The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 9,001-10,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
711845-HT2CCLONEDHUMANUNKNOWNSYA16263>10000Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
5904Alpha2ACLONEDHUMAN3H-RAUWOLSCINEWB 41010.91BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
71440Alpha2BCLONEDHUMAN3H-CLONIDINE4-acetoxy-N,N-diallyltryptamine170Klein LM et al 2018Jan 15, 2025Jan 28, 2025
6160Alpha1CCLONEDBOVINE125I-HEATPRAZOSIN0.37LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64165-HT3CLONEDRAT3H-BIMU-1BIMU 11.6BONHAUS DW, ET AL., 1993Jan 15, 2025Jan 15, 2025
6672D2CLONEDHUMAN3H-NEMONAPRIDEEPIDEPRIDE0.27SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
72208M1CLONEDHUMAN3H-QNB2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
69285-HT2ACLONEDHUMAN3H-KETANSERINTHIORIDAZINE60SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
7184NOPCLONEDMOUSE35S-GTPGammaSAc-RYYKWR-NH21.47Dooley CT, et al., 1997Jan 15, 2025Jan 15, 2025
72720DORCLONEDHUMAN3H-DADLEnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7440BB2CLONEDMOUSE125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14)NMB127Katsuno T, et al., 1999Jan 15, 2025Jan 15, 2025
72976D1CLONEDHUMAN3H-SCH23390catechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7696GABAACLONEDHUMAN3H-MUSCIMOLTHIP102.32Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7952GABAACLONEDHUMAN3H-RO-15-1788152.03He X, et al., 1999Jan 15, 2025Jan 27, 2025
8208SST4CLONEDHUMAN125I-LTT-SST-28SMS 201-9951.36Demchyshyn L, et al., 1993Jan 15, 2025Jan 15, 2025
8464SST5CLONEDHUMAN125I-Tyr3-octreotideBIM 230564.78Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8720SST2CLONEDHUMAN125I-Tyr3-octreotideBIM 23056416.86Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8976SST2CLONEDHUMAN125I-SRIF-28SA2511.88Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74512Beta 1CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9232SST2CLONEDMOUSE125I-MK-678BIM 230590.008Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74768MORCLONEDHUMAN3H-DAMGO(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9488MT2CLONEDHUMAN125I-IodomelatoninN-Acetyltryptamine90Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
75024SERTCLONEDHUMAN3H-CITALOPRAM(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
752805-HT2CCLONEDHUMAN3H-MESULERGINEEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10000CB2CLONEDHUMAN3H-CP-55940JWH-01598.4Griffin G, Tao Q, Abood ME, 2000Jan 15, 2025Jan 15, 2025
75536Beta 1CLONEDHUMAN125I-Pindololpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10256CLONEDHUMAN125I-HEATNOREPINEPHRINE>10000Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75792D3CLONEDHUMAN3H-N-Methylspiperone1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76048M5CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
107685-HT2CCLONEDRAT3H-LSDMELPERONE1258.92ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
763045-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76560Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76816Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77072D2CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77328H1CLONEDHUMAN3H-PYRILAMINE(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77584M1CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77840M5CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78096Sigma 2CLONEDHUMAN3H-DTG(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide9960Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
783525-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
786085-HT2BCLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide400Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788645-HT1ACLONEDHUMAN3H-WAY100635(±)-2,5-Dimethoxy-4-bromoamphetamine2550Ray TS 2010 Jan 15, 2025Jan 15, 2025
791205-HT6CLONEDHUMAN3H-LSD(±)-2,5-Dimethoxy-4-bromoamphetamine5535Ray TS 2010 Jan 15, 2025Jan 15, 2025
79376Alpha1BCLONEDHUMAN3H-PRAZOSINDMT,5-MeO>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14096Alpha2ACLONEDPIG3H-YohimbineGuanabenz57.54Brink CB, et al., 2000Jan 15, 2025Jan 15, 2025
79632CLONEDHUMAN3H-CLONIDINE(±)-2,5-Dimethoxy-4-ethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79888M5CLONEDHUMAN3H-QNB5-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14608D2CLONEDRAT125I-IODOSULPRIDESB-277011-A2818.38Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80144V2CLONEDHUMAN3H-VASOPRESSIN(±)-2,5-Dimethoxy-4-ethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14864D2CLONEDRATUNDEFINEDCLOZAPINE36Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
804005-HT4CLONEDHUMAN3H-GR113808(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15120PTGFRCLONEDHUMAN3H-PGF2AlphaPGF2Alpha,17-phenyl18Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806565-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153765-HT1BCLONEDHUMAN3H-5HTTFMPP114.81BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809125-HT1BCLONEDHUMAN3H-5CT3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine707.946Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
156325-HT2BCLONEDRAT3H-5HTSCH 2339083.17BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
811685-HT3CLONEDHUMAN3H-GR65630N-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158885-HT7CLONEDRATUNDEFINEDSPIPERONE19.95BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81424H1CLONEDHUMAN3H-PYRILAMINE1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-methyl-N-[[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl]methanamine>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16144D1CLONEDHUMAN3H-SCH23390HALOPERIDOL27Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
816805-HT2BCLONEDHUMAN3H-LSD(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
81936M5CLONEDHUMAN3H-QNB(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 15, 2025
16656M2CLONEDHUMAN3H-QNBBiperidine6.3Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
821925-HT2ACLONEDHUMAN3H-KETANSERIN2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one65Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824485-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine0.6Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82704D1CLONEDHUMAN3H-SCH23390(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
17680CLONEDHUMAN125I-VIPVIP [D-Lys15]2Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832165-HT2ACLONEDHUMAN125I-DOISB242087120Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83472M5CLONEDHUMAN3H-NMS1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine2.39883Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83728SERTCLONEDHUMAN3H-CITALOPRAMmethyl (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate372PDSP Certified DataJan 15, 2025Jan 28, 2025
83984KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
18704CGRP1CLONEDPIG125-h alpha-CGRP[N-acetyl]h alpha-CGRP8-371.3Rorabaugh BR et al., 2001Jan 15, 2025Jan 15, 2025
84240KORCLONEDHUMAN3H-U69593(±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide4PDSP Certified DataJan 15, 2025Jan 28, 2025
18960H1CLONEDGUINEA PIG3H-MEPYRAMINE+ 1 mM GTP>10000Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84496KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(2,6-difluorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19216CLONEDRAT125I-VIPAcetyl-His1-PACAP-278Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84752DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19472GPR24CLONEDRAT125I-MCH-(4-19)T-2262968.6Takekawa S et al., 2002Jan 15, 2025Jan 15, 2025
85008DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19728D2CLONEDHUMANUNDEFINEDCHLORPROTHIXENE3.3Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
86032Alpha1ACLONEDHUMAN3H-PRAZOSIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86288A2BCLONEDHUMAN3H-PSB-6038-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
87568D4CLONEDHUMAN3H-N-Methylspiperone2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87824D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline1751Staron J et al 2016Jan 15, 2025Jan 28, 2025
22544D2CLONEDHUMAN3H-MethylspiperoneQuetiapine1000Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88080A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22800H1CLONEDHUMAN3H-PYRILAMINEL-homocysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23056nAChRCLONEDHUMAN3H-EpibatidineL-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
88592D4CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE54Peprah K et al 2012Jan 15, 2025Jan 28, 2025
23568GPR10CLONEDHUMAN125I-PrRP20RFRP-1>10000Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
89360D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide1959Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
240805-HT2ACLONEDHUMAN3H-KETANSERINLOXAPINE2Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89616D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89872nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride192Liu J et al 2010Jan 15, 2025Jan 29, 2025
90128D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxyphenethylamine9000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24848NETCLONEDHUMAN3H-NisoxetineCLOZAPINE3168PDSP Certified DataJan 15, 2025Jan 15, 2025
90384A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25104EP4CLONEDHUMAN3H-PGE2Quetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90640A2BCLONEDHUMAN3H-PSB-6034-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide302 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25360D2CLONEDHUMAN3H-NMSPZOTEPINE25PDSP Certified DataJan 15, 2025Jan 15, 2025
25616D3CLONEDRAT3H-NMSPCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91152A2ACLONEDHUMAN3H-CGS-216802-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methylsulfanyl]-N-(2-methylphenyl)acetamide2360Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91408CB1CLONEDHUMAN3H-CP55940O-6215332Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26128Alpha1BCLONEDHUMAN125I-HEATPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91664A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide129Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26384GAL1CLONEDRAT125I-GALANINGalanin [D-Trp2], porcine407.38Smith KE, et. al., 1998Jan 15, 2025Jan 15, 2025
91920A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(3,4-dichloro-phenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26640D5CLONEDHUMAN3H-SCH23390Rutin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921765-HT6CLONEDHUMAN3H-LSD3-Chloro-N-(1-{2-[(propan-2-yl)-phenyloxy]ethyl} pyrrolidin-3-yl)benzenesulfonamide245Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268965-HT2BCLONEDHUMAN3H-5HTxanomeline19.9526Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92432KORCLONEDHUMAN3H-U6959315,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92688H1CLONEDHUMAN3H-PYRILAMINE9,13-epoxy-15,16-dihydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274085-HT1ACLONEDHUMAN3H-8-OH-DPATLISURIDE0.147911Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929445-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine6Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276645-HT1DCLONEDHUMAN3H-GR-125743MDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279205-HT2ACLONEDHUMAN3H-KETANSERIN5-Hydroxy Tryptamine341Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28176Alpha2BCLONEDHUMAN3H-CLONIDINEMETHYSERGIDE106PDSP Certified DataJan 15, 2025Jan 15, 2025
93712A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester14.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
28432mGluR5CLONEDHUMAN3H-QuisqualateL-CCG-I1500Mutel V, et.al., 2000Jan 15, 2025Jan 28, 2025
93968D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one7.1Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28688DORCLONEDHUMAN3H-DiprenorphineARIPIPRAZOLE>10000Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942245-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-methallyloxyamphetamine61Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29200SST2CLONEDHUMANUNDEFINEDsomatostatin-280.2Patel YC, 1999Jan 15, 2025Jan 15, 2025
947365-HT2BCLONEDHUMAN3H-LSD4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94992D3CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
297125-HT2CCLONEDRAT3H-MESULERGINECLOZAPINE11Liao Y, et.al., 1999Jan 15, 2025Jan 15, 2025
29968H4CLONEDHUMAN3H-HistamineBurimamide180Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30224Calcium channelCLONEDRATUNDEFINEDDuloxetine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 28, 2025
957605-HT7CLONEDHUMAN3H-LSDtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96016SERTCLONEDHUMAN3H-CITALOPRAM6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
30736CLONEDRATUNDEFINEDAtomoxetine1000Bymaster F.P., et. al., 2002Jan 15, 2025Jan 15, 2025
96272Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30992CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
96528M2CLONEDHUMAN[3H]-NMS6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31248D2CLONEDHUMAN3H-NMSPPPP, S(-)-3810PDSP Certified DataJan 15, 2025Jan 15, 2025
96784D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde5.7Mannel B et al 2017Jan 15, 2025Jan 28, 2025
315045-HT1FCLONEDHUMAN3H-5HT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)>10000Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
970405-HT1DCLONEDHUMAN[3H]TiotidineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97296MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol12.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97552A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32784NK3CLONEDHUMAN125I-MePhe7-NKBSR 1428011.7Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98320D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 126Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985765-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
332965-HT7CLONEDHUMAN3H-LSDAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98832Alpha1BCLONEDHUMAN3H-PRAZOSIN1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine94Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
99344D3CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline13.1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34064P2X2, P2X3CLONEDHUMAN3H-A-317491ATP,3'-deoxy22.7Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99600A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine9.25Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34320nAChRCLONEDRAT3H-NICOTINEAlpha-Conotoxin MII3210Grinevich VP, et al., 2004Jan 15, 2025Jan 15, 2025
99856NETCLONEDHUMAN[3H] Nisoxetine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide750Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
100112Alpha2ACLONEDHUMAN3H-RAUWOLSCINEQuetiapine1207PDSP Certified DataJan 15, 2025Jan 28, 2025
34832CB1CLONEDHUMAN3H-CP-55940Rinvanil>10000Jan 15, 2025Jan 15, 2025
100368Alpha2BCLONEDHUMAN3H-RAUWOLSCINEILOPERIDONE11PDSP Certified DataJan 15, 2025Jan 28, 2025
100624CGRPCLONEDHUMANFunctionalN2-[4-Amino-3,5-dibromo-N-(3-phenyl-1-oxopropyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrochloride>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
35600D2CLONEDHUMAN3H-SPIPERONE1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin61Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35856SLC6A4CLONEDHUMAN3H-PAROXETINE5-(2,2,2-Trifluoroacetyl)-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole15Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013925-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione482Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101648GABAACLONEDHUMAN[3H]-MuscimolPerospirone>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
101904H4CLONEDHUMAN[3H]HistamineZiprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
366245-HT2ACLONEDHUMAN125I-R091150HALOPERIDOL435Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102160Alpha2BCLONEDHUMAN[3H]rauwolscineNEMONAPRIDE472PDSP Certified DataMar 25, 2025Jul 28, 2026
37904CDK1CLONEDHUMANFunctional4-[[5-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide8Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38160CLONEDRAT3H-dexamethasoneC55H78NO780von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
38416D3CLONEDHUMAN3H-NEMONAPRIDEMCL-204283Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
39440NETCLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396965-HT2BCLONEDHUMAN3H-5HTVER-332330.1995Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
399525-HT7CLONEDRATFunctionalBW-723C861000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
40464mGluR5CLONEDRATFunctional(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40720mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3-diazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41232CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-cyano-4,4-diphenylbutyl)-4-hydroxy-1-methylpiperidinium Iodide>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42000M1CLONEDHUMAN3H-QNBPAROXETINE300Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42256CLONEDHUMANFunctional1-Benzhydryl-1H-benzotriazole-5-carboxylic acid>10000Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42512CLONEDHUMANUNDEFINED[Nle13]-Motilin0.436516Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43024GAKCLONEDHUMAN3H-StaurosporineZD-6474330Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43280CLK3CLONEDHUMAN3H-StaurosporineEKB-5692100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43536LYNCLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43792ACK1CLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44048JAK1CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44304CSNK1G1CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44560MAPK10CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44816CaMKCLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
45072STK3 mouseCLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45328LCKCLONEDHUMANFunctionalPP260Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45584NETCLONEDHUMAN3H-NisoxetineFemoxetine760Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458405-HT2BCLONEDHUMAN3H-LSDPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46096Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46864M5CLONEDHUMAN3H-QNBPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47376Grik5CLONEDHUMAN3H-Kainic acidLY 2935584200Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47888SST3CLONEDHUMAN3H-thymidineBIM-237451000Zatelli MC, et.al., 2002Jan 15, 2025Jan 15, 2025
48144Y4CLONEDHUMAN3H-Propionyl-NPYPP, human0.06Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48656GNRHRCLONEDHUMANFunctional1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride0.1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
48912Y1CLONEDChicken[125I] - Peptide YYPP, rat>10000Holmberg, SK et al., 2002Jan 15, 2025Jan 15, 2025
49168CCK1CLONEDHUMAN125I-CCK-8LYS3221000Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49680Y2CLONEDChicken[125I] - Peptide YYPP, human1000Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49936mGluR2CLONEDRATFunctional2-amino-suberic acid>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 28, 2025
50192SLC6A3CLONEDRAT3H-dopamineBip-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly1800Ding, J., et, al., 2006Jan 15, 2025Jan 15, 2025
50448NETCLONEDHUMAN3H-NisoxetineN,N-Dimethyl-4-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine8854Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581285-HT2ACLONEDHUMAN125I-DOIN-(3-Methylbenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate1.17Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58384H4CLONEDHUMAN3H-HistamineMRS5697>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58640Sigma 1CLONEDHUMAN3H-Pentazocine(+)Cloperatine20Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58896nAChRCLONEDHUMAN3H-EpibatidineCamel Snus extract177.5Harris A, et al., 2015Jan 15, 2025Jan 28, 2025
591525-HT2ACLONEDHUMAN3H-KETANSERINBROMOCRIPTINE107Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59408D4CLONEDHUMAN3H-N-MethylspiporoneN-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(3-thienyl)benzamide18Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59920M4CLONEDHUMAN3H-QNB4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60176A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-4-(2-((3,4-Difluorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane- 1-carboxamide1.65Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60432GABAACLONEDHUMANFNZWY-TSC-40.007Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60688GABAACLONEDHUMANFNZJYI-192.176Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60944GABAACLONEDHUMANFNZZG69A54.6Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61200GABAACLONEDHUMANFNZJYI-065000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61456GABAACLONEDHUMANFNZRY-05885Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617125-HT2BCLONEDHUMAN3H-LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2,5-dimethoxyphenyl)propan-1-amine36Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62224MORCLONEDHUMAN3H-DAMGOTianeptine768PDSP Certified DataJan 15, 2025Jan 15, 2025
62480SLC6A3CLONEDHUMANWIN354282-methoxy-diphenidine2915Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63504D2CLONEDRAT3H-N-MethylspiperoneRISPERIDONE1.8Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
63760CXCR3CLONEDHUMAN125I-CXCL11CXCL951.1Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
640165-HT6CLONEDHUMAN3H-LSD1-[1-(2,5-Dimethoxybenzenesulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one131.3Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642725-HT2CCLONEDRAT3H-MESULERGINECHLORPROMAZINE15.4882Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64528CLONEDHUMAN3H-Estradiol(+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide0.1Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65296GABAACLONEDHUMAN[3H] FlunitrazepamZG-20810.9Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65553GABAACLONEDHUMAN[3H] FlunitrazepamFG82050.4Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65809GABAACLONEDHUMAN[3H] FlunitrazepamXLI-2TC1.673Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66065Alpha1ACLONEDHUMAN3H-PRAZOSINMellpaladine B1898Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66321DATCLONEDHUMAN3H-WIN35428Finazine59Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
66577SERTCLONEDHUMAN3H-CITALOPRAM3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66833Beta2CLONEDHUMAN3H-CGP12177N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67089Alpha1DCLONEDHUMAN3H-PRAZOSIN1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
673455-HT5ACLONEDHUMAN3H-LSD1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
678575-HT2ACLONEDHUMAN3H-Ketaserin(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline390Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68625UTCLONEDHUMANI125-urotensin IIH-Asp-C[Pen-Phe-DTrp-Lys-Tyr-Cys]Val-OH1.25893Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
33455-HT1ACLONEDHUMAN3H-8-OH-DPATDHE1.5TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68881SST4CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Ala-Thr-Phe-Thr-Ser-Cys}-NH21000Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69137H3CLONEDHUMAN3H-Histamineimmethridine0.794328Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
38575-HT6CLONEDRAT3H-LSDRISPERIDONE1122KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
4113KORCLONEDHUMAN3H-U69,593ETORPHINE - HCI0.2TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69649Alpha2CCLONEDHUMAN3H-RAUWOLSCINEDPH3052Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43695-HT6CLONEDHUMAN3H-LSDTENILAPINE570KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69905D3CLONEDHUMAN3H-N-Methylspiperone4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4625SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDING HIGHLU 19,0053.2PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48815-HT2BCLONEDHUMAN3H-RAUWOLSCINEMETHIOTHEPIN0.58WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704175-HT7CLONEDHUMAN3H-LSDMRP42696.2Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51375-HT2BCLONEDHUMAN3H-5HTM-154341NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70673MORCLONEDHUMAN3H-Diprenorphineoxycodone780Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
53935-HT2BCLONEDRAT3H-5HT5-Hydroxy Tryptamine10BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
70929Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
71185H1CLONEDHUMAN3H-PYRILAMINEARIPIPRAZOLE25.1Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5905Alpha2ACLONEDHUMAN3H-RAUWOLSCINEBAM 13030.39BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
71441Alpha2CCLONEDHUMAN3H-CLONIDINE4-acetoxy-N,N-diallyltryptamine748Klein LM et al 2018Jan 15, 2025Jan 28, 2025
6161Alpha1CCLONEDBOVINE125I-HEATPHENTOLAMINE15.3LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64175-HT3CLONEDRAT3H-BIMU-1BIMU 81BONHAUS DW, ET AL., 1993Jan 15, 2025Jan 15, 2025
72209M2CLONEDHUMAN3H-QNB2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
69295-HT2ACLONEDHUMAN3H-KETANSERINTRIFLUOPERAZINE135SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
7185NOPCLONEDMOUSE35S-GTPGammaSAc-RYYKWK-NH20.72Dooley CT, et al., 1997Jan 15, 2025Jan 15, 2025
7441BB2CLONEDMOUSE125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14)DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14)0.19Katsuno T, et al., 1999Jan 15, 2025Jan 15, 2025
72977D5CLONEDHUMAN3H-SCH23390catechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7697GABAACLONEDHUMAN3H-MUSCIMOLP4S72.44Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7953GABAACLONEDHUMAN3H-RO-15-17881617.3He X, et al., 1999Jan 15, 2025Jan 27, 2025
8209SST4CLONEDHUMAN125I-LTT-SST-28somatostatin-282.2Demchyshyn L, et al., 1993Jan 15, 2025Jan 15, 2025
8465SST5CLONEDHUMAN125I-Tyr3-octreotideBIM 230520.52Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8721SST2CLONEDHUMAN125I-Tyr3-octreotidecycloantagonist SA1698.24Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8977SST2CLONEDHUMAN125I-SRIF-28SMS 201-9950.31Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74513Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9233SST2CLONEDMOUSE125I-MK-678BIM 230600.01Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
9489MT2CLONEDHUMAN125I-IodomelatoninN-Acetyltryptamine,5-Hydroxy210Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
75025NETCLONEDHUMAN3H-Nisoxetine(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
752815-HT3CLONEDHUMAN3H-GR-65630Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10001CB2CLONEDHUMAN3H-CP-55940JWH-0510.33Griffin G, Tao Q, Abood ME, 2000Jan 15, 2025Jan 15, 2025
75537Beta3CLONEDHUMAN125I-Pindololpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10257CLONEDHUMAN125I-HEATOXYMETAZOLINE15.84Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75793D4CLONEDHUMAN3H-N-Methylspiperone1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76049Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10769CLONEDRAT3H-LSDZOTEPINE0.63ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
763055-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76561Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76817Beta 2CLONEDHUMAN3H-CGP12177(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77073D3CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
773295-HT1DCLONEDHUMAN3H-Cimetidine(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77585M2CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77841NETCLONEDHUMAN3H-Nisoxetine(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78097DORCLONEDHUMAN3H-DADLE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide1110Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
783535-HT1BCLONEDHUMAN3H-5-CT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
786095-HT2CCLONEDHUMAN3H-MESULERGINE(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788655-HT1ACLONEDHUMAN3H-WAY100635(±)-3,4-Methylenedioxyamphetamine3762Ray TS 2010 Jan 15, 2025Jan 15, 2025
791215-HT6CLONEDHUMAN3H-LSD(±)-3,4-Methylenedioxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79377Alpha1BCLONEDHUMAN3H-PRAZOSINN,N-Diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14097Alpha2ACLONEDPIG3H-YohimbineOXYMETAZOLINE35.48Brink CB, et al., 2000Jan 15, 2025Jan 15, 2025
79633CLONEDHUMAN3H-CLONIDINE5-Methoxy-N-methyl-N-isopropyltryptamine879.4Ray TS 2010 Jan 15, 2025Jan 15, 2025
79889M5CLONEDHUMAN3H-QNBN,N-Dipropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
146095-HT2ACLONEDHUMAN3H-KETANSERINSB-277011-A>10000Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80145V2CLONEDHUMAN3H-VASOPRESSIN5-Methoxy-N-methyl-N-isopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14865D2CLONEDRATUNDEFINEDOLANZAPINE2.1Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
804015-HT5ACLONEDHUMAN3H-LSD(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15121PTGFRCLONEDHUMAN3H-PGF2AlphaPGF2 Alpha, 1-isopropyl ester3200Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806575-HT1BCLONEDHUMAN3H-5-CT(Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153775-HT1BCLONEDHUMAN3H-5HTTRYPTAMINE524.8BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809135-HT1BCLONEDHUMAN3H-5CT5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine1230.27Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
811695-HT5ACLONEDHUMAN3H-LSDN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158895-HT7CLONEDRATUNDEFINEDDHE151.35BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81425H1CLONEDHUMAN3H-PYRILAMINE2-[(2R)-4-[(5-methyl-2-naphthalen-2-yl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]ethanamine1866Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16145D1CLONEDHUMAN3H-SCH23390CHLORPROMAZINE73Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
816815-HT2CCLONEDHUMAN3H-MESULERGINE(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
81937MORCLONEDHUMAN3H-DAMGO(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16657M2CLONEDHUMAN3H-QNBATR0.9Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
821935-HT2BCLONEDHUMAN3H-LSD2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one10Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824495-HT1BCLONEDHUMAN3H-5-CT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82705D5CLONEDHUMAN3H-SCH23390(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
17681CLONEDHUMAN125I-VIPVIP [D-Leu27]0.43Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832175-HT1ACLONEDHUMAN3H-8-OH-DPATSB2420879300Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
17937CRF1CLONEDHUMAN125-Tyr0 ovineSSR125543A1.86209Gully D et al., 2001Jan 15, 2025Jan 15, 2025
83473M5CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+)69.1831Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83729KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5.3PDSP Certified DataJan 15, 2025Jan 28, 2025
83985KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N,2-bis(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5650PDSP Certified DataJan 15, 2025Jan 28, 2025
18705CGRP1CLONEDPIG125-h alpha-CGRPh alpha-CGRP8-375.7Rorabaugh BR et al., 2001Jan 15, 2025Jan 15, 2025
84241DORCLONEDHUMAN3H-DADLE(±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
18961H1CLONEDGUINEA PIG3H-MEPYRAMINEHISTAMINE>10000Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84497MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19217CLONEDRAT125I-VIP[Phe1]VIP30Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84753MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19473GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHMCH1.5Sailer AW et al., 2001Jan 15, 2025Jan 15, 2025
85009MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19729D2CLONEDHUMAN3H-ClozapineCLOZAPINE44Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
86033Alpha1BCLONEDHUMAN3H-PRAZOSIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86289A3CLONEDHUMAN3H-PSB-118-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
87569DATCLONEDHUMAN3H-WIN 35,4282-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
878255-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline347Staron J et al 2016Jan 15, 2025Jan 15, 2025
22545D2CLONEDHUMAN3H-MethylspiperoneOLANZAPINE31.8Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88081A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22801H1CLONEDHUMAN3H-PYRILAMINEL-cysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23057nAChRCLONEDHUMAN3H-EpibatidineD-methionine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
885935-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE140Peprah K et al 2012Jan 15, 2025Jan 15, 2025
23569GPR10CLONEDHUMAN125I-PrRP20PrRP24-3147Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
893615-HT6CLONEDHUMAN3H-LSDN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide2815Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240815-HT2ACLONEDHUMAN3H-KETANSERINMELPERONE180Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89617D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
24337SLC6A3CLONEDHUMAN3H-dopamineEscitalopram>10000Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89873nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
90129D2CLONEDHUMAN3H-SPIPERONE4-iodo-2,5-dimethoxyphenethylamine2700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24849Alpha2BCLONEDHUMAN3H-CLONIDINECLOZAPINE27PDSP Certified DataJan 15, 2025Jan 15, 2025
90385A2BCLONEDHUMAN3H-PSB-603N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90641A2BCLONEDHUMAN3H-PSB-6034-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25617H4CLONEDHUMAN3H-HistamineCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91153A3CLONEDHUMAN125I-AB-MECA2-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methylsulfanyl]-N-(2-methylphenyl)acetamide4860Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25873Beta2CLONEDHUMAN125I-PindololPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
91409CB1CLONEDHUMAN3H-SR144528O-6215221Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26129H1CLONEDHUMAN3H-PYRILAMINEPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91665A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide25.4Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26385GAL1CLONEDRAT125I-GALANINGalanin [-7 to +29], porcine24.5471Smith KE, et. al., 1998Jan 15, 2025Jan 15, 2025
91921A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(3-trifluoro-methylphenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26641D5CLONEDHUMAN3H-SCH23390Hyperoside>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921775-HT6CLONEDHUMAN3H-LSD3-Chloro-N-({1-[2-(methylsulfanyl)phenyloxy]ethyl}pyrrolidin-3-yl)benzenesulfonamide185Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268975-HT2CCLONEDHUMAN3H-MESULERGINExanomeline39.8107Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92433KORCLONEDHUMAN3H-U695939,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271535-HT2ACLONEDHUMAN125I-DOI5-Hydroxy Tryptamine8.2May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92689H1CLONEDHUMAN3H-PYRILAMINE9,13-epoxylabd-5-ene-7 b,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274095-HT1ACLONEDHUMAN3H-8-OH-DPATPERGOLIDE1.90546Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929455-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine12Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276655-HT1BCLONEDHUMAN3H-GR-125743MDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279215-HT2ACLONEDHUMAN3H-DOB5-Hydroxy Tryptamine14Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28177Beta1CLONEDHUMAN125I-PindololMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93713A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester3.37Federico S et al 2018Jan 15, 2025Jan 15, 2025
28433CLONEDHUMAN3H-Quisqualate1S, 3R-ACPD3200Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93969D2CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile38Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28689KORCLONEDHUMAN3H-BremazocineARIPIPRAZOLE>10000Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942255-HT2ACLONEDHUMAN3H-KETANSERIN4-allyloxy-2,5-dimethoxyamphetamine150Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29201SST2CLONEDHUMANUNDEFINEDSomatostatin-140.2Patel YC, 1999Jan 15, 2025Jan 15, 2025
947375-HT2BCLONEDHUMAN3H-LSD5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94993D4CLONEDHUMAN3H-Methylspiperone4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29969H3CLONEDHUMAN3H-HistamineBurimamide84Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30225Calcium channelCLONEDRATUNDEFINEDVenlafaxine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 28, 2025
957615-HT5ACLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30481CLONEDXenopusUNDEFINED(S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxohexyl)amino]benzenepropaneamide bis(trifluoroacetate) 1000Kromann H, et. al., 2002aJan 15, 2025Jan 15, 2025
96017SERTCLONEDHUMAN3H-CITALOPRAMTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
30737NOSCLONEDRATUNDEFINEDAtomoxetine1000Bymaster F.P., et. al., 2002Jan 15, 2025Jan 15, 2025
96273Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30993CCK1CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
96529M3CLONEDHUMAN[3H]-NMS6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31249D3CLONEDRAT3H-NMSPPPP, S(-)-351.2PDSP Certified DataJan 15, 2025Jan 15, 2025
96785D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)3.4Mannel B et al 2017Jan 15, 2025Jan 28, 2025
315055-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)2515.89Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97041H4CLONEDHUMAN[3H]HistamineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97297MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol6.97Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97553A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate278Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32785EAAT2CLONEDHUMAN3H-D-AspartateWAY-8552570.4Dunlop J, et al., 2003Jan 15, 2025Jan 15, 2025
98321D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985775-HT2CCLONEDHUMAN[3H]-mesulergine2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
33297D1CLONEDHUMAN3H-SCH23390Acetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98833Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine221Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33553CB2CLONEDHUMAN3H-CP-55940Naproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99345D3CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-phenyl-1H-1,2,3-triazol-4-yl)butyl)piperazine5.42Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34065P2X2, P2X3CLONEDHUMAN3H-A-317491ATP,Gamma S24.4Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99601A1CLONEDHUMAN3H-CCPA8-[{4-(2-(Diethylaminoethylamino)-2-oxoethoxy)-3-meth-oxy}-phenyl]-1,3-dimethyl-xanthine10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34321nAChRCLONEDRAT3H-NICOTINELobeline, (-)12.1Grinevich VP, et al., 2004Jan 15, 2025Jan 15, 2025
99857NETCLONEDHUMAN[3H] Nisoxetine(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2400Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
100113Alpha2BCLONEDHUMAN3H-RAUWOLSCINEQuetiapine96PDSP Certified DataJan 15, 2025Jan 28, 2025
34833CB1CLONEDHUMAN3H-CP-55940Rinvanil, Acetyl>10000Jan 15, 2025Jan 15, 2025
100369Beta1CLONEDHUMAN125I-PindololILOPERIDONE>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
35601D2CLONEDHUMAN3H-SPIPERONE1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin110Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35857Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole7.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013935-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione533Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101649H1CLONEDHUMAN[3H] PyrilaminePerospirone10PDSP Certified DataMar 21, 2025Jul 28, 2026
101905Alpha1ACLONEDHUMAN[3H]prazosinZiprasidone44PDSP Certified DataMar 24, 2025Jul 28, 2026
366255-HT2ACLONEDHUMAN125I-R091150CLOZAPINE6.3Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102161Alpha2CCLONEDHUMAN[3H]rauwolscineNEMONAPRIDE710PDSP Certified DataMar 25, 2025Jul 28, 2026
37905CDK1CLONEDHUMANFunctional4-[[5-Amino-1-(2,3,6-trifluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide3.2Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38161CLONEDRAT3H-dexamethasoneC56H80NO8170von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
38417D3CLONEDHUMAN3H-NEMONAPRIDESCH 23390>10000Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
39441SLC6A3CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396975-HT2CCLONEDHUMAN3H-5HT5-CT204.174Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40465mGluR5CLONEDRATFunctional(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40721mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one183Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41233CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)piperazin-1-yl)-2,2-diphenypentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42001M1CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.044Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42257CLONEDHUMANFunctional1-(3’-Methoxybenzyl)-1H-benzotriazole-5-carboxylic acid5011.87Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42513CLONEDHUMANUNDEFINEDerythromycin-A512.861Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43025GAKCLONEDHUMAN3H-StaurosporineCI-103344Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43281CLK3CLONEDHUMAN3H-StaurosporineMLN-5189000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43537MAP3K4CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43793STK6CLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44049PKMYT1CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44305CSNK1G2CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44561KITCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44817CaMKCLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
45073STK36CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45329CSKCLONEDHUMANFunctionalPP2730Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45585SLC6A3CLONEDHUMAN3H-WIN 35,428Femoxetine2050Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458415-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46097Alpha2BCLONEDHUMAN3H-CLONIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46865M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47377Grik5CLONEDHUMAN3H-Kainic acidLY 4677117400Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47889SST4CLONEDHUMAN3H-thymidineBIM-237451000Zatelli MC, et.al., 2002Jan 15, 2025Jan 15, 2025
48145Y4CLONEDHUMAN3H-Propionyl-NPYPYY 3-3615Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48657CLONEDHUMANFunctionalN-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride274Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
48913Y1CLONEDChicken[125I] - Peptide YYPP, human>10000Holmberg, SK et al., 2002Jan 15, 2025Jan 15, 2025
49169CCK2CLONEDHUMAN125I-CCK-8LYS201>10000Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49681Y2CLONEDChicken[125I] - Peptide YYPP, chicken1000Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49937mGluR6CLONEDRATFunctional2-amino-suberic acid>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 15, 2025
50193SLC6A3CLONEDRAT3H-dopamineNal1-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly>10000Ding, J., et, al., 2006Jan 15, 2025Jan 15, 2025
50449NETCLONEDHUMAN3H-NisoxetineN,N-Dimethyl-5-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine667Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581295-HT2ACLONEDHUMAN125I-DOIN-(3-Methylthiobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate2.95Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58385H4CLONEDHUMAN3H-HistamineMRS5678>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58641Sigma 2CLONEDHUMAN3H-DTGCloperatine900Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58897nAChRCLONEDHUMAN3H-EpibatidineKodiak extract168.4Harris A, et al., 2015Jan 15, 2025Jan 28, 2025
591535-HT1ACLONEDHUMAN3H-WAY100635BROMOCRIPTINE12.9Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59409D2CLONEDHUMAN3H-N-MethylspiporoneN-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(3-thienyl)benzamide900Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59921M5CLONEDHUMAN3H-QNB4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60177A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((2-methoxyphenyl)ethynyl)- 6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1- carboxamide0.77Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60433GABAACLONEDHUMANFNZWY-TSC-40.99Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60689GABAACLONEDHUMANFNZJYI-19205Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60945GABAACLONEDHUMANFNZZG69A0.85Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61201GABAACLONEDHUMANFNZJYI-065.48Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61457GABAACLONEDHUMANFNZRY-05840Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617135-HT2BCLONEDHUMAN3H-LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(4-methoxyphenyl)propan-1-amine6.8Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62225KORCLONEDHUMAN3H-U69,593Tianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
62481SLC6A3CLONEDHUMANWIN354283-methoxy-diphenidine88Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63249A1CLONEDHUMAN[3 H]N6 -Rphenylisopropyladenosine(1S,2R,3S,4R,5S)-4-(2-((3,4-Difluorophenyl)ethynyl)-6-methyl-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide5430Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
635055-HT1ACLONEDRAT3H-WAY100635RISPERIDONE250Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
63761CXCR3CLONEDHUMAN125I-CXCL11CXCL1010.4Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64017D3CLONEDMOUSE3H-SPIPERONE(+)-Butaclamol0.14Fishburn CS, et al., 1993Jan 15, 2025Jan 15, 2025
642735-HT2CCLONEDRAT3H-MESULERGINECHLORPROTHIXENE4.46684Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64529CLONEDHUMAN3H-Estradiol2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol9Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65297GABAACLONEDHUMAN[3H] FlunitrazepamZG-2080.38Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65554GABAACLONEDHUMAN[3H] FlunitrazepamFG82052.08Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65810GABAACLONEDHUMAN[3H] FlunitrazepamXLI-2TC44.08Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66066Alpha1DCLONEDHUMAN3H-PRAZOSINMellpaladine B2697Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 28, 2025
66322H1CLONEDHUMAN3H-PYRILAMINEFinazine40Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66578NETCLONEDHUMAN3H-Nisoxetine3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride138Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
66834D1CLONEDHUMAN3H-SCH233930N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67090Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
673465-HT6CLONEDHUMAN3H-LSD1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
678585-HT6CLONEDHUMAN3H-LSD(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline1263Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68626UTCLONEDHUMANI125-urotensin IIH-Asp-C[Cys-Phe-DTrp-Lys-Tyr-Cys]Val-OH1.25893Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68882SST5CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Ala-Thr-Phe-Thr-Ser-Cys}-NH2100Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69138H3CLONEDHUMAN3H-HistamineImetit1.58489Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
38585-HT6CLONEDRAT3H-LSDCLOZAPINE7.1KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
4114KORCLONEDHUMAN3H-U69,593NALORPHINE - HCI0.8TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69650Beta1CLONEDHUMAN125I-iodo-pindolol2-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43705-HT6CLONEDHUMAN3H-LSDTIOSPERONE950KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69906D3CLONEDHUMAN3H-N-Methylspiperone4-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4626SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDING HIGHWIN 35,42810PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48825-HT2BCLONEDHUMAN3H-RAUWOLSCINEMETHYSERGIDE0.64WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704185-HT2BCLONEDHUMAN3H-LSDMRP50286.6Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51385-HT2BCLONEDHUMAN3H-5HTD-367521NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70674MORCLONEDHUMAN3H-DiprenorphineOxymorphone11Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
53945-HT2CCLONEDHUMAN3H-MESULERGINEYOHIMBINE>10000BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
70930Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione3364Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
71186H1CLONEDHUMAN3H-PYRILAMINEHALOPERIDOL440Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5906Alpha2ACLONEDHUMAN3H-RAUWOLSCINEOXYMETAZOLINE3.3BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
71442NETCLONEDHUMAN3H-Nisoxetine4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
6162Alpha1CCLONEDBOVINE125I-HEATCORYNANTHINE142LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64185-HT5ACLONEDMOUSE125I-LSD5-Hydroxy Tryptamine251.18Matthes H, et.al., 1993Jan 15, 2025Jan 15, 2025
6674D2CLONEDHUMAN3H-NEMONAPRIDEHALOPERIDOL9.6SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
72210M3CLONEDHUMAN3H-QNB2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
6930GAL2CLONEDRAT125I-h GalaninGalanin (1-29), rat0.56WANG S, ET AL., 1997Jan 15, 2025Jan 15, 2025
7186NK3CLONEDHUMAN125I-[MePhe7]-NKBNKB0.81Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72722H1CLONEDHUMAN3H-PYRILAMINEnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7442BB2CLONEDMOUSE125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14)Bombesin1.76Katsuno T, et al., 1999Jan 15, 2025Jan 15, 2025
72978D2CLONEDHUMAN3H-N-Methylspiperonecatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7698GABAACLONEDHUMAN3H-MUSCIMOLSR 9553138.01Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7954GABAACLONEDHUMAN3H-RO-15-1788172535He X, et al., 1999Jan 15, 2025Jan 27, 2025
8210SST4CLONEDHUMAN125I-LTT-SST-28MK 6786.5Demchyshyn L, et al., 1993Jan 15, 2025Jan 15, 2025
8466SST5CLONEDHUMAN125I-Tyr3-octreotidecycloantagonist SA5.62Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8722SST2CLONEDHUMAN125I-LTT-SRIF28Somatostatin-140.1Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8978SST2CLONEDHUMAN125I-SRIF-28BIM 230140.5Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74514Beta 2CLONEDHUMAN3H-CGP-12177(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9234SST2CLONEDMOUSE125I-MK-678DC23-600.93Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74770M1CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9490MT2CLONEDHUMAN125I-IodomelatoninN-Acetyltryptamine,5-Methyl41Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
75026NOPCLONEDHUMAN3H-Nociceptin(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
752825-HT5ACLONEDHUMAN3H-LSDEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10002NETCLONEDRAT3H-NorepinephrineDOPAMINE392Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
75538Beta 2CLONEDHUMAN3H-CGP-12177propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10258CLONEDHUMAN125I-HEATUrapidil-5-methyl3.16Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75794DORCLONEDHUMAN3H-DADLE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76050Sigma 2CLONEDHUMAN3H-DTGEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10770CLONEDRAT3H-LSDCLOZAPINE3.98ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
763065-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76562Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76818D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77074D4CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77330H3CLONEDHUMAN3H-Alpha-methylhistamine(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77586M3CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77842SERTCLONEDHUMAN3H-CITALOPRAM(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78098KORCLONEDHUMAN3H-U69593(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide260Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
783545-HT1DCLONEDHUMAN3H-5-CT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
786105-HT3CLONEDHUMAN3H-GR-65630(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788665-HT1ACLONEDHUMAN3H-WAY100635(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
791225-HT6CLONEDHUMAN3H-LSD3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79378Alpha1BCLONEDHUMAN3H-PRAZOSIN5-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
140985-HT2ACLONEDRAT3H-KETANSERINFenfluramine5216Rothman RB, et al, 2000Jan 15, 2025Jan 15, 2025
79634CLONEDHUMAN3H-CLONIDINEN,N-Diisopropyltryptamine356Ray TS 2010 Jan 15, 2025Jan 15, 2025
79890M5CLONEDHUMAN3H-QNB4-Ethylthio-2,5-dimethoxyphenylbutylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
146105-HT2BCLONEDHUMAN3H-5HTSB-277011-A1288.24Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80146V2CLONEDHUMAN3H-VASOPRESSINN,N-Diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14866D2CLONEDRATUNDEFINEDRISPERIDONE0.44Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
804025-HT6CLONEDHUMAN3H-LSD(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806585-HT1DCLONEDHUMAN3H-5-CT(Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153785-HT1BCLONEDHUMAN3H-5HTmCPP363.07BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809145-HT1DCLONEDHUMAN3H-5CT3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine85.1138Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
156345-HT2BCLONEDMOUSE125I-DOI5-Hydroxy Tryptamine1258.92BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
811705-HT6CLONEDHUMAN3H-LSDN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158905-HT7CLONEDRATUNDEFINEDMIANSERIN67.6BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81426D2CLONEDHUMAN3H-N-Methylspiperone2-[(2R)-4-[(5-methyl-2-naphthalen-2-yl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]ethanamine1522Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16146D1CLONEDHUMAN3H-SCH23390CLOZAPINE141Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
816825-HT3CLONEDHUMAN3H-LY278584(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
81938NETCLONEDHUMAN3H-Nisoxetine(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol12Severance AJ et al 2007Jan 15, 2025Jan 15, 2025
16658M2CLONEDHUMAN3H-QNBSCOPOLAMINE0.44Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
821945-HT2CCLONEDHUMAN3H-MESULERGINE2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one543Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824505-HT1DCLONEDHUMAN3H-5-CT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine590Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82706D2CLONEDHUMAN3H-N-Methylspiperone(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
17682CLONEDHUMAN125I-VIPVIP [D-Ile26]38.2Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832185-HT1ACLONEDHUMAN3H-8-OH-DPATCyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide1.21Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83474M4CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+)97.7237Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83730MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide3552PDSP Certified DataJan 15, 2025Jan 28, 2025
83986KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
18706CGRP1CLONEDPIG125-h alpha-CGRP[Pro14]h alpha-CGRP5.5Rorabaugh BR et al., 2001Jan 15, 2025Jan 15, 2025
84242MORCLONEDHUMAN3H-DAMGO(±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide1370PDSP Certified DataJan 15, 2025Jan 28, 2025
18962H1CLONEDHUMAN3H-MEPYRAMINEcis-H2-PAT(-)8.91Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84498DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19218CLONEDRAT125I-VIPPACAP(4-38)800Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84754MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-methyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19474GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCH[Phe13,Tyr19]MCH0.8Sailer AW et al., 2001Jan 15, 2025Jan 15, 2025
85010MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19730D2CLONEDHUMANUNDEFINEDDROPERIDOL0.25Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
86034Alpha1DCLONEDHUMAN3H-PRAZOSIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86546A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione3230Koch P et al 2018Jan 15, 2025Jan 15, 2025
87570DORCLONEDHUMAN3H-DADLE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
878265-HT6CLONEDHUMAN3H-LSD3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline150Staron J et al 2016Jan 15, 2025Jan 15, 2025
225465-HT2ACLONEDHUMAN3H-MethylspiperoneSERTINDOLE0.6Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88082A1CLONEDHUMAN3H-CCPA9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22802H1CLONEDHUMAN3H-PYRILAMINED-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23058nAChRCLONEDHUMAN3H-EpibatidineL-methionine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
885945-HT2ACLONEDHUMAN3H-KETANSERINCLOZAPINE8.9Peprah K et al 2012Jan 15, 2025Jan 15, 2025
23570GPR10CLONEDHUMAN125I-PrRP20PrRP310.68Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
893625-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide6631Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240825-HT2ACLONEDHUMAN3H-KETANSERINMOLINDONE5200Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
24338SLC6A3CLONEDHUMAN3H-dopamineR-citalopram>10000Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89874nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine1820Yu LF et al 2012Jan 15, 2025Jan 29, 2025
90130D2CLONEDHUMAN3H-SPIPERONE2-(2,5- dimethoxy-4-nitro)ethanamine6100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24850D1CLONEDHUMAN3H-SCH23390CLOZAPINE189PDSP Certified DataJan 15, 2025Jan 15, 2025
90386A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25106M5CLONEDHUMAN3H-QNBQuetiapine1942Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90642A2BCLONEDHUMAN3H-PSB-6034-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25362H3CLONEDGUINEA PIG3H-Alpha-Me-histamineZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
25618KORCLONEDHUMAN3H-DiprenorphineCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91154A3CLONEDHUMAN125I-AB-MECAN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide9060Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91410CB1CLONEDHUMAN3H-SR144528O-621456Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26130CCR5CLONEDHUMAN3H-EpibatidinePseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91666A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide6.45Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26386GAL1CLONEDRAT125I-GALANINGalanin (1-16), porcine1.99526Smith KE, et. al., 1998Jan 15, 2025Jan 15, 2025
91922A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(4-methyl-phenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26642D5CLONEDHUMAN3H-SCH23390Miquelianin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921785-HT6CLONEDHUMAN3H-LSD5-Chloro-(R)-N-(1-{2-[(propan-2-yl)-phenyloxy]ethyl} pyrrolidin-3-yl)thiophene-2-sulfonamide200Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268985-HT6CLONEDHUMAN3H-LSDxanomeline1258.93Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
271545-HT2ACLONEDHUMAN125I-DOI1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride28May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92690H1CLONEDHUMAN3H-PYRILAMINE[(8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274105-HT1ACLONEDHUMAN3H-8-OH-DPATPiribedil446.684Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929465-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine17Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276665-HT1ACLONEDHUMAN3H-8-OH-DPATMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279225-HT2CCLONEDRAT3H-MESULERGINEMETHYSERGIDE1Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28178Beta2CLONEDHUMAN125I-PindololMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
93714A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester32.5Federico S et al 2018Jan 15, 2025Jan 15, 2025
28434mGluR5CLONEDHUMAN3H-Quisqualate1S, 3R-ACPD2100Mutel V, et.al., 2000Jan 15, 2025Jan 28, 2025
93970D2CLONEDHUMAN3H-SPIPERONE40 3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one24Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28690SLC6A4CLONEDHUMAN3H-CITALOPRAMARIPIPRAZOLE1080Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942265-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine1900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29202SST3CLONEDHUMANUNDEFINEDSomatostatin-140.3Patel YC, 1999Jan 15, 2025Jan 15, 2025
947385-HT2BCLONEDHUMAN3H-LSD4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94994D4CLONEDHUMAN3H-Methylspiperone4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29970H4CLONEDHUMAN3H-HistamineImpromidine12.3Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30226CLONEDRATUNDEFINEDVenlafaxine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 15, 2025
957625-HT6CLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96018SERTCLONEDHUMAN3H-CITALOPRAMTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96274Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30994CCK2CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
96530Sigma 1CLONEDHUMAN[3H]-Pentazocine6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31250D4CLONEDHUMAN3H-NMSPPPP, S(-)-3532.7PDSP Certified DataJan 15, 2025Jan 15, 2025
96786D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)1.6Mannel B et al 2017Jan 15, 2025Jan 28, 2025
315065-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)1584.89Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97042KORCLONEDHUMAN[3H]U69593Fluorolintane (2-F-DPPy)1278Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97298MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol15.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97554A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate92.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32786EAAT2CLONEDHUMAN3H-D-AspartateWAY-8652570.4Dunlop J, et al., 2003Jan 15, 2025Jan 15, 2025
98322D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985785-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride4440Ofon E et al 2016aJan 15, 2025Jan 15, 2025
33298D2CLONEDHUMAN3H-NMSPAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98834Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine241Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
99346D3CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine3.8Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34066P2X2, P2X3CLONEDHUMAN3H-A-317491ATP,2'-deoxy47.2Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99602A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-methoxy-4-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34322nAChRCLONEDRAT3H-NICOTINEA-853800.09Grinevich VP, et al., 2004Jan 15, 2025Jan 15, 2025
99858SERTCLONEDHUMAN[3H] Citalopram(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide280Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
100114Alpha2CCLONEDHUMAN3H-RAUWOLSCINEQuetiapine166PDSP Certified DataJan 15, 2025Jan 28, 2025
34834CB1CLONEDHUMAN3H-CP-55940PhAR2200Jan 15, 2025Jan 15, 2025
100370D2CLONEDHUMAN3H-N-MethylspiperoneILOPERIDONE369PDSP Certified DataJan 15, 2025Jan 28, 2025
35602D2CLONEDHUMAN3H-SPIPERONE10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin82Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35858Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole5.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013945-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione494Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101650H2CLONEDHUMAN[3H]TiotidinePerospirone244PDSP Certified DataMar 21, 2025Jul 28, 2026
101906Alpha1BCLONEDHUMAN[3H]prazosinZiprasidone37PDSP Certified DataMar 24, 2025Jul 28, 2026
366265-HT2ACLONEDHUMAN125I-R091150OLANZAPINE2.3Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102162Beta1CLONEDHUMAN[125I]-PindololNEMONAPRIDE1882PDSP Certified DataMar 25, 2025Jul 28, 2026
37906CDK1CLONEDHUMANFunctional4-[[5-Amino-1-(2-thienylcarbonyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide4.5Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38162CLONEDRAT3H-dexamethasoneC54H80NO8150von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
38418D3CLONEDHUMAN3H-NEMONAPRIDEMCL-203>10000Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
39442SLC6A4CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396985-HT2CCLONEDHUMAN3H-5HT5-Hydroxy Tryptamine5.7544Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40466mGluR2CLONEDRATFunctional(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40722mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one2160Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41234CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42002M1CLONEDHUMAN3H-QNBSERTRALINE1300Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42258CLONEDHUMANFunctional1-(3’,5’-Difluorobenzyl)-1H-benzotriazole-5-carboxylic acid>10000Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42514CLONEDHUMAN35S-GTPGammaSMotilin1.28825Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43026HCKCLONEDHUMAN3H-StaurosporineStaurosporine12Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43282CLK3CLONEDHUMAN3H-StaurosporineFlavopiridol1000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43538MAP3K5CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43794AURKCCLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44050MAPK14CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44306DAPK2CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44562LCKCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44818CaMKCLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
45074STK38LCLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45330CLONEDRATFunctionalPP21290Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45586SLC6A4CLONEDHUMAN3H-IMIPRAMINEFLUOXETINE0.81Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458425-HT2BCLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46098Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46866M5CLONEDHUMAN3H-QNB(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47378Grik5CLONEDHUMAN3H-Kainic acidLY 525327>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47890SST5CLONEDHUMAN3H-thymidineBIM-237451000Zatelli MC, et.al., 2002Jan 15, 2025Jan 15, 2025
48146Y4CLONEDHUMAN3H-Propionyl-NPYNPY D-Trp32, human, rat1000Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48658CLONEDHUMANFunctionalN-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride0.13Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
48914Y1CLONEDChicken[125I] - Peptide YYPP, chicken>10000Holmberg, SK et al., 2002Jan 15, 2025Jan 15, 2025
49170CCK2CLONEDHUMAN125I-CCK-8TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-1-Adoc560Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49682Y2CLONEDChicken[125I] - Peptide YYBIBP32261000Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49938CLONEDRATFunctionalAMAA>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 15, 2025
50194SLC6A3CLONEDRAT3H-dopamineNal2-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly>10000Ding, J., et, al., 2006Jan 15, 2025Jan 15, 2025
50450NETCLONEDHUMAN3H-NisoxetineN,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine500Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581305-HT2ACLONEDHUMAN3H-KETANSERINN-(3-Methylthiobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate28.2Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58386H4CLONEDHUMAN3H-HistamineMRS5698>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58642H1CLONEDHUMAN3H-PYRILAMINECloperatine4Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58898CCR5CLONEDHUMAN3H-EpibatidineKodiak extract2.9Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
59154D1CLONEDHUMAN3H-SCH23390SR 48692>10000Petrie K, et al., 2005Jan 15, 2025Jan 15, 2025
59410Alpha1ACLONEDHUMAN3H-PRAZOSINN-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(3-thienyl)benzamide170Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59922D3CLONEDHUMAN3H-NMSPN-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-4-[4-(trifluoromethyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60178A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((3-methoxyphenyl)ethynyl)- 6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1- carboxamide0.91Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60434GABAACLONEDHUMANFNZWY-TSC-41.63Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60690GABAACLONEDHUMANFNZJYI-1934Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60946GABAACLONEDHUMANFNZZG69A9.2Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61202GABAACLONEDHUMANFNZJYI-0616.5Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61458GABAACLONEDHUMANFNZRY-05886Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617145-HT2BCLONEDHUMAN3H-LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine4.6Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62226DORCLONEDHUMAN3H-DADLETianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
62482SLC6A3CLONEDHUMANWIN354284-methoxy-diphenidine157Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63250A1CLONEDHUMAN[3 H]N6 -Rphenylisopropyladenosine(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-methoxy-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane1-carboxamide796Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
63506D3CLONEDHUMAN3H-N-MethylspiperoneCariprazine0.085citrome, Leslie et. al, 2013Jan 15, 2025Jan 15, 2025
63762CXCR3CLONEDHUMAN125I-CXCL11CXCL110.03Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64018D3CLONEDMOUSE3H-SPIPERONEHALOPERIDOL4.3Fishburn CS, et al., 1993Jan 15, 2025Jan 15, 2025
642745-HT2CCLONEDRAT3H-MESULERGINECLOZAPINE20.4174Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64530CLONEDHUMAN3H-Estradiol1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol4Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65298GABAACLONEDHUMAN[3H] FlunitrazepamZG-2084.6Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65555GABAACLONEDHUMAN[3H] FlunitrazepamFG82051.16Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65811GABAACLONEDHUMAN[3H] FlunitrazepamXLI-2TC1.21Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66067Alpha2BCLONEDHUMAN3H-RAUWOLSCINEDopargimine5855Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 28, 2025
66323H3CLONEDHUMAN3H-Alpha-methylhistamineFinazine704Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66579DATCLONEDHUMAN3H-WIN354283-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride568Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
66835D2CLONEDHUMAN3H-N-MethylspiperoneN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67091Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
673475-HT7CLONEDHUMAN3H-LSD1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride82Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
678595-HT7CLONEDHUMAN3H-5-CT(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline52Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68627UTCLONEDHUMANI125-urotensin IIH-Asp-C[Pen-Phe-Trp-Orn-Tyr-Cys]Val-OH15.8489Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
33475-HT1ACLONEDHUMAN3H-8-OH-DPATDOPAMINE8248TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68883SST1CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Ala-Phe-Thr-Ser-Cys}-NH26.30957Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69139H3CLONEDHUMAN3H-HistamineVUF83283.16228Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
38595-HT6CLONEDRAT3H-LSDOLANZAPINE27.5KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
4115KORCLONEDHUMAN3H-U69,593NOR-BNI (HCI)20.2TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69651Beta1CLONEDHUMAN125I-iodo-pindolol3-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43715-HT6CLONEDHUMAN3H-LSDAMPEROZIDE1600KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69907D4CLONEDHUMAN3H-N-Methylspiperone4-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4627SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDINGGBR-129093.8PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48835-HT2BCLONEDHUMAN3H-RAUWOLSCINEMIANSERIN5.44WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704195-HT7CLONEDHUMAN3H-LSDMRP50286Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51395-HT2BCLONEDHUMAN3H-5HTQDOB>10000NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70675MORCLONEDHUMAN3H-DiprenorphineTapentadol2100Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
53955-HT2CCLONEDHUMAN3H-MESULERGINESPIPERONE1000BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
70931D4CLONEDHUMAN3H-Methylspiperone4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione1283Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
71187H1CLONEDHUMAN3H-PYRILAMINECLOZAPINE10.8Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5907Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPHENTOLAMINE4.1BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
71443D1CLONEDHUMAN3H-SCH233904-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
6163Alpha1CCLONEDBOVINE125I-HEATWB 41010.68LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64195-HT5ACLONEDMOUSE125I-LSD5-CT15.84Matthes H, et.al., 1993Jan 15, 2025Jan 15, 2025
6675D2CLONEDHUMAN3H-NEMONAPRIDEHALOPERIDOL0.89SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
72211M4CLONEDHUMAN3H-QNB2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
6931GAL2CLONEDRAT125I-h GalaninGalanin (1-13)-SP-(5-11)1.17WANG S, ET AL., 1997Jan 15, 2025Jan 15, 2025
7187NK3CLONEDHUMAN125I-[MePhe7]-NKBNKA539Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
727235-HT1DCLONEDHUMAN125I-aminopotentidinenaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7443BB2CLONEDMOUSE125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14)GRP1.74Katsuno T, et al., 1999Jan 15, 2025Jan 15, 2025
72979D3CLONEDHUMAN3H-N-Methylspiperonecatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7699GABAACLONEDHUMAN3H-MUSCIMOLBicuculline4570.88Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7955GABAACLONEDHUMAN3H-RO-15-1788182167He X, et al., 1999Jan 15, 2025Jan 27, 2025
8211SST3CLONEDHUMAN125I-LTT-SST-28SRIF-D-Trp80.56Corness J, et al., 1993Jan 15, 2025Jan 15, 2025
8467SST3CLONEDHUMAN125I-LTT-SRIF28Somatostatin-140.28Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8723SST2CLONEDHUMAN125I-LTT-SRIF28somatostatin-280.12Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8979SST2CLONEDHUMAN125I-SRIF-28MK 6780.07Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
9235SST2CLONEDMOUSE125I-MK-678BIM 230141.6Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74771M2CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9491MT2CLONEDHUMAN125I-IodomelatoninN-Acetyltryptamine,5-Benzyloxy6.6Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
752835-HT6CLONEDHUMAN3H-LSDEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10003NETCLONEDRAT3H-NorepinephrineMPP+778Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
10259CLONEDHUMAN125I-HEATNiguldipine(+)7.94Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75795KORCLONEDHUMAN3H-U695931S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76051SERTCLONEDHUMAN3H-CITALOPRAMEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10771CLONEDRAT3H-LSDRILAPINE0.63ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
763075-HT3CLONEDHUMAN3H-GR65630(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76563Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76819D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77075DATCLONEDHUMAN3H-WIN 35,428(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77331H4CLONEDHUMAN3H-Histamine(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77587M4CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77843Sigma 1CLONEDHUMAN3H-Pentazocine(+)(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78099MORCLONEDHUMAN3H-DAMGO(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
783555-HT1ECLONEDHUMAN3H-5-HT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
786115-HT5ACLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788675-HT1ACLONEDHUMAN3H-WAY1006353,4,5-Trimethoxyphenethylamine1841Ray TS 2010 Jan 15, 2025Jan 15, 2025
791235-HT6CLONEDHUMAN3H-LSD4-Bromo-2,5-dimethoxyphenethylamine319.9Ray TS 2010 Jan 15, 2025Jan 15, 2025
79379Alpha1BCLONEDHUMAN3H-PRAZOSINN,N-Dipropyltryptamine443.4Ray TS 2010 Jan 15, 2025Jan 28, 2025
140995-HT2ACLONEDRAT3H-KETANSERINFenfluramine (+)>10000Rothman RB, et al, 2000Jan 15, 2025Jan 15, 2025
79635CLONEDHUMAN3H-CLONIDINE5-Methoxy-N,N-diisopropyltryptamine759.5Ray TS 2010 Jan 15, 2025Jan 15, 2025
79891M5CLONEDHUMAN3H-QNB6-Fluoro-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
146115-HT2CCLONEDHUMAN3H-MESULERGINESB-277011-A>10000Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80147V2CLONEDHUMAN3H-VASOPRESSIN5-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14867D2CLONEDRATUNDEFINEDQuetiapine69Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
804035-HT7CLONEDHUMAN3H-LSD(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806595-HT1ECLONEDHUMAN3H-5-HT(Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153795-HT1BCLONEDHUMAN3H-5HT8-OH-DPAT257.03BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809155-HT1DCLONEDHUMAN3H-5CT3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine28.8403Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
156355-HT2BCLONEDMOUSE125I-DOITRYPTAMINE199.52BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
811715-HT7CLONEDHUMAN3H-LSDN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158915-HT7CLONEDRATUNDEFINEDCHLORPROMAZINE70.79BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
814275-HT2ACLONEDHUMAN3H-KETANSERIN2-[(2R)-4-[(5-methyl-2-naphthalen-2-yl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]ethanamine934Weiss DR et al 2018Jan 15, 2025Jan 15, 2025
16147D1CLONEDHUMAN3H-SCH23390THIORIDAZINE100Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
816835-HT5ACLONEDHUMAN3H-LSD(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
16659M2CLONEDHUMAN3H-QNBTrihexyphenidyl7Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
821955-HT3CLONEDHUMAN3H-GR-656302-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one1794Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824515-HT1ECLONEDHUMAN3H-5-HT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82707D3CLONEDHUMAN3H-N-Methylspiperone(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
17683CLONEDHUMAN125I-VIPVIP [D-Ser25]0.65Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832195-HT2ACLONEDHUMAN125I-DOICyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide331Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83475M3CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+)186.209Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83731KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one2950PDSP Certified DataJan 15, 2025Jan 28, 2025
83987KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide3234PDSP Certified DataJan 15, 2025Jan 28, 2025
18707CGRP1CLONEDPIG125-h alpha-CGRP[D-Pen2,7]h alpha-CGRP15.2Rorabaugh BR et al., 2001Jan 15, 2025Jan 15, 2025
842435-HT2BCLONEDHUMAN3H-LSD(±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide134PDSP Certified DataJan 15, 2025Jan 15, 2025
18963H1CLONEDHUMAN3H-MEPYRAMINEtrans-H2-PAT(+)42.4Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84499DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(2,4-dichlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19219CLONEDRAT125I-VIPPACAP(2-38)80Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84755DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-methyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19475GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHSalmon MCH0.2Sailer AW et al., 2001Jan 15, 2025Jan 15, 2025
85011DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19731D2CLONEDHUMANUNDEFINEDEPIDEPRIDE0.01Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
86035Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86547A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1260Koch P et al 2018Jan 15, 2025Jan 15, 2025
87827D2CLONEDHUMAN3H-RACLOPRIDE3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline675Staron J et al 2016Jan 15, 2025Jan 28, 2025
225475-HT2ACLONEDHUMAN3H-MethylspiperonePIMOZIDE77.7Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88083A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22803H1CLONEDHUMAN3H-PYRILAMINEL-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23059MORCLONEDHUMAN3H-DiprenorphineDL-homocysteine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
885955-HT2CCLONEDHUMAN3H-MESULERGINECLOZAPINE17Peprah K et al 2012Jan 15, 2025Jan 15, 2025
23571GPR10CLONEDHUMAN125I-PrRP20NPFF>10000Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
893635-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide108Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240835-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE3.4Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
896195-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1.25893Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
24339SLC6A3CLONEDHUMAN3H-dopamineCITALOPRAM>10000Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89875nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
90131D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-propylphenyl)ethanamine2300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
248515-HT7CLONEDHUMAN3H-LSDCLOZAPINE18PDSP Certified DataJan 15, 2025Jan 15, 2025
90387A2BCLONEDHUMAN3H-PSB-603N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90643A2BCLONEDHUMAN3H-PSB-603(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide119 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25619D2CLONEDHUMAN3H-NMSPCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91155A2ACLONEDHUMAN3H-CGS-21680N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25875Beta1CLONEDHUMAN125I-PindololPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91411CB1CLONEDHUMAN3H-CP55940O-621488Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
261315-HT2CCLONEDRAT3H-MESULERGINEPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91667A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide48.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26387GAL1CLONEDRAT125I-GALANINGalanin (3-29), porcine1000Smith KE, et. al., 1998Jan 15, 2025Jan 15, 2025
91923A1CLONEDHUMAN3H-DPCPX(2-Amino-5-(3,5-dimethylisoxazol-4-yl)-4-(2,2- dimethylpropyl)thiophen-3-yl)(4-chlorophenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26643D5CLONEDHUMAN3H-SCH23390Hyperforin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921795-HT6CLONEDHUMAN3H-LSD5-Chloro-(R)-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3- yl}thiophene-2-sulfonamide202Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268995-HT7CLONEDHUMAN3H-5CTxanomeline125.893Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
271555-HT2ACLONEDHUMAN125I-DOI1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride3.6May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92691H1CLONEDHUMAN3H-PYRILAMINE15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274115-HT1ACLONEDHUMAN3H-8-OH-DPATPramipexole691.831Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929475-HT6CLONEDHUMAN3H-LSD4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine470Sudol S et al 2020Jan 15, 2025Jan 15, 2025
27667M4CLONEDHUMAN3H-QNBMDMA8245PDSP Certified DataJan 15, 2025Jan 15, 2025
279235-HT2CCLONEDRAT3H-5HTMETHYSERGIDE0.8Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28179M1CLONEDHUMAN3H-QNBMETHYSERGIDE5459PDSP Certified DataJan 15, 2025Jan 15, 2025
93715A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester130Federico S et al 2018Jan 15, 2025Jan 15, 2025
28435CLONEDHUMAN3H-Quisqualate3HPG>10000Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93971D2CLONEDHUMAN3H-SPIPERONEcompound 427Ortega R et al 2011Jan 15, 2025Jan 29, 2025
28691NETCLONEDHUMAN3H-NisoxetineARIPIPRAZOLE2090Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942275-HT2ACLONEDHUMAN3H-KETANSERIN4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine980Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29203SST3CLONEDHUMANUNDEFINEDsomatostatin-280.3Patel YC, 1999Jan 15, 2025Jan 15, 2025
947395-HT2BCLONEDHUMAN3H-LSD4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94995D4CLONEDHUMAN3H-Methylspiperone4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29971H3CLONEDHUMAN3H-HistamineImpromidine67Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30227CLONEDRATUNDEFINEDDuloxetine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 15, 2025
957635-HT7CLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30483CLONEDXenopusUNDEFINED(S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-dimethylbutyl)amino]benzenepropaneamide bis(trifluoroacetate)140Kromann H, et. al., 2002aJan 15, 2025Jan 15, 2025
96019SERTCLONEDHUMAN3H-CITALOPRAM6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96275Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30995BZPCLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
96531H1CLONEDHUMAN[3H]-Pyrilamine6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
31251D5CLONEDHUMAN3H-SCH23390PPP, S(-)-32406PDSP Certified DataJan 15, 2025Jan 15, 2025
96787D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)0.91Mannel B et al 2017Jan 15, 2025Jan 28, 2025
315075-HT2BCLONEDHUMAN3H-5HT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)3981.07Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97043M1CLONEDHUMAN[3H]QNBFluorolintane (2-F-DPPy)1597Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97299MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol4.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97555A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate340Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
325315-HT2ACLONEDHUMAN125I-DOI5-Hydroxy Tryptamine14Bentley JM, et al., 2004Jan 15, 2025Jan 15, 2025
32787EAAT2CLONEDHUMAN3H-D-AspartateWAY-879>10000Dunlop J, et al., 2003Jan 15, 2025Jan 15, 2025
98323D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride3578Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985795-HT2CCLONEDHUMAN[3H]-mesulergine2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
33299D3CLONEDRAT3H-NMSPAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98835Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine433Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33555H4CLONEDHUMAN3H-HistamineNaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99091D1CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99347D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2,3-dichlorophenyl)piperazine5.05Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34067P2X2, P2X3CLONEDHUMAN3H-A-317491ADP, Beta S53.8Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99603A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34323nAChRCLONEDRAT3H-NICOTINENicotine0.84Grinevich VP, et al., 2004Jan 15, 2025Jan 15, 2025
99859SERTCLONEDHUMAN[3H] Citalopram(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb5700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
100115D2CLONEDHUMAN3H-N-MethylspiperoneQuetiapine5037PDSP Certified DataJan 15, 2025Jan 28, 2025
34835CB1CLONEDHUMAN3H-CP-55940PhAR, ent2400Jan 15, 2025Jan 15, 2025
100371D3CLONEDHUMAN3H-N-MethylspiperoneILOPERIDONE84PDSP Certified DataJan 15, 2025Jan 28, 2025
35603D2CLONEDHUMAN3H-SPIPERONERISPERIDONE1.4Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35859SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole9.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013955-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione822Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101651H3CLONEDHUMAN[3H]-alpha-methylhistaminePerospirone>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
101907Alpha2ACLONEDHUMAN[3H]rauwolscineZiprasidone162PDSP Certified DataMar 24, 2025Jul 28, 2026
366275-HT2ACLONEDHUMAN125I-R091150RISPERIDONE0.81Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102163Beta2CLONEDHUMAN[3H]-CGP12177NEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
37907CDK1CLONEDHUMANFunctional4-[[5-Amino-1-[(3-methyl-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide4.8Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38163CLONEDRAT3H-dexamethasoneC55H77NO71000von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
38419D3CLONEDHUMAN3H-NEMONAPRIDEMCL-207177Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
39443CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396995-HT2CCLONEDHUMAN3H-5HT8-OH-DPAT2511.89Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
39955D4CLONEDHUMANUNDEFINEDBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
40467mGluR2CLONEDRATFunctional(3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40723mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-methylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one43Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41235CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4,4-diphenylbutyl)piperidin-4-ol 6500Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42003M1CLONEDHUMAN3H-QNBTRAZODONE>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42259CLONEDHUMAN125I-MotilinDelta 2-42.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42515CLONEDHUMAN35S-GTPGammaS[Nle13]-Motilin1.94984Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43027HCKCLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43283CLK4CLONEDHUMAN3H-StaurosporineEKB-5692900Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43539MAP4K5CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43795BMP2KCLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44051MAPK P38CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44307EPHA2CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44563LIMK1CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44819CaMKCLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
45075STK4CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45331CLONEDRATFunctionalPP39900Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45587NETCLONEDHUMAN3H-NisoxetineFLUOXETINE240Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458435-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46099Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46867M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47379CLONEDHUMAN3H-Kainic acidLY 4661958900Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47891P2X1CLONEDXenopusFunctionalNF27919Rettinger J, et.al., 2000Jan 15, 2025Jan 15, 2025
48147Y5CLONEDHUMAN3H-Propionyl-NPYNPY D-Trp32, human, rat35Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48659CLONEDHUMANFunctionalN-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride12.6Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
48915Y1CLONEDChicken[125I] - Peptide YYBIBP322615.8489Holmberg, SK et al., 2002Jan 15, 2025Jan 15, 2025
49171CCK2CLONEDHUMAN125I-CCK-8TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-2-Adoc930Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49683Y2CLONEDChicken[125I] - Peptide YYSR 120819A1000Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49939mGluR2CLONEDRATFunctionalAMAA>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 28, 2025
50195SLC6A3CLONEDRAT3H-dopamineBpa-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly>10000Ding, J., et, al., 2006Jan 15, 2025Jan 15, 2025
50451NETCLONEDHUMAN3H-NisoxetineN,N-Dimethyl-5-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine632Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581315-HT2ACLONEDHUMAN3H-KETANSERINN-(3-Trifluoromethylbenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate8.91Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58387D1CLONEDHUMAN3H-SCH23390MRS5698>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58643H3CLONEDHUMAN3H-Alpha-Me-histamineCloperatine2148Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58899CCR5CLONEDHUMAN3H-EpibatidineCamel Snus extract2.9Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
59155D2CLONEDHUMAN3H-N-MethylspiporoneSR 48692>10000Petrie K, et al., 2005Jan 15, 2025Jan 15, 2025
59411D4CLONEDHUMAN3H-N-MethylspiporoneN-[(3S)-1-Benzyl-3-pyrrolidinyl]-4-(3-thienyl)benzamide2Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59923D4CLONEDHUMAN3H-NMSPN-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-4-[4-(trifluoromethyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60179A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((4-methoxyphenyl)ethynyl)- 6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1- carboxamide0.63Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60435GABAACLONEDHUMANFNZWY-TSC-451.04Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60691GABAACLONEDHUMANFNZJYI-1912.7Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60947GABAACLONEDHUMANFNZZG69A16.3Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61203GABAACLONEDHUMANFNZCM-A50 (S)17Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61459GABAACLONEDHUMANFNZRY-06683Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617155-HT2BCLONEDHUMAN3H-LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2-methoxyphenyl)propan-1-amine5.8Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
622275-HT1ACLONEDHUMAN3H-WAY100635Tianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
62483SLC6A3CLONEDHUMANWIN354282-Cl-diphenidine357Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63251KORCLONEDHUMAN[3H]U69593XLi0932024Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
63507D2CLONEDHUMAN3H-N-MethylspiperoneCariprazine0.49citrome, Leslie et. al, 2013Jan 15, 2025Jan 27, 2025
63763CXCR3CLONEDHUMAN125I-CXCL11NBI-743303.2Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64019D3CLONEDMOUSE3H-SPIPERONEDOMPERIDONE14.1Fishburn CS, et al., 1993Jan 15, 2025Jan 15, 2025
642755-HT2CCLONEDRAT3H-MESULERGINEFLUPHENAZINE977.237Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64531CLONEDHUMAN3H-Estradiol1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol10Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65299GABAACLONEDHUMAN[3H] FlunitrazepamYCT-52.2Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65556GABAACLONEDHUMAN[3H] FlunitrazepamFG82051.54Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65812GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-137.3Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66068Alpha2CCLONEDHUMAN3H-RAUWOLSCINEMellpaladine A3895Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 28, 2025
66324H4CLONEDHUMAN3H-HistamineFinazine>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66580H1CLONEDHUMAN3H-PYRILAMINE3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride312Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66836D3CLONEDHUMAN3H-N-MethylspiperoneN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide1854Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67092Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67348Alpha1ACLONEDHUMAN3H-PRAZOSIN1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride336Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67860D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline22Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
68628UTCLONEDHUMANI125-urotensin IIH-Asp-C[Cys-Phe-Trp-Orn-Tyr-Cys]Val-OH10Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
33485-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT6.9TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68884SST2CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Ala-Phe-Thr-Ser-Cys}-NH21Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69140H3CLONEDHUMAN3H-HistamineClobenpropit2.51189Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
38605-HT6CLONEDRAT3H-LSDQuetiapine1297KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
4116KORCLONEDHUMAN3H-U69,593DYNORPHIN(1-8)-OH0.2TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69652Beta1CLONEDHUMAN125I-iodo-pindolol4-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43725-HT6CLONEDHUMAN3H-LSDRISPERIDONE2400KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69908D4CLONEDHUMAN3H-N-Methylspiperone4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4628SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDINGMETHYLPHENIDATE21PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48845-HT2BCLONEDHUMAN3H-RAUWOLSCINE5-HT,N-ACETYL4170WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70420Sigma 1CLONEDHUMAN3H-Pentazocine(+)MRP50287.9Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51405-HT2CCLONEDHUMAN125I-DOIDMA104NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70676MORCLONEDHUMAN3H-DiprenorphineNALOXONE14Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
53965-HT2CCLONEDHUMAN3H-MESULERGINEKETANSERIN199.52BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
70932D4CLONEDHUMAN3H-Methylspiperone(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
71188H1CLONEDHUMAN3H-PYRILAMINESYA013189Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5908Alpha2ACLONEDHUMAN3H-RAUWOLSCINESPIROXATRINE5.5BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
71444D2CLONEDHUMAN3H-N-Methylspiperone4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
72212M5CLONEDHUMAN3H-QNB2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
6932GAL2CLONEDRAT125I-h GalaninGalanin (2-29), rat3.5WANG S, ET AL., 1997Jan 15, 2025Jan 15, 2025
7188NK3CLONEDHUMAN125I-[MePhe7]-NKBSubstance P1292Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72724H3CLONEDHUMAN3H-Alpha-methylhistaminenaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7444BB2CLONEDMOUSE125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14)NMB134Katsuno T, et al., 1999Jan 15, 2025Jan 15, 2025
72980D4CLONEDHUMAN3H-N-Methylspiperonecatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7700GABAACLONEDHUMAN3H-MUSCIMOLThio-4-PIOL1698.24Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7956GABAACLONEDHUMAN3H-RO-15-17881984He X, et al., 1999Jan 15, 2025Jan 27, 2025
8212SST3CLONEDHUMAN125I-LTT-SST-28Somatostatin-142.09Corness J, et al., 1993Jan 15, 2025Jan 15, 2025
8468SST3CLONEDHUMAN125I-LTT-SRIF28somatostatin-280.22Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8724SST2CLONEDHUMAN125I-LTT-SRIF28seglitide0.1Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8980SST2CLONEDHUMAN125I-SRIF-28RC 1600.07Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74516D1CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9236SST2CLONEDMOUSE125I-MK-678SMS 201-9952.4Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74772M3CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
750285-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
752845-HT7CLONEDHUMAN3H-LSDEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10004NETCLONEDRAT3H-NorepinephrineEPINEPHRINE6500Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
75540D1CLONEDHUMAN3H-SCH23390propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10260CLONEDHUMAN125I-HEATPHENTOLAMINE19.95Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75796MORCLONEDHUMAN3H-DAMGO1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76052NETCLONEDHUMAN3H-NisoxetineEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10772CLONEDRAT3H-LSDFLUPERLAPINE6.3ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
763085-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76564Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76820D2CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77076H1CLONEDHUMAN3H-PYRILAMINE(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77332M1CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77588M5CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77844Sigma 2CLONEDHUMAN3H-DTG(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
781005-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
783565-HT2ACLONEDHUMAN3H-KETANSERIN(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
786125-HT6CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788685-HT1ACLONEDHUMAN3H-WAY1006354-Bromo-2,5-dimethoxyphenethylamine240.8Ray TS 2010 Jan 15, 2025Jan 15, 2025
791245-HT6CLONEDHUMAN3H-LSDDMT487.4Ray TS 2010 Jan 15, 2025Jan 15, 2025
79380Alpha1BCLONEDHUMAN3H-PRAZOSIN4-Ethylthio-2,5-dimethoxyphenylbutylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025