32340 M4 HEART Chick 3H-NMS BTM1086 2.04174 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
354 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT LSD 2.05 HALL ET AL., 1985 Jan 15, 2025 Jan 15, 2025
41064 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-146 2.05 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
83226 5-HT2A CLONED HUMAN 125I-DOI DOM 2.06 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
20314 BRAIN RAT 3H-D-888 NIFEDIPINE 2.06 Reynolds IJ et al., 1986 Jan 15, 2025 Jan 15, 2025
30558 MOR CLONED HUMAN 3H-Diprenorphine Morphine 2.06 Valenzano KJ et. al., 2004 Jan 15, 2025 Jan 15, 2025
66203 D2 STRIATUM RAT 3H-SPIPERONE (-)-7-Chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3] benzothiazepine 2.06 Campiani G, et al., 1998 Jan 15, 2025 Jan 15, 2025
27048 MOR ILEUM GUINEA PIG 3H-DAMGO H-Tyr-Pro-Phe-Phe-NH2 2.06 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
60184 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyridin-4-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide 2.07 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
53036 DOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(thiophen-2'-yl)acetamido]morphinan 2.07 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
38967 nAChR BRAIN RAT 3H-Cytisine 33bMet 2.07 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
16716 M5 CLONED HUMAN 3H-QNB SCOPOLAMINE 2.07 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
99716 D3 CLONED RAT [3H]spiperone (-)-5-OH-DPAT 2.07 Luo D et al 2016 Jan 15, 2025 Jan 28, 2025
18939 H1 CLONED GUINEA PIG 3H-trans-H2-PAT,(-) CLOZAPINE 2.07 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
8704 SST5 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 2.08 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8456 SST5 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 2.08 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
15368 5-HT1B CLONED HUMAN 3H-5HT CGS 12066B 2.08 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
65554 GABAA CLONED HUMAN [3H] Flunitrazepam FG8205 2.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
38722 D3 CLONED RAT 3H-SCH23390 Dihydrexidine, 4-methyl-N-propyl 2.08 Qandil AM, et al., 2003 Jan 15, 2025 Jan 15, 2025
8786 SST5 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 2.08 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
4972 5-HT2A CLONED RAT 3H-KETANSERIN MIANSERIN 2.08 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
60527 GABAA CLONED HUMAN FNZ FG 8205 2.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
8612 SST3 CLONED MOUSE 125I-Tyr11-SRIF BIM 23003 2.08 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
6834 Y4 CLONED HUMAN 125I-PYY NPY, human 2.08 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
15313 5-HT1D CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 2.08 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
26421 GAL3 CLONED RAT 125I-GALANIN M35 2.0893 Smith KE, et. al., 1998 Jan 15, 2025 Jan 15, 2025
32334 M4 HEART Chick 3H-NMS BENZTROPINE 2.0893 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
39764 5-HT2B CLONED HUMAN 3H-5HT METHIOTHEPIN 2.0893 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
63335 CRF1 CLONED HUMAN 3H-NBI 35965 + GTP GammaS NBI 27914 2.0893 Hoare SR, et al., 2003 Jan 15, 2025 Jan 15, 2025
19081 M1 CLONED HUMAN 3H-NMS (R)-Hexbutinol 2.0893 Dorje F et al., 1991 Jan 15, 2025 Jan 15, 2025
39597 5-HT2B CLONED HUMAN Functional 5-Hydroxy Tryptamine 2.0893 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
8212 SST3 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.09 Corness J, et al., 1993 Jan 15, 2025 Jan 15, 2025
58133 5-HT2C CLONED HUMAN 125I-DOI N-(3-Trifluoromethylbenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 2.09 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
6144 Alpha1A CLONED RAT 125I-HEAT WB 4101 2.1 LOMASNEY JW, ET AL., 1991 Jan 15, 2025 Jan 15, 2025
38146 CLONED RAT 3H-dexamethasone C55H77NO7 2.1 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
51717 NR3C1 UNDEFINED HUMAN UNDEFINED dexamethasone 2.1 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
21513 nAChR CLONED Xenopus 3H-Epibatidine NFEP 2.1 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
60687 GABAA CLONED HUMAN FNZ MSA-IV-35 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
55056 5-HT1A UNDEFINED HUMAN UNDEFINED 8-OH-DPAT 2.1 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
14865 D2 CLONED RAT UNDEFINED OLANZAPINE 2.1 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
37909 CDK1 CLONED HUMAN Functional 4-[[5-Amino-1-[(3-fluoro-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 2.1 Lin R, et al., 2005 Jan 15, 2025 Jan 15, 2025
60693 GABAA CLONED HUMAN FNZ Flunitrazepam 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
93979 D2 CLONED HUMAN 3H-SPIPERONE 2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one 2.1 Ortega R et al 2011 Jan 15, 2025 Jan 29, 2025
37659 5-HT1A Hippocampal RAT 3H-8-OH-DPAT 8-OH-DPAT 2.1 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
36383 CLONED HUMAN 3H-SQ 29548 BM 613 2.1 Hanson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
42783 Y2 CLONED HUMAN 125I-PYY PYY 2.1 Kakui N, et al., 2006 Jan 15, 2025 Jan 15, 2025
57887 SLC6A2 UNDEFINED HUMAN UNDEFINED DESIPRAMINE 2.1 O'Neill DJ et al., 2010 Jan 15, 2025 Jan 15, 2025
91424 5-HT2A CLONED HUMAN 125I-DOI 4-((6bR,10aS)-3-Ethyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone 2.1 Li P et al 2014 Jan 15, 2025 Jan 15, 2025
60198 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2S,3R,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiazol-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide 2.1 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
3879 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 2.1 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 27, 2025
7977 GABAA CLONED HUMAN 3H-RO-15-1788 1 2.1 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
47657 GABAA CLONED HUMAN 3H-RO-15-1788 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 2.1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
63786 A1 CLONED RAT 3H-CCPA 8-(4-Iodophenyl)-1,3-dipropylxanthine 2.1 Hayallah AM, et al., 2002 Jan 15, 2025 Jan 15, 2025
12078 5-HT1D CLONED HUMAN 3H-GR-125743 GR 127935 2.1 Domenech T, et al., 1997 Jan 15, 2025 Jan 15, 2025
15151 BRAIN Monkey 3H-KETANSERIN LY 193525 2.1 Nelson et al., 1993 Jan 15, 2025 Jan 15, 2025
97328 DOR CLONED HUMAN [3H]diprenorphine SRI-22138 2.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
53552 SLC6A2 UNDEFINED HUMAN UNDEFINED DESIPRAMINE 2.1 Mahaney PE et al., 2008 Jan 15, 2025 Jan 15, 2025
11058 H3 CLONED HUMAN 3H-methylhistamine R-alpha-methylhistamine 2.1 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
52018 SLC6A4 UNDEFINED RAT UNDEFINED (2-(3,4-dichlorophenoxy)-5-(4-(4-fluoropiperidin-1-yl)but-1-ynyl)phenyl)-N-methylmethanamine 2.1 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
59954 BRAIN RAT 3H-(-)Nicotine 3-(1-Methyl-2-pyrrolidinyl)-5-propylpyridine 2.1 Dukat, M. et. al., 2005 Jan 15, 2025 Jan 15, 2025
24116 V2 CLONED HUMAN 125I-VIP Vasoactive intestinal polypeptide 2.1 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
55605 SLC6A4 UNDEFINED HUMAN UNDEFINED 2-(Aminoethyl)-5-(2'-methoxy-5'-fluorophenethyl)tetrahydrofuran 2.1 Cashman JR et al., 2009 Jan 15, 2025 Jan 15, 2025
24118 V2 CLONED HUMAN 125I-VIP Ro 25-1553 2.1 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
37174 Y5 BRAIN RAT 125I-hPP NPY [Ala31, Aib32], porcine 2.1 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
31548 D1 Striatal Membranes RAT 3H-SCH23390 C23H26ClFN2 dimaleate (24) 2.1 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
60734 GABAA CLONED HUMAN FNZ TG-4-29 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
10816 D3 CLONED HUMAN 125I-IODOSULPRIDE BUTACLAMOL,(+) 2.1 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
24129 V2 Sup T1 HUMAN 125I-VIP VIP Ala2 2.1 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
32839 D4 STRIATUM CANINE 3H-SPIPERONE ETICLOPRIDE 2.1 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
4170 5-HT1D CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 2.1 HAMBLIN AND METCALF, 1991 Jan 15, 2025 Jan 15, 2025
41802 CLONED HUMAN 3H-Estradiol 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 2.1 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
81229 Alpha2C test test 3H-CLONIDINE 5’-Iodo-HEAT HCl 2.1 Petrie EC et al 2012 Jan 15, 2025 Jan 28, 2025
37710 DOR CLONED HUMAN 3H-Diprenorphine HS414 2.1 Tryoen-Toth P, et al., 2005 Jan 15, 2025 Jan 15, 2025
14928 CLONED RAT UNDEFINED OLANZAPINE 2.1 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
59219 D2 CLONED HUMAN 3H-N-Methylspiporone 6-Chloro-3-{3-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 2.1 Smid P, et al., 2005 Jan 15, 2025 Jan 15, 2025
20820 D2 BRAIN CALF 3H-Haloperidol TRIFLUOPERAZINE 2.1 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
70229 MOR CLONED MOUSE 3H-DAMGO DADLE 2.1 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
20821 D2 BRAIN CALF 3H-Haloperidol Triflupromazine 2.1 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
10838 D3 CLONED HUMAN 125I-IODOSULPRIDE BROMOCRIPTINE 2.1 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
12120 H3 BRAIN RAT 3H-RAMHA Thioperamide 2.1 Arrang JM, et al., 1988 Jan 15, 2025 Jan 15, 2025
65625 GABAA CLONED HUMAN [3H] Flunitrazepam Flunitrazepam 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
4697 5-HT1D CLONED HUMAN 3H-5HT CGS 12066B 2.1 WEINSHANK RL, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
14937 D2 STRIATUM RAT UNDEFINED OLANZAPINE 2.1 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
70234 MOR CLONED MOUSE 3H-DAMGO Endomorphin 1 2.1 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
85594 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate 2.1 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
39002 D2 CLONED HUMAN R-SAT BROMPERIDOL 2.1 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
65377 GABAA CLONED HUMAN [3H] Flunitrazepam MSA-IV-35 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
38754 CLONED RAT 3H-dexamethasone (4-{4-[(Benzyl{2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic Acid 2.1 Link JT, et al., 2005 Jan 15, 2025 Jan 15, 2025
29027 SST2 CLONED HUMAN 125I-LTT-SST-28 SMS 201-995 2.1 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
56419 SLC6A4 UNDEFINED UNDEFINED UNDEFINED (Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride 2.1 White JD et al., 2009 Jan 15, 2025 Jan 15, 2025
65124 GABAA CLONED HUMAN [3H] Flunitrazepam TG-4-29 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
99941 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 2.1 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
8550 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 2.1 Yasuda K, et al., 1992 Jan 15, 2025 Jan 15, 2025
7015 Y1 CLONED MOUSE 125I-PYY NPY2-36 2.1 WEINBERG DH, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
35177 D2 STRIATUM RAT 3H-SPIPERONE (R)-(-)-7-chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine 2.1 Campiani G, et al., 2002 Jan 15, 2025 Jan 15, 2025
64106 V2 CLONED HUMAN 3H-AVP AVP 2.1 Macion-Dazard R, et al., 2005 Jan 15, 2025 Jan 15, 2025
31598 D1 Striatal Membranes RAT 3H-SCH23390 C21H24ClFN2 hemifumarate (41) 2.1 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
13423 D3 CLONED HUMAN 125I-IODOSULPRIDE 7-OH-DPAT,(+) 2.1 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
17520 PANCREAS RAT 125I-VIP VIP Ala16 2.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
17524 PANCREAS RAT 125I-VIP VIP Ala21 2.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
56436 SLC6A2 UNDEFINED HUMAN UNDEFINED DESIPRAMINE 2.1 Zhang P et al., 2009 Jan 15, 2025 Jan 15, 2025
2677 5-HT2A FR. CORTEX HUMAN 125I-LSD SPIPERONE 2.1 ELLIOT & KENT, 1989 Jan 15, 2025 Jan 15, 2025
31605 D1 Striatal Membranes RAT 3H-SCH23390 C23H29FN2 (46) 2.1 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
37493 D3 CLONED HUMAN 125I-IABN 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 2.1 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
2935 5-HT2A CORTEX RAT 3H-MESULERGINE MESULERGINE 2.1 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
6263 EP4 CLONED MOUSE 3H-PGE2 PGE1 2.1 Kiriyama M, et al., 1997 Jan 15, 2025 Jan 15, 2025
65402 nAChR CLONED HUMAN [3H] Flunitrazepam XHE-I-037B (S-enriched) 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
90492 D3 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 2.1 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
16771 SLC6A4 CLONED HUMAN 3H-PAROXETINE S33005 2.1 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
63621 KOR BRAIN GUINEA PIG 3H-U69,593 (3R)-N-((1S)-1-{[(3R,4R)-4-(3-Hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide 2.1 Thomas JB, et al., 2003 Jan 15, 2025 Jan 28, 2025
52102 H3 UNDEFINED HUMAN UNDEFINED 4-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-morpholine 2.1 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
51591 Alpha1D UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide 2.1 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
55946 KOR UNDEFINED HUMAN UNDEFINED (1S,2R,6S,14R,15S,16R)-3-(cyclopropylmethyl)-16-[(2R)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.1^{2,8}.0^{1,6}.0^{6,14}.0^{7,12}]icosa-7(12),8,10-triene-11-carboxamide 2.1 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
69515 NMDA WHOLE BRAIN RAT 3H-MK-801 MK-801,(+) 2.1 Kang, H. et, al. 2017 Jan 15, 2025 Jan 28, 2025
72077 nAChR CLONED HUMAN 3H-Epibatidine 2-methoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 2.1 Magnus CJ et al 2019 Jan 15, 2025 Jan 29, 2025
17550 CLONED HUMAN 125I-VIP VIP Ala15 2.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
64916 CB2 CLONED HUMAN 35S-GTPGammaS SR 144528 2.1 Stern E, et al., 2006 Jan 15, 2025 Jan 15, 2025
1175 5-HT1D CORTEX RAT 3H-5HT 5-Hydroxy Tryptamine 2.1 HERRICK-DAVIS & TITELER, 198 Jan 15, 2025 Jan 15, 2025
61080 GABAA CLONED HUMAN FNZ XHE-II-073B (S-ENRICHED) 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
70297 MOR CLONED MOUSE 3H-Diprenorphine dmt1 DALDA 2.1 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
16027 M3 Parotid gland RAT 3H-NMS ATR 2.1 Bockman CS, et al., 2001 Jan 15, 2025 Jan 15, 2025
90779 MOR brain membranes GUINEA PIG 3H-DAMGO NALOXONE 2.1 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
65694 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073B (S enriched) 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
19360 A1 CLONED HUMAN 3H-NECA 6S, (S)-PHPNECA 2.1 Klotz KN et al., 1999 Jan 15, 2025 Jan 15, 2025
55969 KOR UNDEFINED HUMAN UNDEFINED (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide 2.1 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
50338 NET CELLS HUMAN 3H-Nisoxetine DESIPRAMINE 2.1 Deecher, D., et. al. 2006 Jan 15, 2025 Jan 15, 2025
18596 PANCREAS RAT 125I-CCK-33 21 2.1 Evans BE et al., 1986 Jan 15, 2025 Jan 15, 2025
35750 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE A-80426 2.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
52647 CB2 UNDEFINED HUMAN UNDEFINED WIN 55212-2 2.1 Manera C et al., 2007 Jan 15, 2025 Jan 15, 2025
55209 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(bis(2-chlorophenyl)methyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 2.1 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
39086 D3 CLONED HUMAN R-SAT FLUPHENAZINE 2.1 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
96694 D2 STRIATUM RAT [3H]spiperone N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 2.1 Huang L et al 2020 Jan 15, 2025 Jan 28, 2025
51384 M3 UNDEFINED HUMAN UNDEFINED (4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol 2.1 Sonda S et al., 2007 Jan 15, 2025 Jan 15, 2025
14783 D2 Striatal Membranes CALF 3H-Haloperidol Trifluopromazine 2.1 Creese I, et al., 1976 Jan 15, 2025 Jan 15, 2025
14784 D2 Striatal Membranes CALF 3H-Haloperidol TRIFLUOPERAZINE 2.1 Creese I, et al., 1976 Jan 15, 2025 Jan 15, 2025
55237 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 2.1 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
17607 T47D HUMAN 125I-VIP VIP Ala19 2.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
68809 5-HT3 NG108-15 PIG 3H-DAU 6215 QUIPAZINE 2.1 Schiavi, GB et al., 1994 Jan 15, 2025 Jan 15, 2025
13259 Beta2 BRAIN Mammalian 3H-DHA PROPRANOLOL,(-) 2.1 Bylund DB, et al., 1976 Jan 15, 2025 Jan 15, 2025
51151 Alpha1D UNDEFINED HUMAN UNDEFINED 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 2.1 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51411 D3 UNDEFINED HUMAN UNDEFINED (R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine 2.1 Jung JY et al., 2007 Jan 15, 2025 Jan 15, 2025
97748 Y2 CLONED HUMAN 125I-PYY PYY 2.1 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
4053 DOR CLONED HUMAN 3H-DPDPE-Cl Leu-ENKEPHALIN 2.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
51414 D3 UNDEFINED HUMAN UNDEFINED (R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine 2.1 Jung JY et al., 2007 Jan 15, 2025 Jan 15, 2025
9175 SST3 CLONED MOUSE 125I-CGP23996 BIM 23003 2.1 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
29145 SST1 CLONED HUMAN 125I-Tyr11-SRIF Somatostatin-14 2.1 Reisine T, et.al., 1995 Jan 15, 2025 Jan 15, 2025
51679 5-HT1A UNDEFINED HUMAN UNDEFINED 8-OH-DPAT 2.1 Leopoldo M et al., 2007 Jan 15, 2025 Jan 15, 2025
65764 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-70 (C19H13N4F) 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
38116 CLONED RAT 3H-dexamethasone C57H79N2O9Na 2.1 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
48871 KOR BRAIN Frog 3H-EKC EKC 2.1 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
11498 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RITANSERIN 2.1 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
38636 UNDEFINED HUMAN 3H-hypoxanthine N-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl]-2,4,6-trifluoro-benzamide 2.1 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
53996 CHRNA4 UNDEFINED RAT UNDEFINED 3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 2.1 Hansen CP et al., 2008 Jan 15, 2025 Jan 15, 2025
3316 D3 CLONED HUMAN 3H-YM 09151-2 HALOPERIDOL 2.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
53494 MOR UNDEFINED UNDEFINED UNDEFINED 6-desoxymorphine 2.1 Cunningham CW et al., 2008 Jan 15, 2025 Jan 15, 2025
100090 D3 CLONED HUMAN 3H-N-Methylspiperone Cariprazine 2.1 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
11260 H1 CEREBELLUM GUINEA PIG 3H-PYRILAMINE CLOZAPINE 2.1 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
34557 nAChR CLONED RAT 3H-Epibatidine Cytisine 2.1 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
60925 GABAA CLONED HUMAN FNZ JYI-70 2.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
59647 D5 CLONED HUMAN 3H-SCH23390 SK&F 83959 2.1 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
2879 5-HT2A CORTEX RAT 3H-KETANSERIN LSD 2.11 BATTAGLIA ET AL., 1983 Jan 15, 2025 Jan 15, 2025
37506 D3 CLONED HUMAN 3H-YM 09151-2 N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide 2.11 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
101190 5-HT7 CLONED HUMAN 3H-5-HT 5-Hydroxy Tryptamine 2.12 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
41842 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(4-nitrophenyl)amine 2.12 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
13795 NK1 LUNG GUINEA PIG 125I-Bolton Hunter MDL 105,212 (R)-enantiomer 2.12 Kudlacz EM, et al., 1996 Jan 15, 2025 Jan 15, 2025
26350 KOR CLONED RAT 3H-EKC EKC 2.12 Neal, C. R. Jr. , et al. 2003 Jan 15, 2025 Jan 15, 2025
8794 SST5 CLONED HUMAN 125I-LTT-SRIF28 Tyr10-cortistatin 2.13 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8294 SST4 CLONED HUMAN 125I-Tyr10-CST14 CGP 23996 2.13 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
5000 5-HT2C CLONED RAT 3H-MESULERGINE MIANSERIN 2.13 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
90513 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 2.13 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
22433 A2B CLONED HUMAN 3H-ZM241385 33 2.13 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
8400 SST5 CLONED HUMAN 125I-LTT-SRIF28 CST14-Tyr10 2.13 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
42521 CLONED HUMAN Functional [leu13]pMOT(1-16) 2.13796 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
39767 5-HT2B CLONED HUMAN 3H-5HT RITANSERIN 2.13796 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
64141 D3 CLONED RAT 3H-N-Methylspiperone PERPHENAZINE 2.13796 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
32408 5-HT7 CLONED HUMAN 3H-5CT DR4004 2.13796 Kikuchi, C et al., 1999 Jan 15, 2025 Jan 15, 2025
19105 M3 CLONED HUMAN 3H-NMS (R)-Hexbutinol 2.13796 Dorje F et al., 1991 Jan 15, 2025 Jan 15, 2025
28834 SST5 CLONED HUMAN 125I-LTT-SRIF28 Tyr10-cortistatin 2.13796 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
63664 D2 CLONED HUMAN 3H-N-Methylspiperone RISPERIDONE 2.13796 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
28862 SST4 CLONED HUMAN 125I-Tyr10-CST14 CGP 23996 2.13796 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
839 5-HT2C CORTEX RAT 3H-MESULERGINE MESULERGINE 2.14 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
1358 5-HT1D CAUDATE PIG 3H-5HT METERGOLINE 2.14 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
1359 5-HT1D CAUDATE PIG 3H-5HT METERGOLINE 2.14 WAEBER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
16986 D3 CLONED HUMAN 125I-IODOSULPRIDE PD 128,907 2.14 Cussac D, et al., 2000 Jan 15, 2025 Jan 15, 2025
54907 5-HT1A UNDEFINED HUMAN UNDEFINED (3R)-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-3,4-dihydro-2H-chromen- 2.14 Hatzenbuhler NT et al., 2008 Jan 15, 2025 Jan 15, 2025
1176 5-HT1D STRIATUM BOVINE 3H-5HT 5-Hydroxy Tryptamine 2.14 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
22429 A2B CLONED HUMAN 3H-ZM241385 29 2.14 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
36066 DOR Membranes RAT 3H-[Ile5,6]deltorphin II 14-O-Benzyloxymorphone 2.14 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
60183 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyridin-3-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide 2.15 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
10078 MOR BRAIN MOUSE 125I-Endomorphin-2 Alpha-Neoendorphin 2.15 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
35945 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN 4-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine 2.15 Campiani G, et al., 2005 Jan 15, 2025 Jan 15, 2025
50029 SLC6A3 CAUDATE RAT 3H-dopamine RTI-29 2.15 Rothman RB, et al., 2001 Jan 15, 2025 Jan 15, 2025
64929 DOR BRAIN RAT 3H-DPDPE DPDPE 2.15 Amiche M, et al., 1988 Jan 15, 2025 Jan 15, 2025
55216 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(bis(2-chlorophenyl)methyl)-3-(2-(butylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 2.15 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
21960 DOR ILEUM GUINEA PIG 3H-DADLE DALLE 2.15 Leslie FM et al., 1980 Jan 15, 2025 Jan 15, 2025
65595 GABAA CLONED HUMAN [3H] Flunitrazepam XLI-8TC 2.155 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
61285 GABAA CLONED HUMAN FNZ XLI-8TC 2.155 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60181 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((4-(hydroxymethyl)phenyl)- ethynyl)-6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]- hexane-1-carboxamide 2.16 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
34346 nAChR7 CLONED RAT 3H-MLA Alpha-bungarotoxin 2.16 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 15, 2025
15211 D1 Pineal BOVINE 3H-SCH23390 BUTACLAMOL,(+) 2.16 Simonneaux V., et. At., 1990 Jan 15, 2025 Jan 15, 2025
23695 MC4 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH alpha-MSH, [Nle4, D-Phe7] 2.16 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
60066 A3 CLONED HUMAN 125I-AB-MECA (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(2-(4-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,3- triazol-1-yl)-6-(methylamino)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide 2.16 Tosh, Dipip et. al., 2015 Jan 15, 2025 Jan 15, 2025
100948 NET CELLS HEK293 3H-Nisoxetine MAZINDOL 2.17 Reith ME, et al., 2005 Jan 15, 2025 Jan 15, 2025
60688 GABAA CLONED HUMAN FNZ JYI-19 2.176 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65946 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-19 (C23H23N3O3S) 2.176 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
12882 CLONED HUMAN 3H-RX821002 WB 4101 2.18 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
34402 DOR FOREBRAIN RAT 3H-DPDPE Levallorphan 2.18 Codd EE et al, 1995 Jan 15, 2025 Jan 15, 2025
63646 KOR CLONED HUMAN 3H-U69,593 (3R)-N-((1S)-1-{[(3R,4R)-4-(3-Hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide 2.18 Thomas JB, et al., 2003 Jan 15, 2025 Jan 28, 2025
30121 SST5 CLONED HUMAN 125I-SOMATOSTATIN BIM 23268 2.18 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
8386 SST2 CLONED HUMAN 125I-Tyr3-octreotide octreotide-Tyr3 2.18 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
15304 5-HT1D CLONED HUMAN 3H-5HT 5-Methoxytryptamine 2.18 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
89636 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NLX-101 2.18776 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
39793 5-HT2C CLONED HUMAN 3H-5HT SB 221284 2.18776 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
21995 LHRH Pituitary RAT UNDEFINED 3 2.18776 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
2326 5-HT3 NG108-15 NG 3H-ICS 205-930 GRANISETRON 2.19 NEIJT ET AL, 1988 Jan 15, 2025 Jan 15, 2025
86809 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide 2.19 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
16976 D3 CLONED HUMAN 3H-SPIPERONE 7-OH-DPAT,(+) 2.19 Cussac D, et al., 2000 Jan 15, 2025 Jan 15, 2025
16982 D3 CLONED HUMAN 125I-IODOSULPRIDE HALOPERIDOL 2.19 Cussac D, et al., 2000 Jan 15, 2025 Jan 15, 2025
9728 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl-2-Me 2.2 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
66309 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Finazine 2.2 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
17928 CCK2 BRAIN GUINEA PIG 125I-CCK L-365,260 2.2 Lotti VJ et al., 1988 Jan 15, 2025 Jan 15, 2025
50955 KOR UNDEFINED HUMAN UNDEFINED Nalbuphine 2.2 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
17677 CLONED HUMAN 125I-VIP VIP [D-Arg12] 2.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
1806 5-HT2A CORTEX HUMAN 3H-SPIPERONE CYPROHEPTADINE 2.2 PEROUTKA, 1988 Jan 15, 2025 Jan 15, 2025
69391 H1 CLONED HUMAN 3H-PYRILAMINE Quetiapine 2.2 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
73232 Alpha2B test test 3H-RAUWOLSCINE N-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride 2.2 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
32528 KA BRAIN RAT 3H-Kainic acid Kainate 2.2 Shimamoto K,, et. al., 1998 Jan 15, 2025 Jan 15, 2025
8209 SST4 CLONED HUMAN 125I-LTT-SST-28 somatostatin-28 2.2 Demchyshyn L, et al., 1993 Jan 15, 2025 Jan 15, 2025
65299 GABAA CLONED HUMAN [3H] Flunitrazepam YCT-5 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
37141 STRIATUM RAT 3H-CGS-21680 HENECA 2.2 Cristalli G, et al., 1994 Jan 15, 2025 Jan 15, 2025
45589 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Fluvoxamine 2.2 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
47895 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 2.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
60696 GABAA CLONED HUMAN FNZ Flunitrazepam 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60697 GABAA CLONED HUMAN FNZ YCT-5 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
4122 KOR CLONED HUMAN 3H-U69,593 PENTAZOCINE (-) 2.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
541 5-HT1A CELLS C0S-7 125I-NAPS SPIROXATRINE 2.2 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
5152 5-HT2C CLONED HUMAN 125I-DOI DOTB 2.2 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
23585 Spinal cord RAT 125I-1DMe-Y8Fa FMRFamide 2.2 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
34085 P2X2, P2X3 CLONED HUMAN 3H-A-317491 ATP, 2-meS 2.2 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
66089 CB1 CEREBELLUM RAT 3H-CP55940 Arachidonyl cyclopropylamide 2.2 Hillard CJ, et al., 1999 Jan 15, 2025 Jan 28, 2025
57388 CB1 UNDEFINED HUMAN UNDEFINED N-cyclohexyl-4-[(2,6-dichlorophenyl)(phenyl)methyl]piperazine-1-carboxamide 2.2 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
33838 STRIATUM RAT 3H-RX821002 Brimonidine AppNHp 2.2 Bylund DB, et al., 2001 Jan 15, 2025 Jan 15, 2025
2864 5-HT2A CAUDATE BOVINE 125I-LSD KETANSERIN 2.2 HARTIG ET AL., 1985 Jan 15, 2025 Jan 15, 2025
64817 CCR5 CLONED UNDEFINED 125I-RANTES (S)- (-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(4-propyl-4H-1,2,4-tri azol-3-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 2.2 Seto M, et al., 2006 Jan 15, 2025 Jan 28, 2025
65845 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-III-74 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
56373 CB1 UNDEFINED HUMAN UNDEFINED 2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 2.2 Foloppe N et al., 2009 Jan 15, 2025 Jan 15, 2025
67642 STRIATUM RAT 3H-CGS21680 HENECA 2.2 Cristalli G, et al., 1994 Jan 15, 2025 Jan 15, 2025
4156 5-HT1D CLONED HUMAN 3H-5HT 5-Methoxytryptamine 2.2 HAMBLIN AND METCALF, 1991 Jan 15, 2025 Jan 15, 2025
65599 GABAA CLONED HUMAN [3H] Flunitrazepam 6-PBC 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
6975 D3 CLONED HUMAN 125I-IODOSULPRIDE HALOPERIDOL 2.2 LEJEUNE F, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
51266 SLC6A4 UNDEFINED RAT UNDEFINED N,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine 2.2 Keith JM et al., 2007 Jan 15, 2025 Jan 15, 2025
38724 mGluR5 CLONED RAT 3H-SCH23390 Dihydrexidine, DHX 2.2 Qandil AM, et al., 2003 Jan 15, 2025 Jan 27, 2025
29001 SST1 CLONED HUMAN 125I-LTT-SST-28 somatostatin-28 2.2 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
52041 SLC6A4 UNDEFINED HUMAN UNDEFINED FLUOXETINE 2.2 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
66122 D2 CLONED HUMAN 3H-N-Methylspiperone RISPERIDONE 2.2 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 28, 2025
13386 D3 CLONED HUMAN 3H-thymidine APOMORPHINE 2.2 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
64074 CB2 SPLEEN MOUSE 3H-CP-55940 (R)-(+)-AM2233 2.2 Deng H, et al., 2005 Jan 15, 2025 Jan 15, 2025
16204 D2 LZR1 Cells RAT 125I-Epidepride BUTACLAMOL,(+) 2.2 Neve KA, et al., 1990a Jan 15, 2025 Jan 15, 2025
52557 SLC6A4 UNDEFINED HUMAN UNDEFINED FLUOXETINE 2.2 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
42830 ABL1 CLONED HUMAN 3H-Staurosporine Gleevec 2.2 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
48210 Y4 CLONED RAT 125I-hPP NPY13-36, porcine 2.2 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
9301 GABAA CLONED HUMAN 3H-RO-15-1788 Beta CCM 2.2 Hadingham k, et al.,1993 Jan 15, 2025 Jan 27, 2025
65622 GABAA CLONED HUMAN [3H] Flunitrazepam Flunitrazepam 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
94040 Alpha1A CORTEX PIG 3H-PRAZOSIN 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one 2.2 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
41816 CLONED HUMAN 3H-Estradiol 1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 2.2 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
35929 STRIATUM RAT 3H-SPIPERONE (+)-trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione 2.2 Bogeso KP, et al., 1988 Jan 15, 2025 Jan 15, 2025
32603 Striatal Membranes RAT UNDEFINED NNC-756 2.2 Andersen PH, et al., 1992 Jan 15, 2025 Jan 15, 2025
39518 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 2.2 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
51039 CB1 UNDEFINED HUMAN UNDEFINED 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide 2.2 Smith RA et al., 2007 Jan 15, 2025 Jan 15, 2025
56680 KOR UNDEFINED HUMAN UNDEFINED PENTAZOCINE (-) 2.2 Hsin LW et al., 2010 Jan 15, 2025 Jan 15, 2025
11372 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 2.2 Schotte A, et al., 1996 Jan 15, 2025 Jan 27, 2025
56940 DOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-bromo)benzamido]morphinan-oxalate 2.2 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
23405 MOR CLONED HUMAN 3H-DAMGO Morphine 2.2 Gharagozlou P, et al., 2003 Jan 15, 2025 Jan 15, 2025
17774 CLONED RAT 125I-VIP VIP [D-Asn24] 2.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
14963 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 2.2 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 27, 2025
29045 SST5 CLONED HUMAN 125I-LTT-SST-28 NC4-28B 2.2 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
51061 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 2.2 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51575 Alpha1D UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide 2.2 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
60535 GABAA CLONED HUMAN FNZ 6-PBC 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
47999 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
50047 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-CONH2, [MeAla7] 2.2 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
51079 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide 2.2 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
62089 5-HT2A CLONED HUMAN 3H-KETANSERIN 25CN-NBOH 2.2 Halberstadt, AL, et. al. 2016 Jan 15, 2025 Jan 15, 2025
24206 V2 PANC1 RAT 125I-VIP Vasoactive intestinal polypeptide 2.2 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
144 5-HT1A CORTEX RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 2.2 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
19344 NK3 CLONED HUMAN 125I-[MePhe7]-NKB SB 235375 2.2 Hay DW et al., 2002 Jan 15, 2025 Jan 15, 2025
93843 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MW011 2.2 Wrobel MZ et al 2019 Jan 15, 2025 Jan 15, 2025
57748 H3 UNDEFINED HUMAN UNDEFINED 4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole 2.2 Ishikawa M et al., 2010 Jan 15, 2025 Jan 15, 2025
97429 A1 CLONED HUMAN [3H]DPCPX DPCPX 2.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
48278 KOR CLONED HUMAN 3H-Diprenorphine PBR28 2.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
38807 UNDEFINED HUMAN 3H-hypoxanthine Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethylcarbamoyl]-2-hydroxypropylcarbamoyl}-2-methylpropyl)amide 2.2 Johansson P, et al., 2004 Jan 15, 2025 Jan 15, 2025
8089 GABAA CLONED HUMAN 3H-RO-15-1788 27 (6-PBC) 2.2 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
70051 D3 CLONED HUMAN 3H-SPIPERONE (S)-N6-(2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl)-N6-propyl4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine 2.2 Ghosh, B. et, al 2010 Jan 15, 2025 Jan 28, 2025
10921 NK2 CLONED HAMSTER 3H-NEUROKININ A ZM253,270 2.2 Aharony D, et al., 1995 Jan 15, 2025 Jan 15, 2025
17580 CLONED HUMAN 125I-VIP VIP Ala5 2.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
9391 GABAA CEREBRAL CORTEX RAT 3H-PK11195 PK11195 2.2 Yamagishi H, et al., 1998 Jan 15, 2025 Jan 15, 2025
5808 Alpha2A CELLS HT29 3H-RAUWOLSCINE WY 26392 2.2 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
37554 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[2-(4-Phenylpiperazin-1-yl)ethyl]-3-methoxybenzamide 2.2 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
49332 CLONED RAT Functional 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]dodecane 2.2 Boger DL, et al., 2005 Jan 15, 2025 Jan 15, 2025
24245 V2 CLONED RAT 125I-VIP VIP Ala13 2.2 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
29372 nAChR CLONED RAT 3H-Epibatidine Lobeline 2.2 Jensen AA, et al., 2003 Jan 15, 2025 Jan 15, 2025
24257 V2 CLONED RAT 125I-VIP VIP Ala26 2.2 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
52422 SLC6A4 UNDEFINED HUMAN UNDEFINED FLUOXETINE 2.2 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
53704 D2 UNDEFINED HUMAN UNDEFINED RISPERIDONE 2.2 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
51147 Alpha1D UNDEFINED HUMAN UNDEFINED 3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 2.2 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
71117 Sigma 2 CLONED HUMAN 3H-DTG 3-Carboethoxy-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 2.2 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
68558 D3 CLONED HUMAN 125I-IABN 2-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 2.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
47055 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-MPM 2.2 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
3281 D2 CLONED HUMAN 3H-YM 09151-2 PIMOZIDE 2.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
19922 A2A STRIATUM RAT 3H-CGS-21680 HENECA 2.2 Camaioni E et al., 1997 Jan 15, 2025 Jan 15, 2025
47317 5-HT1A CLONED HUMAN 3H-8-OH-DPAT WAY 100,635 2.2 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
50133 A1 CEREBRAL CORTEX RAT 3H-cyclohexyladenosine 8-[4-[[[[[2-[ Ethyl(4-hydroxybenzyl)ammonio]ethyl]-amino]carbonyl]methyl]oxy]phenyl]-1,3-dipropylxanthine Acetate 2.2 Jacobson KA et al., 1985 Jan 15, 2025 Jan 15, 2025
15063 gastrointestinal tract GUINEA PIG 125I-BH Eledoisin eledoisin 2.2 Burcher E, et al., 1986 Jan 15, 2025 Jan 15, 2025
1752 5-HT2A FR. CORTEX RAT 3H-KETANSERIN CINANSERIN 2.2 LEYSEN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
30940 KOR CLONED HUMAN 35S-GTPGammaS U50,488H 2.2 Wang Y, et. al., 2004 Jan 15, 2025 Jan 15, 2025
11485 H1 CLONED HUMAN 3H-PYRILAMINE Quetiapine 2.2 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
61409 GABAA CLONED HUMAN FNZ XHE-III-74 2.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
57060 D2 UNDEFINED UNDEFINED UNDEFINED bifeprunox 2.2 Neves G et al., 2010 Jan 15, 2025 Jan 15, 2025
63973 5-HT6 CLONED HUMAN 3H-LSD N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide 2.2 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
16616 Y1 CLONED HUMAN [125I] - Peptide YY Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26]-NPY 2.2 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
17654 PANC1 RAT 125I-VIP VIP Ala19 2.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
8951 SST5 CLONED RAT 125I-Tyr11-somatostatin-14 AcNH-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH2 2.2 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
38647 UNDEFINED HUMAN 3H-hypoxanthine 3-Deoxy-1,2-O-isopropylidene-D-glucose 2.2 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
7418 MOR CLONED HUMAN 3H-DAMGO NOR-BNI (HCI)2 2.2 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
100955 NET CELLS HEK293 3H-CIT DESIPRAMINE 2.21 Reith ME, et al., 2005 Jan 15, 2025 Jan 15, 2025
49027 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (-)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-1-methyl-propyl]piperidine hydrochloride 2.21 Berardi, F et al., 2003 Jan 15, 2025 Jan 15, 2025
60065 A3 CLONED HUMAN 125I-AB-MECA (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2-(4-(pyrazin-2-yl)-1H-1,2,3- triazol-1-yl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide 2.21 Tosh, Dipip et. al., 2015 Jan 15, 2025 Jan 15, 2025
22430 A2B CLONED HUMAN 3H-ZM241385 30 2.22 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
60188 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-((1H-Pyrazol-3-yl)ethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 2.23 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
86719 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) isonicotinamide 2.23 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
5077 5-HT2C CLONED HUMAN 3H-MESULERGINE CYPROHEPTADINE 2.23 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
98261 DOR BRAIN MOUSE 3H-DPDPE N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide 2.23 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
9463 CEREBELLUM HUMAN 125I-Iodomelatonin Melatonin,6-OH 2.23 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
64519 D2 CLONED HUMAN 3H-N-Methylspiperone PROCHLORPERAZINE 2.23872 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
58166 5-HT2B CLONED HUMAN 3H-LSD METHYLERGONOVINE 2.23872 Wacker D, et al., 2013 Jan 15, 2025 Jan 15, 2025
64646 H1 CLONED HUMAN 3H-PYRILAMINE FLUPHENAZINE 2.23872 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
64651 H1 CLONED HUMAN 3H-PYRILAMINE LOXAPINE 2.23872 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
8200 SST5 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.24 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
2963 5-HT2A CORTEX RAT 125I-LSD METHYSERGIDE 2.24 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
30036 SST1 CLONED HUMAN 125I-SOMATOSTATIN Somatostatin-14 2.25 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
30300 DOR CLONED HUMAN 3H-DPDPE 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-4-nitrobenzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 2.25 Black, SL et al., 2003 Jan 15, 2025 Jan 15, 2025
25482 SLC6A4 CEREBRAL CORTEX RAT 3H-5HT CHLORIMIPRAMINE 2.25 Shank RP, et al., 1988 Jan 15, 2025 Jan 15, 2025
52117 MOR UNDEFINED HUMAN UNDEFINED 6-(4-(2-(benzylamino)ethyl)phenoxy)nicotinamide 2.25 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
55219 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 2.25 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
100939 NET CELLS HEK293 Functional DESIPRAMINE 2.26 Reith ME, et al., 2005 Jan 15, 2025 Jan 15, 2025
29274 KOR BRAIN GUINEA PIG 3H-U69,593 3,4-Dimethoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)-oxy]morphinan-6-one 2.26 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
49572 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 2.26 Shimon I, et.al., 1997 Jan 15, 2025 Jan 15, 2025
2907 5-HT2A CORTEX RAT 3H-KETANSERIN LY 53857 2.27 ROTH ET AL., 1987 Jan 15, 2025 Jan 15, 2025
20313 BRAIN RAT 3H-D-888 Nimodipine 2.28 Reynolds IJ et al., 1986 Jan 15, 2025 Jan 15, 2025
60724 GABAA CLONED HUMAN FNZ JYI-47 2.282 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65500 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-47 2.282 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
15381 5-HT1B CLONED HUMAN 3H-5HT DHE 2.29 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
2327 5-HT3 AMYGDALA HUMAN 3H-ZACOPRIDE GRANISETRON 2.29 BARNES ET AL., 1988 Jan 15, 2025 Jan 15, 2025
1055 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RITANSERIN 2.29 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
1056 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RITANSERIN 2.29 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
1057 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RITANSERIN 2.29 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
47686 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Desmethylsertraline 2.29 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
12897 LUNG RAT 3H-RX821002 ARC-239 2.29 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
2678 5-HT2A CORTEX RAT 125I-LSD SPIPERONE 2.29 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
12975 KA CLONED HUMAN 3H-Kainic acid Kainate 2.29 Kamboj RK, et al., 1994 Jan 15, 2025 Jan 27, 2025
211 5-HT1A CORTEX PIG 3H-8-OH-DPAT CYANOPINDOLOL 2.29 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
15591 5-HT2A CLONED HUMAN 3H-KETANSERIN BUTACLAMOL,(+) 2.29 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
38379 D1 BRAIN RAT 3H-SCH23390 (R)(+)-BrAPB 2.29 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
26933 5-HT6 CLONED HUMAN 3H-LSD LSD 2.29087 Hirst WD, et.al.,2003 Jan 15, 2025 Jan 15, 2025
39742 5-HT2A CLONED HUMAN 125I-DOI METERGOLINE 2.29087 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
26964 5-HT6 CLONED RAT 3H-LSD SB-258585 2.29087 Hirst WD, et.al.,2003 Jan 15, 2025 Jan 15, 2025
27510 5-HT1B STRIATUM GUINEA PIG 3H-GR-125743 5-Hydroxy Tryptamine 2.29087 Millan MJ, et al., 2002a Jan 15, 2025 Jan 15, 2025
32480 NOP CEREBRAL CORTEX MOUSE 35S-GTPGammaS OFQ/N 2.29087 Carra' G., et.al., 2004 Jan 15, 2025 Jan 15, 2025
48897 KOR BRAIN RAT 3H-DHM EKC 2.3 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
42245 CLONED HUMAN 125I-[Ile]Motilin Motilin 2.3 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
62726 SST1 Ovary HAMSTER UNKNOWN Somatostatin-14 2.3 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
47629 ADK recombinant HUMAN Functional 4-N-(4-Chlorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2.3 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
36626 5-HT2A CLONED HUMAN 125I-R091150 OLANZAPINE 2.3 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
42264 CLONED HUMAN 125I-Motilin Delta 21-24 2.3 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
13595 OT Myometrium Rhesus 3H-Oxytocin L-366,875 2.3 Pettibone DJ, et al., 1991 Jan 15, 2025 Jan 15, 2025
32539 5-HT2C CLONED HUMAN 3H-5HT Ro 60-0175 2.3 Bentley JM, et al., 2004 Jan 15, 2025 Jan 15, 2025
60963 GABAA CLONED HUMAN FNZ SVO-8-67 2.3 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
23588 Spinal cord RAT 125I-1DMe-Y8Fa PrRP20 2.3 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
37159 STRIATUM RAT 3H-CGS-21680 N-Ethyl-l-deoxy-1-[6-amino-2-[3-(N,N-dimethylamino)-l-propyn-l-yl]-9H-purin-9-yl]-B-D-ribofuranuronamide 2.3 Cristalli G, et al., 1994 Jan 15, 2025 Jan 15, 2025
95272 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT DPAT 2.3 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
78890 5-HT1A CLONED HUMAN 3H-WAY100635 cis-2a 2.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
3885 D2 CLONED HUMAN 3H-NMS HALOPERIDOL 2.3 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 27, 2025
42287 CLONED HUMAN 125I-Motilin L110A 2.3 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
100656 H1 CLONED HUMAN 3H-PYRILAMINE CYPROHEPTADINE 2.3 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
94002 D4 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one 2.3 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
96825 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 2.3 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
57401 CB1 UNDEFINED HUMAN UNDEFINED 4-[(3-chlorophenyl)(2,4-dichlorophenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 2.3 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
13626 D2 FR. CORTEX HUMAN 125I-Epidepride FLUPENTHIXOL, Alpha 2.3 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
13371 D2 CLONED HUMAN 3H-thymidine APOMORPHINE 2.3 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
98367 D4 CLONED HUMAN [3H]-N-methylspiperone 4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one 2.3 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
90690 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 2.3 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
56130 KOR UNDEFINED HUMAN UNDEFINED (1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide 2.3 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
9539 SLC6A4 CLONED HUMAN 3H-CITALOPRAM NORFLUOXETINE 2.3 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
100676 5-HT2B CLONED HUMAN 3H-LSD Pizotyline 2.3 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
98632 D4 CLONED HUMAN [3H]-N-methylspiperone 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one 2.3 Ofon E et al 2016a Jan 15, 2025 Jan 28, 2025
12107 CLONED HUMAN 125I-hPP PP, BOVINE 2.3 Yan H, et al, 1996 Jan 15, 2025 Jan 15, 2025
3406 MOR CLONED HUMAN 3H-DAMGO CTAP-NH2 2.3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
94031 Alpha1A CORTEX PIG 3H-PRAZOSIN compound 42 2.3 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
9299 GABAA CLONED HUMAN 3H-RO-15-1788 FG 8205 2.3 Hadingham k, et al.,1993 Jan 15, 2025 Jan 27, 2025
96852 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2.3 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
23643 CEREBRAL CORTEX RAT 3H-PRAZOSIN Cyamemazine 2.3 Hameg A. et al., 2003 Jan 15, 2025 Jan 15, 2025
97631 SST5 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
35169 D1 STRIATUM RAT 3H-SCH23390 OCTOCLOTHEPIN 2.3 Campiani G, et al., 2002 Jan 15, 2025 Jan 15, 2025
58977 5-HT2C CLONED HUMAN 3H-MESULERGINE MIANSERIN 2.3 Roth B. et al., 2006 Jan 15, 2025 Jan 15, 2025
23395 NK2 ILEUM GUINEA PIG 125I-Iodohistidyl NKA 2.3 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
50793 SLC6A3 UNDEFINED HUMAN UNDEFINED (RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine 2.3 Froimowitz M et al., 2007 Jan 15, 2025 Jan 15, 2025
93802 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion 2.3 Wrobel MZ et al 2019 Jan 15, 2025 Jan 15, 2025
81259 Alpha1D test test 3H-PRAZOSIN 6-Fluoro-HEAT HCl 2.3 Petrie EC et al 2012 Jan 15, 2025 Jan 28, 2025
98925 A3 HEK293 cells test [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide 2.3 Tosh DK et al 2020 Jan 15, 2025 Jan 15, 2025
36739 D2 CLONED HUMAN 3H-SPIPERONE (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 2.3 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
14725 CysLT1 CLONED HUMAN 3H-LTD4 Montelukast 2.3 Nothacker HP, et al., 2000 Jan 15, 2025 Jan 15, 2025
17541 PANC1 HUMAN 125I-VIP VIP Ala27 2.3 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
14470 BLT2 CLONED HUMAN 3H-LTB4 LTB4 2.3 Wang S., et al., 2000 Jan 15, 2025 Jan 15, 2025
2951 5-HT2B CORTEX BOVINE 3H-KETANSERIN METERGOLINE 2.3 MCKENNA & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
52871 CB1 UNDEFINED HUMAN UNDEFINED 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 2.3 Silvestri R et al., 2008 Jan 15, 2025 Jan 15, 2025
53640 CB1 UNDEFINED HUMAN UNDEFINED 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 2.3 Urbani P et al., 2008 Jan 15, 2025 Jan 15, 2025
16266 M5 CLONED HUMAN 3H-NMS Darifenacin 2.3 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
73101 D4 CLONED HUMAN 3H-N-Methylspiperone . 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl) butan-1-one 2.3 Ofori E et al 2016 Jan 15, 2025 Jan 28, 2025
23694 SLC6A4 CLONED HUMAN 3H-CITALOPRAM Fluvoxamine 2.3 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
37520 D3 CLONED RAT 3H-SPIROPERIDOL N-[3-[4-(2,3-Dichlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 2.3 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
92818 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 2.3 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
57245 CB1 UNDEFINED HUMAN UNDEFINED N-(((3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)naphthalene-1-sulfonamide 2.3 Scott JD et al., 2010 Jan 15, 2025 Jan 15, 2025
39074 D3 CLONED HUMAN R-SAT BROMPERIDOL 2.3 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
10662 M1 CEREBRAL CORTEX RAT 3H-NMS HX 2.3 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
11688 D2 CLONED HUMAN 125I-IODOSULPRIDE CHLORPROMAZINE 2.3 Sokoloff P, et al., 1992 Jan 15, 2025 Jan 15, 2025
94632 CB2 SPLEEN MOUSE 3H-CP55940 6-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 2.3 Pinna G et al 2014 Jan 15, 2025 Jan 28, 2025
7339 DOR CLONED HUMAN 3H-Naltrindole Bremazocine 2.3 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
52395 SLC6A4 UNDEFINED RAT UNDEFINED 2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 2.3 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
56493 CB1 UNDEFINED HUMAN UNDEFINED 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 2.3 Silvestri R et al., 2009 Jan 15, 2025 Jan 15, 2025
21424 A1 BRAIN RAT 3H-cyclohexyladenosine CHA 2.3 Hutchison AJ et al., 1989 Jan 15, 2025 Jan 15, 2025
11698 D3 CLONED HUMAN 125I-IODOSULPRIDE PERGOLIDE 2.3 Sokoloff P, et al., 1992 Jan 15, 2025 Jan 15, 2025
11701 D3 CLONED HUMAN 125I-IODOSULPRIDE TL99 2.3 Sokoloff P, et al., 1992 Jan 15, 2025 Jan 15, 2025
52406 SLC6A4 UNDEFINED RAT UNDEFINED 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline 2.3 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
55222 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(2,6-dichloro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 2.3 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
24249 V2 CLONED RAT 125I-VIP VIP Ala17 2.3 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
30907 BB3 CLONED HUMAN 125I-[D-Tyr6,Beta-Ala11,Phe13,Nle14]Bn(6-14) [D-Tyr6,Beta-Dap11,Phe13,Nle14]Bn(6-14) 2.3 Mantey, SA et. al., 2004 Jan 15, 2025 Jan 15, 2025
3772 MOR BRAIN GUINEA PIG 3H-DAMGO Beta-Endorphin 2.3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
55996 CB1 UNDEFINED HUMAN UNDEFINED 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(piperidin-1-yl)-9H-purine 2.3 Griffith DA et al., 2009 Jan 15, 2025 Jan 15, 2025
6846 Y2 CLONED HUMAN 125I-NPY NPY, human 2.3 Rose et al, 1995 Jan 15, 2025 Jan 15, 2025
59070 MOR CLONED HUMAN 3H-DAMGO DAMGO 2.3 Polepally P, et al., 2014 Jan 15, 2025 Jan 15, 2025
3519 5-HT2A CLONED RAT 3H-KETANSERIN MIANSERIN 2.3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
17600 T47D HUMAN 125I-VIP VIP Ala11 2.3 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
37568 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[4-[4-(1-Naphthalenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 2.3 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
55232 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 2.3 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
65730 GABAA CLONED HUMAN [3H] Flunitrazepam SVO-8-67 2.3 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
55748 5-HT1D UNDEFINED HUMAN UNDEFINED N1,N15-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)pentadecanediamide 2.3 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
3783 MOR BRAIN GUINEA PIG 3H-DAMGO DYNORPHIN(1-11)-OH 2.3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18631 D3 CLONED RAT 3H-RACLOPRIDE THIORIDAZINE 2.3 Strange PG 2001 Jan 15, 2025 Jan 15, 2025
18376 D2 BRAIN RAT 3H-SPIPERONE A 37850 2.3 Hall H et al., 1986 Jan 15, 2025 Jan 27, 2025
68554 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-nitrobenzamide 2.3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
13258 Beta2 BRAIN Mammalian 3H-DHA ALPRENOLOL,(-) 2.3 Bylund DB, et al., 1976 Jan 15, 2025 Jan 15, 2025
18634 D4 CLONED RAT 3H-SPIPERONE HALOPERIDOL 2.3 Strange PG 2001 Jan 15, 2025 Jan 15, 2025
35532 PTGFR CLONED HUMAN 3H-PGF2Alpha FLUPROSTENOL 2.3 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
10701 SUBMAXILLARY GLAND RAT 3H-NMS HX 2.3 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
41677 H2 CLONED HUMAN 3H-TIOTIDINE ORG-5222 2.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
32207 NET Temp. Cortex RAT 3H-Norepinephrine DICLOFENSINE,(+) 2.3 Hyttel J and Larsen J.J., 1985 Jan 15, 2025 Jan 15, 2025
53713 D2 UNDEFINED HUMAN UNDEFINED 1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 2.3 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
49362 CLONED RAT Functional 1-Oxo-1-[5-(4-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 2.3 Boger DL, et al., 2005 Jan 15, 2025 Jan 15, 2025
11222 Total Cortex RAT 3H-PRAZOSIN RISPERIDONE 2.3 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
13014 H1 BRAIN RAT 3H-MEPYRAMINE Carbinoxamine 2.3 Tran VT, et al., 1978 Jan 15, 2025 Jan 15, 2025
30167 A3 CLONED RAT 3H-AB-MECA 2-(methylthio)-N6-(3-Iodobenzyl)adenosine-5'-N-methyluronamide 2.3 Kim HO et al., 1994 Jan 15, 2025 Jan 15, 2025
47831 KOR CLONED HUMAN 3H-U69,593 Levorphanol 2.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
14044 CB1 CEREBELLUM RAT 3H-SR141716A Levonantradol 2.3 Breivogel CS, Childers SR, 2000 Jan 15, 2025 Jan 15, 2025
18908 A3 CLONED HUMAN 3H-MRE 3008F20 MRE 3008F20 2.3 Gessi S et al., 2002 Jan 15, 2025 Jan 15, 2025
27869 5-HT6 CLONED HUMAN 3H-LSD 5-Methoxy-N,N-dimethyl-1-(benzenesulfonyl)tryptamine 2.3 Pullagurla M, et.al.,2003 Jan 15, 2025 Jan 15, 2025
64989 H1 BRAIN RAT 3H-MEPYRAMINE Carbinoxamine 2.3 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
13535 D2 STRIATUM RAT 3H-SPIPERONE BUTACLAMOL,(+) 2.3 Zahniser NR, et al., 1983 Jan 15, 2025 Jan 15, 2025
50402 H1 BRAIN RODENT 3H-MEPYRAMINE (+/-)-p-fluoro-trans-H2-PAT 2.3 Bucholtz E., et.al.1999 Jan 15, 2025 Jan 15, 2025
7396 KOR CLONED HUMAN 3H-U69,593 Naloxone(-) 2.3 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
100325 5-HT6 CLONED HUMAN 3H-LSD SERTINDOLE 2.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
11494 5-HT1E CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 2.3 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
13032 H1 BRAIN RAT 3H-MEPYRAMINE Methdilazine 2.3 Tran VT, et al., 1978 Jan 15, 2025 Jan 15, 2025
98025 SST2 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 2.3 Reubi JC, et.al.,2002 Jan 15, 2025 Jan 15, 2025
9711 MT1 CLONED HUMAN 125I-Iodomelatonin GR 196429 2.3 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
37107 BuChE serum BOVINE Functional N-(1,2,3,4-Tetrahydroacridin-9-yl)-9-[(1,2,3,4-tetrahydro-9-yl)thio]nonan-1-amine 2.3 Campiani G, et al., 2005a Jan 15, 2025 Jan 15, 2025
35829 SLC6A4 CLONED HUMAN 3H-PAROXETINE 7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 2.3 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
48885 KOR BRAIN RAT 3H-NALOXONE Beta-Endorphin 2.3 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
72182 nAChR CLONED HUMAN 3H-Epibatidine 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 2.3 Magnus CJ et al 2019 Jan 15, 2025 Jan 29, 2025
3320 D3 CLONED HUMAN 3H-YM 09151-2 PIMOZIDE 2.3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
82168 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 2.3 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
34297 D1 STRIATUM RAT 3H-SCH23390 Dihydrexidine, DHX 2.3 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
70189 BRAIN Zebrafish 3H-Diprenorphine NALOXONE 2.31 Gonzalez-Nunez V, et al., 2006 Jan 15, 2025 Jan 15, 2025
59326 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[5-(3,4-Dichlorophenyl)-6-fluoro-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2.31 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
12276 Spinal cord RAT 3H-Cytisine Nicotine-L (base) 2.31 Khan IM, et al., 1994 Jan 15, 2025 Jan 15, 2025
2560 5-HT2A CORTEX HUMAN 3H-SPIPERONE THIOTHIXENE,cis- 2.32 ANDORN ET AL., 1984 Jan 15, 2025 Jan 15, 2025
29472 CB1 BRAIN Zebra Finch 3H-CP-55940 HU-210 2.32 Soderstrom, K et al., 2001 Jan 15, 2025 Jan 15, 2025
38441 D5 CLONED HUMAN 3H-SCH23390 MCL-207 2.32 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
41295 D5 CLONED HUMAN Functional 7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide 2.32 Hoefgen B, et al., 2006 Jan 15, 2025 Jan 15, 2025
31112 H3 CEREBRAL CORTEX HUMAN 3H-Alpha-Me-histamine HISTAMINE 2.32 Hancock, AA, et al., 2004 Jan 15, 2025 Jan 15, 2025
50425 SST5 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.32 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
97284 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 2.33 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
309 5-HT1A CORTEX RAT 3H-8-OH-DPAT ICYANOPINDOLOL 2.33 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
88410 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 2.33 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
58116 5-HT2A CLONED HUMAN 125I-DOI N-(2-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 2.34 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
12813 Beta2 Gastrocnemius GUINEA PIG 125I-ICYP TMQ, 3'-Iodo 2.34 Fraundorfer PF, et al., 1994 Jan 15, 2025 Jan 28, 2025
60189 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(2-((1-methyl-1H-pyrazol-4-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)bicyclo[3.1.0]- hexane-1-carboxamide 2.34 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
3925 5-HT6 CLONED RAT 3H-LSD ERGOTAMINE 2.34 BOESS FG, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
8285 SST4 CLONED HUMAN 125I-LTT-SRIF28 BIM 23052 2.34 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
6775 Y2 CLONED HUMAN 125I-PYY NPY2-36, porcine 2.34 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
6804 Y1 CLONED HUMAN 125I-PYY NPY2-36, porcine 2.34 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
56219 SLC6A4 UNDEFINED RAT UNDEFINED (S)-2-((4-(1H-Indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)-methyl)-8-methyl-2,3-dihydro-[1,4]dioxino-[2,3-f]quinoline 2.34 Zhou D et al., 2009 Jan 15, 2025 Jan 15, 2025
21950 MOR ILEUM GUINEA PIG 3H-DHM NALOXONE 2.34 Leslie FM et al., 1980 Jan 15, 2025 Jan 15, 2025
2274 5-HT3 HIPPOCAMPUS HUMAN 3H-ZACOPRIDE BRL 43694 2.34 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
58106 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-Bromobenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 2.34 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
28745 SST4 CLONED HUMAN 125I-LTT-SRIF28 BIM 23052 2.34423 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
63327 CRF1 CLONED HUMAN 125I-Sauvagine DMP696 2.34423 Hoare SR, et al., 2003 Jan 15, 2025 Jan 15, 2025
32366 M4 HEART Chick 3H-NMS PrBCh 2.34423 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
67722 D2 STRIATUM PIG 3H-SPIPERONE Flupenthixol 2.34423 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
26794 GAL2 CLONED HUMAN 125I-GALANIN Galanin, Human 2.34423 Borowsky Beth, et. al., 1998 Jan 15, 2025 Jan 15, 2025
24755 Y2 CLONED HUMAN 125I-PYY NPY2-36, porcine 2.34423 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
18665 H3 CLONED HUMAN 3H-Alpha-Me-histamine VUF5202 2.34423 Wieland K et al., 2001 Jan 15, 2025 Jan 15, 2025
65603 GABAA CLONED HUMAN [3H] Flunitrazepam YT-III-271 2.35 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
61261 GABAA CLONED HUMAN FNZ YT-III-271 2.35 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
10064 MOR BRAIN MOUSE 125I-Endomorphin-1 Morphine 6-glucuronide 2.35 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
12685 KOR BE(2)-C HUMAN 3H-NalBzoH Bremazocine 2.35 Standifer KM, et al., 1994 Jan 15, 2025 Jan 27, 2025
22432 A2B CLONED HUMAN 3H-ZM241385 32 2.35 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
70066 D3 CLONED HUMAN 3H-SPIPERONE 7-OH-DPAT 2.35 Ghosh, B. et, al 2010 Jan 15, 2025 Jan 28, 2025
51991 DOR UNDEFINED HUMAN UNDEFINED 1'-(o-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 2.36 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
41843 H3 CLONED RAT 3H-Alpha-Me-histamine 2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone 2.36 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
5578 5-HT2C CLONED HUMAN 125I-DOI DOI 2.36 WAINSCOTT DB, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
52247 Beta1 UNDEFINED HUMAN UNDEFINED (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 2.37 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
63213 KOR CEREBELLUM GUINEA PIG 3H-Bremazocine Tyr-Met-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) 2.37 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
55106 H1 UNDEFINED HUMAN UNDEFINED CLOZAPINE 2.38 von Coburg Y et al., 2009 Jan 15, 2025 Jan 15, 2025
30037 SST1 CLONED HUMAN 125I-SOMATOSTATIN somatostatin-28 2.38 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
65898 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-49 (C20H12N3O2F4Br) 2.38 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
12205 BRAIN HUMAN UNDEFINED ATR 2.38 Richelson E., 1988 Jan 15, 2025 Jan 15, 2025
60665 GABAA CLONED HUMAN FNZ JYI-49 2.38 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60706 GABAA CLONED HUMAN FNZ TJH-IV-51 2.39 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
8249 SST1 CLONED HUMAN 125I-Tyr10-CST14 BIM 23052 2.39 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
50235 Y2 CLONED GUINEA PIG 125I-PYY NPY18-36, porcine 2.39 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
65600 GABAA CLONED HUMAN [3H] Flunitrazepam 6-PBC 2.39 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
30559 MOR CLONED HUMAN 3H-Diprenorphine Naltrexone 2.39 Valenzano KJ et. al., 2004 Jan 15, 2025 Jan 15, 2025
60534 GABAA CLONED HUMAN FNZ 6-PBC 2.39 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
8312 SST4 CLONED HUMAN 125I-CGP23996 CGP 23996 2.39 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
65404 GABAA CLONED HUMAN [3H] Flunitrazepam TJH-IV-51 2.39 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
6023 M4 ADRENAL BOVINE 3H-QNB TRIPITRAMINE 2.39 CHELALA JL, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
8591 SST2 CLONED MOUSE 125I-Tyr11-SRIF SMS 201-995 2.39 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
8617 SST3 CLONED MOUSE 125I-Tyr11-SRIF BIM 23027 2.39 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
23731 MC5 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH alpha-MSH, [Nle4, D-Phe7] 2.39 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
22511 MC5 CLONED HUMAN 125I-NDP-MSH NDP-MSH 2.39 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
15353 5-HT1D CLONED RAT 3H-5HT 5-Methoxytryptamine 2.39 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
23552 H3 BRAIN CORTEX GUINEA PIG 3H-NAMH A-317920 2.39883 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
83471 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 2.39883 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83472 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 2.39883 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
64288 5-HT2C CLONED RAT 3H-MESULERGINE SERTINDOLE 2.39883 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
28740 SST1 CLONED HUMAN 125I-Tyr10-CST14 BIM 23052 2.39883 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
69262 H3 CLONED RAT 3H-Alpha-Me-histamine proxyfan 2.39883 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
26823 GAL1 CLONED HUMAN 125I-GALANIN M40 2.39883 Borowsky Beth, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11524 GABAA FOREBRAIN RAT FNZ Clonazepam 2.4 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
53255 D2 UNDEFINED HUMAN UNDEFINED 1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 2.4 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
62727 SST1 Ovary HAMSTER UNKNOWN somatostatin-28 2.4 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
17930 CCK2 BRAIN HUMAN 125I-CCK L-365,260 2.4 Lotti VJ et al., 1988 Jan 15, 2025 Jan 15, 2025
61455 GABAA CLONED HUMAN FNZ RY-058 2.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
9236 SST2 CLONED MOUSE 125I-MK-678 SMS 201-995 2.4 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
35860 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 2.4 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
5144 5-HT2C CLONED HUMAN 125I-DOI DOI 2.4 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
93211 D4 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 2.4 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
9248 SST2 CLONED MOUSE 125I-MK-678 BIM 23057 2.4 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
32803 D2 CLONED RAT 3H-SPIPERONE PIMOZIDE 2.4 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
42791 CLONED HUMAN 125I-ghrelin 5-(4-{[3,5-Difluoro-4-(methylsulfonyl)benzyl]amino}phenyl)-6-ethylpyrimidine-2,4-diamine 2.4 Serby MD, et al., 2006 Jan 15, 2025 Jan 15, 2025
12072 5-HT1D CLONED HUMAN 3H-GR-125743 5-CT 2.4 Domenech T, et al., 1997 Jan 15, 2025 Jan 15, 2025
24104 5-HT2A CLONED HUMAN 3H-SPIPERONE THIORIDAZINE 2.4 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
70187 BRAIN RAT 3H-MEGY Met-enkephalin 2.4 Gonzalez-Nunez V, et al., 2005 Jan 15, 2025 Jan 15, 2025
1838 5-HT2A CORTEX RAT 3H-KETANSERIN DHE 2.4 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
16176 D2 CLONED RAT 125I-IODOSULPRIDE PIMOZIDE 2.4 Sokoloff P, et al., 1990 Jan 15, 2025 Jan 15, 2025
52016 SLC6A4 UNDEFINED RAT UNDEFINED (2-(3,4-dichlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine 2.4 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
2865 5-HT2B CORTEX BOVINE 3H-KETANSERIN KETANSERIN 2.4 MCKENNA & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
11057 H3 CLONED HUMAN 3H-methylhistamine N-methylhistamine 2.4 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
30513 M2 CLONED HUMAN 3H-QNB Arecoline 2.4 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
16690 M4 CLONED HUMAN 3H-QNB Biperidine 2.4 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
64818 CCR5 CLONED UNDEFINED 125I-RANTES (S)- (-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 2.4 Seto M, et al., 2006 Jan 15, 2025 Jan 28, 2025
91446 5-HT2A CLONED HUMAN 125I-DOI (6bR,10aS)-8-[3-(4-Fluorophenoxy)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahy-dro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxaline 2.4 Li P et al 2014 Jan 15, 2025 Jan 15, 2025
94007 5-HT1A CORTEX PIG [3H]WAY 600135 compound 42 2.4 Ortega R et al 2011 Jan 15, 2025 Jan 15, 2025
54839 SLC6A4 UNDEFINED RAT UNDEFINED 8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}-N-methylchromane-5-carboxamide 2.4 Hatzenbuhler NT et al., 2008 Jan 15, 2025 Jan 15, 2025
4409 5-HT1D CLONED RAT 3H-5HT 5-Methoxytryptamine 2.4 HAMBLIN MW, ET AL., 5/1992 Jan 15, 2025 Jan 15, 2025
7994 GABAA CLONED HUMAN 3H-RO-15-1788 18 2.4 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
6973 D3 CLONED HUMAN 125I-IODOSULPRIDE 7-OH-DPAT,(+) 2.4 LEJEUNE F, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
31551 D1 Striatal Membranes RAT 3H-SCH23390 C21H24ClFN2 dimaleate (27) 2.4 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
47935 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 2.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
2880 5-HT2A CORTEX RAT 3H-KETANSERIN LSD 2.4 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
49473 KOR CLONED HUMAN 3H-Diprenorphine Dynorphin A(1-11)-NH2,[Pro3] 2.4 Schlechtingen, G et al., 2003 Jan 15, 2025 Jan 15, 2025
3146 5-HT7 CLONED RAT 3H-LSD ACETOPHENAZINE 2.4 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
78923 5-HT1B CLONED HUMAN 3H-5-CT S,S-2c 2.4 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
90447 D2 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 2.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
17488 PANCREAS GUINEA PIG 125I-VIP VIP Ala11 2.4 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
88656 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 2.4 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
42321 SLC6A3 Striatal Membranes RAT 3H-LBT-999 GBR-12935 2.4 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
62801 Brain caudate nucleus HUMAN 3H-QNB ATR 2.4 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 15, 2025
2899 5-HT2A CORTEX RAT 3H-KETANSERIN LSD 2.4 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
50003 SLC6A4 WHOLE BRAIN MINUS CEREBELLUM RAT 3H-5HT CITALOPRAM 2.4 Rothman RB, et al., 2001 Jan 15, 2025 Jan 15, 2025
2900 5-HT2A CORTEX RAT 3H-KETANSERIN LSD 2.4 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
25173 Alpha1B CLONED HUMAN 125I-HEAT THIORIDAZINE 2.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94042 Alpha1A CORTEX PIG 3H-PRAZOSIN 3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 2.4 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
5725 Alpha2C KIDNEY OPOSSUM 3H-RAUWOLSCINE IDAZOXAN 2.4 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
23646 PDE4 CEREBRAL CORTEX RAT 3H-Rolipram Roflumilast 2.4 Zhao, Y et. al., 2003 Jan 15, 2025 Jan 15, 2025
10335 nAChR T.Californica electric organ RAT 125I-Alpha-bgt Epibatidine 2.4 Bannon AW, et al., 1998 Jan 15, 2025 Jan 15, 2025
17503 PANCREAS GUINEA PIG 125I-VIP VIP Ala27 2.4 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
16992 M1 CLONED HUMAN 3H-NMS NNC 11-1607 2.4 Christopoulos A, et al., 2001 Jan 15, 2025 Jan 15, 2025
17760 CLONED RAT 125I-VIP VIP [D-Tyr10] 2.4 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
21856 5-HT1B CLONED RAT 3H-GR-125743 S,S-2c 2.4 Nichols DE, et al., 2002 Jan 15, 2025 Jan 15, 2025
17505 PANCREAS RAT 125I-VIP Vasoactive intestinal polypeptide 2.4 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
101222 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-([1,1'-biphenyl]-2-yl)piperazin-1-yl)-1-(3,4-dichlorophenyl)ethanol hydrochloride 2.4 Gu, Zheng-Song, et al., 2017 Jan 15, 2025 Jan 15, 2025
72298 Sigma 2 test test 3H-DTG 10-(Cyclopropylmethoxy)-3,9-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 2.4 Gadhiya S et al 2016 Jan 15, 2025 Jan 28, 2025
20330 BRAIN RAT 3H-D-888 D888,(-) 2.4 Reynolds IJ et al., 1986 Jan 15, 2025 Jan 15, 2025
9324 GABAA CLONED HUMAN 3H-RO-15-1788 Bretazenil 2.4 Hadingham k, et al.,1993 Jan 15, 2025 Jan 27, 2025
36716 5-HT2C CLONED HUMAN 3H-MESULERGINE (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-chloro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 2.4 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
9071 SST4 CLONED RAT 125I-CGP23996 BIM 23066 2.4 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
68977 GABAA CLONED RAT 3H-Ro15-1788 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3-fluoropyridin-2-yl)pyridazine 2.4 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
32882 D2 CLONED HUMAN 3H-domperidone HALOPERIDOL 2.4 Grandy DK, et al., 1989 Jan 15, 2025 Jan 15, 2025
54133 TRPV1 UNDEFINED RAT UNDEFINED [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1,10}.0^{2,6}.0^{11,15}]octadeca-3,8-dien-8-yl]methyl 2-(3-fluorophenyl)acetate 2.4 Choi HK et al., 2009 Jan 15, 2025 Jan 15, 2025
57721 NR3C1 UNDEFINED HUMAN UNDEFINED prednisolone 2.4 Onnis V et al., 2010 Jan 15, 2025 Jan 15, 2025
47738 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY 28-36, [P30, Y32, L34] 2.4 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
39036 D2 CLONED HUMAN R-SAT PIMOZIDE 2.4 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
59260 CLONED RAT 3H-5HT (2R)-8-{4-[3-(7-Fluoro-1H-indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one 2.4 Smid P, et al., 2005 Jan 15, 2025 Jan 15, 2025
1921 5-HT2A CORTEX RAT 3H-SPIPERONE DROPERIDOL 2.4 LEYSEN ET AL., 1978 Jan 15, 2025 Jan 15, 2025
24196 V2 CLONED HUMAN 125I-VIP VIP Ala19 2.4 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
70277 MOR CLONED MOUSE 3H-DAMGO DADLE 2.4 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
39560 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 2.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
35211 D3 olfactory tubercle RAT 3H-7-OH-DPAT OCTOCLOTHEPIN 2.4 Campiani G, et al., 2002 Jan 15, 2025 Jan 15, 2025
39052 D2 CLONED HUMAN R-SAT RACLOPRIDE 2.4 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
20621 BRAIN RAT 3H-WB4101 Dihydro-alpha-ergocryptine 2.4 U'Prichard DC et al., 1977 Jan 15, 2025 Jan 15, 2025
1167 5-HT1D CAUDATE C0S-7 3H-5HT 5-CT 2.4 HOYER, 1987 Jan 15, 2025 Jan 15, 2025
20623 BRAIN RAT 3H-WB4101 Dihydroergocristine 2.4 U'Prichard DC et al., 1977 Jan 15, 2025 Jan 15, 2025
1168 5-HT1D CAUDATE CALF 3H-5HT 5-CT 2.4 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
1169 5-HT1D CAUDATE CALF 3H-5HT 5-CT 2.4 WAEBER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
29075 SST5 CLONED HUMAN 125I-LTT-SST-28 BIM 23060 2.4 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
51603 Alpha1D UNDEFINED HUMAN UNDEFINED 2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2.4 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
53395 CB1 UNDEFINED HUMAN UNDEFINED Rimonabant 2.4 Wang H et al., 2008 Jan 15, 2025 Jan 15, 2025
94613 CB2 SPLEEN MOUSE 3H-CP55940 7-Methyl-1-(4-methylbenzyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 2.4 Pinna G et al 2014 Jan 15, 2025 Jan 28, 2025
88475 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 2.4 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
16029 M3 Parotid gland RAT 3H-NMS 4-DAMP 2.4 Bockman CS, et al., 2001 Jan 15, 2025 Jan 15, 2025
100766 PDE4c CLONED HUMAN Functional L-826,141 2.4 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
99743 DOR CLONED HUMAN 3H-DPDPE [D-Ala2, Leu5] enkephalin amide 2.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
39078 D3 CLONED HUMAN R-SAT PROCHLORPERAZINE 2.4 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
935 5-HT2C C. PLEXUS TUM MOUSE 125I-LSD MIANSERIN 2.4 YAGALOFF ET AL., 1986 Jan 15, 2025 Jan 15, 2025
57257 CB1 UNDEFINED HUMAN UNDEFINED Rimonabant 2.4 Scott JD et al., 2010 Jan 15, 2025 Jan 15, 2025
51373 M2 UNDEFINED HUMAN UNDEFINED 3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 2.4 Sonda S et al., 2007 Jan 15, 2025 Jan 15, 2025
16046 D2 Striatal Membranes RAT 3H-sulpiride Sultopride 2.4 Imafuku J, 1987 Jan 15, 2025 Jan 15, 2025
20656 BRAIN RAT 3H-CLONIDINE DHE 2.4 U'Prichard DC et al., 1977 Jan 15, 2025 Jan 15, 2025
39089 D3 CLONED HUMAN R-SAT RISPERIDONE 2.4 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
36018 BRAIN RAT 3H-3-PPP,(+) HALOPERIDOL 2.4 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
5811 Alpha2A CELLS HT29 3H-RAUWOLSCINE SKF 86466 2.4 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
66228 Ghrelin CLONED HUMAN 125I-ghrelin 5-(4-{[3,5-Difluoro-4-(methylsulfonyl)benzyl]amino}phenyl)-6-ethylpyrimidine-2,4-diamine 2.4 Serby MD, et al., 2006 Jan 15, 2025 Jan 15, 2025
70324 MOR CLONED MOUSE 3H-Diprenorphine Diprenorphine 2.4 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
19892 A1 BRAIN RAT 3H-cyclohexyladenosine 8 2.4 Bridges AJ et al., 1987 Jan 15, 2025 Jan 15, 2025
90805 DOR brain membranes RAT 3H-DPDPE NALOXONE 2.4 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
30133 SST5 CLONED RAT 125I-SOMATOSTATIN BIM 23052 2.4 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
70070 MOR CLONED HUMAN 3H-DAMGO c2,2′(Tyr-DCys-Gly-Phe)2-cystamine 2.4 Remesic, M. et, al 2018 Jan 15, 2025 Jan 28, 2025
1720 5-HT2A CORTEX RAT 3H-KETANSERIN BUTACLAMOL,(+) 2.4 LYON ET AL., 1987 Jan 15, 2025 Jan 15, 2025
30393 B2 CLONED HUMAN 3H-BRADYKININ (2E)-N-{2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(2-pyridinylmethoxy)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl}-3-{6-[(4-pyridinylacetyl)amino]-3-pyridinyl}-2-propenamide 2.4 Sawada, Y et al., 2004 Jan 15, 2025 Jan 15, 2025
19387 A3 CLONED HUMAN 3H-NECA 1, HENECA 2.4 Klotz KN et al., 1999 Jan 15, 2025 Jan 15, 2025
63420 D2 STRIATUM RAT 3H-SPIPERONE HALOPERIDOL 2.4 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
11713 D3 CLONED HUMAN 125I-IODOSULPRIDE Amisulpride 2.4 Sokoloff P, et al., 1992 Jan 15, 2025 Jan 15, 2025
19395 A3 CLONED HUMAN 3H-NECA 7 2.4 Klotz KN et al., 1999 Jan 15, 2025 Jan 15, 2025
8134 GABAA CLONED HUMAN 3H-RO-15-1788 27 (6-PBC) 2.4 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
29897 GABAB CEREBELLUM CAT 3H-BACLOFEN CGP27492 2.4 Froestl W, et. al., 1995 Jan 15, 2025 Jan 15, 2025
56521 CB2 UNDEFINED HUMAN UNDEFINED (S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide 2.4 Silvestri R et al., 2009 Jan 15, 2025 Jan 15, 2025
42442 GABAA WHOLE BRAIN RAT FNZ CGS 9896 2.4 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
51661 D2 UNDEFINED HUMAN UNDEFINED 2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2.4 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
60370 GABAA CLONED HUMAN FNZ WYS13 2.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
9176 SST3 CLONED MOUSE 125I-CGP23996 BIM 23027 2.4 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
48606 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
89828 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 2.4 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
81381 Sigma 2 test test 3H-DTG 5’-Bromo-4’-OMethyl-HEAT HCl 2.4 Petrie EC et al 2012 Jan 15, 2025 Jan 28, 2025
69352 D2 CLONED HUMAN 3H-NMSP HALOPERIDOL 2.4 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
22259 5-HT1A CEREBRAL CORTEX RABBIT 3H-8-OH-DPAT SPIROXATRINE 2.4 Weber JT, et al., 1997 Jan 15, 2025 Jan 15, 2025
32500 5-HT2C CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 2.4 Kimura Y, et al., 2004 Jan 15, 2025 Jan 15, 2025
99832 DOR CLONED HUMAN [3H]DPDPE DALEA 2.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
38136 CLONED RAT 3H-dexamethasone C57H79N2O9Na 2.4 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
65016 H1 BRAIN GUINEA PIG 3H-MEPYRAMINE PROMAZINE 2.4 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
17146 5-HT1D BRAIN HUMAN 3H-5CT Ziprasidone 2.4 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
11771 CAUDATE NUCLEUS HUMAN 3H-QNB ATR 2.4 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
32507 5-HT2B CLONED HUMAN 3H-5HT Ro 60-0175 2.4 Kimura Y, et al., 2004 Jan 15, 2025 Jan 15, 2025
98043 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pyridin-2-amine 2.4 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
35839 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 2.4 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
99644 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-3-methoxy}-phenyl]-xanthine 2.41 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
53080 KOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan 2.41 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
145 5-HT1A CORTEX PIG 3H-8-OH-DPAT 5-Hydroxy Tryptamine 2.41 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
205 5-HT1A CORTEX RAT 3H-8-OH-DPAT CYANOPINDOLOL 2.41 FOZARD ET AL., 1987 Jan 15, 2025 Jan 15, 2025
99595 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 2.43 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
30298 DOR CLONED HUMAN 3H-DPDPE 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-benzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 2.43 Black, SL et al., 2003 Jan 15, 2025 Jan 15, 2025
54865 SLC6A4 UNDEFINED RAT UNDEFINED (-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide 2.44 Hatzenbuhler NT et al., 2008 Jan 15, 2025 Jan 15, 2025
60707 GABAA CLONED HUMAN FNZ WYS13 2.442 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65320 nAChR CLONED HUMAN [3H] Flunitrazepam WYS13-C20H18N2O3 2.442 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
2866 5-HT2A CORTEX HUMAN 3H-KETANSERIN KETANSERIN 2.45 HOYER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
52788 5-HT2A UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide 2.45 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
883 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHYSERGIDE 2.45 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4989 5-HT2C CLONED RAT 3H-MESULERGINE ERGOTAMINE 2.45 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
4998 5-HT2C CLONED RAT 3H-MESULERGINE METHIOTHEPIN 2.45 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
90511 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 2.45 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
6803 Y1 CLONED HUMAN 125I-PYY NPY2-36, human 2.45 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
5027 5-HT2A CLONED HUMAN 3H-KETANSERIN METHYSERGIDE 2.45 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
6828 Y4 CLONED HUMAN 125I-PYY PP,SALMON 2.45 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
39772 5-HT2B CLONED HUMAN 3H-5HT SB 221284 2.45471 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
32370 M4 HEART Chick 3H-NMS TELENZEPINE 2.45471 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
64663 H1 CLONED HUMAN 3H-PYRILAMINE THIORIDAZINE 2.45471 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
64664 H1 CLONED HUMAN 3H-PYRILAMINE MESORIDAZINE 2.45471 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
24734 Y1 CLONED HUMAN 125I-PYY NPY2-36, human 2.45471 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
19103 M3 CLONED HUMAN 3H-NMS (R)-Trihexyphenidyl 2.45471 Dorje F et al., 1991 Jan 15, 2025 Jan 15, 2025
47282 Beta2 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, dl 2.45471 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
50375 Y1 CLONED HUMAN 125I-PYY NPY2-36, human 2.45471 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
63717 D3 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 2.45471 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
26346 DOR CLONED RAT 3H-EKC EKC 2.46 Neal, C. R. Jr. , et al. 2003 Jan 15, 2025 Jan 15, 2025
36077 KOR Membranes RAT 3H-U69,593 14-Benzyloxymetopon 2.46 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
38440 D5 CLONED HUMAN 3H-SCH23390 MCL-203 2.47 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
10087 MOR BRAIN MOUSE 125I-Endomorphin-2 Morphine 6-glucuronide 2.47 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
22431 A2B CLONED HUMAN 3H-ZM241385 31 2.47 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
52134 KOR UNDEFINED HUMAN UNDEFINED 6-(4-((benzylamino)methyl)phenoxy)nicotinamide 2.47 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
10061 MOR BRAIN MOUSE 125I-Endomorphin-1 DADLE-OH 2.49 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
92826 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 2.49 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
18933 H1 CLONED HUMAN 3H-trans-H2-PAT,(-) trans-H2-PAT(+/-) 2.49 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
36610 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 2.5 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
37129 A1 BRAIN RAT 3H-cyclohexyladenosine N-Ethyl-l-deoxy-1-[6-amino-2-(3-hydroxy-3-phenyl-l-propyn-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide 2.5 Cristalli G, et al., 1994 Jan 15, 2025 Jan 15, 2025
38669 UNDEFINED HUMAN 3H-hypoxanthine Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcarbamoyl}-2-methyl-propyl)-amide 2.5 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
53778 5-HT1A UNDEFINED HUMAN UNDEFINED Ziprasidone 2.5 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
13588 OT Mammary RAT 3H-Oxytocin L-366,875 2.5 Pettibone DJ, et al., 1991 Jan 15, 2025 Jan 15, 2025
7447 BB2 CELLS MOUSE 125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14) GRP 2.5 Katsuno T, et al., 1999 Jan 15, 2025 Jan 15, 2025
55575 MOR UNDEFINED HUMAN UNDEFINED N-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone 2.5 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
60695 GABAA CLONED HUMAN FNZ Flunitrazepam 2.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
14616 H4 CLONED HUMAN 3H-Histamine HISTAMINE 2.5 Zhu, Yand, et al., 2001 Jan 15, 2025 Jan 15, 2025
72475 5-HT1B test test 3H-GR125743 METHYSERGIDE 2.5 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
56094 MOR UNDEFINED HUMAN UNDEFINED (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide 2.5 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
24095 5-HT2A CLONED HUMAN 3H-SPIPERONE LOXAPINE 2.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
61216 GABAA CLONED HUMAN FNZ ZG-224 2.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
88609 D3 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 2.5 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
1058 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RITANSERIN 2.5 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
31782 M1 CLONED HUMAN 3H-NMS OLANZAPINE 2.5 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
13607 WHOLE BRAIN GUINEA PIG 3H-SR 48692 SR 48692 2.5 Betancur C, et al., 1995 Jan 15, 2025 Jan 15, 2025
20775 D2 BRAIN CALF 3H-Haloperidol 2-Bromo-alpha-ergocryptine 2.5 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
56619 NR3C1 UNDEFINED HUMAN UNDEFINED (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-m-tolylethanol 2.5 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
54829 D3 UNDEFINED HUMAN UNDEFINED N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine 2.5 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
56622 NR3C1 UNDEFINED HUMAN UNDEFINED 4-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonitrile 2.5 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
48689 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 2.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
32052 CORTEX RAT 3H-IDAZOXAN R 50 970 2.5 Megens et al., 1986 Jan 15, 2025 Jan 15, 2025
35124 BRAIN RAT 3H-Cytisine 2-Chloro-3-(2(S)-azetidinylmethoxy)pyridine 2.5 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
4406 5-HT1D CLONED RAT 3H-5HT 5-Hydroxy Tryptamine 2.5 HAMBLIN MW, ET AL., 5/1992 Jan 15, 2025 Jan 15, 2025
36662 CLONED RAT 3H-PRAZOSIN RISPERIDONE 2.5 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
3127 5-HT6 CLONED RAT 3H-LSD OLANZAPINE 2.5 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
91449 5-HT2C CLONED HUMAN 125I-DOI (6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline 2.5 Li P et al 2014 Jan 15, 2025 Jan 15, 2025
94009 5-HT1A CORTEX PIG [3H]WAY 600135 3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 2.5 Ortega R et al 2011 Jan 15, 2025 Jan 15, 2025
65850 GABAA CLONED HUMAN [3H] Flunitrazepam ZG-224 2.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
13630 D2 Temp. Cortex HUMAN 125I-Epidepride FLUPENTHIXOL, Alpha 2.5 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
13886 A1 CEREBELLUM Chick 125I-Aba CHA 2.5 Leung E, et al., 1987 Jan 15, 2025 Jan 15, 2025
56640 NR3C1 UNDEFINED HUMAN UNDEFINED 1-((S)-4-Fluoro-phenyl)-1-[(4aR,5S)-1-(4-fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-ethanol 2.5 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
57408 CB1 UNDEFINED HUMAN UNDEFINED N-cyclohexyl-4-[(2,4-dichlorophenyl)(4-fluorophenyl)methyl]piperazine-1-carboxamide 2.5 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
2881 5-HT2A CORTEX RAT 3H-KETANSERIN LSD 2.5 LEYSON ET AL., 1982 Jan 15, 2025 Jan 15, 2025
17478 PANCREAS GUINEA PIG 125I-VIP Vasoactive intestinal polypeptide 2.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
63047 MC3 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Oic-DNal(2') Arg-Trp-Lys]-NH2 2.5 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
23625 D3 CLONED HUMAN 3H-Butaclamol(+) Cyamemazine 2.5 Hameg A. et al., 2003 Jan 15, 2025 Jan 15, 2025
48713 CLONED HUMAN Functional TAK-013 2.5 Betz SF, et al., 2006 Jan 15, 2025 Jan 15, 2025
53835 5-HT1A UNDEFINED RAT UNDEFINED 2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole 2.5 Siracusa MA et al., 2008 Jan 15, 2025 Jan 15, 2025
37708 DOR CLONED HUMAN 3H-Diprenorphine N,N(CH3)2-Dmt-Tic-NH2 2.5 Tryoen-Toth P, et al., 2005 Jan 15, 2025 Jan 15, 2025
2893 5-HT2A CORTEX RAT 3H-SPIROPERIDOL LSD,2-Bromo 2.5 PEROUTKA & SNYDER, 1979 Jan 15, 2025 Jan 15, 2025
65103 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-4513 2.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
31825 5-HT2A CLONED HUMAN 35S-GTPGammaS OLANZAPINE 2.5 Bymaster F.P., et. al., 1999 Jan 15, 2025 Jan 15, 2025
16212 D2 CORTEX RAT 125I-Epidepride BUTACLAMOL,(+) 2.5 Neve KA, et al., 1990a Jan 15, 2025 Jan 15, 2025
31829 M1 CLONED HUMAN 3H-NMS OLANZAPINE 2.5 Bymaster F.P., et. al., 1999 Jan 15, 2025 Jan 15, 2025
42581 Alpha1B CLONED UNDEFINED UNDEFINED WB 4101 2.5 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
52054 SLC6A4 UNDEFINED HUMAN UNDEFINED N-methyl(2-(4-(methylthio)phenoxy)-5-(4-thiomorpholinobut-1-ynyl)phenyl)methanamine 2.5 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
65623 GABAA CLONED HUMAN [3H] Flunitrazepam Flunitrazepam 2.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
42584 Alpha1C CLONED UNDEFINED UNDEFINED Terazosin 2.5 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
63065 MC3 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Acpc-DNal(2') Arg-Trp-Lys]-NH2 2.5 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
63834 A2B CLONED HUMAN 3H-ZM241385 8-(4-Iodophenyl)-1,3-dipropylxanthine 2.5 Hayallah AM, et al., 2002 Jan 15, 2025 Jan 15, 2025
49506 KOR CLONED HUMAN 3H-Diprenorphine Dynorphin A(1-9)-OH 2.5 Schlechtingen, G et al., 2003 Jan 15, 2025 Jan 15, 2025
55907 MOR UNDEFINED HUMAN UNDEFINED (1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide 2.5 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
11365 5-HT2A CLONED HUMAN 125I-R091150 OLANZAPINE 2.5 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
100965 5-HT2A CLONED HUMAN 3H-KETANSERIN OLANZAPINE 2.5 Snyder et al., 2015 Jan 15, 2025 Jan 15, 2025
34918 CCR5 CLONED UNDEFINED 3H-Epibatidine A-84543 2.5 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
17767 CLONED RAT 125I-VIP VIP [D-Met17] 2.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
34919 CCR5 CLONED UNDEFINED 3H-Epibatidine 5-(1-Ethynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 2.5 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
17512 PANCREAS RAT 125I-VIP VIP Ala8 2.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
31593 D1 Striatal Membranes RAT 3H-SCH23390 C22H27FN2 fumarate (39, -) 2.5 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
100714 MT1 C.H.O. HUMAN 2-I125 iodomelatonin N-Allyl-3-(5-methoxy-1H-indol-3-yl)propanamide 2.5 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
56939 DOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-trimethylfluoro)benzamido]morphinan-oxalate 2.5 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
14956 D4 CLONED HUMAN UNDEFINED HALOPERIDOL 2.5 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 27, 2025
60780 GABAA CLONED HUMAN FNZ Ro15-4513 2.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
7021 Y2 CLONED MOUSE 125I-PYY NPY2-36 2.5 WEINBERG DH, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
50031 Y2 CLONED RABBIT 125I-PYY PYY, human 2.5 Matsumoto M, et al.,1996 Jan 15, 2025 Jan 15, 2025
4720 5-HT1D CLONED BOVINE 3H-5HT 5-CT 2.5 WEINSHANK RL, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
101489 D4 CLONED HUMAN [3H]N-methylspiperone Asenapine 2.5 PDSP Certified Data Mar 20, 2025 Mar 20, 2025
19826 D4 CLONED HUMAN UNDEFINED ILOPERIDONE 2.5 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
66164 5-HT1A CLONED HUMAN 3H-WAY100635 Ziprasidone 2.5 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
884 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHYSERGIDE 2.5 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
32122 CORTEX RAT 3H-Yohimbine R 51 562 2.5 Megens et al., 1986 Jan 15, 2025 Jan 15, 2025
21372 A1 CLONED HUMAN 3H-CPX CPX 2.5 Linden J et al., 1999 Jan 15, 2025 Jan 15, 2025
66175 D3 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 2.5 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 28, 2025
31873 M1 CLONED HUMAN 3H-QNB OLANZAPINE 2.5 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
7043 D4 CLONED HUMAN 3H-NGD 94-1 NGD 94-1 2.5 TALLMAN JF, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
32131 FOREBRAIN RAT 3H-WB4101 Metopimazine 2.5 Megens et al., 1986 Jan 15, 2025 Jan 15, 2025
19844 D3 CLONED HUMAN UNDEFINED RISPERIDONE 2.5 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
63365 CLONED HUMAN 3H- Ketanserin l-(2,5-Dimethoxy-4-hexylphenyl)-2-aminopropane Hydrochloride 2.5 Seggel, Mark R., et al, 1990 Jan 15, 2025 Jan 15, 2025
1670 5-HT2A FR. CORTEX RAT 3H-KETANSERIN ALTANSERIN 2.5 LEYSEN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
49546 retina RABBIT 125I-Iodomelatonin Melatonin,2-Iodo 2.5 Morgan PJ, et al., 1994 Jan 15, 2025 Jan 15, 2025
3724 KOR CLONED HUMAN 3H-U69,593 Naloxone(-) 2.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
4494 D2 BRAIN RAT 3H-SPIPERONE PIMOZIDE 2.5 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
50574 5-HT4A CLONED HUMAN 3H-5HT Prucalopride 2.5 Briejer MR, et al., 2001 Jan 15, 2025 Jan 15, 2025
93841 SERT CLONED HUMAN 3H-IMIPRAMINE IMIPRAMINE 2.5 Wrobel MZ et al 2019 Jan 15, 2025 Jan 28, 2025
51601 Alpha1D UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide 2.5 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
1170 5-HT1D CAUDATE CALF 3H-5HT 5-CT 2.5 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
23954 D3 CLONED HUMAN UNDEFINED RISPERIDONE 2.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
10387 nAChR M10 membranes Mammalian 3H-Epibatidine Anatoxin-a 2.5 Whiteaker P, Sharples CG, Wonnacott S, 1998 Jan 15, 2025 Jan 15, 2025
63379 NMDA FOREBRAIN RAT 3H-MK-801 (+)-MK-801 2.5 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
2964 5-HT2A CORTEX RAT 3H-KETANSERIN METHYSERGIDE 2.5 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
14996 5-HT6 CLONED RAT 3H-Risperidone OLANZAPINE 2.5 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
23956 D3 CLONED HUMAN UNDEFINED SERTINDOLE 2.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
11673 BRAIN HUMAN 3H-KETANSERIN KETANSERIN 2.5 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
35738 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE A-80426 2.5 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
47517 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY NPY [Ala31, Aib32], porcine 2.5 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
159 5-HT1A CORTEX RAT 3H-8-OH-DPAT 5-Methoxytryptamine 2.5 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
15008 5-HT6 CLONED RAT 3H-LSD OLANZAPINE 2.5 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
23716 MC1 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH ACTH-(1-39) 2.5 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
1189 5-HT1D STRIATUM BOVINE 3H-5HT 5-Methoxytryptamine 2.5 HEURING & PEROUTKA, 1987 Jan 15, 2025 Jan 15, 2025
11173 5-HT6 CLONED RAT 3H-Risperidone OLANZAPINE 2.5 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
5800 Alpha2A CELLS HT29 3H-RAUWOLSCINE BAM 1303 2.5 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
4528 5-HT2A BRAIN RAT 3H-SPIPERONE FLUPHENAZINE 2.5 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
17585 T47D HUMAN 125I-VIP VIP Ala27 2.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
70068 MOR CLONED HUMAN 3H-DAMGO c2,2′(Dmt-DCys-Gly-Phe)2-piperazine 2.5 Remesic, M. et, al 2018 Jan 15, 2025 Jan 28, 2025
57780 D2 UNDEFINED HUMAN UNDEFINED (R)-3-((4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one 2.5 Yan Y et al., 2010 Jan 15, 2025 Jan 15, 2025
23990 D3 CLONED HUMAN 3H-SPIPERONE THIORIDAZINE 2.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
17079 BRAIN HUMAN 3H-RAUWOLSCINE RAUWOLSCINE 2.5 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
70843 5-HT2C test test 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)ethanamine 2.5 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
36539 Alpha1A CLONED HUMAN 3H-PRAZOSIN 9-OH-risperidone 2.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
18620 D2 CLONED RAT 3H-RACLOPRIDE SULPIRIDE,(-) 2.5 Strange PG 2001 Jan 15, 2025 Jan 15, 2025
54972 5-HT2A UNDEFINED UNDEFINED UNDEFINED 2-(4-Hexyl-2,5-dimethoxy-phenyl)-1-methyl-ethylamine : (Hydrochloride) 2.5 Runyon SP et al., 2008 Jan 15, 2025 Jan 15, 2025
30397 B2 CLONED HUMAN 3H-BRADYKININ Ethyl {4-[(3-{[({(2E)-3-[6-(Acetylamino)-3-pyridinyl]-2-propenoyl}amino)acetyl](methyl)amino}-2,6-dichlorobenzyl) 2.5 Sawada, Y et al., 2004 Jan 15, 2025 Jan 15, 2025
4543 5-HT2A BRAIN RAT 3H-SPIPERONE RMI 81,582 2.5 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
38591 D3 CLONED RAT 3H-SCH23390 Dinapsoline,(+/-)-4-Methyl-N-propyl 2.5 Qandil AM, et al., 2003 Jan 15, 2025 Jan 15, 2025
51392 M3 UNDEFINED HUMAN UNDEFINED 3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 2.5 Sonda S et al., 2007 Jan 15, 2025 Jan 15, 2025
30404 MOR thalamus CALF 3H-DAMGO Morphine 2.5 Gilbert AK et al., 2004 Jan 15, 2025 Jan 27, 2025
462 5-HT1A CORTEX RAT 3H-8-OH-DPAT RU 24969 2.5 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
19919 A1 BRAIN RAT 3H-cyclohexyladenosine R,S-PHPNECA 2.5 Camaioni E et al., 1997 Jan 15, 2025 Jan 15, 2025
6099 5-HT3 HIPPOCAMPUS GUINEA PIG 3H-PPP-3 PPP, R(+)-3 2.5 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
17107 H1 BRAIN HUMAN 3H-PYRILAMINE PYRILAMINE 2.5 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
68564 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-nicotinamide 2.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
53716 D3 UNDEFINED HUMAN UNDEFINED HALOPERIDOL 2.5 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54230 CB1 UNDEFINED UNDEFINED UNDEFINED 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-isopropyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2.5 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
49623 SST4 CLONED HUMAN 125I-LTT-SST-28 Cortistatin 2.5 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
54231 CB1 UNDEFINED UNDEFINED UNDEFINED 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-isobutyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2.5 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
3804 5-HT7 CLONED HUMAN 3H-LSD CLOZAPINE 2.5 STAM NJ, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
17886 CCK2 BRAIN RAT 125I-CCK-8 Gastrin I 2.5 Nishida A et al., 1994 Jan 15, 2025 Jan 15, 2025
36318 NMDA CORTEX RAT 3H-MK-801 MK-801,(+) 2.5 Bresink I, et al., 1995 Jan 15, 2025 Jan 28, 2025
12512 M1 CLONED HUMAN 3H-MQNB(-) OXO-M 2.5 Mei L, et al., 1991 Jan 15, 2025 Jan 15, 2025
22496 MC1 CLONED HUMAN 125I-NDP-MSH ACTH-(1-39) 2.5 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
62949 CAUDATE CALF 3H-Haloperidol HALOPERIDOL 2.5 Creese, I et al., 1976a Jan 15, 2025 Jan 15, 2025
4588 5-HT2A BRAIN RAT 3H-KETANSERIN FLUPHENAZINE 2.5 ROTH BL, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
98028 SST5 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 2.5 Reubi JC, et.al.,2002 Jan 15, 2025 Jan 15, 2025
62956 CAUDATE CALF 3H-Haloperidol FLUPHENAZINE 2.5 Creese, I et al., 1976a Jan 15, 2025 Jan 15, 2025
91886 A1 CLONED HUMAN 3H-CCPA (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methylphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone 2.5 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
97006 NMDA FOREBRAIN RAT [3H]MK-801 (+)-MK-801 2.5 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
24305 SLC6A4 CLONED HUMAN 3H-5HT Escitalopram 2.5 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
18932 H1 CLONED HUMAN 3H-MEPYRAMINE trans-H2-PAT(-) 2.5 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
98036 SST3 CLONED HUMAN 125I-LTT-SRIF28 KE119 2.5 Reubi JC, et.al.,2002 Jan 15, 2025 Jan 15, 2025
8952 SST5 CLONED RAT 125I-Tyr11-somatostatin-14 AcNH-4-NO2-Phe-c[D-Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH2 2.5 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
48888 KOR BRAIN RAT 3H-NALOXONE DAMGO 2.5 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
32505 5-HT2B CLONED HUMAN 3H-5HT YM348 2.5 Kimura Y, et al., 2004 Jan 15, 2025 Jan 15, 2025
28154 5-HT1B CLONED HUMAN 3H-GR-125743 METHYSERGIDE 2.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
10495 nAChR T.Californica electric organ RAT 125I-Alpha-bgt Epibatidine-(+) 2.5 Sullivan, et al., 1996 Jan 15, 2025 Jan 27, 2025
10754 D2 CLONED RAT 3H-LSD PIMOZIDE 2.51 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
34326 nAChR CLONED RAT 3H-NICOTINE MCC 2.51 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 15, 2025
11037 H1 CLONED HUMAN 3H-MEPYRAMINE CHLORPHENIRAMINE 2.51 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
19492 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(2-Amino-4-chlorophenyl)-1,3-dipropylxanthine 2.51 Bruns RF et al., 1986 Jan 15, 2025 Jan 15, 2025
8493 SST3 CLONED HUMAN 125I-Tyr10-CST14 octreotide 2.51 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
9018 SST5 CLONED HUMAN 125I-SRIF-28 CGP 23996 2.51 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
6459 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 SDZ 205557 2.51 HEGDE SS, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
11864 5-HT1B STRIATUM GUINEA PIG 3H-5CT 5-Hydroxy Tryptamine 2.51 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
15452 5-HT1B CLONED RAT 3H-5HT OXYMETAZOLINE 2.51 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
17004 NOP CLONED HUMAN Leucyl-3H-NC Ro65-6570 2.51 Hashiba E, et al., 2001 Jan 15, 2025 Jan 15, 2025
15477 5-HT1B CLONED MOUSE 3H-5HT CYANOPINDOLOL 2.51 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
41849 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-5-ylamine 2.51 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
11906 H1 CLONED HUMAN 3H-MEPYRAMINE CHLORPHENIRAMINE 2.51 Moguilevsky N, et al., 1995 Jan 15, 2025 Jan 15, 2025
49029 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) AC 915‚HCl 2.51 Berardi, F et al., 2003 Jan 15, 2025 Jan 15, 2025
11918 5-HT1D CLONED HUMAN 35S-GTPGammaS GR 127935 2.51 Price GW, et al., 1997 Jan 15, 2025 Jan 15, 2025
41873 H3 CLONED RAT 3H-Alpha-Me-histamine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine 2.51 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
146 5-HT1A CORTEX RAT 3H-WB4101 5-Hydroxy Tryptamine 2.51 NORMAN ET AL., 1985 Jan 15, 2025 Jan 15, 2025
6296 5-HT7 CLONED GUINEA PIG 3H-5CT OCTOCLOTHEPIN 2.51 TO ZP, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
14258 D3 CLONED RAT 3H-SPIPERONE CHLORPROMAZINE 2.51 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 15, 2025
4030 5-HT4 CLONED RAT 3H-5HT RS 57639 2.51 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
15567 5-HT2A CLONED RAT 125I-DOI DOI 2.51 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
11987 H3 CORTEX RAT 3H-NAMH HISTAMINE 2.51 Brown JD, et al., 1996 Jan 15, 2025 Jan 15, 2025
10713 CLONED RAT 3H-LSD CHLORPROMAZINE 2.51 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
10719 CLONED RAT 3H-LSD PERPHENAZINE 2.51 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
12262 5-HT1D CLONED HUMAN 35S-GTPGammaS GR 127935 2.51 Selkirk JV, et al., 1998 Jan 15, 2025 Jan 15, 2025
15358 5-HT1D CLONED RAT 3H-5HT 5-Hydroxy Tryptamine 2.51 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
23561 H3 CLONED RAT 3H-NAMH A-304121 2.51189 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
69140 H3 CLONED HUMAN 3H-Histamine Clobenpropit 2.51189 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
26400 GAL2 CLONED RAT 125I-GALANIN Galanin (-7 +29), porcine 2.51189 Smith KE, et. al., 1998 Jan 15, 2025 Jan 15, 2025
26403 GAL2 CLONED RAT 125I-GALANIN Galanin, Human 2.51189 Smith KE, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18748 Alpha1D CLONED HUMAN 125I-BE2254 BMY 7378 2.51189 Vicentic A et al., 2002 Jan 15, 2025 Jan 15, 2025
40280 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHYSERGIDE 2.51189 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
25438 M3 CLONED HUMAN 3H-QNB 3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxy-delta2-isoxazoline sesquifumarate 2.51189 De Amici M, et al., 2003 Jan 15, 2025 Jan 15, 2025
40290 5-HT2C Choroid Plexus PIG 3H-KETANSERIN RITANSERIN 2.51189 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
86634 5-HT4 CLONED HUMAN 3H-GR113808 2-Methyl-4-[[1-(2-morpholin-4-ylethyl)-4-piperidinyl]methoxy]- 2H-pyrrolo[3,4-c]quinoline 2.51189 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
28784 SST3 CLONED HUMAN 125I-Tyr10-CST14 octreotide 2.51189 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
63344 Y5 CLONED HUMAN 125I-PYY PP, human 2.51189 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
27260 D3 CLONED HUMAN 125I-IODOSULPRIDE TL99 2.51189 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
63654 5-HT1A CLONED HUMAN 3H-WAY100635 Ziprasidone 2.51189 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
69289 D3 CLONED HUMAN 125I-IODOSULPRIDE trans-3-(2-(4-((1-Naphthalenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine 2.51189 Macdonald G, et al., 2003 Jan 15, 2025 Jan 15, 2025
69295 D3 CLONED HUMAN 125I-IODOSULPRIDE trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine 2.51189 Macdonald G, et al., 2003 Jan 15, 2025 Jan 15, 2025
69319 D3 CLONED HUMAN 125I-IODOSULPRIDE trans-3-(2-(4-((3-(2,6-Difluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine 2.51189 Macdonald G, et al., 2003 Jan 15, 2025 Jan 15, 2025
34767 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[3-(2,4-dimethyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 2.51189 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
34794 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[5-phenyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 2.51189 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
22000 LHRH Pituitary RAT UNDEFINED 8 2.51189 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
17394 H1 CLONED HUMAN 3H-MEPYRAMINE l-Chlorpheniramine 2.51189 Gillard M, et al., 2002 Jan 15, 2025 Jan 15, 2025
68855 SST3 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Ala-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 2.51189 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
27600 Alpha2C CLONED HUMAN 3H-RX821002 Dexmedetomidine 2.5119 Millan MJ, et al., 2000a Jan 15, 2025 Jan 15, 2025
192 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT DMT,5-OH 2.52 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
5553 5-HT2A CLONED HUMAN 125I-DOI OLANZAPINE 2.53 WAINSCOTT DB, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
27060 DOR vas deferens MOUSE 3H-DSLET Leu5-Enkephalin 2.53 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
60708 GABAA CLONED HUMAN FNZ YT-III-25 2.531 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65201 GABAA CLONED HUMAN [3H] Flunitrazepam YT-III-25 2.531 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
12313 AORTA Dog 125I-HEAT PHENTOLAMINE 2.55 Jones SB, et al., 1987 Jan 15, 2025 Jan 15, 2025
41076 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-186 2.55 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
55210 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(bis(2-chlorophenyl)methyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 2.55 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
27086 MOR BRAIN MOUSE 3H-DAMGO Tyr-d-Arg-Phe-A2pr-NH2 2.55 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
56564 MOR UNDEFINED HUMAN UNDEFINED Morphine 2.55 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
542 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIROXATRINE 2.56 ALEXANDER & WOOD, 1988 Jan 15, 2025 Jan 15, 2025
2901 5-HT2A CORTEX HUMAN 3H-SPIPERONE LSD 2.56 PIERCE & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
15449 5-HT1B CLONED RAT 3H-5HT RU 24969 2.57 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
348 5-HT1A CORTEX PIG 3H-8-OH-DPAT LSD 2.57 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
358 5-HT1A CORTEX PIG 3H-8-OH-DPAT LSD 2.57 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
17000 M4 CLONED HUMAN 3H-NMS NNC 11-1585 2.57 Christopoulos A, et al., 2001 Jan 15, 2025 Jan 15, 2025
89613 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 2.5704 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
34095 H3 BRAIN CORTEX GUINEA PIG 3H-Alpha-Me-histamine ABT-239 2.5704 Esbenshade TA, et al., 2004 Jan 15, 2025 Jan 15, 2025
64078 H3 CORTEX GUINEA PIG 3H-Alpha-Me-histamine ABT-239 2.5704 Esbenshade TA, et al., 2004 Jan 15, 2025 Jan 15, 2025
26959 5-HT6 CLONED HUMAN 3H-LSD SB-357134 2.5704 Hirst WD, et.al.,2003 Jan 15, 2025 Jan 15, 2025
32345 M4 LUNG RABBIT 3H-NMS Cyclopentolate 2.5704 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
64658 H1 CLONED HUMAN 3H-PYRILAMINE PERPHENAZINE 2.5704 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
69273 H3 CLONED HUMAN 3H-Alpha-Me-histamine GT 2331 2.5704 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
27292 Alpha1A CLONED HUMAN 3H-PRAZOSIN Roxindole 2.5704 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
34012 NET STRIATUM RAT 3H-Noradrenaline DESIPRAMINE 2.5704 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
36366 MOR BRAIN RAT 3H-DAMGO (2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]-3-phenylpropanoic acid bis(tetrafluoroborate) 2.58 Spetea M, et al., 2004 Jan 15, 2025 Jan 15, 2025
8545 SST4 CLONED RAT 125I-Tyr11-SRIF Somatostatin-14 2.58 O'Carroll AM, et al., 1993 Jan 15, 2025 Jan 15, 2025
343 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT LISURIDE 2.59 HALL ET AL., 1985 Jan 15, 2025 Jan 15, 2025
99719 D3 CLONED RAT [3H]spiperone 4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol 2.59 Luo D et al 2016 Jan 15, 2025 Jan 28, 2025
17149 5-HT2A BRAIN HUMAN 3H-KETANSERIN CLOZAPINE 2.59 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
72448 5-HT1D test test 3H-GR125743 2-(5-Bromo-1H-indol-3-yl)-N,N-dimethylethanamine 2.6 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
17161 5-HT2A BRAIN HUMAN 3H-KETANSERIN ZOTEPINE 2.6 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
17162 5-HT2A BRAIN HUMAN 3H-KETANSERIN KETANSERIN 2.6 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
35850 SLC6A4 CLONED HUMAN 3H-PAROXETINE 3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester 2.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
11790 FR. CORTEX HUMAN 3H-PRAZOSIN CHLORPROMAZINE 2.6 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
6673 D2 ANTERIOR PITUITARY PIG 3H-NEMONAPRIDE HALOPERIDOL 2.6 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
17684 CLONED HUMAN 125I-VIP VIP [D-Asn24] 2.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
4373 5-HT6 CLONED HUMAN 3H-LSD OCTOCLOTHEPIN,(+) 2.6 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
42262 CLONED HUMAN 125I-Motilin Delta 13-16 2.6 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
61462 GABAA CLONED HUMAN FNZ RY-066 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
30488 M4 CLONED HUMAN 3H-QNB 3-Ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 2.6 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
21534 A1 BRAIN RAT 3H-cyclohexyladenosine 10 2.6 Bridges AJ et al., 1988 Jan 15, 2025 Jan 15, 2025
100643 5-HT2B CLONED HUMAN 3H-LSD CYPROHEPTADINE 2.6 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
10792 D2 CLONED HUMAN 125I-IODOSULPRIDE HALOPERIDOL 2.6 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
98090 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-(4-fluorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide 2.6 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
19756 D2 CLONED HUMAN 3H-Sertindole SERTINDOLE 2.6 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
60716 GABAA CLONED HUMAN FNZ XHE-III-14 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
30767 SST5 CLONED RAT 125I-Tyr11-SRIF Somatostatin-14 2.6 Viollet, C et. al., 1997 Jan 15, 2025 Jan 15, 2025
16693 M4 CLONED HUMAN 3H-QNB Trihexyphenidyl 2.6 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
56123 DOR UNDEFINED HUMAN UNDEFINED CCDC 710249, HCl salt 2.6 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
56635 NR3C1 UNDEFINED HUMAN UNDEFINED (R)-1-Cyclopropyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol 2.6 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
16444 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE PHENTOLAMINE 2.6 Naselsky DP, et al., 2001 Jan 15, 2025 Jan 15, 2025
9277 GABAA CLONED HUMAN 3H-RO-15-1788 Ro15-4513 2.6 Hadingham K, et al., 1995 Jan 15, 2025 Jan 27, 2025
57405 CB1 UNDEFINED HUMAN UNDEFINED N-cyclohexyl-4-[(2,4-dichlorophenyl)(4-methoxyphenyl)methyl]piperazine-1-carboxamide 2.6 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
48711 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 2.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
17480 PANCREAS GUINEA PIG 125I-VIP VIP Ala2 2.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
65102 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-4513 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
90961 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (S)-5-((3-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate 2.6 Sun H et al 2016 Jan 15, 2025 Jan 28, 2025
20819 D2 BRAIN CALF 3H-Haloperidol Teflutixol 2.6 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
37463 D3 CLONED HUMAN 3H-YM 09151-2 butylamide benzthiophene 2.6 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
34137 Beta1 CLONED HUMAN 125I-CYP PINDOLOL,(+/-) 2.6 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
40538 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine 2.6 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
30299 DOR CLONED HUMAN 3H-DPDPE 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-4-chlorobenzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 2.6 Black, SL et al., 2003 Jan 15, 2025 Jan 15, 2025
33883 D2 FR. CORTEX RAT 3H-SPIPERONE HALOPERIDOL 2.6 Andersen PH, et al., 1985 Jan 15, 2025 Jan 15, 2025
14943 D3 CLONED RAT UNDEFINED SERTINDOLE 2.6 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
12387 KOR CORTEX RAT 3H-flumazenil Bretazenil 2.6 Giusti P, et al., 1993 Jan 15, 2025 Jan 27, 2025
3684 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl NALMEFENE-HCl 2.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
38758 Sf9 HUMAN 3H-dexamethasone (2-Chloro-5-{4-[((2,4-difluorobenzyl){2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic Acid 2.6 Link JT, et al., 2005 Jan 15, 2025 Jan 15, 2025
91751 A2B CLONED HUMAN 3H-MRS-1754 8-(1-{2-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 2.6 Basu S et al 2017 Jan 15, 2025 Jan 15, 2025
55911 MOR UNDEFINED HUMAN UNDEFINED (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide 2.6 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
13930 5-HT2C CLONED HUMAN 3H-MESULERGINE ZOTEPINE 2.6 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 27, 2025
24170 V2 PANC1 HUMAN 125I-VIP VIP Ala19 2.6 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
60779 GABAA CLONED HUMAN FNZ Ro15-4513 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
68972 GABAA CLONED RAT 3H-Ro15-1788 5-[3-(3,5-Difluoropyridin-2-yl)-4-fluorophenyl]-3-(2,4,6-trifluorophenyl)pyridazine 2.6 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
56944 DOR UNDEFINED UNDEFINED UNDEFINED 4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-yl]benzamide; oxalic acid 2.6 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
11391 D2 CLONED HUMAN 3H-SPIPERONE ORG-5222 2.6 Schotte A, et al., 1996 Jan 15, 2025 Jan 27, 2025
9606 CORTEX RAT 3H-NMS AMITRIPTYLINE 2.6 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
65676 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-III-14 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
16271 M3 CLONED RAT 3H-PIRENZEPINE a 2.6 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
10896 D2 CLONED RAT 3H-SPIPERONE BUTACLAMOL,(+) 2.6 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
2965 5-HT2A CORTEX RAT 3H-SPIROPERIDOL METHYSERGIDE 2.6 PEROUTKA & SNYDER, 1979 Jan 15, 2025 Jan 15, 2025
65686 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-59 (C22H13N3O2F4) 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
17564 CLONED HUMAN 125I-VIP VIP Ala26 2.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
35740 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 2.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
32925 D2 BRAIN MOUSE 3H-SPIROPERIDOL HALOPERIDOL 2.6 Andersen PH, et al., 1988 Jan 15, 2025 Jan 15, 2025
47523 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY CP760524 2.6 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
70053 D3 CLONED HUMAN 3H-SPIPERONE S)-N6-Propyl-N6-(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)-4, 5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine 2.6 Ghosh, B. et, al 2010 Jan 15, 2025 Jan 28, 2025
17063 BRAIN HUMAN 3H-PRAZOSIN Ziprasidone 2.6 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
66476 5-HT7 CLONED HUMAN 3H-LSD N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride 2.6 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
60591 GABAA CLONED HUMAN FNZ JYI-59 2.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
68534 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-chlorobenzamide 2.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
73398 5-HT7 test test 3H- LSD N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride 2.6 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
1721 5-HT2A CORTEX RAT 3H-SPIPERONE BUTACLAMOL,(+) 2.6 PEROUTKA & SNYDER, 1980 Jan 15, 2025 Jan 15, 2025
17081 D2 BRAIN HUMAN 3H-SPIPERONE HALOPERIDOL 2.6 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
17091 D2 BRAIN HUMAN 3H-SPIPERONE Ziprasidone 2.6 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025