36716 5-HT2C CLONED HUMAN 3H-MESULERGINE (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-chloro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 2.4 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
58220 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(8-Chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-1-ethylpiperazine N-oxide 5100 Chen X, et al., 2015 Jan 15, 2025 Jan 15, 2025
62316 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
877 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ICYANOPINDOLOL >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
1133 5-HT2C CORTEX PIG 3H-MESULERGINE SUMATRIPTAN >10000 McCARTHY & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
13933 5-HT2C CLONED HUMAN 3H-MESULERGINE OLANZAPINE 7.8 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 27, 2025
36717 5-HT2C CLONED HUMAN 3H-MESULERGINE (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-bromo-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 17 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
58221 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(8-Chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-1-isopropylpiperazine N-oxide 6700 Chen X, et al., 2015 Jan 15, 2025 Jan 15, 2025
62317 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-Cl-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
878 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ICYANOPINDOLOL 9770 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
1134 5-HT2C Choroid Plexus RAT 3H-MESULERGINE SUMATRIPTAN >10000 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
70766 5-HT2C test test 3H-MESULERGINE D-lysergic acid diethylamide (LSD) 45.3 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
78190 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
13934 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 10 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 27, 2025
80494 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one 2354 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
25198 5-HT2C CLONED RAT 3H-MESULERGINE THIORIDAZINE 69 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
36718 5-HT2C CLONED HUMAN 3H-MESULERGINE (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-bromo-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 8.9 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
58222 5-HT2C CLONED HUMAN 3H-MESULERGINE 8-Chloro-11-[4-(1,1-dideutrioethyl)piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 280 Chen X, et al., 2015 Jan 15, 2025 Jan 15, 2025
58990 5-HT2C CLONED HUMAN 3H-MESULERGINE SERTRALINE 1000 Roth B. et al., 2006 Jan 15, 2025 Jan 15, 2025
879 5-HT2C CORTEX RAT 3H-MESULERGINE ICYANOPINDOLOL >10000 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
1135 5-HT2C Choroid Plexus PIG 3H-MESULERGINE SUMATRIPTAN >10000 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
1903 5-HT2A CORTEX RAT 3H-MESULERGINE DOMPERIDONE 278 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
76143 5-HT2C CLONED HUMAN 3H-MESULERGINE 2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
13935 5-HT2C CLONED HUMAN 3H-MESULERGINE RISPERIDONE 24 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 27, 2025
36719 5-HT2C CLONED HUMAN 3H-MESULERGINE (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 0.65 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
58223 5-HT2C CLONED HUMAN 3H-MESULERGINE 11-(Piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 170 Chen X, et al., 2015 Jan 15, 2025 Jan 15, 2025
880 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ICYANOPINDOLOL >10000 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
1136 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TFMPP 50.1 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
13936 5-HT2C CLONED HUMAN 3H-MESULERGINE FLUPERLAPINE 56 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 27, 2025
83568 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
33136 5-HT2C CLONED RAT 3H-MESULERGINE valeryl salicylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
59504 5-HT2C BRAIN RAT 3H-MESULERGINE 4-{[(4-Iodobenzyl)sulfanyl]methyl}-1H-imidazole >10000 Hough, L. et. al., 2007 Jan 15, 2025 Jan 15, 2025
59760 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)-1-butanone 872.1 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
881 5-HT2C Choroid Plexus PIG 3H-MESULERGINE INDORENATE 324 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
1137 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TFMPP 50.1 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
2929 5-HT2A CORTEX RAT 3H-MESULERGINE MEPYRAMINE 952 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
13937 5-HT2C CLONED HUMAN 3H-MESULERGINE TENILAPINE 151 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 27, 2025
48241 5-HT2C CLONED RAT 3H-MESULERGINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
58993 5-HT2C CLONED HUMAN 3H-MESULERGINE BUPROPION >10000 Roth B. et al., 2006 Jan 15, 2025 Jan 15, 2025
1138 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TFMPP 61.7 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
77938 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
13938 5-HT2C CLONED HUMAN 3H-MESULERGINE LOXAPINE 17 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
883 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHYSERGIDE 2.45 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
1139 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TFMPP 61.8 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
13939 5-HT2C CLONED HUMAN 3H-MESULERGINE CHLORPROMAZINE 6.1 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
82035 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(1,3-Benzodioxol-4-ylmethyl)-4-(2-methylphenyl)piperazine 868 DeRuiter J et al 2018 Jan 15, 2025 Jan 15, 2025
24691 5-HT2C CEREBRAL CORTEX RAT 3H-MESULERGINE 8-OH-DPAT >10000 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
25459 5-HT2C CLONED HUMAN 3H-MESULERGINE MDL 100907 136 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
58995 5-HT2C CLONED HUMAN 3H-MESULERGINE Nefazodone 72 Roth B. et al., 2006 Jan 15, 2025 Jan 15, 2025
884 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHYSERGIDE 2.5 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
1140 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TFMPP 63 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
13940 5-HT2C CLONED HUMAN 3H-MESULERGINE THIORIDAZINE 46 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
24948 5-HT2C CLONED RAT 3H-MESULERGINE HALOPERIDOL >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
1141 5-HT2C CORTEX PIG 3H-MESULERGINE TFMPP 120 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
74869 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
13941 5-HT2C CLONED HUMAN 3H-MESULERGINE PROCHLORPERAZINE 122 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
66166 5-HT2C CLONED HUMAN 3H-MESULERGINE Ziprasidone 0.72 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
886 5-HT2C Choroid Plexus HUMAN 3H-MESULERGINE METITEPIN 1.35 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
1142 5-HT2C CORTEX PIG 3H-MESULERGINE TMA,2,3,5- 5710 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
13942 5-HT2C CLONED HUMAN 3H-MESULERGINE PERPHENAZINE 132 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
80758 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 970 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
16502 5-HT2C CLONED RAT 3H-MESULERGINE Fluorocarazolol,(S) >10000 Roth BL, et al., 2001 Jan 15, 2025 Jan 15, 2025
82294 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
25462 5-HT2C CLONED HUMAN 3H-MESULERGINE SR 46349B 8.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
58998 5-HT2C CLONED HUMAN 3H-MESULERGINE Duloxetine 916 Roth B. et al., 2006 Jan 15, 2025 Jan 15, 2025
61814 5-HT2C CLONED HUMAN 3H-MESULERGINE FECIMBI-36 1.7 Prabhakaran, Jaya et. al. 2015 Jan 15, 2025 Jan 15, 2025
887 5-HT2C CORTEX RAT 3H-MESULERGINE METITEPIN 1.74 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
1143 5-HT2C CORTEX PIG 3H-MESULERGINE TMA,2,3,5- 2666 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
2935 5-HT2A CORTEX RAT 3H-MESULERGINE MESULERGINE 2.1 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
13943 5-HT2C CLONED HUMAN 3H-MESULERGINE MESORIDAZINE 157 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
25719 5-HT2C CLONED RAT 3H-MESULERGINE Ephedrine,(-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
1144 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TRYPTAMINE 46.8 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
68984 5-HT2C CLONED RAT 3H-MESULERGINE HALOPERIDOL 1000 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
4984 5-HT2C CLONED RAT 3H-MESULERGINE 5-Methoxytryptamine 63.09 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
73080 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 2623 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
13944 5-HT2C CLONED HUMAN 3H-MESULERGINE TRIFLUOPERAZINE 378 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
49784 5-HT2C CLONED RAT 3H-MESULERGINE PSILOCYBIN >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
58488 5-HT2C CLONED HUMAN 3H-MESULERGINE MRS5678 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
59512 5-HT2C CLONED HUMAN 3H-MESULERGINE Nantenin 1069 LeGendre, O. et. al., 2009 Jan 15, 2025 Jan 15, 2025
1145 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TRYPTAMINE 46.8 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4985 5-HT2C CLONED RAT 3H-MESULERGINE BUSPIRONE 6025.59 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
75897 5-HT2C CLONED HUMAN 3H-MESULERGINE Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
13945 5-HT2C CLONED HUMAN 3H-MESULERGINE FLUPHENAZINE 579 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
82041 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(1,3-Benzodioxol-4-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperazine 753 DeRuiter J et al 2018 Jan 15, 2025 Jan 15, 2025
88697 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
58489 5-HT2C CLONED HUMAN 3H-MESULERGINE MRS5697 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
59001 5-HT2C CLONED HUMAN 3H-MESULERGINE Venlafaxine >10000 Roth B. et al., 2006 Jan 15, 2025 Jan 15, 2025
1146 5-HT2C Choroid Plexus PIG 3H-MESULERGINE TRYPTAMINE 50.1 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
4986 5-HT2C CLONED RAT 3H-MESULERGINE CLOZAPINE 17.37 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
77434 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
13946 5-HT2C CLONED HUMAN 3H-MESULERGINE SPIPERONE 1108 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
82554 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-2-(2-((3-chlorophenoxy)methyl)morpholino)-1-(indolin-1-yl)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
86650 5-HT2C CLONED HUMAN 3H-MESULERGINE N-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide >10000 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
58490 5-HT2C CLONED HUMAN 3H-MESULERGINE MRS5676 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
1147 5-HT2C Choroid Plexus PIG 3H-MESULERGINE URAPIDIL >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
4987 5-HT2C CLONED RAT 3H-MESULERGINE CYPROHEPTADINE 6.3 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
13947 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL 5000 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
80507 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one 320 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
24699 5-HT2C CEREBRAL CORTEX RAT 3H-MESULERGINE BUSPIRONE 2089.3 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
31355 5-HT7 BRAIN RAT 3H-MESULERGINE 5-CT 0.00398107 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
39803 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Hydroxy Tryptamine 18.197 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
58491 5-HT2C CLONED HUMAN 3H-MESULERGINE MRS5755 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
892 5-HT2C Choroid Plexus PIG 3H-MESULERGINE BUSPIRONE 8320 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
1148 5-HT2C Choroid Plexus PIG 3H-MESULERGINE URAPIDIL >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4988 5-HT2C CLONED RAT 3H-MESULERGINE DP-5-CT >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
13948 5-HT2C CLONED HUMAN 3H-MESULERGINE PIMOZIDE 874 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
31356 5-HT7 BRAIN RAT 3H-MESULERGINE 5-Hydroxy Tryptamine 0.125893 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
39804 5-HT2C CLONED HUMAN 3H-MESULERGINE mCPP 85.1138 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
58492 5-HT2C CLONED HUMAN 3H-MESULERGINE MRS5923 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
893 5-HT2C Choroid Plexus PIG 3H-MESULERGINE BUTACLAMOL,(+) 160 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
66429 5-HT2C CLONED HUMAN 3H-MESULERGINE N-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
1149 5-HT2C Choroid Plexus PIG 3H-MESULERGINE URAPIDIL >10000 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
4989 5-HT2C CLONED RAT 3H-MESULERGINE ERGOTAMINE 2.45 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
13949 5-HT2C CLONED HUMAN 3H-MESULERGINE PENFLURIDOL 2079 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
83581 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
25981 5-HT2C CLONED RAT 3H-MESULERGINE Norephedrine, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
31357 5-HT7 BRAIN RAT 3H-MESULERGINE 5-Methoxytryptamine 0.630957 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
100989 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-fluorophenyl)-N-(3,4- dimethoxyphenethyl)propan-1-amine 126 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39293 5-HT2C CLONED RAT 3H-MESULERGINE 1-Methylpsilocin 48 Sard H, et al., 2005 Jan 15, 2025 Jan 15, 2025
39805 5-HT2C CLONED HUMAN 3H-MESULERGINE MK 212 891.251 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
48253 5-HT2C CLONED RAT 3H-MESULERGINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
1150 5-HT2C Choroid Plexus PIG 3H-MESULERGINE WB 4101 398 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
4990 5-HT2C CLONED RAT 3H-MESULERGINE FLUOXETINE 23.98 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
77182 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-N,2-dibutyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
13950 5-HT2C CLONED HUMAN 3H-MESULERGINE THIOTHIXENE 1311 Herrick-Davis K, et al., 2000 Jan 15, 2025 Jan 15, 2025
23422 5-HT2C BRAIN RAT 3H-MESULERGINE ABT-702 >10000 Jarvis MF, et. al., 2000 Jan 15, 2025 Jan 15, 2025
24446 5-HT2C CLONED HUMAN 3H-MESULERGINE Agomelatine 707.946 Millan MJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
31358 5-HT7 BRAIN RAT 3H-MESULERGINE SUMATRIPTAN 25.1189 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
33406 5-HT2C CLONED RAT 3H-MESULERGINE ibuprofen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
39806 5-HT2C CLONED HUMAN 3H-MESULERGINE Ro 600332 13.8038 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
58238 5-HT2C CLONED HUMAN 3H-MESULERGINE 8-Chloro-11-(4-ethylpiperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 24 Chen X, et al., 2015 Jan 15, 2025 Jan 15, 2025
895 5-HT2C CORTEX PIG 3H-MESULERGINE BUTACLAMOL,(+) 200 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
1151 5-HT2C Choroid Plexus PIG 3H-MESULERGINE WB 4101 437 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
68991 5-HT2C CLONED RAT 3H-MESULERGINE CLOZAPINE 11 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
4991 5-HT2C CLONED RAT 3H-MESULERGINE GR 113808 >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
82047 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(1,3-Benzodioxol-4-ylmethyl)-4-[4-(trifluoromethyl)phenyl]piperazine 1000 DeRuiter J et al 2018 Jan 15, 2025 Jan 15, 2025
82815 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
24447 5-HT2C CLONED HUMAN 3H-MESULERGINE MELATONIN >10000 Millan MJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
31359 5-HT7 BRAIN RAT 3H-MESULERGINE RISPERIDONE 5.01187 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
33663 5-HT2C CLONED RAT 3H-MESULERGINE PARECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
39807 5-HT2C CLONED HUMAN 3H-MESULERGINE DOI 18.6209 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
896 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CARAZOLOL 6310 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
1152 5-HT2C Choroid Plexus PIG 3H-MESULERGINE WY 26392 1000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
66688 5-HT2C CLONED HUMAN 3H-MESULERGINE ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4992 5-HT2C CLONED RAT 3H-MESULERGINE HALOPERIDOL >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72320 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-Aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 15, 2025
24448 5-HT2B CLONED HUMAN 3H-MESULERGINE Agomelatine 257.04 Millan MJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
31360 5-HT7 BRAIN RAT 3H-MESULERGINE LSD 7.94328 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
100992 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 235 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39808 5-HT2C CLONED HUMAN 3H-MESULERGINE BW-723C86 114.815 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
897 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CF 25-397 32.4 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
1153 5-HT2C Choroid Plexus PIG 3H-MESULERGINE WY 26392 1050 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4993 5-HT2C CLONED RAT 3H-MESULERGINE KETANSERIN 48.97 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72833 5-HT2C CLONED HUMAN 3H-MESULERGINE isoginkgetin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
73089 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride >10000 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
24449 5-HT2B CLONED HUMAN 3H-MESULERGINE MELATONIN 5754.4 Millan MJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
31361 5-HT7 BRAIN RAT 3H-MESULERGINE METERGOLINE 10 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
39809 5-HT2C CLONED HUMAN 3H-MESULERGINE Ro 60-0175 26.9153 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59009 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(2-(Benzo[d][1,3]dioxol-4-ylmethylamino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride 138.038 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
898 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CGS 12066B 1290 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
1154 5-HT2C Choroid Plexus PIG 3H-MESULERGINE YOHIMBINE >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
2946 5-HT2A CORTEX RAT 3H-MESULERGINE METERGOLINE 0.48 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
4994 5-HT2C CLONED RAT 3H-MESULERGINE LISURIDE 15.84 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
76930 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80770 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one 1870 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
31362 5-HT7 BRAIN RAT 3H-MESULERGINE MESULERGINE 10 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
37250 5-HT2C CLONED RAT 3H-MESULERGINE AMITRIPTYLINE 8 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39298 5-HT2C CLONED HUMAN 3H-MESULERGINE GR 127935 105 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
39810 5-HT2C CLONED HUMAN 3H-MESULERGINE LISURIDE 6.45654 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59010 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(2-(2-Hydroxybenzylamino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride 131.826 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
66179 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL 4700 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
899 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CGS 12066B >10000 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
1155 5-HT2C Choroid Plexus PIG 3H-MESULERGINE YOHIMBINE >10000 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
4995 5-HT2C CLONED RAT 3H-MESULERGINE mCPP 114.81 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72579 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,3-dihydroamentoflavone 1828 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
75651 5-HT2C CLONED HUMAN 3H-MESULERGINE benzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76675 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
17027 5-HT7 CLONED HUMAN 3H-MESULERGINE ILOPERIDONE 112 Kalkman HO, et al., 2001 Jan 15, 2025 Jan 15, 2025
31363 5-HT7 BRAIN RAT 3H-MESULERGINE RITANSERIN 25.1189 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
100995 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 219 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
37251 5-HT2C CLONED RAT 3H-MESULERGINE FLUOXETINE 160 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39811 5-HT2C CLONED HUMAN 3H-MESULERGINE Ro 600869 2.75423 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59011 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(2,5-dimethoxy-4-(trifluoromethyl)phenyl)- ethanamine hydrochloride 11.749 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
900 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CGS 12066B >10000 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
1156 5-HT2C Choroid Plexus PIG 3H-MESULERGINE YOHIMBINE >10000 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
4996 5-HT2C CLONED RAT 3H-MESULERGINE MESULERGINE 1.9 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
74628 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
87684 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
31364 5-HT7 BRAIN RAT 3H-MESULERGINE PINDOLOL,(+/-) >10000 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
37252 5-HT2C CLONED RAT 3H-MESULERGINE PAROXETINE >10000 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39812 5-HT2B CLONED HUMAN 3H-MESULERGINE 5-Hydroxy Tryptamine 2.81838 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59012 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-((2,5-Dimethoxy-4-(trifluoromethyl)phenethylamino)methyl)phenol hydrochloride 3.23594 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
1157 5-HT2C Choroid Plexus PIG 3H-MESULERGINE YOHIMBINE >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4997 5-HT2C CLONED RAT 3H-MESULERGINE METERGOLINE 1.99 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
82053 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(1,3-Benzodioxol-5-ylmethyl)-4-(2-methylphenyl)piperazine 924 DeRuiter J et al 2018 Jan 15, 2025 Jan 15, 2025
86149 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167) 4815 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
31365 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE 5-CT 0.000794328 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
37253 5-HT2C CLONED RAT 3H-MESULERGINE Fluvoxamine 6700 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39813 5-HT2B CLONED HUMAN 3H-MESULERGINE mCPP 12.0226 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59013 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-((2,5-Dimethoxy-4-(trifluoromethyl)phenethylamino)methyl)phenol hydrochloride 12.0226 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
1158 5-HT2C Choroid Plexus PIG 3H-MESULERGINE YOHIMBINE >10000 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68998 5-HT2C CLONED RAT 3H-MESULERGINE ISOCLOZAPINE 2.9 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
4998 5-HT2C CLONED RAT 3H-MESULERGINE METHIOTHEPIN 2.45 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
24454 5-HT2C Choroid Plexus PORCINE 3H-MESULERGINE Agomelatine 407.38 Millan MJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
91270 5-HT2C CLONED HUMAN 3H-MESULERGINE 17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan >10000 Zheng Y et al 2018 Jan 15, 2025 Jan 15, 2025
31366 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE 5-Hydroxy Tryptamine 0.1 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
98950 5-HT2C CLONED HUMAN 3H-MESULERGINE C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 15, 2025
100998 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 224 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
37254 5-HT2C CLONED RAT 3H-MESULERGINE CITALOPRAM 630 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39814 5-HT2B CLONED HUMAN 3H-MESULERGINE MK 212 151.356 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59014 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-((4-Ethyl-2,5-dimethoxyphenethylamino)methyl)phenol hydrochloride 3.38844 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
903 5-HT2C CORTEX PIG 3H-MESULERGINE CHLORPROMAZINE 30 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
4999 5-HT2C CLONED RAT 3H-MESULERGINE METHYSERGIDE 1.02 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
80519 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one 1078 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
24455 5-HT2C Choroid Plexus PORCINE 3H-MESULERGINE MELATONIN >10000 Millan MJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
31367 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE 5-Methoxytryptamine 0.251189 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
37255 5-HT2C CLONED RAT 3H-MESULERGINE BUPROPION >10000 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39815 5-HT2B CLONED HUMAN 3H-MESULERGINE Ro 600332 15.8489 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59015 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-((2,5-Dimethoxy-4-propylphenethylamino)methyl)phenol hydrochloride 3.0903 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
66952 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5000 5-HT2C CLONED RAT 3H-MESULERGINE MIANSERIN 2.13 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
73352 5-HT2C test test 3H-MESULERGINE N-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
86664 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide >10000 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
31368 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE SUMATRIPTAN 100 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
37256 5-HT2C CLONED RAT 3H-MESULERGINE Venlafaxine >10000 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39816 5-HT2B CLONED HUMAN 3H-MESULERGINE DOI 7.07946 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59016 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(2,5-dimethoxy-4-(methylthio)phenyl)ethanamine hydrochloride 27.5423 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
5001 5-HT2C CLONED RAT 3H-MESULERGINE NORFLUOXETINE 30.9 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
31369 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE RISPERIDONE 0.398107 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
101001 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 167 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
35977 5-HT2C BRAIN CORTEX GUINEA PIG 3H-MESULERGINE 8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 3.8 Campiani G, et al., 2005 Jan 15, 2025 Jan 15, 2025
37257 5-HT2C CLONED RAT 3H-MESULERGINE Nefazodone 72 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
39817 5-HT2B CLONED HUMAN 3H-MESULERGINE BW-723C86 3.16228 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59017 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(4-(ethylthio)-2,5-dimethoxyphenyl)-ethanamine hydrochloride 9.12011 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
906 5-HT2C CORTEX PIG 3H-MESULERGINE CINANSERIN 160 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
5002 5-HT2C CLONED RAT 3H-MESULERGINE OXYMETAZOLINE 645.65 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
73098 5-HT2C CLONED HUMAN 3H-MESULERGINE . 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl) butan-1-one >10000 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
73610 5-HT2C test test 3H-MESULERGINE ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74378 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11146 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RISPERIDONE 63 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
82314 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-(4-(Pyridin-2-yl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
88714 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1498 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
31370 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE METERGOLINE 1.58489 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
35978 5-HT2C BRAIN CORTEX GUINEA PIG 3H-MESULERGINE 3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 15 Campiani G, et al., 2005 Jan 15, 2025 Jan 15, 2025
39818 5-HT2B CLONED HUMAN 3H-MESULERGINE Ro 60-0175 0.549541 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
59018 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(2,5-dimethoxy-4-(propylthio)phenyl)-ethanamine hydrochloride 8.70964 Hansen M, et al., 2014 Jan 15, 2025 Jan 15, 2025
5003 5-HT2C CLONED RAT 3H-MESULERGINE PAROXETINE >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
6027 5-HT2C Choroid Plexus PIG 3H-MESULERGINE SDZ 205557 3981.07 BUCHHEIT KH, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
75403 5-HT2C CLONED HUMAN 3H-MESULERGINE Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,2-dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d]- [1,3]dioxole-3b(3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11147 5-HT2C Choroid Plexus PIG 3H-MESULERGINE 9-OH-risperidone 71 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
82059 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(1,3-Benzodioxol-5-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperazine 430 DeRuiter J et al 2018 Jan 15, 2025 Jan 15, 2025
83595 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
31371 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE LSD 0.398107 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
39819 5-HT2B CLONED HUMAN 3H-MESULERGINE LISURIDE 1.38038 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
908 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 200 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
67212 5-HT2C CLONED HUMAN 3H-MESULERGINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 916 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69004 5-HT2C CLONED RAT 3H-MESULERGINE 2-(Trifluoromethanesulfonyloxy)-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 620 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
5004 5-HT2C CLONED RAT 3H-MESULERGINE RITANSERIN 2.69 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
76428 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11148 5-HT2C Choroid Plexus PIG 3H-MESULERGINE HALOPERIDOL 5000 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
81292 5-HT2C test test 3H-MESULERGINE 6-[Me2]N-HEAT HCl 475 Petrie EC et al 2012 Jan 15, 2025 Jan 15, 2025
31372 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE MESULERGINE 12.5893 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
101004 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 206 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39820 5-HT2B CLONED HUMAN 3H-MESULERGINE Ro 600869 7.94328 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
50572 5-HT2C CLONED HUMAN 3H-MESULERGINE Prucalopride >10000 Briejer MR, et al., 2001 Jan 15, 2025 Jan 15, 2025
909 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 200 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
5005 5-HT2C CLONED RAT 3H-MESULERGINE ZACOPRIDE,S 3388.44 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
11149 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIPAMPERONE 120 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
89741 5-HT2C CLONED HUMAN 3H-MESULERGINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
31373 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE RITANSERIN 5.01187 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
39821 5-HT2C CLONED HUMAN 3H-MESULERGINE RS-102221 1.47911 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
910 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 200 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
5006 5-HT2C CLONED RAT 3H-MESULERGINE SER-084 54.95 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
11150 5-HT2C Choroid Plexus PIG 3H-MESULERGINE FLUSPIRILENE 1830 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
80782 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one 885 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82574 5-HT2C CLONED HUMAN 3H-MESULERGINE (S)-2-(2-((3-Chlorophenoxy)methyl)morpholino)-1-(indolin-1-yl)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
31374 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE PINDOLOL,(+/-) 501.187 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
39822 5-HT2C CLONED HUMAN 3H-MESULERGINE SB 242084 0.47863 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
911 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 204 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
1679 5-HT2A CORTEX RAT 3H-MESULERGINE APOMORPHINE 1670 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
5007 5-HT2C CLONED RAT 3H-MESULERGINE 5-Hydroxy Tryptamine 87.09 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
11151 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CLOZAPINE 13 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
78735 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
101007 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 143 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
36751 5-HT2C CLONED HUMAN 3H-MESULERGINE (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 0.42 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39823 5-HT2C CLONED HUMAN 3H-MESULERGINE KETANSERIN 16.9824 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
41615 5-HT2C CLONED RAT 3H-MESULERGINE N-DESMETHYLCLOZAPINE 11.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
912 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 204 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
5008 5-HT2C CLONED RAT 3H-MESULERGINE SPIPERONE 870.96 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
73872 5-HT2C test test 3H-MESULERGINE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 764 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
11152 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ZOTEPINE 2.9 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
36752 5-HT2C CLONED HUMAN 3H-MESULERGINE (-)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 0.21 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39824 5-HT2C CLONED HUMAN 3H-MESULERGINE MESULERGINE 1.12202 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
913 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 204 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
5009 5-HT2C CLONED RAT 3H-MESULERGINE SUMATRIPTAN >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
11153 5-HT2C Choroid Plexus PIG 3H-MESULERGINE OLANZAPINE 7.1 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
82065 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(1,3-Benzodioxol-5-ylmethyl)-4-[4-(trifluoromethyl)phenyl]piperazine 1000 DeRuiter J et al 2018 Jan 15, 2025 Jan 15, 2025
98193 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Desalkylquetiapine 107 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
36753 5-HT2C CLONED HUMAN 3H-MESULERGINE (+)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 1.5 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39825 5-HT2C CLONED HUMAN 3H-MESULERGINE METERGOLINE 0.467735 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
914 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 204 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
2962 5-HT2A CORTEX RAT 3H-MESULERGINE METHYSERGIDE 1.9 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
5010 5-HT2C CLONED RAT 3H-MESULERGINE TRYPTAMINE 56.23 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
11154 5-HT2C Choroid Plexus PIG 3H-MESULERGINE Quetiapine 3820 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
88466 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
28050 5-HT2C CLONED RAT 3H-MESULERGINE Fenfluramine (+) 6245 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98194 5-HT2C CLONED HUMAN 3H-MESULERGINE Quetiapine 2502 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
101010 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 154 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39826 5-HT2C CLONED HUMAN 3H-MESULERGINE SB 206553 3.16228 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
915 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CINANSERIN 204 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
69011 5-HT2C CLONED RAT 3H-MESULERGINE 2-(Trifluoromethanesulfonyloxy)-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 34 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
5011 5-HT2C CLONED RAT 3H-MESULERGINE YOHIMBINE >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
11155 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ORG-5222 0.17 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
78483 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-butyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80531 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one 2275 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
39827 5-HT2C CLONED HUMAN 3H-MESULERGINE MIANSERIN 1.51356 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
916 5-HT2C CORTEX RAT 3H-MESULERGINE CINANSERIN 363 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
70548 5-HT2C CLONED HUMAN 3H-MESULERGINE MRP3160 5.4 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
73108 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one 603 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
11156 5-HT2C Choroid Plexus PIG 3H-MESULERGINE SERTINDOLE 1.3 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
86676 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid >10000 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
99988 5-HT2C CLONED HUMAN 3H-MESULERGINE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
39828 5-HT2C CLONED HUMAN 3H-MESULERGINE RITANSERIN 1.62181 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
75157 5-HT2C CLONED HUMAN 3H-MESULERGINE methyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11157 5-HT2C Choroid Plexus PIG 3H-MESULERGINE Ziprasidone 13 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
99989 5-HT2C CLONED HUMAN 3H-MESULERGINE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
101013 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 79 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39829 5-HT2C CLONED HUMAN 3H-MESULERGINE SB-215505 11.2202 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
918 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CK 204-933 23.4 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
69526 5-HT2C CLONED HUMAN 3H-MESULERGINE Ephenidine >10000 Kang, H. et, al. 2017 Jan 15, 2025 Jan 15, 2025
39830 5-HT2C CLONED HUMAN 3H-MESULERGINE SB204741 2137.96 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
919 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CORYNANTHINE 2880 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4759 5-HT2C CLONED RAT 3H-MESULERGINE 5-Hydroxy Tryptamine 159 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
74135 5-HT2C test test 3H-MESULERGINE naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
39831 5-HT2C CLONED HUMAN 3H-MESULERGINE S33526 457.088 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
41367 5-HT2C CLONED RAT 3H-MESULERGINE 2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione 99.6 Kumar JS, et al., 2006 Jan 15, 2025 Jan 15, 2025
920 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CORYNANTHINE 3160 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
4760 5-HT2C CLONED RAT 3H-MESULERGINE 5-Methoxytryptamine 215 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
76184 5-HT2C CLONED HUMAN 3H-MESULERGINE (2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
78232 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
85400 5-HT2C test test 3H-MESULERGINE 2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole >10000 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
88472 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
101016 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 92 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39832 5-HT2C CLONED HUMAN 3H-MESULERGINE LY 266097 67.6083 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
921 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYANOPINDOLOL >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4761 5-HT2C CLONED RAT 3H-MESULERGINE mCPP 300 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
83609 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
39833 5-HT2B CLONED HUMAN 3H-MESULERGINE RS-102221 234.423 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
922 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYANOPINDOLOL >10000 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
69018 5-HT2C CLONED RAT 3H-MESULERGINE 2-Methoxy-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 21 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
4762 5-HT2C CLONED RAT 3H-MESULERGINE TFMPP 299 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
71834 5-HT2C CLONED HUMAN 3H-MESULERGINE SAS-0132 245 Yi B et al 2017 Jan 15, 2025 Jan 15, 2025
80794 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 80 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82074 5-HT2C CLONED HUMAN 3H-MESULERGINE Donepezil >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
30618 5-HT2C CLONED HUMAN 3H-MESULERGINE SB-269970 >10000 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
33178 5-HT2C CLONED RAT 3H-MESULERGINE Naproxen sodium,(-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
39834 5-HT2B CLONED HUMAN 3H-MESULERGINE SB 242084 45.7088 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
923 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYANOPINDOLOL >10000 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
4763 5-HT2C CLONED RAT 3H-MESULERGINE TRYPTAMINE 772 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
88731 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1861 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
24987 5-HT2C CLONED RAT 3H-MESULERGINE LOXAPINE 21 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
101019 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 124 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39835 5-HT2B CLONED HUMAN 3H-MESULERGINE KETANSERIN 234.423 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
924 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYANOPINDOLOL >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
4764 5-HT2C CLONED RAT 3H-MESULERGINE MK 212 2552 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
77980 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
26012 5-HT2C CLONED RAT 3H-MESULERGINE Cathinone, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
39836 5-HT2B CLONED HUMAN 3H-MESULERGINE MESULERGINE 1.94984 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
925 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYPROHEPTADINE 8.32 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
4765 5-HT2C CLONED RAT 3H-MESULERGINE QUIPAZINE 1344 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
72349 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 15, 2025
11933 5-HT2C CLONED HUMAN 3H-MESULERGINE GR 127935 100 Price GW, et al., 1997 Jan 15, 2025 Jan 15, 2025
39837 5-HT2B CLONED HUMAN 3H-MESULERGINE METERGOLINE 0.707946 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
926 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYPROHEPTADINE 8.32 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
4766 5-HT2C CLONED RAT 3H-MESULERGINE 5-CT 5810 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
73118 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile 443 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
74910 5-HT2C CLONED HUMAN 3H-MESULERGINE 1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11934 5-HT2C CLONED HUMAN 3H-MESULERGINE SB 216641 158.48 Price GW, et al., 1997 Jan 15, 2025 Jan 15, 2025
16542 5-HT2C CLONED RAT 3H-MESULERGINE Fluorocarazolol,(R) >10000 Roth BL, et al., 2001 Jan 15, 2025 Jan 15, 2025
82334 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-(4-(Pyridin-2-yl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85406 5-HT2C test test 3H-MESULERGINE 2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole 1420 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
88478 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
25758 5-HT2C CLONED RAT 3H-MESULERGINE Ephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34718 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[(5-phenyl-3-pyridyl)carbamoyl-6-triflouromethylindoline 5.01187 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
101022 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 68 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39838 5-HT2B CLONED HUMAN 3H-MESULERGINE SB 206553 5.49541 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
927 5-HT2C CORTEX PIG 3H-MESULERGINE METITEPIN 13 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
4767 5-HT2C CLONED RAT 3H-MESULERGINE METHYSERGIDE 1 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
11935 5-HT2C CLONED HUMAN 3H-MESULERGINE BRL 15572 630.95 Price GW, et al., 1997 Jan 15, 2025 Jan 15, 2025
80543 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one 2208 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
25247 5-HT2C CLONED RAT 3H-MESULERGINE THIOTHIXENE 1593 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34719 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[5-(4-fluorophenyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 6.30957 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
39839 5-HT2B CLONED HUMAN 3H-MESULERGINE MIANSERIN 5.49541 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
928 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METITEPIN 16 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
69024 5-HT2C CLONED RAT 3H-MESULERGINE 8-methoxy-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 86 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
4768 5-HT2C CLONED RAT 3H-MESULERGINE MESULERGINE 0.9 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
77728 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
23200 5-HT2C CLONED RAT 3H-MESULERGINE DL-homocysteine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
28320 5-HT2C CLONED RAT 3H-MESULERGINE Norfenfluramine (-) 814 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34720 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[5-(3,5-Difluorophenyl)-3-pyridyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 79.4328 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
39840 5-HT2B CLONED HUMAN 3H-MESULERGINE RITANSERIN 1.25893 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
929 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METITEPIN 18.6 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
4769 5-HT2C CLONED RAT 3H-MESULERGINE CYPROHEPTADINE 21 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70817 5-HT2C CLONED HUMAN 3H-MESULERGINE D-578 73 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
23201 5-HT2C CLONED RAT 3H-MESULERGINE L-cysteine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
34721 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[5-(2,6-Difluorophenyl)-3-pyridyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 25.1189 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
101025 5-HT2C CLONED HUMAN 3H-MESULERGINE RITANSERIN 1.8 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39841 5-HT2B CLONED HUMAN 3H-MESULERGINE SB-215505 1.47911 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
930 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METITEPIN 27.5 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
4770 5-HT2C CLONED RAT 3H-MESULERGINE CLOZAPINE 39 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
75938 5-HT2C CLONED HUMAN 3H-MESULERGINE Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
23202 5-HT2C CLONED RAT 3H-MESULERGINE D-homocysteine thiolactone >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
34722 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[5-(4-pyridyl)-3-pyridyl]carbamoyl-6-trifluoromethylindoline 0.630957 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
39842 5-HT2B CLONED HUMAN 3H-MESULERGINE SB204741 51.2861 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
931 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METITEPIN 27.5 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
82595 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-2-((3-Chlorophenoxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85667 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-phenylpiperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
23203 5-HT2C CLONED RAT 3H-MESULERGINE L-homocysteine thiolactone >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
34723 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[5-(3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 0.794328 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
36771 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CLOZAPINE 9.5 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
39843 5-HT2B CLONED HUMAN 3H-MESULERGINE S33526 4.0738 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
932 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METITEPIN 27.5 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
4772 5-HT2C CLONED RAT 3H-MESULERGINE KETANSERIN 94 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
77476 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
85668 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
86692 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid >10000 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
88484 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
23204 5-HT2C CLONED RAT 3H-MESULERGINE D-homocysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
92324 5-HT2C CLONED HUMAN 3H-MESULERGINE (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
33444 5-HT2C CLONED RAT 3H-MESULERGINE Ketorolac tris salt >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34724 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[5-(4-methyl-3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 0.398107 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
101028 5-HT2C CLONED HUMAN 3H-MESULERGINE 1,2-dimethoxy-4-propylbenzene; 2-(2H-1,3-benzodioxol-5-yl)ethan-1-amine; butylbenzene 399 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
39844 5-HT2B CLONED HUMAN 3H-MESULERGINE LY 266097 0.199526 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
933 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METOCLOPRAMIDE 3980 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
4773 5-HT2C CLONED RAT 3H-MESULERGINE DOB 152 HERRICK-DAVIS K, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
5285 5-HT2C CLONED HUMAN 3H-MESULERGINE SB 206553 12.02 Kennett GA, et al., 1996 Jan 15, 2025 Jan 15, 2025
23205 5-HT2C CLONED RAT 3H-MESULERGINE L-homocysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
92325 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13:15,16-diepoxylabdane-6β,15α-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
33701 5-HT2C CLONED RAT 3H-MESULERGINE ROFECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34725 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[6-(3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5.01187 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
69030 5-HT2C CLONED RAT 3H-MESULERGINE 2-Hydroxy-11-(4-methylpiperazine)-5H-dibenzo[b,e][1,4]diazepine 81 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
80806 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one 4348 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
85414 5-HT2C test test 3H-MESULERGINE 1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one >10000 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
85926 5-HT2C CLONED HUMAN 3H-MESULERGINE delta9 -tetrahydrocannabinol (THC) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
23206 5-HT2C CLONED RAT 3H-MESULERGINE L-cysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
92326 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13:15,16-diepoxylabdane-6β,16β-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
1703 5-HT2A CORTEX RAT 3H-MESULERGINE DMT,5-OH 230 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
69799 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
83623 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
87463 5-HT2C CLONED HUMAN 3H-MESULERGINE FK881 >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
23207 5-HT2C CLONED RAT 3H-MESULERGINE DL-homocysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
92327 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13:15,16-diepoxylabdane-6β,16α-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
66472 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69800 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
73128 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide 1892 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
77224 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
23208 5-HT2C CLONED RAT 3H-MESULERGINE D-homocysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
92328 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13-epoxylabd-5-en-7-on-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
63656 5-HT2C CLONED HUMAN 3H-MESULERGINE Ziprasidone 0.724436 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
69801 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[1-(4-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
85673 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
23209 5-HT2C CLONED RAT 3H-MESULERGINE L-homocysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
90025 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Bromo-2,5-dimethoxyphenethylamine 47 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
92329 5-HT2C CLONED HUMAN 3H-MESULERGINE 15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
62889 5-HT2C CLONED RAT 3H-MESULERGINE Ketamine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
938 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 6.3 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
69802 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
85674 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88490 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
23210 5-HT2C CLONED RAT 3H-MESULERGINE L-cysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
90026 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-chloro-2,5-dimethoxy)ethanamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
92330 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13-epoxy-15,16-dihydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
36778 5-HT2C Choroid Plexus PIG 3H-MESULERGINE HALOPERIDOL >10000 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
939 5-HT2C Choroid Plexus HUMAN 3H-MESULERGINE MIANSERIN 6.61 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
69803 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-[1-(3-methylphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
72619 5-HT2C CLONED HUMAN 3H-MESULERGINE tetrahydroamentoflavone 9890 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
80555 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
23211 5-HT2C CLONED RAT 3H-MESULERGINE D-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
90027 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-methyl) ethanamine 150 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
92331 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13-epoxylabd-5-ene-7 β,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
63147 5-HT2C CLONED RAT 3H-MESULERGINE Mitragynine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
940 5-HT2C CORTEX RAT 3H-MESULERGINE MIANSERIN 7.94 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
66732 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride 110 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69036 5-HT2C CLONED RAT 3H-MESULERGINE 8-hydroxy-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 440 Liao Y, et.al., 1997 Jan 15, 2025 Jan 15, 2025
69804 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(1-phenylcyclohexyl)morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
72876 5-HT2C CLONED HUMAN 3H-MESULERGINE 2″-glucosylvitexin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
75692 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76972 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-butyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
23212 5-HT2C CLONED RAT 3H-MESULERGINE L-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88748 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1122 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
90028 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
91308 5-HT2C CLONED HUMAN 3H-MESULERGINE 17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan >10000 Zheng Y et al 2018 Jan 15, 2025 Jan 15, 2025
92332 5-HT2C CLONED HUMAN 3H-MESULERGINE (8S,9R,10S)-15,16-epoxy-9α-hydroxylabda-5,13(16),14-trien-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
941 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 8.32 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
76717 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
85421 5-HT2C test test 3H-MESULERGINE 1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one 5920 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
86701 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-phenylpiperazin-1-yl)ethyl)isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
23213 5-HT2C CLONED RAT 3H-MESULERGINE D-methionine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
90029 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,5-dimethoxyphenethylamine 4100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
92333 5-HT2C CLONED HUMAN 3H-MESULERGINE 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
96173 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
74670 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
82094 5-HT2C CLONED HUMAN 3H-MESULERGINE 6-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
86702 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide 0.933 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
23214 5-HT2C CLONED RAT 3H-MESULERGINE L-methionine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
90030 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-iodo-2,5-dimethoxyphenethylamine 40 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
92334 5-HT2C CLONED HUMAN 3H-MESULERGINE 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
96174 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
63406 5-HT2C CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 15 Keck, Paul e. et. al, 2003 Jan 15, 2025 Jan 15, 2025
943 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
67503 5-HT2C CLONED RAT 3H-MESULERGINE YOHIMBINE 1000 Song, Gang et., al. 2017 Jan 15, 2025 Jan 15, 2025
85679 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
90031 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5- dimethoxy-4-nitro)ethanamine 370 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96175 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
944 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
67504 5-HT2C CLONED RAT 3H-MESULERGINE mirtazapine 24 Song, Gang et., al. 2017 Jan 15, 2025 Jan 15, 2025
2736 5-HT2A CORTEX RAT 3H-MESULERGINE QUIPAZINE 635 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
85680 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl) picolinamide 140 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88496 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
90032 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 40 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96176 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
98992 5-HT2C CLONED HUMAN 3H-MESULERGINE [[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 15, 2025
945 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
67505 5-HT2C CLONED RAT 3H-MESULERGINE PROPRANOLOL 574 Song, Gang et., al. 2017 Jan 15, 2025 Jan 15, 2025
90033 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 69 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96177 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
59569 5-HT2C CLONED HUMAN 3H-MESULERGINE 8-Fluoro-N-phenyl-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide 5171 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
946 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
73138 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl) butan-1-one hydrochloride 1404 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
73394 5-HT2C test test 3H-MESULERGINE N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
80818 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one 2094 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81330 5-HT2C test test 3H-MESULERGINE 6-Iodo-HEAT HCl >10000 Petrie EC et al 2012 Jan 15, 2025 Jan 15, 2025
16818 5-HT2C CLONED HUMAN 3H-MESULERGINE S33005 >10000 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
82354 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-1-(Indolin-1-yl)-2-(2-((pyridin-2-yloxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85426 5-HT2C test test 3H-MESULERGINE FLUOXETINE 72 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
86194 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
90034 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,5-dimethoxy-4-isopropylthiophenethylamine 130 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96178 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
947 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
66995 5-HT2C CLONED HUMAN 3H-MESULERGINE [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2995 5-HT2A CORTEX RAT 3H-MESULERGINE MIANSERIN 4.6 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
74419 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75443 5-HT2C CLONED HUMAN 3H-MESULERGINE Ethyl(1S,2R,3S,4R,5S)-4-(2-((5-bromothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
16819 5-HT2C CLONED HUMAN 3H-MESULERGINE Venlafaxine >10000 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
86707 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide 1330 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90035 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 39 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96179 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
948 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
16820 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOMIPRAMINE 64.6 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
86708 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide 5.1 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90036 5-HT2C CLONED HUMAN 3H-MESULERGINE MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96180 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
48564 5-HT2C CLONED RAT 3H-MESULERGINE mCPP 108 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
59572 5-HT2C CLONED HUMAN 3H-MESULERGINE 8-Fluoro-N-isopropyl-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
949 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
76469 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
16821 5-HT2C CLONED HUMAN 3H-MESULERGINE CITALOPRAM 617 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
83637 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
85685 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
90037 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96181 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
63669 5-HT2C CLONED HUMAN 3H-MESULERGINE RISPERIDONE 10.4713 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
950 5-HT2C CORTEX PIG 3H-MESULERGINE MIANSERIN 13 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
16822 5-HT2C CLONED HUMAN 3H-MESULERGINE Reboxetine 457 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
85686 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)picolinamide 268 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88502 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
90038 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 5.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
25782 5-HT2C CLONED RAT 3H-MESULERGINE Pseudoephedrine, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96182 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
36534 5-HT2C CLONED RAT 3H-MESULERGINE 9-OH-risperidone 100.315 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
49078 5-HT2C CLONED RAT 3H-MESULERGINE TRAZODONE 1999 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
695 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYPROHEPTADINE 12.6 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
80567 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((4-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one 2762 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82615 5-HT2C CLONED HUMAN 3H-MESULERGINE (S)-2-((3-chlorophenoxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine 3386 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
90039 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 13 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
96183 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 15, 2025
59575 5-HT2C CLONED HUMAN 3H-MESULERGINE 8-Fluoro-N-propyl-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
696 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYPROHEPTADINE 13.8 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
952 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MK 212 692 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
67256 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
85432 5-HT2C test test 3H-MESULERGINE 2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride 4647 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
90040 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
100280 5-HT2C CLONED HUMAN 3H-MESULERGINE Asenapine 0.24 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
697 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CYPROHEPTADINE 13.8 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
953 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MK 212 692 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
73657 5-HT2C test test 3H-MESULERGINE N-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride 110 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73913 5-HT2C test test 3H-MESULERGINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 916 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
78777 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
86713 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90041 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 130 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
100281 5-HT2C CLONED HUMAN 3H-MESULERGINE SERTINDOLE 1.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
59833 5-HT2C CLONED HUMAN 3H-MESULERGINE N-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-4-(2-methoxyphenyl)-1-piperazinecarboxamide 1937 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
698 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DIHYDROERGOCRYPTINE 100 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
954 5-HT2C Choroid Plexus PIG 3H-MESULERGINE OXPRENOLOL >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
72122 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 15, 2025
72378 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-methoxy-6-methyl-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 15, 2025
80314 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((1H-indol-3-yl)methylene)-2-amino-1H-imidazol-4(5H)-one 349 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
86714 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(o-tolyl)piperazin-1-yl)ethyl)isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90042 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
25274 5-HT2C CLONED RAT 3H-MESULERGINE Ziprasidone 68 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100282 5-HT2C CLONED HUMAN 3H-MESULERGINE ZOTEPINE 3.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
59578 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Cyclohexyl-8-fluoro-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
699 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DIHYDROERGOCRYPTINE 126 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
955 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PAPP 603 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
70843 5-HT2C test test 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)ethanamine 2.5 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
85691 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)picolinamide 90.9 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
90043 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 21 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27835 5-HT2B CLONED HUMAN 3H-MESULERGINE S33084 158.489 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100283 5-HT2C CLONED HUMAN 3H-MESULERGINE Ziprasidone 4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
700 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DHE 31.6 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
956 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PAPP 603 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
73148 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl) butan-1-one hydrochloride >10000 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
85692 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide 564 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
85948 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
88508 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
90044 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27836 5-HT2B CLONED HUMAN 3H-MESULERGINE GR218231 1000 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100284 5-HT2C CLONED HUMAN 3H-MESULERGINE Perospirone 5.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
58044 5-HT2C CLONED HUMAN 3H-MESULERGINE Memantine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
701 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DHE 33.1 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
70845 5-HT2C test test 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 39 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
78525 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
81085 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
90045 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27837 5-HT2B CLONED HUMAN 3H-MESULERGINE L741,626 630.957 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100285 5-HT2C CLONED HUMAN 3H-MESULERGINE OLANZAPINE 16 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
59581 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Butyl-8-fluoro-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
702 5-HT2C CORTEX PIG 3H-MESULERGINE DHE 39 McCARTHY & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
958 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PHENTOLAMINE 891 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
75198 5-HT2C CLONED HUMAN 3H-MESULERGINE ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
80830 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 426 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
90046 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 16 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27838 5-HT2C Choroid Plexus PIG 3H-MESULERGINE S33084 199.526 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100286 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 19 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
35774 5-HT2C CLONED HUMAN 3H-MESULERGINE A-80426 1000 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
703 5-HT2C CORTEX PIG 3H-MESULERGINE DMA,2,4- 3152 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
959 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PHENTOLAMINE 891 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
70847 5-HT2C test test 3H-MESULERGINE N-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 18 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
85439 5-HT2C test test 3H-MESULERGINE 2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole 6210 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
86719 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) isonicotinamide 2.23 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90047 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 6.4 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27839 5-HT2C Choroid Plexus PIG 3H-MESULERGINE GR218231 1000 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100287 5-HT2C CLONED HUMAN 3H-MESULERGINE RISPERIDONE 24 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
35775 5-HT2C CLONED HUMAN 3H-MESULERGINE S-34324 1000 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
704 5-HT2C CORTEX PIG 3H-MESULERGINE DMA,2,5- 1217 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
960 5-HT2C CORTEX RAT 3H-MESULERGINE PHENTOLAMINE 1120 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
86720 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide 6.79 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90048 5-HT2C CLONED HUMAN 3H-MESULERGINE Mescaline-NBOMe 640 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27840 5-HT2C Choroid Plexus PIG 3H-MESULERGINE L741,626 3981.07 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100288 5-HT2C CLONED HUMAN 3H-MESULERGINE Paliperidone 38 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
35776 5-HT2C CLONED HUMAN 3H-MESULERGINE (+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 1000 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
59584 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Phenyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
705 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DMT,5-MeO 87.1 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
961 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PHENTOLAMINE 1150 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
70849 5-HT2C test test 3H-MESULERGINE 2-(4-chloro-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 67 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
76225 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
85697 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
90049 5-HT2C CLONED HUMAN 3H-MESULERGINE LSD 15 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
27841 5-HT2C CLONED HUMAN 3H-MESULERGINE S33084 79.4328 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
33217 5-HT2C CLONED RAT 3H-MESULERGINE Diclofenac sodium salt >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100289 5-HT2C CLONED HUMAN 3H-MESULERGINE ILOPERIDONE 46 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
35777 5-HT2C CLONED HUMAN 3H-MESULERGINE (+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 1000 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
706 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DMT,5-MeO 100 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
74178 5-HT2C test test 3H-MESULERGINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 2664 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
78274 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
82114 5-HT2C CLONED HUMAN 3H-MESULERGINE 5,6-dimethoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)isoindolin-1-one 3428 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85698 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88514 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
27842 5-HT2C CLONED HUMAN 3H-MESULERGINE GR218231 1000 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100290 5-HT2C CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 62 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
35778 5-HT2C CLONED HUMAN 3H-MESULERGINE (+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 1000 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
59842 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(2-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 1241 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
63682 5-HT2C CLONED HUMAN 3H-MESULERGINE OLANZAPINE 10.2329 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
707 5-HT2C CORTEX PIG 3H-MESULERGINE DOB 69 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
963 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(+/-) >10000 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
70851 5-HT2C test test 3H-MESULERGINE 2-(2,5-dimethoxy-4-nitrophenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 250 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
80579 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((5-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one 1265 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
83651 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
27843 5-HT2C CLONED HUMAN 3H-MESULERGINE L741,626 1000 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
100291 5-HT2C CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 86 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
35779 5-HT2C CLONED HUMAN 3H-MESULERGINE (+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 1000 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
59587 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Isopropyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
708 5-HT2C CORTEX PIG 3H-MESULERGINE DOB 69 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
5316 5-HT2C Choroid Plexus RAT 3H-MESULERGINE RS 67333 794.32 EGLEN RM, ET AL, 1995 Jan 15, 2025 Jan 15, 2025
100292 5-HT2C CLONED HUMAN 3H-MESULERGINE Blonanserin 251 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
709 5-HT2C CORTEX PIG 3H-MESULERGINE DOB,R(-) 47 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
965 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(+) >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
70853 5-HT2C test test 3H-MESULERGINE 4-(2-((4-fluoro-2-methoxybenzyl)amino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride >10000 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
86725 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide 0.156 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
100293 5-HT2C CLONED HUMAN 3H-MESULERGINE Lurasidone HCl 481 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
710 5-HT2C CORTEX PIG 3H-MESULERGINE DOB,S(+) 81 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
966 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(+) >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
73158 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl) butan-1-one hydrochloride 2976 Ofori E et al 2016 Jan 15, 2025 Jan 15, 2025
78022 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
12742 5-HT2C BRAIN RAT 3H-MESULERGINE LY 293284 1000 Foreman MM, et al., 1994 Jan 15, 2025 Jan 15, 2025
80326 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one 604 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82374 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-4-(2-(Indolin-1-yl)ethyl)-2-((pyridin-2-yloxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85446 5-HT2C test test 3H-MESULERGINE 1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol >10000 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
86726 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
100294 5-HT2C CLONED HUMAN 3H-MESULERGINE NEMONAPRIDE 481 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
59590 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Propyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
711 5-HT2C CORTEX PIG 3H-MESULERGINE DOBU 26 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
967 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(+) >10000 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
85703 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl)picolinamide 79.4 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
100295 5-HT2C CLONED HUMAN 3H-MESULERGINE GMC 1-116 615 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
712 5-HT2C CORTEX PIG 3H-MESULERGINE DOET 101 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
968 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(+) >10000 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
74952 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
85704 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88520 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
24776 5-HT2C CLONED RAT 3H-MESULERGINE CHLORPROMAZINE 26 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
28104 5-HT2C CLONED RAT 3H-MESULERGINE Fenfluramine (-) 3415 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100296 5-HT2C CLONED HUMAN 3H-MESULERGINE Remoxapride 3574 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41672 5-HT2C CLONED RAT 3H-MESULERGINE ORG-5222 0.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
63432 5-HT2C Choroid Plexus PIG 3H-MESULERGINE Y-931 0.89 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
969 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(+) >10000 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
70601 5-HT2C CLONED HUMAN 3H-MESULERGINE MRP3172 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
34761 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methylthio-1-[[3-(4-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 3.16228 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
59593 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Cyclohexyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
62665 5-HT2C CLONED RAT 3H-MESULERGINE (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-methyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one 1679 Mcleod, Michael C. et. al., 2016 Jan 15, 2025 Jan 15, 2025
63433 5-HT2C Choroid Plexus PIG 3H-MESULERGINE OLANZAPINE 2.7 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
714 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOI 18.6 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
970 5-HT2C CORTEX PIG 3H-MESULERGINE PINDOLOL,(+/-) >10000 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
77770 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80842 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((6-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
33482 5-HT2C CLONED RAT 3H-MESULERGINE Meloxicam sodium >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33738 5-HT2C CLONED RAT 3H-MESULERGINE VALDECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34762 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methylthio-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 1.58489 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
63434 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CLOZAPINE 2.9 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
715 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOI 18.6 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
75979 5-HT2C CLONED HUMAN 3H-MESULERGINE Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
82635 5-HT2C CLONED HUMAN 3H-MESULERGINE (S)-1-(Indolin-1-yl)-2-(2-((3-methoxyphenoxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
86731 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
34763 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[3-(2-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 19.9526 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
63435 5-HT2C Choroid Plexus PIG 3H-MESULERGINE HALOPERIDOL 5700 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
716 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOI 18.6 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
972 5-HT2C CORTEX RAT 3H-MESULERGINE PINDOLOL,(-) >10000 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
86732 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide 100 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
26060 5-HT2C CLONED RAT 3H-MESULERGINE Methcathinone, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34764 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 1 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
59596 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-Methyl-2-propanyl)-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
63436 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RISPERIDONE 22 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
717 5-HT2C CORTEX PIG 3H-MESULERGINE DOI 30 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
85709 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
34765 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[3-(4-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 0.630957 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
718 5-HT2C CORTEX PIG 3H-MESULERGINE DOM 193 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
974 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(-) >10000 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
77518 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80590 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((6-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one 1704 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
85454 5-HT2C test test 3H-MESULERGINE 2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride >10000 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
85710 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(piperonyl)piperazin-1-yl)ethyl)picolinamide 61.2 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88526 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
34766 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[3-(2-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5.01187 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
719 5-HT2C CORTEX PIG 3H-MESULERGINE DOM,R(-) 94 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
975 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(-) >10000 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
25551 5-HT2C CLONED HUMAN 3H-MESULERGINE pdspTestCompound3 63.44 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34767 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[3-(2,4-dimethyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 2.51189 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
59599 5-HT2C CLONED HUMAN 3H-MESULERGINE N-Butyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
63695 5-HT2C CLONED HUMAN 3H-MESULERGINE Quetiapine 1412.54 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
720 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOMPERIDONE >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
976 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(-) >10000 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
79056 5-HT2C CLONED HUMAN 3H-MESULERGINE Salvinorin A >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
98768 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
34768 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[4-methyl-3-(4-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 0.316228 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
721 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOMPERIDONE >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
977 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(-) >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
79057 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-2,5-Dimethoxy-4-bromoamphetamine 41.5 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
83665 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
86737 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
34769 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[4-Chloro-3-(4-methyl-3pyridyl)phenyl]carbamoyl-5-methoxy-6-trifluoromethylindoline 0.630957 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
978 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PINDOLOL,(-) >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
5074 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxytryptamine 52.48 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
77266 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
79058 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-3,4-Methylenedioxyamphetamine 6418 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80338 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one 35 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
86738 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
22226 5-HT2C CLONED RAT 3H-MESULERGINE Salvinorin A >10000 Roth BL, et al., 2002 Jan 15, 2025 Jan 15, 2025
34770 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[4-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 15.8489 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
38866 5-HT2C CLONED RAT 3H-MESULERGINE MDL 11,939 853.6 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
59602 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-Methylphenyl)-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide >10000 Kwon, Y. et. al., 2010 Jan 15, 2025 Jan 15, 2025
979 5-HT2C CORTEX RAT 3H-MESULERGINE PIRENPERONE 15.15 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
66515 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5075 5-HT2C CLONED HUMAN 3H-MESULERGINE BUSPIRONE 489.77 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
6355 5-HT2C Choroid Plexus PORCINE 3H-MESULERGINE GR 113808 >10000 GALE JD, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
79059 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-3,4-Methylenedioxymethamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85715 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(furoyl)piperazin-1-yl)ethyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
34771 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[4-(4-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5.01187 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
38867 5-HT2C CLONED RAT 3H-MESULERGINE SR 46349B 8.243 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
980 5-HT2C CORTEX PIG 3H-MESULERGINE PIRENPERONE 20 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
5076 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 4.26 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
79060 5-HT2C CLONED HUMAN 3H-MESULERGINE 3,4,5-Trimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85716 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) picolinamide 49.8 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87508 5-HT2C CLONED HUMAN 3H-MESULERGINE 1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
88532 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
38868 5-HT2C CLONED RAT 3H-MESULERGINE MDL 100907 88 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
725 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOPAMINE >10000 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
981 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 25 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
5077 5-HT2C CLONED HUMAN 3H-MESULERGINE CYPROHEPTADINE 2.23 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
75733 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
79061 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Bromo-2,5-dimethoxyphenethylamine 89.5 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
25045 5-HT2C CLONED RAT 3H-MESULERGINE OLANZAPINE 24 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
982 5-HT2C Choroid Plexus HUMAN 3H-MESULERGINE PIRENPERONE 52.5 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
3542 5-HT2C CLONED RAT 3H-MESULERGINE Amphetamine,(+) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5078 5-HT2C CLONED HUMAN 3H-MESULERGINE DP-5-CT 1000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
77014 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
79062 5-HT2C CLONED HUMAN 3H-MESULERGINE DMT 334.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80854 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((6-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one 4367 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82134 5-HT2C CLONED HUMAN 3H-MESULERGINE 6-methoxy-2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)isoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85462 5-HT2C test test 3H-MESULERGINE 2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate 6265 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
28374 5-HT2C CLONED RAT 3H-MESULERGINE ERGOTAMINE 12 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
727 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOPAMINE >10000 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
983 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 56.2 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
3543 5-HT2C CLONED RAT 3H-MESULERGINE SKF 82958 4626 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5079 5-HT2C CLONED HUMAN 3H-MESULERGINE ERGOTAMINE 9.77 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
5335 5-HT2C Choroid Plexus RAT 3H-MESULERGINE RS 67506 1995.26 EGLEN RM, ET AL, 1995 Jan 15, 2025 Jan 15, 2025
72407 5-HT2C CLONED HUMAN 3H-MESULERGINE 5,6-methylenedioxy-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 15, 2025
74711 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
79063 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Hydroxy-N,N-dimethyltryptamine 141.2 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86743 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
59863 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(2-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 1077 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
728 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOPAMINE >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
66776 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 2664 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
3544 5-HT2C CLONED RAT 3H-MESULERGINE APOMORPHINE 1103 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5080 5-HT2C CLONED HUMAN 3H-MESULERGINE FLUOXETINE 112.2 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72920 5-HT2C CLONED HUMAN 3H-MESULERGINE vicenin-2 >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
79064 5-HT2C CLONED HUMAN 3H-MESULERGINE DMT,5-MeO 538 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86744 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(piperonyl)piperazin-1-yl)ethyl)isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
729 5-HT2C Choroid Plexus PIG 3H-MESULERGINE DOPAMINE >10000 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
985 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 60.3 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
3545 5-HT2C CLONED RAT 3H-MESULERGINE BROMOCRIPTINE,(+) 4674 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5081 5-HT2C CLONED HUMAN 3H-MESULERGINE GR 113808 >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
79065 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Ethyl-2,5-dimethoxyphenethylamine 104.1 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85721 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) picolinamide 0.8 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
59609 5-HT2C BRAIN RAT 3H-MESULERGINE LP-211 91 Hedlund, P. et. al., 2010 Jan 15, 2025 Jan 15, 2025
986 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 50 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
3546 5-HT2C CLONED RAT 3H-MESULERGINE BUTACLAMOL,(+) 1064 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5082 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
73178 5-HT2C test test 3H-MESULERGINE 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
76762 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
79066 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Ethylthio-2,5-dimethoxyphenethylamine 53.9 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80602 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-5-((7-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one 3013 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82394 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-1-(Indolin-1-yl)-2-(2-(((4-methylpyridin-2-yl)oxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85722 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl)picolinamide 116 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88538 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-Phenoxypropyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
47322 5-HT2C CLONED RAT 3H-MESULERGINE WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
987 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 50.1 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3547 5-HT2C CLONED RAT 3H-MESULERGINE CARBAMAZEPINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69595 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-CI-DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5083 5-HT2C CLONED HUMAN 3H-MESULERGINE KETANSERIN 47.86 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
74459 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
79067 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-4-Ethylthio-2,5-dimethoxyamphetamine 50.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
81371 5-HT2C test test 3H-MESULERGINE 5’-Bromo-4’-OMethyl-HEAT HCl 711 Petrie EC et al 2012 Jan 15, 2025 Jan 15, 2025
50651 5-HT2C CLONED RAT 3H-MESULERGINE MDMA >10000 Setola V, et al., 2003 Jan 15, 2025 Jan 15, 2025
988 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 50.1 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
3548 5-HT2C CLONED RAT 3H-MESULERGINE CGS 12066B 6601 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69596 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5084 5-HT2C CLONED HUMAN 3H-MESULERGINE LISURIDE 5.88 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
75484 5-HT2C CLONED HUMAN 3H-MESULERGINE propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
79068 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-2,5-Dimethoxy-4-ethoxyamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
25564 5-HT2C CLONED HUMAN 3H-MESULERGINE pdspTestCompound4 50 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
63708 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 17.378 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
66013 5-HT2C CLONED RAT 3H-MESULERGINE Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
989 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIRENPERONE 50.1 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
3549 5-HT2C CLONED RAT 3H-MESULERGINE CHLORPROMAZINE 39 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69597 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5085 5-HT2C CLONED HUMAN 3H-MESULERGINE mCPP 104.71 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
73437 5-HT2C test test 3H-MESULERGINE N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
79069 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-N-methyl-N-isopropyltryptamine 2186 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86749 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(furoyl)piperazin-1-yl)ethyl)isonicotinamide 331 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
3550 5-HT2C CLONED RAT 3H-MESULERGINE CLOMIPRAMINE 52 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69598 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5086 5-HT2C CLONED HUMAN 3H-MESULERGINE MESULERGINE 1.69 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
76510 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
79070 5-HT2C CLONED HUMAN 3H-MESULERGINE N,N-Diisopropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86750 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) isonicotinamide 55 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
36574 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RISPERIDONE 48 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
735 5-HT2C CORTEX PIG 3H-MESULERGINE DOPR 14 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
991 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIZOTIFEN 7.9 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
67039 5-HT2C CLONED HUMAN 3H-MESULERGINE {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
3551 5-HT2C CLONED RAT 3H-MESULERGINE COCAINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69599 5-HT2C CLONED HUMAN 3H-MESULERGINE DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
5087 5-HT2C CLONED HUMAN 3H-MESULERGINE METERGOLINE 0.18 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
79071 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Ethylthio-2,5-dimethoxyphenylbutylamine 468 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
82655 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
83679 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
85727 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(3-(4-phenylpiperazin-1-yl)propyl)picolinamide 111 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
86239 5-HT2C CLONED HUMAN 3H-MESULERGINE JWH-391 1899 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
992 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIZOTIFEN 8.32 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
3552 5-HT2C CLONED RAT 3H-MESULERGINE CYPROHEPTADINE 15 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5088 5-HT2C CLONED HUMAN 3H-MESULERGINE METHIOTHEPIN 0.34 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70880 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine 343 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
79072 5-HT2C CLONED HUMAN 3H-MESULERGINE N,N-Dipropyltryptamine 1567 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85472 5-HT2C test test 3H-MESULERGINE 2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride >10000 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
85728 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) picolinamide 128 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88544 5-HT2C CLONED HUMAN 3H-MESULERGINE (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
34784 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[2-Fluoro-5-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1995.26 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
737 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ERGOMETRINE 31.6 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
993 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIZOTIFEN 8.32 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
3553 5-HT2C CLONED RAT 3H-MESULERGINE DEPRENYL >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5089 5-HT2C CLONED HUMAN 3H-MESULERGINE METHYSERGIDE 0.95 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70881 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine 338 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
79073 5-HT2C CLONED HUMAN 3H-MESULERGINE 6-Fluoro-N,N-dimethyltryptamine 674.2 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
34785 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[2-methyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 25.1189 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
738 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ERGOTAMINE 50 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
994 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIZOTIFEN 8.32 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
3554 5-HT2C CLONED RAT 3H-MESULERGINE DESIPRAMINE 748 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5090 5-HT2C CLONED HUMAN 3H-MESULERGINE MIANSERIN 1.38 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70882 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
79074 5-HT2C CLONED HUMAN 3H-MESULERGINE LISURIDE >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80866 5-HT2C CLONED HUMAN 3H-MESULERGINE )-5-((6-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 980 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
34786 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[2-Chloro-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 10 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
59106 5-HT2C CLONED RAT 3H-MESULERGINE Beta-LT >10000 Buhler A, et al., 2007 Jan 15, 2025 Jan 15, 2025
739 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ERGOTAMINE 56.2 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
995 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PRAZOSIN >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
1763 5-HT2A CORTEX RAT 3H-MESULERGINE CINANSERIN 7.9 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
3555 5-HT2C CLONED RAT 3H-MESULERGINE DHE 298 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
3811 5-HT2C CLONED HEK293 3H-MESULERGINE SB 242084 1 Kennett GA, et al., 1997 Jan 15, 2025 Jan 15, 2025
5091 5-HT2C CLONED HUMAN 3H-MESULERGINE NORFLUOXETINE 91.2 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70883 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine 32 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
78819 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
79075 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-2,5-Dimethoxy-4-iodoamphetamine 45.8 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86755 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide 28.7 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
21987 5-HT2C CLONED RAT 3H-MESULERGINE CYPROHEPTADINE 11 Runyon S.P. et al., 2001 Jan 15, 2025 Jan 15, 2025
34787 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[4-methyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
740 5-HT2C Choroid Plexus PIG 3H-MESULERGINE FENOLDOPAM 2140 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
67300 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 113 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
3556 5-HT2C CLONED RAT 3H-MESULERGINE L-DOPA >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5092 5-HT2C CLONED HUMAN 3H-MESULERGINE OXYMETAZOLINE 120.22 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70884 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
79076 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane 10.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85476 5-HT2C test test 3H-MESULERGINE 1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride >10000 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
86756 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl) isonicotinamide 385 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
21988 5-HT2C CLONED RAT 3H-MESULERGINE IMIPRAMINE 160 Runyon S.P. et al., 2001 Jan 15, 2025 Jan 15, 2025
34788 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[4-tert-Butyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 3.16228 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
3557 5-HT2C CLONED RAT 3H-MESULERGINE DOPAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5093 5-HT2C CLONED HUMAN 3H-MESULERGINE PAROXETINE >10000 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70885 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
73701 5-HT2C test test 3H-MESULERGINE [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
79077 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-2,5-Dimethoxy-4-methylamphetamine 3980 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
81125 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
85733 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
21989 5-HT2C CLONED RAT 3H-MESULERGINE AMDA 43 Runyon S.P. et al., 2001 Jan 15, 2025 Jan 15, 2025
33253 5-HT2C CLONED RAT 3H-MESULERGINE nimesulide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34789 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[4-Chloro-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 5.01187 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
59621 5-HT2C BRAIN RAT 3H-MESULERGINE RA-7 171 Hedlund, P. et. al., 2010 Jan 15, 2025 Jan 15, 2025
998 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PROPRANOLOL 589 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67558 5-HT2C KIDNEY HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)amino)- 9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol 84 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
3558 5-HT2C CLONED RAT 3H-MESULERGINE DOPAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5094 5-HT2C CLONED HUMAN 3H-MESULERGINE RAUWOLSCINE 645.65 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70886 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
73958 5-HT2C test test 3H-MESULERGINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
79078 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-3,4,5-Trimethoxamphetamine 4599.5 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80614 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-4-((1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
85734 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl)picolinamide 80 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88550 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 8829 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
99046 5-HT2C CLONED HUMAN 3H-MESULERGINE (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 15, 2025
34790 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[4-Methoxy-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 0.501187 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
36582 5-HT2C Choroid Plexus PIG 3H-MESULERGINE 9-OH-risperidone 47 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
743 5-HT2C Choroid Plexus PIG 3H-MESULERGINE FLUPHENAZINE 2570 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
3559 5-HT2C CLONED RAT 3H-MESULERGINE 8-OH-DPAT >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5095 5-HT2C CLONED HUMAN 3H-MESULERGINE RITANSERIN 0.25 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
70887 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine 24 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
75239 5-HT2C CLONED HUMAN 3H-MESULERGINE ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
78567 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
79079 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-2,5-Dimethoxy-4-ethylamphetamine 107.2 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
99047 5-HT2C CLONED HUMAN 3H-MESULERGINE (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 15, 2025
34791 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[3-Fluoro-5-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
744 5-HT2C Choroid Plexus PIG 3H-MESULERGINE GEPIRONE >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
1000 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PROPRANOLOL,(-) 158 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
3560 5-HT2C CLONED RAT 3H-MESULERGINE ETICLOPRIDE,S(-) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5096 5-HT2C CLONED HUMAN 3H-MESULERGINE ZACOPRIDE,S 794.32 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
79080 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-2,4,5-Trimethoxamphetamine 4062 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
32744 5-HT2C CLONED RAT 3H-MESULERGINE 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+/-) 0.21 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
99048 5-HT2C CLONED HUMAN 3H-MESULERGINE (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 15, 2025
34792 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[5-Bromo-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1.99526 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
745 5-HT2C Choroid Plexus PIG 3H-MESULERGINE GEPIRONE >10000 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
1001 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PROPRANOLOL,(-) 178 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
3561 5-HT2C CLONED RAT 3H-MESULERGINE FLUPENTHIXOL, Alpha 295 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5097 5-HT2C CLONED HUMAN 3H-MESULERGINE SB200646a 398.1 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
79081 5-HT2C CLONED HUMAN 3H-MESULERGINE LYSERGIC ACID 30.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86761 5-HT2C FR. CORTEX RAT 3H-MESULERGINE MESULERGINE 1.9 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
32745 5-HT2C CLONED RAT 3H-MESULERGINE 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+) 0.16 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
34793 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-[[5-Ethyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 0.630957 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
63721 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL 4677.35 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
1002 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PROPRANOLOL,(-) 407 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
3562 5-HT2C CLONED RAT 3H-MESULERGINE FLUPHENAZINE 1011 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5098 5-HT2C CLONED HUMAN 3H-MESULERGINE SB204741 1995.26 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
76266 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11498 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RITANSERIN 2.1 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
79082 5-HT2C CLONED HUMAN 3H-MESULERGINE cis-2a 105.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80362 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one 841 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82154 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
86762 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(3-(4-phenylpiperazin-1-yl)propyl)isonicotinamide 29.8 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
32746 5-HT2C CLONED RAT 3H-MESULERGINE 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(-) 0.39 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
34794 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methoxy-1-[[5-phenyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 2.51189 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
1003 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PROPRANOLOL,(-) 457 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
67563 5-HT2C KIDNEY HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)amino)- 9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(pentan-3-ylamino)-9H-purin-9- yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol 703 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
3563 5-HT2C CLONED RAT 3H-MESULERGINE GBR-12909 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
5099 5-HT2C CLONED HUMAN 3H-MESULERGINE SER-084 22.9 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
79083 5-HT2C CLONED HUMAN 3H-MESULERGINE R,R-2b 471.7 Ray TS 2010 Jan 15, 2025 Jan 15, 2025