutyl)oxy]styryl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-[[4-[[(tert-butyloxy)carbonyl]amino]butyl]oxy]styryl]xanthine 1,3,7-Trimethyl-8-[3-(acetylamino)styryl]xanthine 1,3,7-Trimethyl-8-[3-(trifluoromethyl)styryl]xanthine 1,3,7-Trimethyl-8-[3-[(3-carboxy-1-oxopropyl)amino]styryl]xanthine 1,3,7-Trimethyl-8-[3-[(tert-butyloxy)carbonyl]amino]-styryl]xanthine 1,3,7-Trimethyl-8-[3-[(tert-butyloxy)carbonyl]amino]styryl]xanthine 1,3,7-Trimethyl-8-[3-[bis[(tert-butyloxy)carbonyl]amino]-styryl]xanthine 1,3,7-Trimethyl-8-[3-[bis[(tert-butyloxy)carbonyl]amino]styryl]xanthine 1,3,9-trimethyl 1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}-5-methylbenzene 1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene 1,3-di-o-tolyl-guanidine 1,3-diallyl-7-methylxantine 1,3-Diallylxantine 1,3-dibenzylxantine 1,3-DibutylX-7-riboside 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1,3-Diethyl-3-(4-hydroxybutyl)-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1,3-diethyl-8-phenyl 1,3-diethyl-8-phenylxanthine 1,3-diethyl-8phenyl 1,3-Diethylxanthine 1,3-diethylxantine 1,3-DihexylX 1,3-dihydro-1-[2-[4-[3-(trifluoromethyl)phenyl-1-piperazinyl]-ethyl]-2H-benzimidol-2-one 1,3-diisobutylxantine 1,3-dimethyl 1,3-Dimethyl-8(3,4-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(2,3-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(2-methoxystyryl)xanthine 1,3-Dimethyl-8-(3,4-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(3,5-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(3-aminostyryl)xanthine 1,3-Dimethyl-8-(3-nitrostyryl)xanthine 1,3-Dimethyl-8-(4-methoxystyryl)xanthine 1,3-dimethyl-8-phenyl 1,3-Dimethyl-8-[3-(trifluoromethyl)styryl]xanthine 1,3-Dimethyl-8-[4-(dimethylamino)styryl]xanthine 1,3-dimethyl-8phenyl 1,3-Dimethyl-8[4-(dimethylamino)styryl]xanthine 1,3-dimethyl-9-(2-(p-tolyloxy)ethyl)-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-dimethyl-9-(2-(pyridin-2-yl)ethyl)-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-dimethyl-9-(pyridin-2-ylmethyl)-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-dipropyl 1,3-Dipropyl-7-methyl-8-styrylxanthine 1,3-Dipropyl-8-(4-hydroxyphenyl)xanthine 1,3-Dipropyl-8-(p-hydroxyphenyl)xanthine 1,3-Dipropyl-8-phenylxanthine 1,3-DipropylX-7-riboside 1,3-Dipropylxanthine 1,3-n-dipropyl-7-propargyl 1,3-n-dipropylxantine 1,4-bis[3-(1,2,3,4-Tetrahydroacridin-9-yl)aminopropyl]piperazine 1,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene 1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1Hpyrazole-3-carboxamide 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1,7-dimethyl-3-isobutylxantine 1,7-dimethyl-3-n-propylxantine 1,7-Dimethylxanthine 1,9-DimethylX 1,N6-Ehteno-2-oxoado 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-(3,3-dimethylbutyl)piperazine 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-(cyclopropylsulfonyl)piperazine 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-(methylsulfonyl)piperazine 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazine 1-((1-((1H-Imidazol-1-yl)methyl)cyclopropyl)methyl)-3-(3,4-dimethoxyphenyl)thiourea 1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride 1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((5-bromopyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((5-ethynylpyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((6-bromopyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride 1-((6-bromopyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride 1-((6-chloropyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride 1-((R)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea 1-((S)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea 1-((S)-4-Fluoro-phenyl)-1-[(4aR,5S)-1-(4-fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-ethanol 1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-(2-fluorophenyl)-2-(2-methoxyphenyl)ethyl)piperazine 1-(1-(3-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-(3-fluorophenyl)-2-(2-methoxyphenyl)ethyl)piperazine 1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone 1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-(4-fluorophenyl)-2-(2-methoxyphenyl)ethyl)piperazine 1-(1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo-[1,5-b]isoquinolin-6-yl)but-3-en-1-ol 1-(1-adamantylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(1-NAPHTHYL)PIPERAZINE 1-(1-phenyl-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-phenyl-2-(2-propoxyphenyl)ethyl)piperazine 1-(1H-indol-4-yloxy)-3-(cycloheptylamino)propan-2-ol 1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 1-(1H-indol-4-yloxy)-3-(cyclopentylamino)propan-2-ol 1-(1H-indol-4-yloxy)-3-(pentan-3-ylamino)propan-2-ol 1-(1H-indol-4-yloxy)-4-(cyclohexylamino)butan-2-ol 1-(1H-indol-5-yloxy)-3-(cyclohexylamino)propan-2-ol 1-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)-4,4-difluoropiperidine 1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-4-(4-fluoro-phenyl)-1,2,3,6-tetrahydro-pyridine 1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-piperidine 1-(2,4,5-trimethoxyphenyl)-2-aminopropane HCI 1-(2,4-dichlorophenyl)-4-(hydroxymethyl)-N-(piperidin-1-yl)-5-(4-(pyridin-3-yl)phenyl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-(fluoromethoxy)phenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-morpholino-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-morpholino-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(pyrrolidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-morpholino-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-N-piperidin-1-yl-1H-pyrazole-4-carboxamide 1-(2,4-Dichlorophenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,4-Difluorophenyl)-3-[4-(3-pyridylethynyl)-2-thiazolyl]urea 1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,4-Dimethyl-phenyl)-4-(2-phenyl-cyclopropylmethyl)-piperazine; hydrobromide 1-(2,4-dimethylphenyl)-4-(((1R,2S)-2-phenylcyclopropyl)methyl)piperazine 1-(2,4-dimethylphenyl)-4-(((1S,2R)-2-phenylcyclopropyl)methyl)piperazine 1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,5-dimethoxy-4-ethoxyphenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-fluorophenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane, (+) 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane, (-) 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane 1-(2,5-dimethoxy-4-n-hexylphenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-n-propylphenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-nitrophenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-t-butylphenyl)-2-aminopropane HCI 1-(2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,6-Dimethoxypyridin-3-yl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-(1H-Imidazol-1-yl)ethyl)-3-(3,4-dimethoxyphenyl)thiourea 1-(2-(2,3-dihydrobenzofuran-7-yl)-1-phenylethyl)piperazine 1-(2-(2-(cyclopropylmethoxy)phenyl)-1-phenylethyl)piperazine 1-(2-(2-(difluoromethoxy)-6-fluorophenyl)-1-phenylethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-(2-fluorophenyl)ethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-(3-fluorophenyl)ethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-(4-fluorophenyl)ethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine 1-(2-(2-cyclopropoxyphenyl)-1-phenylethyl)piperazine 1-(2-(2-fluoro-6-methoxyphenyl)-1-phenylethyl)piperazine 1-(2-(2-isopropoxyphenyl)-1-phenylethyl)piperazine 1-(2-(2-methoxyphenyl)-1-phenylethyl)piperazine 1-(2-(3-fluoro-2-methoxyphenyl)-1-phenylethyl)piperazine 1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride 1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride 1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-bromo-2-phenylethyl)-N-(2-ethoxyethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-bromo-2-phenylethyl)-N-butyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-Bromo-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2-bromophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2-Bromophenyl)-5-(4-methoxyphenyl)-N3-(piperidin-1-yl)-1H-pyrazole-3,4-dicarboxamide 1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-chlorophenyl)ethyl)-N,N-diethyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(2-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(3-fluorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(4-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-Chloro-2-phenyl-ethyl)-6-methylsulfanyl-4-morpholin-4-yl-1H-pyrazolo[3,4-d]pyrimidine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-dimethyl-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-6-amine 1-(2-chloro-2-phenylethyl)-N-(2-fluorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N-propyl-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N6,N6-dimethyl-N4-propyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 1-(2-Chloro-4-cyanophenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-Chloro-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2-Chloro-4-methanesulfonylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-Chloro-4-methylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(1-cyclopropyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(1-isopropyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-methyl-3-(1-(2-phenylpropan-2-yl)-1H-imidazol-4-yl)-1H-pyrazole 1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-methyl-3-(1-phenyl-1H-imidazol-4-yl)-1H-pyrazole 1-(2-Dimethylaminoethyl)-4-hydroxyindole 1-(2-Methoxy-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(2-Methoxyphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrotrifluoroacetate 1-(2-Methoxyphenyl)piperazine 1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin 1-(2’-Butyl)-1H-benzotriazole-5-carboxylic acid 1-(2’-Ethoxy-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(2’-Ethylsulfanyl-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(2’-Methoxy-1’-methyl-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(3-(1H-Imidazol-1-yl)-propyl)-3-(4-methylsulfanyl-phenyl)-thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,3-dihydrobenzo[b][1,4]dioxin-7-yl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,4-dimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4,5-trimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxybenzyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)-1-methylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)urea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,5-dimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3-methoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(benzyloxy)phenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(dimethylamino)phenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-acetylphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-ethylphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-fluorophenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methylphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-nitrophenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(benzo[d][1,3]dioxol-6-yl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-benzylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-butylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-cyclohexylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-isopropylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-methylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-naphthalen-1-ylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-phenylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-tert-butylthiourea 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidine-4-carbonitrile 1-(3-(trifluoromethyl)phenyl)piperazine 1-(3-Chloro-4-fluorophenyl)-4-(morpholin-4-yl)-1,5-dihydro-pyrrole-2-one 1-(3-Chlorophenyl) piperazine 1-(3-chlorophenyl)-2-(cyclobutylamino)propan-1-one 1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(3-Hydroxypropyl)uracil 1-(3-Isopropoxypropyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(3-Methoxyphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(3-Methylphenyl)-4-morpholin-1-yl-2,4-dihydro-pyrrol-2-one 1-(3-tert-Butyldimethylsilyloxypropyl)uracil 1-(3-Triphenylsilyloxypropyl)uracil 1-(3-Tritylaminopropyl)uracil 1-(3-Trityloxypropyl)uracil 1-(3’,5’-Difluorobenzyl)-1H-benzotriazole-5-carboxylic acid 1-(3’-Methoxybenzyl)-1H-benzotriazole-5-carboxylic acid 1-(3’-Pentyl)-1H-benzotriazole-5-carboxylic acid 1-(4,4-Bis(4-chlorophenyl)butyl)-4-(4-chlorophenyl)piperidin-4-ol Hydrochloride 1-(4,5-Dimethyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(4,5-Diphenyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(4-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazin-1-yl)-3,3-dimethylbutan-1-one 1-(4-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazin-1-yl)ethanone 1-(4-(1-pyrrolidinyl)-2-butynyl)-2-pyrrolidinone 1-(4-(1H-Imidazol-1-yl)butyl)-3-(3,4-dimethoxyphenyl)thiourea 1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-(2-methoxyphenyl)piperazin-1-yl)-2-(4-phenyl-6-(trifluoromethyl)pyrimidin-2-ylthio)propan-1-one 1-(4-(3-(2,4-dimethoxyphenyl)-1-m-tolyl-1H-pyrazole-5-carbonyl)piperazin-1-yl)ethanone 1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)-2-methylpropan-1-one 1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)ethanone 1-(4-(3-(piperidin-1-yl)propoxy)benzyl)piperidine 1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea 1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea 1-(4-(4-chlorophenyl)-5,6-dihydropyridin-1(2H)-yl)-3,3-diphenylpropan-1-one 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-(N-hydroxyl)aminobenzenesulfonyl)naphthalene 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-olol 1-(4-acetyl-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-amino-3-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one 1-(4-aminobenzenesulfonyl)naphthalene 1-(4-aminobenzyl)indene 1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-aminophenyl)-2-pyrrolidin-1-yl-pentan-1-one 1-(4-azio-3-iodophenyl)-2-pyrroldin-1-yl-pentan-1-one 1-(4-benzhydrylpiperazin-1-yl)-3-(3-methyl-1H-indol-4-yloxy)propan-2-ol 1-(4-benzyl-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-Biphenyl-4-y)-4-(4-chlorophenyl)butyl]-4-(4-chlorophenyl)piperidin-4-ol 1-(4-bromo-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-Bromophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 1-(4-Bromophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-(4-chloro-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-Chloro-2,6-dimethylphenyl)-5-(1-methoxymethylpropyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochlorid... 1-(4-Chloro-2-cyanophenyl)-5-(1-ethylpropyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Chloro-2-cyanophenyl)-5-(1-methoxymethylpropyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Chloro-2-cyanophenyl)-5-(1-propylbutyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(4-Chloro-2-cyanophenyl)-5-(2-methoxy-1-methoxy-methylethyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triaza-acenaphthylene 1-(4-Chloro-2-methylbenzyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid cyclohexylamide 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 1-(4-Chloro-phenyl)-5-cyano-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(ethylthio)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(hydroxymethyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfonyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylthio)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylthio)-N-(pyrrolidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-fluoro-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-iodo-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(morpholin-4-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(pyrrolidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-[4-(trifluoromethyl)benzyl]-1H-imidazole-4-carbox-amide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N,N-diethyl-5-methyl-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1R,2R)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1S,2S)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2-(1H)yl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N-(trans-4-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carbox-amide 1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-Chlorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione 1-(4-Chlorophenyl)-3-pyrrolidin-1-yl-pyrrole-2,5-dione 1-(4-chlorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 1-(4-Chlorophenyl)-4-azepan-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-azepan-1-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-piperidin-1-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine 1-(4-Chlorophenyl)-4-{[1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Chlorophenyl)-4-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazine 1-(4-Chlorophenyl)-5-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-1,2,4-triazole-3-carboxamide Dihydrochloride 1-(4-Chlorophenyl)-5-cyano-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-N-cycloheptyl-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-N-cyclohexyl-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-difluorophenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,5-dichlorophenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2-ethylphenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2-methoxyphenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-phenyl-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-N-cyclopentyl-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-Cyano-4,4-diphenylbutyl)-4-phenylpiperidine-4-carbonitrile 1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Amide 1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Ethyl Ester Hydrochloride 1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Hydrochloride 1-(4-Ethoxy-phenyl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea 1-(4-ethylphenyl)-3-methyl-6-(4-(4-(1-phenylvinyl)cyclohexyl)butyl)-1,2,3,4-tetrahydronaphthalene 1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one 1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-Fluorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione 1-(4-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 1-(4-fluorophenyl)-4-(3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 1-(4-fluorophenyl)-4-(8-phenyl-3,8-diaza-bicyclo[3.2.1]octan-3-yl)butan-1-one 1-(4-Fluorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 1-(4-Fluorophenyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine 1-(4-Fluorophenyl)-4-{[1-(4-fluorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Fluorophenyl)-4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazine 1-(4-Hydroxyphenyl)-4-{[1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Iodophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-(4-Methoxy-2-methylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydromethanesulfonate 1-(4-Methoxyphenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Methoxyphenyl)-4-{[1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Methylphenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 1-(4-Methylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-p-Tolyl-butyl)-piperidine 1-(4-Phenyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(4-tert-butylbenzyl)-3-(1-(3-fluoro-4-(methylsulfonamido)phenyl)ethyl)thiourea 1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 1-(4-{[4-(2,4-Diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanone 1-(4-{[4-(2,4-Diamino-6-ethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanol 1-(4-{[4-(2,4-Diamino-6-ethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanone 1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(5-Chloropyridin-2-yl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(5-Oxohexyl)theobromine (pentoxifylline) 1-(5-Phenyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(5-Triphenylsilyloxypentyl)uracil 1-(5-Tritylaminopentyl)uracil 1-(5-Trityloxypentyl)uracil 1-(6-chloro-pyridin-3-yloxymethyl)-cyclopropylamine; hydrochloride 1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 1-(adamantan-1-ylamino)-3-(1H-indol-5-yloxy)-propan-2-ol 1-(adamantan-1-ylamino)-4-(1H-indol-4-yloxy)-butan-2-ol 1-(benzo[d]thiazol-2-yl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine 1-(benzo[d]thiazol-2-ylmethyl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine 1-(Bicyclo[2.2.1]hept-5-en-2-yl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea 1-(bis(4-chlorophenyl)methyl)-3-((3,5-difluorophenyl)(methylsulfonyl)methylene)azetidine 1-(cyano-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(cyclobutylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(cyclohexylcarbonyl)-4-(diphenylmethyl)-1,4-diazepane 1-(Cyclohexylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(cyclopentylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 1-(oxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(pyridin-3-yloxymethyl)-cyclopropylamine; hydrochloride 1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(4-[trifluoromethyl]-benzoyl)amino-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(alpha-toluenesulfonyl)amino-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-6-(4-n-propylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-6-(4-phenylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-6-(phenylaminocarbonyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(2-furoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(2-[4-methoxyphenyl]ethylamino)carbonyl-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-chlorobenzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-tert-butylbenzyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-[2-phenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-[3-phenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-[4-tert-butylphenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(tert-butoxymethylcarbonyl)aminophenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-phenylethoxy-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 1-Adrenaline 1-allyl-3,7-dimethylxantine 1-Amino-2-phenylethane 1-Benzhydryl-1H-benzotriazole-5-carboxylic acid 1-Benzoylpiperazine 1-Benzyl-1H-benzotriazole-5-carboxylic acid 1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-Benzyl-2-pyridin-2-yl-1H-benzoimidazole 1-Benzyl-2-thiazol-4-yl-1H-benzoimidazole 1-benzyl-3-(N,N-dimethylaminoethyl)indene 1-Benzyl-4-(3-hydroxyphenyl)piperidine 1-benzyl-4-(4-methoxybenzyl)piperazine 1-benzyl-4-methyl-6-phenyl-3-(phenylsulfonyl)pyridin-2(1H)-one 1-Benzyl-4-[3-(methylsulfonyl)phenyl]piperazine 1-Benzyl-4-[3-(methylsulfonyl)phenyl]piperidine 1-benzyl-5,6-dimethoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 1-Benzyl-N-(2-cyclohexylidene-2-fluoroethyl)-4-piperidinamine 1-Benzyl-N-(2-cyclopentylidene-2-fluoroethyl)-4-piperidinamine 1-benzyl-N-cycloheptyl-4-oxo-1,4-dihydroquinoline-3-carboxamide 1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide 1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide 1-Benzylpiperazine 1-beta-hydroxyethyl-3-methylxantine 1-Butyl-1H-benzotriazole-5-carboxylic acid 1-Butylpsilocin 1-Butylpsilocybin 1-Butyltheobromine 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1-Cyclobutyl-1H-benzotriazole-5-carboxylic acid 1-Cyclohexyl-1H-benzotriazole-5-carboxylic acid 1-Cyclohexyl-3-(4-phenyl-1H-imidazol-2-yl)-9H-Beta-carboline 1-Cyclopentyl-1H-benzotriazole-5-carboxylic acid 1-Cyclopropyl-1H-benzotriazole-5-carboxylic acid 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 1-deaza-2-Cl-CHA (2c) 1-deaza-2-Cl-CPA (2b) 1-deaza-2-Cl-PIA (2a) 1-deazaadenosine 1-deazaCHA (3c) 1-deazaCPA (3b) 1-deazaNECA (10) 1-deazaPIA (3a) 1-Deoxysalvinorin A 1-Ethoxy-4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-4-aza-tricyclo[5.2.2.0*2,6*]undecane-3,5,8-trione 1-ethyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1-ethyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin 1-Ethyl-1H-benzotriazole-5-carboxylic acid 1-ethyl-1H-benzo[d]imidazol-2(3H)-one 1-Ethyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-10-ol 1-Ethyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol 1-ethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-Ethyl-3,3-dimethyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1-ethyl-3-methylxantine 1-Ethyl-3-{(1,4-cis)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 1-Ethyl-3-{(1,4-trans)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 1-ethyl-5-methoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 1-Ethyl-8-(4-(4-(3-fluorobenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-fluorobenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-methoxybenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-methoxyphenyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-methylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-phenethylpiperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(piperidine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 1-Ethyltheobromine 1-Hydroxy-1-[5-(2-pyridyl)oxazol-2-yl]-7-phenylheptane 1-Hydroxy-1-[5-(2-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1-Hydroxymethyl-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Isopropoxymethyl-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Isopropyl-1H-benzotriazole-5-carboxylic acid 1-isopropyl-4-(4-(3-((methylamino)methyl)-4-(4-(methylthio)phenoxy)phenyl)but-3-ynyl)piperazin-2-one 1-Isopropyl-5-Methoxytryptamine 1-Isopropyl-5-Methyltryptamine 1-Isopropyltryptamine 1-Me-Tet-AMPA 1-Methoxy-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1-Methoxy-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1-Methoxy-4-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.2.0*2,6*]undec-8-ene-3,5-dione 1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-Methyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-10-ol 1-Methyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol 1-Methyl-2-(2,4,5-trimethoxy-phenyl)-ethylamine 1-Methyl-2-oxoado 1-methyl-2-phenylethylamine 1-Methyl-2-thiazol-4-yl-1H-benzoimidazol 1-Methyl-3-phenyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1-Methyl-4-naphthalen-2-yl-piperidine-4-carbonitrile 1-Methyl-4-naphthalen-2-yl-piperidine-4-carboxylic Acid Ethyl Ester 1-methyl-4-phenylpyridinium ion 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole 1-Methyl-5-(2-thioxo-1,2-dihydrospiro[3,1-benzoxazine-4,1'-cyclobutan]-6-yl)-1H-pyrrole-2-carbonitrile 1-methyl-5-(4-methyl-4-thien-3-yl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)- 1H-pyrrole-2-carbonitrile 1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole 1-Methyl-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-methyl-serotonin 1-Methylenoxime-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Methylpsilocin 1-Methylpsilocybin 1-Methylxanthine 1-N-Allyl-7, 8-dihydro-14-hydroxymorphinone 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 1-Naphthalenamine, 4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-, (1S-cis)- 1-NP 1-oleoyl 2-acetyl glycerol 1-Oxo-1-[4-(2-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[4-(3-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[4-(4-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-furyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-oxazolyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-oxazolyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-pyrazinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-pyrazinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-10-phenyldecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-11-phenylundecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-2-phenylethane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-3-phenylpropane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-4-phenylbutane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-5-phenylpentane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-6-(phenyl)hex-5-yne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-6-heptyne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-6-phenylhexane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-7-(phenyl)hept-6-yne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-7-(trimethylsilyl)hept-6-yne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-8-phenyloctane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-decene 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-decyne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-octadecyne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-phenylnonane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]butane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]decane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]dodecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]ethane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]heptane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]hexadecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]hexane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]nonane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]octadecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]octane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]pentane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]propane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]tetradecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]undecane 1-Oxo-1-[5-(2-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-pyrimidinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-thiazolyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-thiazolyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-thienyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-thienyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(3-pyridazinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(3-pyridazinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(3-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(3-thienyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(4-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(4-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(4-pyrimidinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(5-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(phenyl)oxazol-2-yl]-7-phenylheptane 1-Pentyl-1H-benzotriazole-5-carboxylic acid 1-phenlsemicarbazide 1-phenyl-1-(piperidin-2-yl)propan-2-one 1-Phenyl-2-amino-athan (GERMAN) 1-phenyl-2-aminopropane 1-phenyl-2-aminopropane,(+) 1-phenyl-4-((1-phenyl-1H-1,2,3-triazol-4-yl)methyl)piperazine 1-phenyl-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 1-Phenyl-4-(2-phenyl-3H-imidazol-4-ylmethyl)-piperazine 1-Phenyl-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-PP 1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-Propyl-1H-benzotriazole-5-carboxylic acid 1-Propyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-10-ol 1-Propyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol 1-Propyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Propyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-t-Butyl-1H-benzotriazole-5-carboxylic acid 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 1-thiocarbamoyl-3,5-di-(4-methylphenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydropyrazole 1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-methylphenyl)-5-(furan-2-yl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-methylphenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(furan-2-yl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(thiopen-2-yl)-4,5-dihydropyrazole 1-TMT 1-[(1-(4-Chlorophenyl)-1H-1,2,3-triazol-4-yl)methyl]-4-phenylpiperazine 1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-phenylpiperazine 1-[(1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazol-4-yl)carbonyl]-THIQ 1-[(1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazol-4-yl)carbonyl]piperidin-4-ol 1-[(1-(4-Fluorophenyl)-1H-pyrazol-4-yl)methyl]-4-phenylpiperazine 1-[(2,4-dichlorophenyl)(phenyl)methyl]-4-(piperidin-1-ylcarbonyl)piperazine 1-[(E)-4-trityloxy-2-butenyl]uracil 1-[(Z)-4-Trityloxy-2-butenyl]uracil 1-[1-(2-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol(HCl) 1-[1-(3-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol (HCl) 1-[1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(3-Fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(3-Fluorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(3-Methoxyphenyl)-2-(4-methyl-1-piperazinyl)ethyl]cyclohexanol Dihydrochloride 1-[1-(3-Methoxyphenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(4-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol (HCl) 1-[1-(4-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(4-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(4-Fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(4-Fluorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(4-Methoxyphenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[2-(4-Benzoyl-1-piperazinyl)ethyl]-2-imidazolidinone 1-[2-(4-Benzyl-1-piperazinyl)ethyl]-2-imidazolidinone 1-[2-(Azidomethyl)-4-(trityloxy)butyl]uracil 1-[2-(Benzoyloxyethoxy)methyl]uracil 1-[2-(Hydroxymethyl)-4-(trityloxy)butyl]uracil 1-[2-(Trityloxy)ethoxymethyl]uracil 1-[2-Dimethylamino-1-(3-methoxy-phenyl)-ethyl]-cyclohexanol (HCl) 1-[2-Dimethylamino-1-(3-trifluoromethyl-phenyl)-ethyl]-cyclohexanol (HCl) 1-[2-[4-(1-Indanyl)-1-piperazinyl]ethyl]-2-imidazolidinone 1-[3-(Methylsulfonyl)phenyl]-4-propylpiperazine 1-[3-[N-(4-Bromobenzyl)-N-(pyrid-2-yl)amino]propyl]-3-[3-(1H-imidazol-4-yl)propyl]thiourea Dihydrochloride 1-[4-(4-methylcyclohexyl)butyl]alpha,alpha-diphenyl-4-piperdinemethanol 1-[4-(4-methylphenyl)butyl]-alpha,alpha-diphenyl-4-piperdine-methanol 1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 1-[4-(tert-Butoxycarbonylamino)-3-(trityloxymethyl)butyl]-uracil 1-[4-Acetyloxy-3-(tritylaminomethyl)butyl]uracil 1-[4-Hydroxy-2-(trityloxymethyl)butyl]uracil 1-[4-Hydroxy-3-(tritylaminomethyl)butyl]uracil 1-[5-(1-Methylimidazol-2-yl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(1-Methylpyrrol-2-yl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(2-Furyl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(2-Pyridyl)oxazol-2-yl]-7-phenylheptane 1-[5-(2-Pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-[5-(2-Pyrimidinyl)oxazol-2-yl]-7-phenylheptan-1-ol 1-[5-(3-Furyl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(3-Pyridazinyl)oxazol-2-yl]-7-phenylheptan-1-ol 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride 1-[[2,3-Dihydro-7-(3-pyridyl)benzofuran-5-yl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[2-Chloro-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[2-Fluoro-5-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[3-Fluoro-5-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid 1-[[4-Chloro-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[4-Chloro-3-(4-methyl-3pyridyl)phenyl]carbamoyl-5-methoxy-6-trifluoromethylindoline 1-[[4-Methoxy-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[4-tert-Butyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-(2,6-Difluorophenyl)-3-pyridyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-(3,5-Difluorophenyl)-3-pyridyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-Bromo-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-Ethyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-{2-(3-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride 1-{2-(3-Methylpiperazin-1-yl)-1-[3-(trifluoromethyl)phenyl]ethyl}cyclohexanol Dihydrocholoride 1-{2-(4-Methylpiperazin-1-yl)-1-[4-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride 1-{2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride 1-{2-Piperazin-1-yl-1-[3-(trifluoromethyl)phenyl]ethyl}cyclohexanol Dihydrochloride 1-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-4-(3-phenyl-propyl)-piperazine 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid 1-{[1-(4-Chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methoxyphenyl)piperazine 1-{[1-(4-Fluorophenyl)-1H-1,2,3-triazol-4-yl]methyl}-4-phenylpiperazine 1-{[1-(4-Nitrophenyl)-1H-1,2,3-triazol-4-yl]methyl}-4-phenylpiperazine 10 10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 10-(1-ethyl-1,2,3,6-tetrahydro-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin 10-(2-Butenyl)-11-hydroxy-N-propylnoraporphine 10-(2-Methylallyl)-11-hydroxy-N-propylnoraporphine 10-(4-(5-(4-fluorobenzamido)-1H-indol-3-yl)piperidin-1-yl)decanoic acid 10-(4-methylpiperazino)-5H-dibenz[b,f]oxepin 10-Allyl-11-hydroxy-N-methylaporphine 10-Allyl-11-hydroxy-N-propylnoraporphine 10-[1,2,3,6-tetrahydro-1(2-propenyl)-4-pyridinyl]-5H-dibenzo[a,d]cycloheptene 10-[1-methyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin 103 104 105 108 109 10a-homo-9,11-ethano PGH2 10alpha,11alpha-oxido PGA2 10S-hydroxylobel-7-ene 11 11,9-epoxymethano PGH2 11-(1-Methylallyloxy)-N-methylaporphine 11-(2-Butynyloxy)-N-propylnoraporphine 11-(2-Hexyl-5-hydroxyphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(2-Hexyl-5-hydroxyphenoxy)undecanoic Acid (4-Hydroxyphenyl)amide 11-(2-Hexyl-5-hydroxyphenoxy)undecanoic Acid Cyclopropylamide 11-(3-Hydroxy-4-hexylphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(3-Hydroxy-4-hexylphenoxy)undecanoic Acid (4-Hydroxyphenyl)amide 11-(3-Hydroxy-4-hexylphenoxy)undecanoic Acid Cyclopropylamide 11-(3-Hydroxy-5-pentylphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(3-Hydroxy-5-pentylphenoxy)undecanoic Acid (4-Hydroxyphenyl)amide 11-(3-Hydroxy-5-pentylphenoxy)undecanoic Acid Cyclopropylamide 11-(3-Hydroxyphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(3-Hydroxyphenoxy)undecanoic Acid (4-Hydroxy-phenyl)amide 11-(3-Hydroxyphenoxy)undecanoic Acid Cyclopropilamide 11-(4-Methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 11-Allyloxy-N-methylaporphine 11-Amino-9,10-dihydro-9,10-ethanoanthracene Oxalate 11-Hydroxy-N-propylnoraporphine 11-Propargyloxy-N-methylaporphine 11-Propargyloxy-N-propylnoraporphine 11-valeryloxynoraporphine 110 111 112 113 116 117 118 119 11f 11Z,14Z,17Z-eicosatrienoic acid 12 12'-hydroxy-2',5'-diisopropyl-3',6',18-trioxoergotaman 12(R)-HETE 12-Deoxyphorbol 13-phenylacetate 12-METHOXYIBOGAMINE 12-oxo-LTB4 120 121 122 1229U91 124 125I-NCQ 298 127 128 12a 12b 12c 13 13,14,15,16-Tetrahydrosalvinorin A 130 134 136 137 138 13a 13b 13c 13d 13e 14 14-Benzyloxymetopon 14-ethoxy-3-hydroxy-5-methyl- 17-(2-phenylethyl)morphinan-6-one 14-Hydroxydihydromorphinone 14-methoxymetopon 14-O-(1-naphthylmethyl)oxymorphone 14-O-(2,6-dichlorobenzyloxy)oxymorphone 14-O-Allyloxymorphone 14-O-Benzyloxymorphone 14-O-methyloxymorphone 14-O-phenylpropylnaltrexone 14-phenylpropoxymetopon 14a 14b 14beta-(2'-chlorocinnamoylamino)-7,8-dihydromorphinone 14beta-(p-chlorocinnamoylamino)-7,8-dihydrocodeinone 14Beta-(p-nitrocinnamoylamino)-7,8-dihydrocodeinone 14c 14d 14e 14f 14g 14h 14i 14j 14k 14l 15 15-(2-hydroxyethyl)-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-ethyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl PGF2alpha 15-methyl-N-(1,3,4-thiadiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl-N-(4-methyl-1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl-N-(5-methyl-1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15a 15b 15c 15d 15e 15f 15g 15h 16 16,16-dimethyl PGF2alpha 16-(2-Hexyl-5-hydroxyphenoxy)hexadecanoic Acid (4-Hydroxyphenyl)amide 16-(2-Hexyl-5-hydroxyphenoxy)hexadecanoic Acid Cyclopropylamide 16-(3-Hydroxy-4-hexylphenoxy)hexadecanoic Acid (4-Hydroxyphenyl)amide 16-(3-Hydroxy-5-pentylphenoxy)hexadecanoic Acid (2-Hydroxyethyl)amide 16-(3-Hydroxy-5-pentylphenoxy)hexadecanoic Acid (4-Hydroxyphenyl)amide 16-(3-Hydroxy-5-pentylphenoxy)hexadecanoic Acid Cyclopropylamide 16-(3-Hydroxyphenoxy)hexadecanoic Acid (2-Hydroxy-ethyl)amide 16-(3-Hydroxyphenoxy)hexadecanoic Acid (4-Hydroxy-phenyl)amide 16-(3-Hydroxyphenoxy)hexadecanoic Acid Cyclopropylamide 16a 16b 16c 17 17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate 17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(2',3',4',6'-tetra-O-benzyl-D-glucopyranosyl)acetamido]morp... 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3'-methoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(D-glucopyranosyl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(thiophen-2'-yl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzylacetamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(cinnamoylacetamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(D-glucopyranosyl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)phenylacetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-nitro)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-amino)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carboxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-methoxy)benzylacetamido]morphinan ( 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-tert-butoxycarbonylamino)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(thiophen-2'-yl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-[(3'-dimethylamino)benzamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-bromo)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-iodo)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-methyl)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-t-butyl)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-trimethylfluoro)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-naphthalyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-isoquinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(4'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(2'-naphthalyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(2'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-isoquinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(4'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-6,7-didehydro-4,5-alpha-epoxy-5'-guanidinyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-4-chlorobenzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphi... 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-4-nitrobenzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphin... 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-benzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-guanidinylmethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 17-deoxysalvinorin A 17-Hydroxy-13-methyl-10-(4-methyl-benzyl)-17-prop-1-ynyl-1,2,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-cyclopenta[a]phen... 17a 17b 17beta-Estradiol 18 19 19a 19b 19c 1alpha H, 3 alpha, 5 alpha H-tropan-3-yl-3,5dichlorobenzoate 1b 1c 1d 1DMe-Y8Fa 1e 1H-Benzimidazol-2-yl-thiourea 1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 1R,3R-ACPD 1R,3S-ACPD 1S, 3R-ACPD 1S, 3S-ACPD 2 2 (BCCT) 2',3'-Dihydro-(3R)-(4-Phenyl-1H-imidazol-2-yl)spiro[Beta-carboline-1,2'-1H-indene] 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 2'-Deoxy-N6-methylado 2'-Deoxyadenosine 2'-O-Methyladenosine 2'-Oxopyrrolidino-1-pyrrolidino-4-butyne 2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone 2,2-Dimethyl-1-(oxazol-2-yl)-1-oxo-9(Z)-octadecene 2,2-Dimethyl-propionic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-(2,2-dimethyl-propionyloxymethyl)-propyl Ester 2,2-Dimethyl-propionic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phosphono-oxymethyl-propyl Ester, Ammonium Salt 2,2-Dimethyl-propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3... 2,2-Diphenyl-ethylamine 2,2-diphenylethylamine 2,3,4,5-Tetrahydro-1H-2-benzazepine 2,3,4,5-Tetrahydro-5H-1,4-benzothiazepine 2,3,4,5-Tetrahydro-5H-1,4-benzoxazepine 2,3,7,11b-Tetrahydrodibenzo[d,e,h]isoquinoline Oxalate 2,3-dichloro-alpha-methyl benzylamine 2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-1H-benzimidazole-1-carboxamide 2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-6-methoxy-1H-benzimidazole-1-carboxylate 2,3-Dihydroisoindole 2,3-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 2,3-DIMETHYLPHENYLPIPERAZINE 2,3-O-(4 benzoylbenzoyl)-ATP 2,4,5-TMA 2,4,9-trimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione 2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione 2,4-Diaminobutyric acid 2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine 2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2,4-dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-DIMETHYLPHENYLPIPERAZINE 2,4-DMA 2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine 2,5,7-Trimethyl-3-[4-(phenylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine 2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,5-bis(GSyl)-alpha-MethylDopamine 2,5-Dihydro-6-methoxy-2-(2-methoxyphenyl)-5-[2-(4-morpholinyl)ethyl]-1H-pyrido[4,3-b]indol-1-one 2,5-Dihydro-6-methoxy-5-[2-(4-morpholinyl)ethyl]-2-[(1S,2S)-1,33-trimethylbicyclo[2.2.1]heptan-2-yl]-1H-pyrido[4,3-b]indol-1-... 2,5-Dimethoxy-4-bromoamphetamine 2,5-Dimethoxy-4-bromoamphetamine, benzyloxy 2,5-Dimethoxy-4-bromoamphetamine, R(-) 2,5-Dimethoxy-4-bromoamphetamine, S(+) 2,5-Dimethoxy-4-ethyl-amphetamine,(+/-) 2,5-DIMETHOXY-4-ETHYLAMPHETAMINE 2,5-DIMETHOXY-4-ETHYLAMPHETAMINE, (-) 2,5-DIMETHOXY-4-IODOAMPHETAMINE , (+) 2,5-DIMETHOXY-4-IODOAMPHETAMINE , (-) 2,5-Dimethoxy-4-methylamphetamine 2,5-Dimethoxy-4-methylamphetamine, R(-) 2,5-dimethoxy-4-methylphenylisopropylamine 2,5-dimethyoxy-4-iodophenylisopropylamine 2,6-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}pyridine 2,6-Difluorobenzoic Acid 2-(2,6-difluorobenzoyloxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester 2,N,N-TMT 2,N,N-TRIMETHYLTRYPTAMINE 2-((2-(2-fluorophenyl)-7-methoxybenzofuran-4-yl)methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline 2-((2-(furan-2-yl)-7-methoxybenzofuran-4-yl)methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline 2-((3R)-3-Methyl-4-{[(2S)-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}pipera-zin-1-yl)quinoline-6-carbonitril... 2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethanamine 2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)acetic acid 2-(-3-pyridinyl)-1-azabicyclo[2.2.2]octane 2-(1-(3,5-diethoxy-4-(1H-pyrrol-1-yl)benzyl)piperidin-4-ylamino)-N,N-dimethylbenzo[d]oxazole-5-sulfonamide 2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-carboxamide 2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-carboxylic acid 2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)-N,N-dimethylbenzo[d]oxazole-5-sulfonamide 2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide 2-(1-(4-(4-chlorophenyl)-2,2,4-trimethyl-3,4-dihydroquinolin-1(2H)-yl)-1-oxopropan-2-yl)hexahydro-1H-isoindole-1,3(2H)-dione 2-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide 2-(1-(4-chloro-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-carboxylic acid 2-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-carboxylic acid 2-(1H-Benzoimidazol-2-yl)-phenol 2-(1H-Benzoimidazol-2-yl)-pyridin-3-ol 2-(1H-Indol-3-yl)-2-oxo-N-(1-phenyl-ethyl)-acetamide 2-(1H-Indol-3-yl)-N-(4-methoxy-benzyl)-2-oxo-acetamide 2-(1H-Indol-3-yl)-N-(4-nitro-benzyl)-2-oxo-acetamide 2-(2,4-Dichlorophenyl)-1-(4-fluorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 2-(2,4-Dichlorophenyl)-1-(4-methoxyphenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 2-(2,4-Dichlorophenyl)-4-methyl-6-(1-propylbutyl)-2,6,7,8-tetrahydro-1,2,3,6-tetraazaacenaphthylene 2-(2,4-Dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1-(4-(trifluoromethyl)phenyl)-1H-imidazole-4-carbox-amide 2-(2,5-Dimethoxy-phenyl)-1-methyl-ethylamine 2-(2,6-bis(2-(diethylamino)ethoxy)phenoxy)-N,N-diethylethanamine 2-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2-azaspiro[4.5]decane-1,3-dione 2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole 2-(2-benzylphenyl)-ethylamine 2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-isopropyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-N-methyl-1H-imidazole-4-carboxamide 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-methyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoropropyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-c]pyridine hydrochloride 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoropropyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2-methoxy-2-methylpropyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-cyclopentyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-ethyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-isobutyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-isopropyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-(pyridin-3-yl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imidazole-4-carboxamide 2-(2-Dimethylaminomethyl-phenylsulfanyl)-5-methyl-phenylamine 2-(2-Thiazolyl)ethanamine 2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl-cyclohexyl)-acetamide 2-(3,5-Difluorophenyl)-4-(3-fluorophenylethynyl)thiazole 2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)acetamide 2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-isopropoxyphenyl)piperazin-1-yl)ethyl)acetamide 2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)acetamide 2-(3-(2-(cyclopropylamino)pyrimidin-4-yl)piperidin-1-yl)-1-(1H-indol-3-yl)ethanone 2-(3-Bromophenyl)histamine 2-(3-Chlorophenyl)histamine 2-(3-Iodophenyl)histamine 2-(3-pyridinyl)-2,5-diazabicyclo[2.2.2]octane 2-(4'-Methylaminophenyl)Benzothiazole 2-(4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxy-5-fluorophenoxy)ethanol 2-(4-(2-(benzylamino)ethyl)phenoxy)isonicotinamide 2-(4-(2-(benzylamino)ethyl)phenoxy)nicotinamide 2-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)phenol 2-(4-(3-(tert-butylamino)-2-hydroxypropoxy)-1H-indol-3-yl)acetamide 2-(4-(4-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)piperazin-1-yl)butyl)-6-(1H-imidazol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)piperazin-1-yl)butyl)-6-(1H-indol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)-4-oxobutyl)-6-(1H-imidazol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)butyl)-6-(1H-imidazol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)butyl)-6-(1H-indol-1-yl)pyridazin-3(2H)-one 2-(4-(5-(aminomethyl)pyridin-2-yloxy)phenyl)-N-benzylethanamine 2-(4-(benzyloxy)phenyl)-3-(2-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta... 2-(4-(benzyloxy)phenyl)-3-(8-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta... 2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Bromobenzyl)-3-{4-[2-(4-(dimethylamino)phenyl)vinyl]phenoxy}propan-1-ol 2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-bromophenyl)-2-phenylethanamine 2-(4-bromophenyl)ethylamine 2-(4-Chloro-1,3-dihydro-isoindol-2-ylamino)-4,5-dihydro-3H-imidazol-1-ium 2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 2-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Chlorophenyl)-5-phenyl-4-isoxazolin-3-one 2-(4-Fluoro-phenyl)-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-acetamide 2-(4-Fluorophenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-(4-Hexyl-2,5-dimethoxy-phenyl)-1-methyl-ethylamine : (Hydrochloride) 2-(4-hexylphenyl)-2-phenylethanamine 2-(4-hexylphenyl)ethanamine 2-(4-Hydroxyphenyl)-1-p-tolyl-3H-inden-5-ol 2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol 2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Methoxyphenyl)ado (CV-1674) 2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Nitro-phenyl)-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-acetamide 2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}-1,4-diazepan-1-yl)-quinoline-6-carbonitrile 2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile 2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)quino-line-6-carboxamide 2-(5-benzyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)-N-isopropylpropanamide 2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8atetrahydro-2H-phthalazin-1-one 2-(5-Nitro-1H-indol-3-yl)-2-oxo-N-(1-phenyl-ethyl)-acetamide 2-(5-{2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethoxy}-1H-indol-3-yl)-ethylamine 2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine 2-(6-chloro-3-pyridinyl)-2,6-diazabicyclo[3.2.1]octane 2-(6-chloro-4-methylpyridin-3-yl)-7-azabicyclo[2.2.1]heptane 2-(6-Chloro-pyridazin-3-yl)-2,5-diaza-bicyclo[2.2.1]heptane 2-(6-chloropyridin-3-yl)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene 2-(6-chloropyridin-3-yl)-2,7-diazaspiro[4.4]nonane 2-(6-fluoro-5-phenylpyridin-3-yl)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene 2-(6-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane 2-(6-Phenylpyridazin-4-yl)benzonitrile 2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,3-d]pyrimidin-4-ylthio)-N-(2-methoxyphenyl)propanamide 2-(Aminoethyl)-5-(2'-methoxy-5'-fluorophenethyl)tetrahydrofuran 2-(Aminomethyl)-4-hydroxy-3-methyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one hydrochloride 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide 2-(dimethylamino)-6-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-3H-pyrrolo[2,3-d]pyrimidin-4(7H)-one 2-(Dimethylamino)tetralin 2-(methylamino)-N6-(3-Iodobenzyl)adenosine-5'-N-methyluronamide 2-(methylthio)-N6-(3-Iodobenzyl)adenosine-5'-N-methyluronamide 2-(N,N-Diethylamino)-3'-chloropropiophenone 2-(N,N-Dimethylamino)-3'-chloropropiophenone 2-(N-(2-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-(4-chlorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-(4-fluorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-(4-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-Cyclopentylamino)-3'-chloropropiophenone 2-(N-Cyclopropylamino)-3-chloropropiophenone 2-(N-dipropylamino)quinoline 2-(N-Isopropylamino)-3'-chloropropiophenone 2-(N-Methyl-N-tert-butylamino)-3'-chloropropiophenone 2-(N-Propylamino)-3'-chloropropiophenone 2-(N-tert-Butylamino)-1-(2'-thienyl)-1-propanone 2-(N-tert-Butylamino)-3',4'-dichloropropiophenone 2-(N-tert-Butylamino)-3'-bromopropiophenone 2-(N-tert-Butylamino)-3'-chloro-4'-methylpropiophenone 2-(N-tert-Butylamino)-3'-chlorobutyrophenone 2-(N-tert-Butylamino)-3'-chloroheptanophenone 2-(N-tert-Butylamino)-3'-chlorohexanophenone 2-(N-tert-Butylamino)-3'-chlorooctanophenone 2-(N-tert-Butylamino)-3'-chloropentanophenone 2-(N-tert-Butylamino)-3'-chlorophenyl-4-cyclohexylbutanophenone 2-(N-tert-Butylamino)-3'-chlorophenyl-4-methylpentanophenone 2-(N-tert-Butylamino)-3'-methylpropiophenone 2-(N-tert-Butylamino)-4'-bromo-5'-methylpropiophenone 2-(N-tert-Butylamino)-4'-bromopropiophenone 2-(N-tert-Butylamino)-4'-chloropropiophenone 2-(N-tert-Butylamino)-4'-methylpropiophenone 2-(N-tert-Butylamino)propiophenone 2-(Phenylamino)ado (CV-1808) 2-(pyridin-3-yl)-2,7-diazaspiro[4.4]nonane 2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 2-(tert-Butylamino)-3',4'-dichlorobutyrophenone 2-(tert-Butylamino)-3',4'-dichloropentanophenone 2-(tert-Butylamino)-3',5'-dichloropropiophenone 2-(tert-Butylamino)-3',5'-difluoropropiophenone 2-(tert-Butylamino)-3'-fluoropropiophenone 2-(tert-butylamino)-7-chloro-3,4-dihydronaphthalen-1(2H)-one 2-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 2-1sopropyl-l.2,3,4-tetrahydro[2.7]naphthyridine oxalate 2-AG 2-amino-2-(3-hydoxy-5-methylisoxazol-4-yl)acetic acid, (RS) 2-amino-2-(3-hydoxy-5-methylisoxazol-4-yl)propionic acid 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 2-amino-3-phosphonopropionate 2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate 2-Amino-4-(3-difluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-fluorophenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-hydroxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-methoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-methylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-trifluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-trifluoromethylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-(dimethylamino)phenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-difluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-fluorophenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-hydroxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-methoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-methylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-trifluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-trifluoromethylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-benzo[1,3]dioxol-5-yl-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-amino-4-oxo-6-methyl-5-substituted pyrrolo[2,3-d]pyrimidine 2-Amino-4-phenyl-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride 2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate 2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 2-Amino-6-(3-hydroxy-5-methylisoxazol-4-yl)hexanoic Acid 2-Amino-6-ethyl-5-[(1'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(2',6'-dimethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(2'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3',4'-dichlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3',5'-trifluoromethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]p-yrimidine 2-Amino-6-ethyl-5-[(3'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-fluorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-methyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-N6- (3-iodobenzyl)-adenosine 2-amino-suberic acid 2-Aminoethyl-5-(3'-(2''-methoxy-5''-fluorophenyl)-1'-propyl)tetrahydrofuran 2-Aminoquinoline 2-Arachidonyl glycerol + PMSF 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 2-Biphenyl-2-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-Biphenyl-4-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-Bromo-3-(2(S)-azetidinylmethoxy)pyridine 2-Bromo-3-ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Bromo-4-(3-fluorophenylethynyl)thiazole 2-Bromo-4-hydroxy-3-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Bromo-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Bromo-alpha-ergocryptine 2-Bromomelatonin 2-CADO 2-carboxymethylbenzenesfulfonamide 2-CH3-5-HT 2-Chloro-3-(2(S)-azetidinylmethoxy)pyridine 2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(R)-pyrrolidinyl)methoxy)pyridine 2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine 2-Chloro-3-cyclohexyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-cyclopropyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-cyclopropyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-ethyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-hexyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-Chloro-4-hydroxy-3-hydroxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-isopropyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-isopropyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-thione 2-Chloro-4-hydroxy-3-isopropyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-isopropyl-5-phenylthieno[2,3-b]pyridin-6(7H)-thione 2-Chloro-4-hydroxy-3-methoxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-methyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-5-(3-phenoxyphenyl)-3-propylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine 2-Chloro-5'-methylthioado 2-chloro-5,5a,6,7,8,10-hexahydro-5,8-methanopyrrolo[2,1-g][1,7]naphthyridine 2-chloro-5-(2-prpylidene)-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 2-Chloro-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-Chloro-9-methyladenines 2-Chloro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-benzamide 2-Chloro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)acetamide 2-Chloro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-7-yl)-benzamide 2-chloro-N-(2,6-dimethylphenyl)-N-(2-morpholino-2-(4-nitrophenyl)acetyl)benzamide 2-Chloro-N6-(3-iodobenzyl)-adenosine 2-Chloro-N6-(3-iodobenzyl)adenosine-5'-N-methyluronamide 2-chloro-N6-cyclopentyladenosine 2-Chloroadenosine 2-Chloroado 2-Chloroethyldibenzylamine 2-Chloromelatonin 2-CI Adenosine 2-Cl-CPA 2-CPP 2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-cyclohexyl-3-(4-methoxyphenyl)-N-(6-methylpyridin-2-yl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-4-carboxamide 2-cyclohexyl-5-(2-morpholinoethyl)-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 2-dimethylamino-2-(3-hydroxy-5-methyl-isoxazol-4-yl)acetic acid zwitterion monohydrate, (RS) 2-dimethylamino-2-(3-hydroxy-5-methyl-isoxazol-4-yl)acetic acid zwitterion monohydrate, (RS) 2-dimethylamino-3-(3-hydroxy-5-methyl-isoxalzol-4-yl)-propionic acid zwitterion 2-Ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Ethyl-l,2,3,4-tetrahydro[2,7]naphthyrtdme oxalate 2-Ethynyl-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-Ethynyl-4-(3-fluorophenylethynyl)thiazole 2-exo-(5-(6-Hydroxy-1-hexynyl)-3-pyridyl)-7-azabicyclo[2.2.1]heptane 2-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 2-Fluoro-5'-MethylthioAdo 2-Fluoro-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-FluoroAdo 2-Fluorobenzoic Acid 2-(2-fluorobenzoyloxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester 2-Fluoromethyl-3-{4-[2-(4-methylaminophenyl)vinyl]phenoxy}propan-1-ol 2-fluoronorepinehprine 2-Hydrazinobenzenesulfonamide 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 2-hydroxydibenzodiazepine 2-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 2-Iodomelatonin 2-Me-Tet-AMPA 2-Methoxy-10-allyl-11-hydroxy-N-methylaporphine 2-Methoxy-11-allyloxy-N-methylaporphine 2-methoxy-11-hydroxy-N-propylnoraporphine 2-Methoxy-11-hydroxyaporphine 2-Methoxy-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-methoxy-4-amino-5-chlorobenzoic acid 2-(diethylamino)ethyl ester 2-Methoxy-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-Methoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 2-methoxyapomorphine 2-methoxydibenzodiazepine 2-METHOXYPHENYLPIPERAZINE 2-Methyl- 2.3-dihydro-l H-pyrrolo[3,4-c]pyrMine oxalate 2-Methyl-1-(oxazol-2-yl)-1-oxo-9(Z)-octadecene 2-Methyl-3-(4-phenylpiperazinylmethyl)imidazo[1,2-a]-pyridine 2-Methyl-3-[4-(4-chlorophenyl)piperazinylmethyl]imidazo-[1,2-a]-pyridine 2-Methyl-4-(2-thienylethynyl)thiazole 2-Methyl-4-(3-thienylethynyl)thiazole 2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 2-Methyl-4-(m-tolylethynyl)thiazole 2-Methyl-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2-methyl-4-phenyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 2-Methyl-4-[4-(3-methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine 2-Methyl-4-[[3-(trifluoromethoxy)phenyl]ethynyl]thiazole 2-Methyl-4-[[3-(trifluoromethyl)phenyl]ethynyl]thiazole 2-Methyl-l,2,3.4-tetrahydro[2,7]naphthyridine oxalate 2-methyl-serotonin 2-METHYLPHENYLPIPERAZINE 2-Methylsulfonyloxy-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 2-Methylsulfonyloxy-11-(4-methyl-1-piperazinyl)-dibenz[b,f][1,4]oxazepine 2-Methylthiazole-4-carboxylic Acid 3-Fluorophenylamide 2-Methylthiazole-4-carboxylic Acid 3-Pyridylamide 2-methylthio-ATP 2-MPP 2-MsO-11-(4-methl-1-piperazinyl)-5H-dibenzo [b,e] [1,4]diazepine 2-MsO-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 2-MsO-11-(4-methyl-1-piperazinyl)-dibenz[b,f][1,4]oxazepine 2-NAP 2-NP 2-Oxoado (isoguanosine) 2-Oxoquazepam 2-Phenethylamine 2-Phenylethylamine 2-Phenylmelatonin 2-Piperidino-3'-chloropropiophenone 2-Propyl-l,2,3,4-tetrahydro[2,7]naphthyrMme oxalate 2-Pyrazin-2-yl-1H-benzoimidazol 2-Pyridin-2-yl-1H-benzoimidazol 2-Pyridin-2-yl-3H-benzoimidazol-5-ylamine 2-Pyridin-2-yl-3H-benzoimidazole-5-carbonitrile 2-Pyridin-3-yl-1H-benzoimidazol 2-Pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane 2-Pyrrolidinone, {1-[4-(1-pyrrolidinyl)-2-butynyl]-} 2-Sulfamoylbenzoic acid hydrazide 2-tert-butyl-3-methyl-2,3-dihydroisoquinolin-4(1H)-one 2-tert-Butylamino-3',4'-difluoropropiophenone 2-Thio-3-propylX 2-Thiophen-2-yl-1H-benzoimidazol 2-[ [ 4-(2-Carbomethoxyethyl)phenethyl]amino]-adenosine-5’-N-ethylcarboxamide Hydrochloride 2-[(1R,11S,13S,17S,18R,20R,27S,29R,30R,31S,35E)-19-phenyl-21-oxa-8,14,19,26-tetraazadecacyclo[24.5.2.2^{11,14}.0^{1,27}.0^{2,... 2-[(2-butoxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[(2-methoxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[(2-Methyl-4-thiazolyl)ethynyl]pyrazine 2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]acetic acid bis(tetrafluoroborate) 2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]acetic acid bis(tetrafluoroborate) 2-[1-(2-Bromophenyl)methylidene]-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-[1-(2-Bromophenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 2-[1-(4-Hydroxyphenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 2-[2,5-Dimethoxy-4-(3-phenyl-propyl)-phenyl]-1-methyl-ethylamine 2-[2-(2,4,6-Trimethyl-phenoxy)-acetylamino]-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid (1,1-dioxo-tetrahydro-1lam... 2-[2-(ethoxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[2-(hydroxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)ethanone 2-[4-(2,3-Dimethyl-1H-imidazolium-1-yl)-2-butynyl]isoxazolidin-3-one iodide 2-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]isoxazolidin-3-one sesquifumarate 2-[4-(3-Phenyl-propyl)-phenyl]-ethylamine 2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[p-(2-carboxyethyl)-phenethylamino]-5'-N-ethylcarboxamido adenosine 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-mesitylenepiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-naphthalen-1-ylpiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-o-tolylpiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-o-xylylpiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-[(2,3-dimethoxyphenyl)piperazin-1-yl]ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-[4-(benzodioxan-5-yl)piperazin-1-yl]ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-[4-(o-cyanophenyl)piperazin-1-yl]ethanone 2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]1H-benzimidazole 2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]benzothiazole 2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]benzoxazole 2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]1H-benzimidazole 2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]benzothiazole 2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]benzoxazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]-1-methyl-1H-benzimidazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]1H-benzimidazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]1H-benzimidazole 2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[4-(2-Carboxyethyl)phenethyl]amino]adenosine-5'-N-ethylcarboxamide Hydrochloride 2-[[4-(2-Carboxyethyl)phenethyl]amino]adenosine-5'-N-ethylcarboxamide Hydrochloride 2-[[4-[4-(2-Methoxyphenyl)-1-piperazinyl]butyl]thio]benzothiazole 2-[[4-[4-(2-Methoxyphenyl)-1-piperazinyl]butyl]thio]benzoxazole 2-[[6-[4-(2-Methoxyphenyl)-1-piperazinyl]hexyl]thio]benzothiazole 2-[[6-[4-(2-Methoxyphenyl)-1-piperazinyl]hexyl]thio]benzoxazole 2-{(1H-Pyrrolo[2,3-b]pyridin-3-yl)methyl}-5-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane 2-{1-[2,5-Di(trifluoromethyl)phenyl]methylidene}-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 2-{1-[4-(Dimethylamino)phenyl]methylidene}-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(3,4-dihydroisoquinoline) 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2'-pyrimidil)piperazine 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3'-chlorophenyl)piperazine 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3'-trifluoromethyl)piperazine 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(N-methyl)piperazine 2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-2-aza-spiro[4.5]decane-1,3-dione 2-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol 2-{4-[2-(4-Methylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol 2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione 2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-methyl-amine 20 20-COOH-LTB4 20-OH-LTB4 20a 20b 21 21-nitro-7alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 21-nitro-8alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 21a 21b 21c 22 22-nitro-7apha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 22-nitro-8alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 227I-BOP 22a 22b 23 24 24c 25 26 26A 26B 26c 27 27 (6-PBC) 27a 27b 28 28g 28h 28i 28j 28k 28l 29 29a 29b 2a 2b 2e 2f 2g 2Me4CPG 2R, 4R-APDC 2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2'-methoxyphenyl)piperazine 2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(4'-fluorophenyl)piperazine 3 3 (BCCE) 3'-(3-Aminophenyl)epibatidine 3'-(3-Bromophenyl)epibatidine 3'-(3-Chlorophenyl)epibatidine 3'-(3-Dimethylaminophenyl)epibatidine 3'-(3-Fluorophenyl)epibatidine 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 3'-(3-nitrophenyl)epibatidine 3'-(4-Aminophenyl)epibatidine 3'-(4-Chlorophenyl)epibatidine 3'-(4-fluorophenyl)deschloroepibatidine 3'-(4-Methoxylphenyl)epibatidine 3'-(4-Nitrophenyl)epibatidine 3'-(7-Methyl-imidazo[1,2-b]pyridazin-3-yl)-biphenyl-2-carbonitrile 3'-Deoxyadenosine (cordycepin) 3(R)-Amino-2-(R,S)-hydroxybutyl)phosphinic Acid 3, 4-Dihydroxyphenethylamine 3, {4-Dihydroxy-alpha-[(methylamino)methyl]benzyl} alcohol 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}furan 3,4-dichloro amphetamine 3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7... 3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-Dihydro-2-[4-(3,4-dihydro-6-methoxypyrazino[1,2-a]indol-2(1H)-yl)butyl]pyrazino[1,2-a]indol-1(2H)-one 3,4-Dihydroxyphenylethylamine 3,4-Dimethoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)-oxy]morphinan-6-one 3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-DNH 3,4CTMP 3,5-DHPG 3,5-dihydroxyphenylglycine 3,5-diphenylpyridazine 3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 3,6-diacetyldihydromorphine 3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine 3,7-dimethyl-1-n-propylxantine 3,7-dimethyl-1-proporgylxantine 3,7-Dimethyl-8-(m-hydroxystyryl)-1-propargylxanthine 3,7-dimethylxanthine 3,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine 3,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine 3,9-DimethylX 3-((1-(pyrrolidin-1-yl)cyclopropyl)methoxy)pyridine 3-((1-Methyl-2(R)-azetidinyl)methoxy)pyridine Dihydrochloride 3-((1-Methyl-2(R)-pyrrolidinyl)methoxy)pyridine Dihydrochloride 3-((1-Methyl-2(S)-azetidinyl)methoxy)pyridine Dihydrochloride 3-((1H-Pyrrole-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol 3-((2,2-Dimethylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((2,6-dichlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-fluorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3,3-Difluoroazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3,3-Dimethylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3R,4R)-1-((S)-3-cyclohexyl-3-hydroxypropyl)-3,4-dimethylpiperidin-4-yl)phenol 3-((4-chlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((4-isopropylphenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((Acetoxy)-1-methylpropyl)dimethylammonium Oxalate 3-((Azetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((Benzoyloxy)-1-methylpropyl)dimethylammonium Chloride 3-((Cyclobutanecarbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((Cyclopropanecarbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((Isobutyryloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonit... 3-((S)-1-Azetidin-2-ylmethoxy)-2-fluoro-pyridine 3-(1-methyl-2-pyrrolidinyl)pyridine 3-(1-methyl-2-pyrrolidinyl)pyridine, (+) 3-(1-methyl-2-pyrrolidinyl)pyridine, (-) 3-(1-methyl-2-pyrrolidinyl)pyridine, (S) 3-(1-Methylcyclopropyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine1,1-Dioxide 3-(2(R)-Azetidinylmethoxy)pyridine Dihydrochloride 3-(2(R)-Pyrrolidinylmethoxy)pyridine Dihydrochloride 3-(2(s)-Azetidinylmethoxy) Pyridine 3-(2,4-dithioxo-1,3-thiazolidin-3-yl)propanoic acid 3-(2-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-yl)eth... 3-(2-(allylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(benzylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(5-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(6,7-dichloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-... 3-(2-(butylamino)ethyl)-8-(6-chloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-on... 3-(2-(butylamino)ethyl)-8-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclobutylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclohexylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclohexylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-... 3-(2-(cyclopentylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclopropylmethylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclopropylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4... 3-(2-(diisopropylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(S)-Pyrrolidinylmethoxy)pyridine Fumarate 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide 3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(2-Aminoethyl)-2-chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one hydrochloride 3-(2-Aminoethyl)-2-chloro-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one hydrochloride 3-(2-aminoethyl)-8-(bis(2-chlorophenyl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-Dimethylaminoethyl)-4-hydroxy 2-methylindole 3-(2-Dimethylaminoethyl)-6-hydroxyindole 3-(2-DIMETHYLAMINOETHYL)INDOL-5-OL 3-(2-Hydroxyethyl)-8-(m-methoxystyryl)-7-methyl-1-propargylxanthine 3-(2-Methoxy-phenyl)-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-acrylamide 3-(3-hydroxypentyl)-N-(1-propyl)piperidine 3-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane 3-(4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxybenzofuran-2-yl)-N-(2-(dimethylamino)ethyl)benzamide 3-(4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-ylamino)propan-1-ol 3-(4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl)benzoic acid 3-(4-(3-(methoxymethyl)-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-(4-fluorophenyl)naphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-(4-hydroxyphenyl)naphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-(4-methoxyphenyl)naphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-6-hydroxy-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-cyclopropyl-6-hydroxy-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(4-cyclohexylpiperazin-1-yl)butyl)benzo[d]thiazole-2(3H)-thione 3-(4-(6-hydroxy-3-isobutyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(6-hydroxy-3-octyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(6-hydroxy-3-pentyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-aminobenzyl)indene 3-(4-aminobenzyl)indole 3-(4-aminophenethyl)-7-(2-(ethyl(2-hydroxyethyl)amino)ethyl)-1-propyl-1H-purine-2,6(3H,7H)-dione 3-(4-Benzyl-piperazin-1-yl)-phenol 3-(4-Chlorophenyl)-1-(1H-indol-3-ylmethyl)pyrrolidin-3-ol 3-(4-Chlorophenyl)-1-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrrolidin-3-ol 3-(4-Chlorophenyl)-1-[2-(1H-indol-3-yl)ethyl]pyrrolidin-3-ol 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2,2-trifluoroethyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2-difluorobutyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2-difluoropropyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-isopropyl-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-5-morpholin-4-yl-1,2,4-oxadiazole 3-(4-Chlorophenyl)-8-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-Chlorophenyl)-8-(4-fluorobenzyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-(2-hydroxy-2-methylpropyl)-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidin... 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[3-(dimethylamino)propyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine... 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(methyl)-piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidi... 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(pyrrolidin-1-yl)butyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidin... 3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide 3-(4-chlorophenyl)deschloroepibatidine 3-(4-Fluorophenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-(4-Methoxyphenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-(4-Propyl-1-piperazinyl)phenol 3-(4-tert-butylbenzoyl)-2-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)thiazolidine-4-carboxamide 3-(5-Benzoyl-2-isobutoxyphenyl)propionic Acid 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluor... 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(propylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Phenylpyridazin-3-yl)benzonitrile 3-(6-Ethoxypyridazin-4-yl)benzonitrile 3-(6-ethylaminopyridazin-4-yl)-benzonitrile 3-(6-methylpyridin-2-ylcarbamoyl)phenyl methanesulfonate hydrobromide 3-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester 3-(6-Phenyl-pyridazine-4-yl)-benzoic acid methyl ester 3-(6-Phenylpyridazin-4-yl)benzonitrile 3-(8-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-yl)oct... 3-(8-(3,4-dichlorophenyl)-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)-N,N-diethylpropan-1-amine 3-(8-(3,4-dichlorophenyl)-6-methyl-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)-N,N-diethylpropan-1-amine 3-(azepan-1-yl)-N,5-dicyclopropyl-2-methylbenzenamine 3-(benzo[d][1,3]dioxol-5-yl)-N-(2-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-2-oxo-1-p-tolylethyl)-N-methylacrylamide 3-(Benzyloxy)-5-(3-bromophenyl)pyridazine 3-(Benzyloxy)-5-(3-cyanophenyl)pyridazine 3-(benzyloxy)-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3-(dimethylamino) butyl pyrrolidine-1-carboxylate 3-(dimethylamino)butyl dimethylcarbamate 3-(dimethylamino)butyl methylcarbamate 3-(dimethylamino)butyl piperidine-1-carboxylate 3-(Dimethylamino)fluoranthene 3-(N-Cyclopropyl-N-methylaminornethyl)pyrMine oxalate 3-(N-Formylcarbamoyl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-(N-Methyl-N-n-peno, laminomethyl)pyrtdine oxalate 3-(N-Methyl-N-n-propylaminomethyl)pyridine oxalate 3-(N-Methyl-N-n-propylammomethyl)-2-methylpyridine oxalate 3-(N-n-Butyl-N-methylaminornethyl)pyridine oxalate 3-(N-propylpiperidin-4-yl)phenol 3-(Phenylsulfonyl)-4-(2-piperidin-1-ylethyl)-1H-indole 3-(Phenylsulfonyl)-4-(2-pyrrolidin-1-ylethyl)-1H-indole 3-(Phenylsulfonyl)-4-(3-piperidin-1-ylpropyl)-1H-indole 3-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 3-(pyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane 3-(Pyrrol-1-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-(tert-butylamino)-1-(3-chlorophenyl)-2-methylpropan-1-one 3-(Thien-2-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-(Thien-3-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)benzonitrile 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyrazine-2-carbonitrile 3-allyl-8-benzhydryl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-Amino-5-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carbothioamide 3-amino-6-ethyl-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propylthio)thieno[2,3-d]pyrimidin-4(3H,4aH,7aH)-one 3-Aminofluoranthene 3-AMTBI 3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester 3-benzyl-5-cyclopentyl-1-propylxanthine 3-benzyl-N1-(N,N-dimethylaminoethyl)indole 3-Benzylamino-6-chloro-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 3-beta-hydroxyethyl-1-methylxantine 3-Bromo-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-bromo-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-bromoboldine 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3-chloro-5,7,8,9,9a,10-hexahydro-7,10-methanopyrrolo[1,2-b][2,6]naphthyridine 3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 3-Chloro-N-(1,2,3,4-tetrahydro-1,3,4-trioxoisoquinolin-6-yl)propanamide 3-chloro-N-(4-methylthiazol-2-yl)benzamide hydrobromide 3-chloro-N-(6-chloropyridin-2-yl)benzamide hydrobromide 3-chloro-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-CPP 3-cyano-N-(6-methylpyridin-2-yl)benzamide 3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one 3-Cyclopropyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 3-Deoxy-1,2-O-isopropylidene-D-glucose 3-desoxy-3-carboxamidonaltrexone 3-Ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 3-ethyl-1-NP 3-ethyl-2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-1H-benzimidazole-1-carboxamide 3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid (8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-amide 3-Ethyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 3-Ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 3-ethyl-THIQ 3-Ethynyl-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-Fluoromethyl-7-bromo-THIQ 3-Fluoromethyl-7-cyano-THIQ 3-Fluoromethyl-7-N-(4-chlorophenyl)aminosulfonyl-THIQ 3-Fluoromethyl-7-nitro-THIQ 3-fluoromethyl-THIQ 3-Heptanone, 6-(dimethylamino)-4,4-diphenyl-, (+-)- 3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid, (RS) 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3-Hydroxy-9-aminomethyl-9,10-dihydroanthracene 3-Hydroxymethyl-7-nitro-THIQ 3-Hydroxymethyl-THIQ 3-Hydroxytyramine 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine4-oxide 3-iodo-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-Iodoboldine 3-isobutyl-1-methyl 3-isobutyl-1-methyl-7-n-propylxantine 3-isobutyl-1-methyl-7-propargylxantine 3-Isobutyl-1-methylxanthine 3-isobutyl-1-methylxantine 3-isopropyl-1-methyl 3-isopropyl-2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-1H-benzimidazole-1-carboxamide 3-methoxy-4-((S)-((S)-morpholin-2-yl)(phenyl)methoxy)benzonitrile 3-methoxy-9-aminomethyl-9,10-dihydroanthracene 3-methoxy-dibenz[d,g]azecine 3-methoxy-N-(4-methylthiazol-2-yl)benzamide hydrobromid 3-methoxy-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-Methoxymethyl-THIQ 3-METHOXYPHENYLPIPERAZINE 3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 3-Methyl-2-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-benzonitrile 3-Methyl-2-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-phenol 3-methyl-2-(4-(3-(pyrrolidin-1-yl)propoxy)phenyl)quinazolin-4(3H)-one 3-Methyl-2-morpholin-4-yl-7-[(4-phenylpiperazin-1-yl)methyl]-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 3-Methyl-6-phenyl-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole 3-Methyl-7-nitro-THIQ 3-Methyl-7-[(4-phenylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 3-Methyl-7-[(4-pyridin-2-ylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 3-methyl-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-methyl-THIQ 3-N,N-dimethylaminobutyl-N,N-dimethylcarbamate 3-n-Hexyl-6-methoxy-9-aminomethyl-9,10-dihydroanthracene 3-n-Pentyloxy-9-aminomethyl-9,10-dihydroanthracene fumarate 3-phenyl-1-NP 3-Phenyl-2-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-propionic acid te... 3-Phenyl-4-N-phenylamino-1-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrazolo[3,4-d]pyrimidine 3-Phenyl-4-N-phenylamino-1-alpha-L-lyxofuranosylpyrazolo[3,4-d]pyrimidine 3-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine 3-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine 3-Phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 3-Propylxanthine (enprofylline) 3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)urea 3-tert-Butyl-2-chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]-pyridin-6(7H)-one 3-Trifluoromethylphenylpiperazine 3-[(1,4-cis)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-cis)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-cis)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-trans)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-trans)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-trans)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(2,4-dimethoxy)benzylidene]-anabaseine 3-[(2,5-Dimethyl-4-thiazolyl)ethynyl]pyridine 3-[(2-Methyl-4-oxazolyl)ethynyl]pyridine 3-[(2-Methyl-4-thiazolyl)ethynyl]-5-vinylpyridine 3-[(2-Methyl-4-thiazolyl)ethynyl]benzamide 3-[(2-Methyl-4-thiazolyl)ethynyl]benzonitrile 3-[(2-Methyl-4-thiazolyl)ethynyl]phenol 3-[(2-Methyl-4-thiazolyl)ethynyl]quinoline 3-[(2-Methyl-5-phenyl-4-thiazolyl)ethynyl]pyridine 3-[(5-Ethyl-2-methyl-4-thiazolyl)ethynyl]pyridine 3-[2-(DIMETHYLAMINO)ETHYL]-2-METHYLINDOLE 3-[2-(DIMETHYLAMINO)ETHYL]-2-METHYLINDOLE 3-[2-Benzyloxy-5-(4-isobutoxybenzoyl)phenyl]propionic Acid 3-[2-Isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propionic Acid 3-[2-Isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propionic Acid 3-[2-Isobutoxy-5-(4-propoxybenzoyl)phenyl]propionic Acid 3-[3-(4-Isobutoxybenzoyl)phenyl]propionic Acid 3-[3-(Imidazol-4(5)-yl)propyl]-1-[3-[N-(4-bromobenzyl)-N-(pyrid-2-yl)amino]propyl]-S-methylisothiourea Hydroiodide Dihydrochl... 3-[4-(2,3-Dimethyl-1H-imidazolium-1-yl)-2-butynyl]oxy-delta2-isoxazoline iodide 3-[4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl]benzoic acid methyl ester 3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxy-delta2-isoxazoline sesquifumarate 3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxyisoxazole sesquifumarate 3-[4-(2-Methyl-3-(4-bromobenzyl)-1H-imidazolium-1-yl)-2-butynyl]oxyisoxazole bromide 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(3-Aminopropoxy)-3-bromophenyl]-N-[2-(4-chlorophenyl)ethyl]-2- hydroxyiminopropanamide 3-[4-(3-Fluorophenylethynyl)-2-thiazolyl]-2-propyn-1-ol 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Es... 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylami... 3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(methylsulfonyl)phenyl]-5-(trifluoromethyl)(2-pyridyl) phenyl ketone 3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 3-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butoxy]isoquinoline 3-[5-(4-Isobutoxybenzoyl)-2-propoxyphenyl]propionic Acid 3-[5-[(2-Methyl-4-thiazolyl)ethynyl]-3-pyridyl]-2-propyn-1-ol 3-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyloxy]isoquinoline 3-[6-(2,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[6-(2-Fluorophenyl)-pyridazin-4-yl]benzonitrile 3-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[6-(4-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclo-hexyl]-1H-indole 3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclohexyl]-2-methyl-1H-indole 3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-1H-indole 3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-2-methyl-1H-indole 3-[[3-(5-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide 3-[[3-(7-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide 3-{(1,4-cis)-4-[(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine 3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-isopropyl-1H-indole-5-carbonitrile 3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile 3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile 3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-pipera-zin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile 3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile 3-{(1,4-trans)-4-[4-(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine 3-{(4-(Pyrimidin-2-yl)piperazin-1-yl)methyl}-1H-pyrrolo[2,3-b]pyridine 3-{(Cyclopropylmethyl)[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Cyclopropylmethyl)[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Cyclopropylmethyl)[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Cyclopropylmethyl)[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid 3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid Methyl Ester 3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(3,4-dihydroisoquinoline) 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(2'-methoxyphenyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(2'-pyrimidyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3'-chlorophenyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3'-methyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3'-trifluoromethylphenyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(4'-fluorophenyl)piperazine 3-{4-Amino-5-[4-(3-m-tolylureido)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N,N-dimethylpropionamide 3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N-methylpropanamide 3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}propanamide 3-{4-[(1,4-cis)-4-(1H-Indol-4-yl)-pipera-zinyl-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 3-{4-[(1,4-trans)-4-(1H-indol-4-yl)-pipera-zinyl-1-yl]cyclohexyl}-1H-indole-5-carbonitrile 3-{4-[2-(4-Aminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol 3-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N,N-dimethylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-isopropylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-propylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxylic Acid 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-(cyclopropylmethyl)-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopentyl-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopropyl-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-ethyl-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide 3-{Cyclobutyl[3-(5-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(6-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(7-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{[(1S)-1-(4-Bromophenyl)ethyl]amino}-6-chloro-4H-thieno-[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 3-{[3-(5-Fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide 3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine 3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-5,7-dimethylimidazo[1,2-c]pyrimidine 3-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]methyl}-1Hpyrrolo[2,3-b]pyridine 3-{[4-(4-Chlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}2,5,7-rimethylimidazo[1,2-c]pyrimidine 3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3- carbonyl]-amino}-butyric acid 1-ethyl-1-me... 3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid 1-ethyl-1-m... 3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid 1-isobutyl-... 3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid ethyl ester 3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid tert-butyl ... 30 30a 30b 30m 30n 30o 30p 31 31 (ZK 93423) 31a 31b 32 32 (abecarnil) 32a 32b 32D-W-NPY 33 33a 33b 33bMet 34 34a 34b 35 36 37 38 39 3a 3alpha-Hydroxy-3beta-octyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-phenyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-phenylethyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-phenylmethyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-propyl-5alpha-androstan-17-one 3b 3beta-4-ChloroBZT 3beta-Cyclohexyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-Cyclohexylethyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-Cyclohexylmethyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-n-Butyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-n-Hexyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-s-Butyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-tert-Butyl-3alpha-hydroxy-5alpha-androstan-17-one 3c 3C4HPG 3CTMP 3CTMPNMe 3d 3e 3f 3FLB 3g 3h 3H-GR113808 3HPG 3i 3j 3k 3l 3m 3PPP(+/-) 3PPP,(+) 3PPP,(-) 3PPP,(R) 3PPP,(S) 4 4 (3EBC) 4'deoxy EM-A enolether 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 4, 9-DB-3-4-3 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 4,4'-DifluoroBZT 4,5a-Epoxy-3-methoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)oxy]morphinan-6-one 4,5a-Epoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)oxy]3-[(prop-2-ynyl)oxy]morphinan-6-one 4,5alpha-Epoxy-3-hydroxy-5beta,17-dimethyl-14beta-[(3-phenylpropyl)oxymorphinan-6-one 4-((1-Bromo-2-naphthyl)methyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxyphenol 4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-cyclohexylpiperazine-1-carboxamide 4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxy-N-(quinuclidin-3-yl)benzofuran-2-carboxamide 4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-N-(2-(dimethylamino)ethyl)-7-methoxybenzofuran-2-carboxamide 4-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonit... 4-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-6-ylcarbamoyl)-butyric acid 4-(1-(1-(1H-indol-3-yl)propan-2-yl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(2-methoxyethyl)pyrimidin-2-amine 4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(3-methoxypropyl)pyrimidin-2-amine 4-(1-(2-(1H-pyrazol-4-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(5-chloro-1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(benzo[b]thiophen-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-bromo-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 4-(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 4-(1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 4-(1-hydroxy-2-(4-(4-hydroxyphenyl)butan-2-ylamino)ethyl)phenol 4-(1-hydroxy-2-(methylamino)ethyl)-1,2-benzenediol 4-(1H-imidazol-1-yl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide 4-(1H-indol-4-yloxy)-1-(cyclohexylamino)butan-2-ol 4-(1H-indol-4-yloxy)-1-(isopropylamino)butan-2-ol 4-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)morpholine 4-(2,2-Diphenyl-1-ethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-(2,4-Dichloro-5-methoxyanilino)-7-methoxy-8-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyanilino)-8-methoxy-7-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyphenylamino)-7-[2-(4-hydroxypiperidin-1-yl)ethoxy]-8-methoxybenzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyphenylamino)-8-[2-(4-hydroxypiperidin-1-yl)ethoxy]-7-methoxybenzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloroanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloroanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,5-dichlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexanol 4-(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-ylsulfonyl)morpholine 4-(2-(3,4-Dimethylphenylamino)ethyl)-1H-imidazole 4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole 4-(2-(4-Cyclohexylphenylamino)ethyl)-1H-imidazole 4-(2-(4-Methoxyphenylamino)ethyl)-1H-imidazole 4-(2-(4-Methylphenylamino)ethyl)-1H-imidazole 4-(2-(4-tert-Butylphenylamino)ethyl)-1H-imidazole 4-(2-(4-Trifluoromethylphenylamino)ethyl)-1H-imidazole 4-(2-(Cyclohexylamino)ethyl)-1H-imidazole 4-(2-(Phenylamino)ethyl)-1H-imidazole 4-(2-acetylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-amino-1-hydroxyethyl)-1,2-benzenediol 4-(2-Amino-propyl)-2,5-dimethoxy-phenol 4-(2-aminoethyl)-1,2-benzenediol 4-(2-Aminoethyl)pyrocatechol 4-(2-aminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Azepan-1-ylethyl)-3-(phenylsulfonyl)-1H-indole 4-(2-butylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-carboxamidophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Chloro-4-fluoro-5-methoxyanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2-Chloro-5-methoxy-4-methylanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2-Chloro-5-methoxy-4-methylanilino)-8-[2-(4-hydroxypiperidin-1-yl)ethoxy]-7-methoxybenzo[g]quinoline-3-carbonitrile 4-(2-chlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(2-chlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(2-chlorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-cyanophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-dimethylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-(2-ethylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-fluorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(2-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Fluorophenylethynyl)-2-methylthiazole 4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-(2-Methoxyphenylethynyl)-2-methylthiazole 4-(2-methylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-methylsulfonamidophenyl)-N-(1,2,3,tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-(2-Naphthylmethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-(2-nitrophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)cyclohexanol 4-(2-propylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-pyridinyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-pyridinyl-N-oxide)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(3,3-Diphenyl-1-propyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-(3,4-Dichlorophenyl)-1-methylpiperidine-4-carbonitrile 4-(3,4-Dichlorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(3,4-dichlorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dichlorophenyl)-7-((1-isopropylpiperidin-4-yl)methoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dichlorophenyl)-7-((1-isopropylpiperidin-4-yl)methoxy)-2-methyl-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dichlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(3,4-dichlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one 4-(3,4-dimethoxyphenyl)-2-(5-((R)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1... 4-(3,4-dimethoxyphenyl)-2-(5-((S)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1... 4-(3,5-Difluorophenylethynyl)-2-methylthiazole 4-(3-(4-(piperidin-1-yl)but-1-ynyl)benzyl)morpholine 4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 4-(3-chloro-4-methoxyphenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(3-chlorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3-chlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(3-Chlorophenylethynyl)-2-methylthiazole 4-(3-Fluorophenylethynyl)-2-methylthiazole 4-(3-Fluorophenylethynyl)-2-thiazolylamine 4-(3-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3-Methoxyphenylethynyl)-2-methylthiazole 4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester 4-(3-piperidin-1-yl-propoxy)-benzonitrile 4-(3-piperidin-1-ylpropoxy)benzonitrile 4-(3-Pyridylethynyl)-2-thiazolylamine 4-(4-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)piperazin-1-yl)indolin-2-one 4-(4-((phenethylamino)methyl)phenoxy)benzamide 4-(4-(3-((methylamino)methyl)-4-(4-(methylthio)phenoxy)phenyl)but-3-ynyl)piperazin-2-one 4-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)benzonitrile 4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-1-phenylbutan-1-one 4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(difluoromethoxy)phenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-N-phenylbenzamide 4-(4-aminobenzenesulfonyl)-1-NP 4-(4-Bromo-2-chlorophenylamino)-5,6-dichloro-N-(2-hydroxyethoxy)nicotinamide 4-(4-Bromo-2-chlorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-6-methoxynicotinamide 4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-5-fluoro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-chloro-3-fluorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Chloro-5-methoxy-2-methylanilino)-7-methoxy-8-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-5-methoxy-2-methylanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-5-methoxy-2-methylanilino)-8-methoxy-7-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-5-methoxy-2-methylanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-phenyl)-1-(1H-indol-3-ylmethyl)-piperidin-4-ol 4-(4-Chlorophenyl)-1-(3-phenoxypropyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4,4-diphenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-(3,4-dichlorophenyl)-4-phenylbutyl)piperidin-4-ol Hydrochloride 4-(4-Chlorophenyl)-1-(4-(4-chlorophenyl)-4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-(4-methoxyphenyl)-4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-cyano-4,4-diphenylbutyl)-4-hydroxy-1-methylpiperidinium Iodide 4-(4-Chlorophenyl)-1-(4-hydroxy-4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-phenyl-4-m-tolylbutyl)piperidin-4-ol Hydrochloride 4-(4-Chlorophenyl)-1-(4-phenyl-4-p-tolylbutyl)piperidin-4-ol Hydrochloride 4-(4-Chlorophenyl)-1-(4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Chlorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-Chlorophenyl)-1-pyrid-2-yl-pyrazole 4-(4-chlorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Chlorophenyl)-5-(2,4-dichlorophenyl)-N-(piperidin-1-yl)thiazolecarboxamide 4-(4-chlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(4-chlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-ethoxyphenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(4-Fluorophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Fluorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Easter 4-(4-Fluorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-fluorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Fluorophenylethynyl)-2-methylthiazole 4-(4-Idophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Iodophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Iodophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)ethyl)azetidin-2-one 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(pyridin-4-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(thiazol-2-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(trifluoromethyl)piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-methoxyphenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine 4-(4-Methylphenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Methylphenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(6-(4-chlorophenyl)-2,6-diazabicyclo[2.2.1]heptan-2-yl)-1-(4-fluorophenyl)butan-1-one 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzamide 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoic Acid 4-(6-methoxy-2-(4-methoxyphenyl)benzofuran-3-carbonyl)benzonitrile 4-(6-Phenylpyridazin-4-yl)benzonitrile 4-(7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)benzonitrile 4-(8-benzyl-5-cyano-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-propylpiperazine-1-carboxamide 4-(adamantan-1-ylamino)-1-(1H-indol-4-yloxy)-butan-2-ol 4-(Bis(2-bromoethyl)amino)-2,3,5-trifluorobenzoic Acid 4-(Bis(2-bromoethyl)amino)-3,5-difluorobenzoic Acid 4-(Bis(2-chloroethyl)amino)-2,3,5,6-tetrafluorobenzoic Acid 4-(Bis(2-chloroethyl)amino)-2,3,5-trifluorobenzoic Acid 4-(Bis(2-chloroethyl)amino)-3,5-difluorobenzoic Acid 4-(Bis(2-iodoethyl)amino)-2,3,5,6-tetrafluorobenzoic Acid 4-(Bis(2-iodoethyl)amino)-2,3,5-trifluorobenzoic Acid 4-(Bis(2-iodoethyl)amino)-3,5-difluorobenzoic Acid 4-(Diacetylamino)-l-ethyl-[ 1,2,4]triazolo[4,3-a]quinoxaline 4-(diethylamino) [ 1,2,4]triazolo[4,3-a]quinoxaline 4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 4-(Dimethylaminomethyl)-6-methoxy-1,2,3,4-tetrahydrocarbazole Oxalate 4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzamide 4-(N-(2-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(3,4-dichlorophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-acetylphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-benzyloxyphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-biphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-bromophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-chlorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-ethyloxycarbonylphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfona mide 4-(N-(4-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-nitrophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-phenoxyphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-fluorenylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-phenylsulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile 4-({4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazin-1-yl}carbonyl)morpholine 4-({[4-(2,4-Diamino-6-ethylpyrimidin-5-yl)phenyl]amino}methyl)benzonitrile 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 4-Amino Phosphonobutyrate 4-Amino-1-(2-hydroxy-3-nonyl)pyrazolo[3,4-d]pyrimidine 4-Amino-1-(beta-hydroxyethyl)pyrazolo[3,4-d]pyrimidine 4-amino-2-decylpyrazolo[3,4-d]pyrimidine 4-Amino-3-bromo-1-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrazolo[3,4-d]pyrimidine 4-Amino-3-bromo-1-alpha-L-lyxofuranosylpyrazolo[3,4-d]pyrimidine 4-Amino-4'-hydroxystilbene 4-Amino-5-bromo-7-(5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-bromo-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(4'-C-spirocyclopropyl-beta-D-erythro-pentofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(5-O-methyl-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine 4-Amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Aminobutanoic acid 4-aminobutanoic acid 4-Aminobutyric acid 4-ARA-127 4-benzenesulfonyl-1-NP 4-benzhydryl-N-butylpiperazine-1-carboxamide 4-benzhydryl-N-cyclohexylpiperazine-1-carbothioamide 4-benzhydryl-N-cyclohexylpiperazine-1-carboxamide 4-benzoyl-1-NP 4-benzyl-1-NP 4-Benzyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-bromo-1-NP 4-carboxybenzenesulfonamide 4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-chloro-3-hydroxy-dibenz[d,g]azecine 4-Chloro-N-(1,2,3,4-tetrahydro-1,3,4-trioxoisoquinolin-6-yl)butanamide 4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}... 4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl]-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptylamino]-methy... 4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl][4-(1,2,3,4-tetrahydroacridin-9-ylamino)butylamino]methylen... 4-ChloroBZT 4-CPP 4-cyano-1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 4-Cyano-N-ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]benzamide 4-DAMP 4-diphenylacetoxy-N-methyl-piperadine 4-Ethyl-5-(4-piperidyl)-3-isoxazolol 4-fluoro-2,3,7,11b-tetrahydro-1H-pyrido[3,4,5-k]acridin-8,9-diol 4-Fluoro-3-(2-dimethylaminoethyl)indole 4-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 4-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenylthio)benzylamine 4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-fluoro-N-(3-(1-(2-(piperidin-1-yl)ethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide 4-fluoro-N-(3-(1-(2-hydroxyethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide 4-fluoro-N-(3-(1-octylpiperidin-4-yl)-1H-indol-5-yl)benzamide 4-fluoro-N-(3-{1-[(2E)-4-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)but-2-en-1-yl]piperidin-4-yl}-1H-indol-5... 4-fluoro-N-(3-{1-[10-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)decyl]piperidin-4-yl}-1H-indol-5-yl)benzamid... 4-fluoro-N-(3-{1-[11-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)undecyl]piperidin-4-yl}-1H-indol-5-yl)benzam... 4-fluoro-N-(3-{1-[12-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)dodecyl]piperidin-4-yl}-1H-indol-5-yl)benzam... 4-fluoro-N-(3-{1-[2-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethoxy)ethyl]piperidin... 4-fluoro-N-(3-{1-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)benzamide 4-fluoro-N-(3-{1-[3,3,3-trifluoro-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-ind... 4-fluoro-N-(3-{1-[3-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-indol-5-yl)benzamid... 4-fluoro-N-(3-{1-[6-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)hexyl]piperidin-4-yl}-1H-indol-5-yl)benzamide 4-fluoro-N-(3-{1-[7-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)heptyl]piperidin-4-yl}-1H-indol-5-yl)benzamid... 4-fluoro-N-(3-{1-[9-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)nonyl]piperidin-4-yl}-1H-indol-5-yl)benzamide 4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-benzamide 4-fluoro-N-{3-[1-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethyl)piperidin-4-yl]-1H-... 4-fluoro-N-{3-[1-({3-[(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)methyl]phenyl}methyl)piperidin-4-yl]-1H-ind... 4-fluorodinapsoline hydrobromide 4-HPCA 4-HT 4-Hydrazino-3-chlorobenzenesulfonamide 4-Hydrazino-3-fluorobenzenesulfonamide 4-Hydroxy-1-methylgramine 4-Hydroxy-2,3-dimethyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-2-methyl-5-(2-thienyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-2-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-(2-dimethylaminopropyl)indole 4-Hydroxy-3-(2-pyrrolidin-1-ylethyl)indole 4-Hydroxy-3-(2-thienyl)-5,6,7,8-tetrahydrobenzo[b]thieno[2,3-b]pyridin-2(1H)-one 4-Hydroxy-3-(2-[N-1,2,3,4 tetrahydroquinolino]ethyl)indole 4-Hydroxy-3-(2-[N-methylpiperazino]ethyl)indole 4-Hydroxy-3-(3-dimethylaminopropyl)indole 4-Hydroxy-3-(3-phenoxyphenyl)-1,5,6,7-tetrahydrocyclopenta[4,5]thieno[2,3-b]pyridin-2-one 4-Hydroxy-3-(3-phenoxyphenyl)-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-b]pyridin-2(1H)-one 4-Hydroxy-3-isopropyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methoxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methyl-5-(2-thienyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-phenylquinolin-2(1H)-one 4-Hydroxy-3-phenylthieno[3,4-b]pyridin-2(1H)-one 4-Hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-hydroxydinapsoline hydrobromide 4-hydroxyduloxetine 4-hydroxyduloxetine glucuronide 4-hydroxyduloxetine glucuronide 4-Hydroxygramine 4-Iodo-2,5-dimethoxyphenylisopropylamine 4-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 4-MB-3-3 4-METHOXY-N,N-DIMETHYLTRYPTAMINE 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benzamide 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide 4-METHOXYPHENYLPIPERAZINE 4-Methyl-1-[2-(4-chlorophenoxy)ethyl]piperidine hydrochloride 4-Methyl-1-[3-(4-chlorophenoxy)propyl]piperidine hydrochloride 4-Methyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-methyl[1]benzofuro[3,2-g]quinolin-2-ol 4-N,N'-Dimethylamino-4'-hydroxystilbene 4-N-(2-Methoxyphenyl)amino-5-(4-ethoxyphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3,4-Ethylenedioxyphenyl)amino-5-(2-methylphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3,4-Ethylenedioxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3-Ethoxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3-Pyridyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Bromophenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Chlorophenyl)amino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Chlorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-(4-chlorophenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-(4-ethoxyphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-(4-methoxyphenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Ethoxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-(3-aminophenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-(4-fluorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(4'-C-spirocyclopropyl-beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine 4-N-(4-Hydroxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Hydroxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methoxyphenyl)amino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methoxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methoxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methylphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(Cyanoyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Benzylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Benzylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Cyclohexylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Cyclohexylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Methylamino-4'-hydroxystilbene, SB-13 4-N-Phenylamino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-iodo-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(2,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(2-deoxy-beta-D-erythropentofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(3,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5'-deoxy-4'-C-methyl-beta-D-ribo-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5-amino-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5-azido-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 4-OH-TRYPTAMINE 4-Oxo-4-piperidin-1-yl-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-butyramide 4-P-ADOT 4-P-CADOT 4-P-PDOT 4-phenyl-1-NP 4-phenyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-phenylpiperidine 4-PIOL 4-Piperazino[ 1,2,4]triazolo[4,3-a ]quinoxaline 4-Sulfamoylbenzoic acid hydrazide 4-TrifluoromethylBZT 4-[(1E)-3-({2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(1-pyrrolidinyl)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl}amino)-3-oxo... 4-[(1E)-3-[[2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(2-pyridinylmethoxy)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl]amino]-3... 4-[(2,4-Dichlorophenyl)(p-tolyl)methyl]-N-piperidin-1-ylpiperazine-1-carboxamide 4-[(2,4-Dichlorophenyl)(phenyl)methyl]-N-piperidin-1-ylpiperazine-1-carboxamide 4-[(2-chloro-4-fluorophenyl)(phenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(2-fluoro-4-chlorophenyl)(phenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(3-chlorophenyl)(2,4-dichlorophenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(3-Fluorophenyl)ethynyl]-2-methyloxazole 4-[(4-bromo-2-fluorophenyl)(phenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(5-Amino-1-benzoyl-1H-1,2,4-triazol-3-yl)amino]-benzenesulfonamide 4-[2-(1,1-dimethylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-[2-(1-methylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-[2-(1-Pyrrolidinyl)ethyl]-imidazole 4-[2-(2-Methylpiperidin-1-yl)ethyl]-3-(phenylsulfonyl)-1H-indole 4-[2-(3,4-Dichloro-phenyl)-acetyl]-3-pyrrolidin-1-ylmethyl-piperazine-1-carboxylic acid methyl ester(GR89696) 4-[2-(3-Methylpiperidin-1-yl)ethyl]-3-(phenylsulfonyl)-1H-indole 4-[2-(methylsulfonyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-(1-pyrrolidinyl)pyridine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-fluoropyridine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-methylpyridine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine 4-[3-(4-Benzhydryl-piperazin-1-yl)-2-hydroxy-propoxy]-1H-indole-2-carbonitrile 4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one 4-[3-(4-Phenylpiperazin-1-yl)propoxy]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[3-(4-Phenylpiperazin-1-yl)propoxy]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[3-(4-Phenylpiperazin-1-yl)propyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[3-(4-Phenylpiperazin-1-yl)propyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine 4-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-morpholine 4-[4-(2,4-Diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenoxymethyl]-benzonitrile 4-[4-(3-Methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine 4-[4-(4-Benzylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[4-(4-Benzylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one 4-[4-(4-Phenylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[4-(4-Phenylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[4-(4-Phenylpiperazinilmetil)-1H-1,2,3-triazol-4-yl]acetamide 4-[4-[4-[hydroxy(diphenyl)methyl]-1-piperidinyl]butyl]benzoic acid 4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one 4-[5-Amino-1-(2,6-difluoro-benzenesulfonyl)-1H-[1,2,4]triazol-3-ylamino]-benzenesulfonamide 4-[5-Amino-1-(2,6-difluoro-benzoyl)-1H-[1,2,4]triazol-3-ylamino]-N-(2-dimethylaminoethyl)-benzenesulfonamide 4-[5-Amino-1-(2,6-difluoro-benzyl)-1H-[1,2,4]triazol-3-ylamino]-benzenesulfonamide 4-[6-fluoro-2,2-bis-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-ylmethyl]-morpholine 4-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-butyric acid 4-[[3-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-5-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2,3,6-trifluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2-thienylcarbonyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-[(3,5-dimethyl-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-[(3-fluoro-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-[(3-methyl-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}butyric Acid Methyl Ester 4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2'-pyrimidyl)piperazine 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3'-trifluoromethylphenyl)piperazine 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(N-methyl)piperazine 4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(2-Pyridyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate 4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)] undecane-3,5,8-trione 4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate 4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole 4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole 4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-methyl-1H-benzimidazole 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]piperazin-1-yl}-2-methyl-1H-benzimidazole 4-{[(4-{2,4-Diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}phenyl)amino]methyl}benzonitrile 4-{[4-(3-{4-[(Benzyl{2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)butanoyl]amino}butanoic Acid 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 40 40 (DMCM) 41 42 43 43a 43b 44 44a 44b 44c 44d 44e 44f 45 45a 45b 46 47 48 49 4a 4a-Benzyl-2-chloroethynyl-1,2,3,4,4a,9,10,10a-octahydro-phenanthrene-2,7-diol(CP-394531) 4a-Benzyl-7-hydroxy-3,4,4a,9,10,10a-hexahydro-1H-phenanthren-2-one 4aH-8, {9c-Iminoethanophenanthro[4,5-bcd]furan-5(6H)-one,} N-allyl-7,7a,8, 9-tetrahydro-3,7a-dihydroxy- 4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aR,9aS-(+)-cis-4a-Ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro-[2,3-c]pyridin-6-ol 4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aS,9aR-(-)-cis-4a-Ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro-[2,3-c]pyridin-6-ol 4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4ATMP 4b 4c 4C3HPG 4CPG 4d 4e 4f 4FTMP 4g 4h 4i 4j 4k 4MeTMP 4MeTMPNMe 4OHBA 4OHMNA 4Z,7Z,10Z,13Z,16Z,19Z-Docosahexaenoic acid 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(3,4-dihydroisoquinoline) 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2'-methoxyphenyl)piperazine 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3'-trifluoromethylphenyl)piperazine 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(4'-fluorophenyl)piperazine 5 5'-(Dimethylamino)methyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 5'-(N-ethyl-carbamoyl)adenosine 5'-(N-ethylcarboxamido)adenosine 5'-(Trimethylammonium)methyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]-morphinan Iodi... 5'-Amidinomethyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 5'-amino-5'-deoxy- 5-iodotubercidin 5'-benzyl-12'-hydroxy-2'-isopropyl-3',6',18-trioxoergotaman 5'-benzyl-12'-hydroxy-2'-methyl-3',6',18-trioxoergotaman 5'-ChloroAdo 5'-Deoxy-5'-aminoadenosine 5'-Deoxy-5'-iodoado 5'-Deoxy-5'-isobutylthioadenosine 5'-deoxy-5-iodotubercidin 5'-Deoxyadenosine 5'-guanidinonaltrindole 5'-Methylthioado 5'-N-Biguanidino-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 5'-O-Acetylado 5'-O-Nitroado 5(S)-HETE 5, 6-Dehydroarachidonic acid 5,5-Bis-(4-bromo-phenyl)-3-(2-morpholin-4-yl-ethyl)-imidazolidine-2,4-dione 5,5a,6,7,8,10-hexahydro-5,8-methanopyrrolo[2,1-g][1,7]naphthyridin-2-amine 5,6,7,9-Tetrahydro-8H-pyrldo[3,4-c]azepine oxalate 5,6-DHT 5,6-difluoroindol-methylethylamine 5,6-DIHYDROXY TRYPTAMINE 5,6-dihydroxy-2-(N,N-di-n-propylamino)tetralin ((-)-5,6-diOH-DPAT 5,6-DIHYDROXY-DPAT 5,6-Dihydroxyduloxetine glucuronide 5,6-Dihydroxytryptamine 5,6-dimethoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5,6-dimethoxy-1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5,6-dimethoxy-1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5,6-Dimethyl-2-pyridin-2-yl-1H-benzoimidazole 5,6-Dimethyl-2-thiazol-4-yl-1H-benzoimidazole 5,7,8,9,9a,10-hexahydro-7,10-methanopyrrolo[1,2-b][2,6]naphthyridin-3-amine 5,7-DCKA 5,7-DHT 5,7-DIHYDROXY TRYPTAMINE 5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine 5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-N,N,6-trimethyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 5-(1,2,3,4-Tetrahydro-acridin-9-ylamino)-pentanoic acid [3-(acridin-9-ylsulfanyl)-propyl]-amide 5-(1,4,4-trimethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1H- pyrrole-2-carbonitrile 5-(1-Ethylpropyl)-7-methyl-1-(2-methyl-4-trifluoromethoxyphenyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 5-(1-Ethynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(1-Hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(10-Hydroxy-1-decynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (1,5-dimethyl-hexyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (1-methyl-hexyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (2-diisopropylcarbamoyl-1-methy... 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (3,3-dimethyl-butyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (3-tert-butoxy-propyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid diisobutylamide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid isobutyl-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid isobutyl-methyl-amide 5-(2,2,2-Trifluoroacetyl)-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide 5-(2-Azetidnylmethoxy)-2-Chloropyridine, (R) 5-(2-isopropylidene)-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 5-(2-morpholinoethyl)-2-phenyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 5-(2-Phenyl-1-ethynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole 5-(3,5-dimethyl-piperidine-1-sulfonyl)-3-methyl-benzofuran-2-carboxylic acid 4-methyl-benzylamide 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzofuran-2-carboxamide 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethyl-N-phenethylbenzofuran-2-carboxamide 5-(3-Bromophenyl)-3-ethoxy pyridazine 5-(3-Bromophenyl)-3-isopropoxypyridazine 5-(3-Bromophenyl)-3-methoxypyridazine 5-(3-Bromophenyl)-3-phenyl pyridazine 5-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine 5-(3-Hydroxy-1-propargyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(3-Hydroxy-3-methyl-1-butynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 5-(4,4-diethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile 5-(4,4-Dimethyl-2-thioxo-1,4-dihydro-2H-3, 1-benzoxazin-6-yl)-1H-pyrrole-2-carbonitrile 5-(4-((phenethylamino)methyl)phenoxy)picolinamide 5-(4-(3,4-Dichlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(3-Chloro-4-trifluoromethylphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-(4-Bromophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Chlorophenyl)piperazin-1-yl)-2,2-diphenypentanenitrile 5-(4-(4-Chlorophenyl)piperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Methoxyphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(Diphenylmethylene)piperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Aminophenyl)-6-methylthieno[2,3-d]pyrimidin-4-amine 5-(4-Benzyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Bromophenyl)-1-(2,4-dichlorophenyl)-N-(4-methylpiperazin-1-yl)-1H-pyrazole-4-carboxamide 5-(4-Bromophenyl)-N-cycloheptyl-1-(2,4-dichlorophenyl)-1H-pyrazole-4-carboxamide 5-(4-Bromophenyl)-N-cyclopropyl-1-(2,4-dichlorophenyl)-1H-pyrazole-4-carboxamide 5-(4-Butyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide 5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide 5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide 5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(1-isopropyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(1-isopropyl-5-methyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(2-isopropyl-1H-imidazol-5-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-isopropyl-1H-imidazol-2-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-dihydro-1H-pyrazole-3-carboxylic acid morpholin-4-ylamide bisulphate salt 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylsulfinyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylthio)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylthio)-N-(pyrrolidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-(1-(2-phenylpropan-2-yl)-1H-imidazol-4-yl)-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(7-(N-(1-phenethylpiperidin-4-yl)propionamido)heptyl)-1H-pyrazole-3-carb... 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(4-methylpiperazin-1-yl)-1H-pyrazole-4-carboxamide 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-1,2,4-triazole-3-carboxamide Dihydrochloride 5-(4-chlorophenyl)-3-(1-cyclobutyl-1H-imidazol-4-yl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-3-(1-cyclohexyl-1H-imidazol-4-yl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole 5-(4-Chlorophenyl)-4-(2,4-dichlorophenyl)-N-(piperidin-1-yl)thiazolecarboxamide 5-(4-chlorophenyl)-4-cyano-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-Chlorophenyl)-N-cyclopropyl-1-(2,4-dichlorophenyl)-1H-pyrazole-4-carboxamide 5-(4-ethyl-4-methyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile 5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Hydroxy-4-p-tolylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Hydroxy-4-phenylpiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-Hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-Piperidyl)-4-propylisothiazol-3-ol Hydrobromide 5-(4-{[3,5-Difluoro-4-(methylsulfonyl)benzyl]amino}phenyl)-6-ethylpyrimidine-2,4-diamine 5-(6-Fluoro-1-hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(6-Hydroxy-1-hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(GSyl)-alpha-MethylDopamine 5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methyl-2-butenyl)dihydro-2(3H)-furanone 5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methylbutyl)dihydro-2(3H)-furanone 5-(N-Ethyl)amino-5,0,7,8-tetrahydroquinoline maleate 5-2-Azetidnylmethoxy)-2-Chloropyridine, (R) 5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene-9-carboxylic acid methyl ester 5-Amino-2-thiazol-4-yl-1H-benzimidazol 5-amino-3-(N-methylpiperidin-4-yl)-1H-indole 5-Amino-3-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carboamide 5-Amino-3-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carbothioamide 5-Aminosalicylic acid 5-APT 5-Benzoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-Benzoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-benzyl-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 5-benzyl-7-chloro-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 5-Benzyloxytryptamine 5-Br-T 5-Br-T, 1-Isopropyl 5-Bromo-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 5-bromo-2-(((1R)-3-bromo-2,2-dimethyl-6-methylenecyclohexyl)methyl)-4-methoxyphenol 5-bromo-2-(((1S)-3-bromo-2,2-dimethyl-6-methylenecyclohexyl)methyl)-4-methoxyphenol 5-Bromo-2-((R)-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol 5-bromo-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 5-Bromo-3-(1-methyl-2-pyrrolidinyl)pyridine 5-Bromo-3-(2(S)-azetidinylmethoxy)pyridine 5-bromo-4-methoxy-2-(((1S)-2,2,5-trimethyl-6-methylenecyclohexyl)methyl)phenyl acetate 5-Bromo-4-methoxy-2-((1S,4R)-2,2,4-trimethyl-6-methylene-cyclohexylmethyl)-phenol 5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-Bromotryptamine 5-Butyl-1-(4-chloro-2-cyanophenyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 5-BZT 5-carboxamidotryptamine 5-Carboxyamido Tryptamine 5-Carboxyamido Tryptamine, Dipropyl 5-carboxyl-2,4-di-benzamidobenzoic acid 5-Chlor-2-thiazol-4-yl-1H-benzimidazol 5-Chloro-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 5-Chloro-1H-indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 5-chloro-2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide 5-chloro-2-(1-(3-ethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide 5-chloro-2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide 5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-Chloro-2-pyridin-2-yl-1(3)H-benzoimidazole 5-Chloro-2-[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]thio]benzothiazole 5-Chloro-2-[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]thio]benzoxazole 5-Chloro-3-(2(S)-azetidinylmethoxy)pyridine 5-Chloro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-Chloro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine 5-Chlorotryptamine 5-Cl-T 5-CT 5-CT,DP 5-CT,N,N-DiMe 5-ethyl-3-(1-methyl-2-pyrrolidinyl)pyridine 5-F-6-F3C, 1-(1-indolinyl)-2-propylamines 5-F-6-I, 1-(1-indolinyl)-2-propylamines 5-F-T 5-Fluor-2-thiazol-4-yl-1H-benzimidazol 5-Fluoro-2-[(2-methyl-4-thiazolyl)ethynyl]pyridine 5-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 5-Fluoro-3-[(1,4-cis)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole 5-Fluoro-3-[(1,4-trans)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole 5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole 5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole 5-Fluoro-3-{cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole 5-Fluoro-3-{trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole 5-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-Fluorotryptamine 5-Fluorowillardiine-(S) 5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-HMMP 5-HPCA 5-HT 5-HT, alpha,Omega-dimethyl 5-HT,1-Me 5-HT,2-Me 5-HT,20Me 5-HT,a-Me 5-HT,a-Me-,S(+) 5-HT,b-Me 5-HT,N,N-DIMETHYL 5-HT,N,N-DIPROPYL 5-HT,N-ACETYL 5-HT,o-N 5-HT,omega-N-Me 5-HT,x-Me 5-HTP dipeptide 5-HTQ 5-Hydroxy Tryptamine 5-HYDROXY TRYPTAMINE, 1-Me 5-Hydroxy Tryptamine, 2-Me 5-Hydroxy Tryptamine, Alpha-methyl 5-HYDROXY TRYPTAMINE, b-Me 5-HYDROXY TRYPTAMINE, Omega-N-Me 5-Hydroxy-6-(3-phenoxyphenyl)-3,4-dihydro-2H,8H-1,9-dithia-8-azafluoren-7-one 5-hydroxy-6-methoxyduloxetine 5-hydroxy-6-methoxyduloxetine glucuronide 5-hydroxy-6-methoxyduloxetine sulfate 5-Hydroxy-N,N-dimethyl-1-(benzenesulfonyl)tryptamine 5-HYDROXY-N,N-DIMETHYLTRYPTAMINE 5-hydroxyduloxetine 5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isobutyl-5-methyl-hexanoyloxymethyl)tetrahydro-2-furanone 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 5-hydroxypentanoic acid 5-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 5-M-DMT 5-M-N,N-DMT 5-MCA-NAT 5-ME-URAPIDIL 5-MeOT 5-MeOT,N,N tryptamine 5-MeOT,N,N-DIPROPYL 5-MeOT-N-butanyl 5-MeOT-N-hexanyl 5-MeOT-N-pentanyl 5-MeOT-N-propionyl 5-MET 5-methoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5-Methoxy-1-(2-propyl)-DMT Maleate 5-methoxy-1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5-methoxy-1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5-Methoxy-1-[(5-phenyl-3-pyridyl)carbamoyl-6-triflouromethylindoline 5-Methoxy-1-[[2-methyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[2-[(3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(2,4-dimethyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(2-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(2-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(4-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[4-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[4-(4-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[4-methyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 5-Methoxy-1-[[4-methyl-3-(4-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(4-fluorophenyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(4-methyl-3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(4-pyridyl)-3-pyridyl]carbamoyl-6-trifluoromethylindoline 5-Methoxy-1-[[5-fluoro-4-methyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-phenyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[6-(3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-2-n-propyl-DMT Oxalate 5-Methoxy-2-phenyl-DMT Oxalate 5-Methoxy-3-(di-n-propylamino)chroman 5-METHOXY-3-[2-(DIMETHYLAMINO)ETHYL]INDOLE 5-Methoxy-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-Methoxy-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-Methoxy-N,N-diethyl-1-(4-acetamidobenzenesulfonyl)tryptamine 5-Methoxy-N,N-diethyl-1-(4-aminobenzenesulfonyl)tryptamine 5-Methoxy-N,N-diethyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N,N-dimethyl-1-(4-acetamidobenzenesulfonyl)tryptamine 5-Methoxy-N,N-dimethyl-1-(4-aminobenzenesulfonyl)tryptamine 5-Methoxy-N,N-dimethyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N,N-Dimethyltryptamine 5-Methoxy-N-benzyl-N-methyl-1-(4-aminobenzenesulfonyl)tryptamine 5-Methoxy-N-benzyl-N-methyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N-methyl-1-(benzenesulfonyl)tryptamine 5-Methoxytryptamine 5-Methyl-(3R)-3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-hexanoic aci... 5-Methyl-(3S)-3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-hexanoic aci... 5-Methyl-1-[[2-{(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-methyl-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 5-methyl-10-(4-methylpiperazino)-5H-dibenzo[a,d]cycloheptene 5-Methyl-2-pyridin-2-yl-1(3)H-benzoimidazol 5-Methyl-2-thiazol-4-yl-1(3)H-benzoimidazole 5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 5-Methyl-3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-hexanoic acid ter... 5-Methyl-N,N-Dimethyltryptamine 5-methyl-urapidil 5-Methylthio-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methylthio-1-[[3-(4-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methyltryptamine 5-MOT 5-MT 5-NH2T 5-Nitro-2-pyridin-2-yl-1(3)H-benzoimidazol 5-Nitro-2-thiazol-4-yl-1(3)H-benzoimidazole 5-Nitro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-isophthalamic acid methyl ester 5-OBzlTRYPTAMINE 5-OH-DMT 5-OH-ME-Nw Tryptamine 5-OME-3-ADTN 5-Phenyl-4-N-phenylamino-7-(5-amino-5-deoxy-alpha-L- lyxofuranosylpyrrolo[2,3-d]pyrimidine 5-Phenyl-4-N-phenylamino-7-(5-deoxy-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine 5-Phenyl-4-N-phenylamino-7-(5-O-methyl-alpha-L-lyxofuranosyl)pyrrolo[2,3- d]pyrimidine 5-Phenyl-4-N-phenylamino-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine 5-Propyl-5-normetazocine 5-tert-Butyl-2-pyridin-2-yl-1H-Benzoimidazole 5-tert-Butyl-2-thiazol-4-yl-1H-benzimidazol 5-[(2-Methyl-4-thiazolyl)ethynyl]-1H-indole 5-[(2-Methyl-4-thiazolyl)ethynyl]-2-vinylpyridine 5-[(2-Methyl-4-thiazolyl)ethynyl]pyrimidine 5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(Z)-3-isobutyl-5 -methylhexylidene]tetrahydro-2-furanone 5-[(Z)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine 5-[3-Bromo-4-(4-methanesulfonyl-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 5-[3-Chloro-4-(4-methanesulfonyl-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 5-[4-(1,3-Benzoxazol-2-ylamino)phenyl]-6-methylthieno[2,3-d]pyrimidin-4-amine 5-[4-(2-Amino-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(2-Bromo-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-5-[4-(4-iodo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-5-[4-(4-methoxy-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-piperazin-1-yl-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-carboxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-2-thioxo-dihydro-pyrimidine-4,6-dione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(3-iodo-benzoyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-iodo-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-nitro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-trimethylsilyl-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(isopropyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(4-Chloro-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 5-[4-(4-Chloro-benzylamino)-phenyl]-6-phenethyl-pyrimidine-2,4-diamine 5-[4-(Benzylamino)phenyl]-6-[(benzyloxy)methyl]pyrimidine-2,4-diamine 5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid 5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-(3,4-dihydroisoquinoline) 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2'-methoxyphenyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2'-pyrimidyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(3'-chlorophenyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(4'-fluorophenyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(N-methyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 5-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline 5-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline 5-{4-[(2-Chloro-pyridin-4-ylmethyl)-amino]-phenyl}-6-ethyl-pyrimidine-2,4-diamine 5-{4-[(5-Chloro-thiophen-3-ylmethyl)-amino]-phenyl}-6-ethyl-pyrimidine-2,4-diamine 5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid 5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester 50 50a 50b 51 51a 51b 52 52a 52b 53 53a 53b 54 54a 54b 55 55a 55b 56 56a 56b 57 58 5a 5b 5c 5d 5e 5f 5g 5h 5i 5j 5k 5Z,8Z,11Z,14Z,17Z-eicosapentaenoic acid 6 6'-methylepibatidine 6, PHPNECA 6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6