47836 KOR CLONED HUMAN 3H-U69,593 MCL-135 0.1 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
3293 D2 CLONED HUMAN 3H-YM 09151-2 SPIPERONE 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
36061 MOR Membranes RAT 3H-DAMGO 14-O-methyloxymorphone 0.1 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
47070 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-MPM 0.1 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
3296 D2 CLONED HUMAN 3H-YM 09151-2 YM-09151-2 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
29152 SST4 CLONED HUMAN 125I-Tyr11-SRIF somatostatin-28 0.1 Reisine T, et.al., 1995 Jan 15, 2025 Jan 15, 2025
38113 CLONED RAT 3H-dexamethasone RU-486 0.1 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
8678 SST2 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.1 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
63974 5-HT6 CLONED HUMAN 3H-LSD N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide 0.1 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
31977 D2 CORTEX RAT 125I-Epidepride EPIDEPRIDE 0.1 Kessler, R.M., et. al., 1993 Jan 15, 2025 Jan 15, 2025
48875 KOR BRAIN Frog 3H-EKC CAM 0.1 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
8940 SST2 CLONED RAT 125I-Tyr11-somatostatin-14 AcNH-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH2 0.1 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
8943 SST3 CLONED RAT 125I-Tyr11-somatostatin-14 Somatostatin-14 0.1 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
3312 D3 CLONED HUMAN 3H-YM 09151-2 ETICLOPRIDE,S(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
29168 SST1 CLONED HUMAN UNDEFINED Somatostatin-14 0.1 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
2545 5-HT3 CORTEX RAT 3H-BRL 43694 ZACOPRIDE,RS 0.1 NELSON & THOMAS, 1989 Jan 15, 2025 Jan 15, 2025
29169 SST1 CLONED HUMAN UNDEFINED somatostatin-28 0.1 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
48625 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
57075 D2 UNDEFINED HUMAN UNDEFINED Bifeprunox 0.1 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
8949 SST5 CLONED RAT 125I-Tyr11-somatostatin-14 H2N-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2 0.1 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
9468 Colliculus Neurons GUINEA PIG 125I-Iodomelatonin S 20098 0.1 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
5117 5-HT2A CLONED HUMAN 125I-DOI DOHx 0.1 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
28157 5-HT2B CLONED HUMAN 3H-LSD METHYSERGIDE 0.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48893 KOR BRAIN Frog 3H-NALOXONE CAM 0.1 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
36350 MOR BRAIN RAT 3H-DAMGO 14-O-methyloxymorphone 0.1 Spetea M, et al., 2004 Jan 15, 2025 Jan 15, 2025
48639 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
23708 MC1 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH alpha-MSH, [Nle4] 0.102 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
55857 D3 UNDEFINED UNDEFINED UNDEFINED N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one 0.105 Butini S et al., 2009 Jan 15, 2025 Jan 15, 2025
28767 SST2 CLONED HUMAN 125I-LTT-SRIF28 seglitide 0.109648 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
27503 5-HT1B STRIATUM GUINEA PIG 3H-GR-125743 GR46,611 0.109648 Millan MJ, et al., 2002a Jan 15, 2025 Jan 15, 2025
8199 SST5 CLONED HUMAN 125I-LTT-SST-28 LTT-SST-28 0.11 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
16394 CB1 WHOLE BRAIN RAT 3H-CP-55940 CP-55244 0.11 Breivogel CS, et al., 2001 Jan 15, 2025 Jan 15, 2025
34572 FOREBRAIN RAT 3H-Epibatidine A-85380-I 0.11 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
7445 BB2 CLONED MOUSE 125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14) DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14) 0.11 Katsuno T, et al., 1999 Jan 15, 2025 Jan 15, 2025
56086 MOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.11 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
18725 CGRP Coronary artery PIG 125-h alpha-CGRP h alpha-CGRP 0.11 Rorabaugh BR et al., 2001 Jan 15, 2025 Jan 15, 2025
17959 CCK2 BRAIN RAT 125I-CCK-8 15g 0.11 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
17961 CCK2 BRAIN RAT 125I-CCK-8 15f 0.11 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
17969 CCK2 BRAIN RAT 125I-CCK-8 14g 0.11 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
19764 D3 CLONED HUMAN UNDEFINED FLUPHENAZINE 0.11 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
54069 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(2'-quinolyl)acetamido]morphinan 0.11 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
17975 CCK2 BRAIN RAT 125I-CCK-8 2 0.11 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
8504 SST3 CLONED HUMAN 125I-CGP23996 somatostatin-28 0.11 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
60476 GABAA CLONED HUMAN FNZ PWZ-007A 0.11 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
63049 MC5 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Oic-DNal(2') Arg-Trp-Lys]-NH2 0.11 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
9805 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Bromo 0.11 Nonno,Pannacci,Lucini, Angeloni,Fraschini,Stankov Jan 15, 2025 Jan 15, 2025
37711 DOR CLONED HUMAN 3H-Diprenorphine HS464 0.11 Tryoen-Toth P, et al., 2005 Jan 15, 2025 Jan 15, 2025
29010 SST5 CLONED HUMAN 125I-LTT-SST-28 D-Trp8 SST-14 0.11 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
16211 D2 CORTEX RAT 125I-Epidepride Spiroperidol 0.11 Neve KA, et al., 1990a Jan 15, 2025 Jan 15, 2025
55894 MOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.11 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
33884 D2 FR. CORTEX RAT 3H-SPIPERONE SPIPERONE 0.11 Andersen PH, et al., 1985 Jan 15, 2025 Jan 15, 2025
11106 5-HT2A CLONED HUMAN 3H-KETANSERIN ILOPERIDONE 0.11 CINP 2000 PROCEEDING Jan 15, 2025 Jan 15, 2025
47729 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY, zebrafish 0.11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
56948 KOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-methyl)benzamido]morphinan-oxalate 0.11 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
12920 CELLS OPOSSUM 3H-RAUWOLSCINE RAUWOLSCINE 0.11 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
47745 Y1 CLONED RAT [125I] - Peptide YY PYY,[leu31,Pro34], human 0.11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
7813 GABAA CLONED HUMAN 3H-RO-15-1788 12 0.11 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
30854 NTSR1 CLONED MOUSE 125I-Neurotensin Neurotensin 2 0.11 Pettibone, DJ et al., 2001 Jan 15, 2025 Jan 15, 2025
60552 GABAA CLONED HUMAN FNZ SH-I-048A 0.11 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
23945 D3 CLONED HUMAN UNDEFINED FLUPHENAZINE 0.11 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
41865 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrazin-2-ylamine 0.11 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41877 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine 0.11 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
11670 BRAIN HUMAN 3H-PRAZOSIN PRAZOSIN 0.11 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
32926 D2 BRAIN MOUSE 3H-SPIROPERIDOL Spiroperidol 0.11 Andersen PH, et al., 1988 Jan 15, 2025 Jan 15, 2025
8870 GABAA CLONED HUMAN 3H-15-4513 CGS 8216, 1 0.11 Scholze P, et al., 1996 Jan 15, 2025 Jan 27, 2025
65448 GABAA CLONED HUMAN [3H] Flunitrazepam PWZ-007A 0.11 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
16299 D1 CLONED RAT 125I-SCH 23982 SCH 23390 0.11 Tiberi M, et al., 1991 Jan 15, 2025 Jan 27, 2025
9900 nAChR ADRENAL RAT 3H-Epibatidine IPH 0.11 Mukhin, et al, 1999 Jan 15, 2025 Jan 27, 2025
6833 Y4 CLONED HUMAN 125I-PYY P34-PYY,human 0.11 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
34489 CCR5 CLONED RAT 3H-Epibatidine Epibatidine-I,(+/-) 0.11 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
31164 NK3 BRAIN CORTEX GUINEA PIG 125I-Iodohistidyl [MePhe7]NKB SR 142801 0.11 Emonds-Alt X., et.al., 1995 Jan 15, 2025 Jan 15, 2025
68798 5-HT3 NG108-15 PIG 3H-DAU 6215 ZACOPRIDE,S 0.11 Schiavi, GB et al., 1994 Jan 15, 2025 Jan 15, 2025
55757 5-HT1D UNDEFINED HUMAN UNDEFINED 2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine 0.11 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
65498 nAChR CLONED HUMAN [3H] Flunitrazepam SH-I-048A 0.11 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
17884 CCK2 BRAIN RAT 125I-CCK-8 Racemate 0.11 Nishida A et al., 1994 Jan 15, 2025 Jan 15, 2025
38367 D1 BRAIN RAT 3H-SCH23390 MCL-204 0.11 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
47073 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-03I 0.11 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
68086 Y1 CLONED HUMAN [125I] - Peptide YY NPY Leu31, Pro34, human 0.11 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
26871 KOR CLONED RAT 3H-Diprenorphine [D-Ala8]Dyn A (1-11) NH2 0.11 Vig BS, et al., 2003 Jan 15, 2025 Jan 15, 2025
37112 BuChE serum BOVINE Functional N-[3-(1,2,3,4-Tetrahydroacridin-9-ylamino)propyl]-N'-[4-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)butyl]acetamide 0.11 Campiani G, et al., 2005a Jan 15, 2025 Jan 15, 2025
34110 H3 CLONED RAT 3H-Alpha-Me-histamine Cipralisant 0.112202 Esbenshade TA, et al., 2004 Jan 15, 2025 Jan 15, 2025
26820 GAL1 CLONED HUMAN 125I-GALANIN M35 0.112202 Borowsky Beth, et. al., 1998 Jan 15, 2025 Jan 15, 2025
98284 KOR CEREBELLUM GUINEA PIG 3H-U69593 N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide 0.113 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
16479 Beta1 CLONED HUMAN 125I-Pindolol Fluorocarazolol,(S) 0.114 Roth BL, et al., 2001 Jan 15, 2025 Jan 15, 2025
30357 KOR CLONED RAT 3H-Diprenorphine [ D-Ala8]Dyn A-(1-11)NH2 0.114 Aldrich JV, et.al.,2001 Jan 15, 2025 Jan 15, 2025
54955 Beta2 UNDEFINED HUMAN UNDEFINED CARAZOLOL 0.114 Sabio M et al., 2008 Jan 15, 2025 Jan 28, 2025
27415 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Roxindole 0.114815 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
50238 Y2 CLONED GUINEA PIG 125I-PYY NPY8-20, Ahx 0.117 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
60446 GABAA CLONED HUMAN FNZ XLI-286 0.118 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65455 nAChR CLONED HUMAN [3H] Flunitrazepam XLI-286 0.118 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
55672 AChE UNDEFINED HUMAN UNDEFINED N-(2-Hydroxyethyl)-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine 0.1191 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
15878 5-HT7 CLONED RAT UNDEFINED 5-CT 0.12 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
50951 KOR UNDEFINED HUMAN UNDEFINED 17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate 0.12 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
17160 5-HT2A BRAIN HUMAN 3H-KETANSERIN Ziprasidone 0.12 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
10250 CLONED HAMSTER 125I-HEAT PRAZOSIN 0.12 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
51210 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(5-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.12 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
8723 SST2 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 0.12 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
10261 CLONED HUMAN 125I-HEAT PRAZOSIN 0.12 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
53013 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan 0.12 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
9494 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Bromo 0.12 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
53272 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(6-fluoro-5-(3-methoxyphenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.12 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
53018 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)benzamido]morphinan 0.12 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
60442 GABAA CLONED HUMAN FNZ QH-II-090 0.12 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
13861 MOR Striatal Membranes BOVINE 3H-DAMGO CAM 0.12 McLaughlin, et al., 1998 Jan 15, 2025 Jan 15, 2025
93990 D3 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one 0.12 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
93992 D3 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one 0.12 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
53291 CHRNA4 UNDEFINED RAT UNDEFINED varenicline 0.12 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
6701 D2 ANTERIOR PITUITARY PIG 3H-SPIPERONE EPIDEPRIDE 0.12 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
19760 D2 CLONED HUMAN UNDEFINED Thiothixene-cis 0.12 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
54068 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-quinolyl)acetamido]morphinan 0.12 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
5951 Alpha2C CELLS OK 3H-RAUWOLSCINE RAUWOLSCINE 0.12 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
8767 SST2 CLONED HUMAN 125I-Tyr3-octreotide octreotide 0.12 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
11843 FR. CORTEX RAT 3H-PRAZOSIN PRAZOSIN 0.12 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
19782 5-HT2A CLONED HUMAN UNDEFINED ILOPERIDONE 0.12 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
6729 D2 ANTERIOR PITUITARY PIG 3H-RACLOPRIDE EPIDEPRIDE 0.12 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
16203 D2 LZR1 Cells RAT 125I-Epidepride Spiroperidol 0.12 Neve KA, et al., 1990a Jan 15, 2025 Jan 15, 2025
10830 D2 CLONED HUMAN 125I-IODOSULPRIDE R(-)NPA 0.12 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
55630 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(3-Pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride 0.12 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
9552 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 0.12 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
37712 DOR CLONED HUMAN 3H-Diprenorphine HS510A 0.12 Tryoen-Toth P, et al., 2005 Jan 15, 2025 Jan 15, 2025
60497 GABAA CLONED HUMAN FNZ PWZ-0071 0.12 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
2645 5-HT2A CORTEX RAT 3H-KETANSERIN SPIPERONE 0.12 ROTH ET AL., 1987 Jan 15, 2025 Jan 15, 2025
13143 D2 STRIATUM RAT 3H-SPIPERONE SPIPERONE 0.12 Billard W, et al., 1984 Jan 15, 2025 Jan 15, 2025
55902 MOR UNDEFINED HUMAN UNDEFINED Butorphanol 0.12 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
10092 MOR BRAIN MOUSE 125I-Endomorphin-2 NALBzoH 0.12 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
14700 LUNG RABBIT 3H-PZ Dexetimide 0.12 Bloom JW, et al., 1987 Jan 15, 2025 Jan 15, 2025
10096 MOR BRAIN MOUSE 125I-Endomorphin-2 Diprenorphine 0.12 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
29302 AT1 CLONED RAT 125I-Angiotensin II CANDESARTAN 0.12 Inada Y, et al., 2002 Jan 15, 2025 Jan 28, 2025
5242 5-HT7 CLONED RAT 3H-5HT 5-CT 0.12 RUAT M, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
29306 AT1 CLONED RAT 125I-Angiotensin II CANDESARTAN 0.12 Inada Y, et al., 2002 Jan 15, 2025 Jan 28, 2025
99964 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.12 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
41342 CLONED HUMAN UNDEFINED SKF 29661 0.12 Wu Q, et al., 2005 Jan 15, 2025 Jan 15, 2025
8324 SST2 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 0.12 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
55968 KOR UNDEFINED HUMAN UNDEFINED nalmefene 0.12 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
5025 5-HT2A CLONED HUMAN 3H-KETANSERIN METERGOLINE 0.12 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
51362 M2 UNDEFINED HUMAN UNDEFINED 7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 0.12 Sonda S et al., 2007 Jan 15, 2025 Jan 15, 2025
65442 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-077 0.12 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
16556 CLONED HUMAN 3H-SP ZD6021 0.12 Rumsey et al., 2001 Jan 15, 2025 Jan 15, 2025
65459 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-090 (CGS-8216) 0.12 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65464 nAChR CLONED HUMAN [3H] Flunitrazepam PWZ-0071 0.12 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7870 GABAA CLONED HUMAN 3H-RO-15-1788 CGS 8216, 1 0.12 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
56000 CB1 UNDEFINED HUMAN UNDEFINED 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride 0.12 Griffith DA et al., 2009 Jan 15, 2025 Jan 15, 2025
53953 D3 UNDEFINED HUMAN UNDEFINED 6-(4-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butoxy)phenyl)-5,6-dihydroimidazo[2,1-b]thiazole 0.12 Leopoldo M et al., 2009 Jan 15, 2025 Jan 15, 2025
6597 5-HT7 CLONED Mammalian 3H-5HT 5-CT 0.12 SEBBEN M, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
50118 SST5 CLONED HUMAN 125I-Tyr11-SRIF-14 Somatostatin-14 0.12 Poitout L., et.al., 2001 Jan 15, 2025 Jan 15, 2025
7885 GABAA CLONED HUMAN 3H-RO-15-1788 16 0.12 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
7378 KOR CLONED HUMAN 3H-U69,593 U50,488H 0.12 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
36056 MOR Membranes RAT 3H-DAMGO 14-O-Benzyloxymorphone 0.12 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
7642 5-HT1D CLONED HUMAN 3H-5HT GR 127935 0.12 Skingle M, et al., 1996 Jan 15, 2025 Jan 15, 2025
38368 D1 BRAIN RAT 3H-SCH23390 SCH 23390 0.12 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
7906 GABAA CLONED HUMAN 3H-RO-15-1788 2 0.12 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
34030 KOR CLONED RAT 3H-Diprenorphine Nor-BNI 0.12 Jones, RM et. al., 1998 Jan 15, 2025 Jan 15, 2025
31985 D2 HIPPOCAMPUS RAT 125I-Epidepride EPIDEPRIDE 0.12 Kessler, R.M., et. al., 1993 Jan 15, 2025 Jan 15, 2025
63473 5-HT1A CLONED HUMAN 3H-WAY100635 Brexpiprazole 0.12 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
37621 D2 CLONED HUMAN 3H-SPIROPERIDOL HALOPERIDOL 0.12 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
16377 Y2 CLONED RAT [125I] - Peptide YY PYY 3-36, porcine 0.12 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
17406 NOP BRAIN MOUSE 125I-Tyr14-OFQ OFQ/N,Iodo[Tyr14] 0.12 Mogil JS, Pasternak GW., 2001 Jan 15, 2025 Jan 15, 2025
28761 SST2 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 0.120226 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
59266 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-azabicyclo[2.2.1]heptane 0.122 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
67547 nAChR FOREBRAIN RAT 3H-Epibatidine Cytisine-(-) 0.123 Gohlke, H et al., 2003 Jan 15, 2025 Jan 15, 2025
32880 D2 CLONED HUMAN 3H-domperidone SPIPERONE 0.125 Grandy DK, et al., 1989 Jan 15, 2025 Jan 15, 2025
39971 CEREBRAL CORTEX RAT 3H-RX821002 ATIPAMEZOLE 0.125893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
68937 SST5 CLONED HUMAN 125I-SRIF Cyclo[(diaminoethylcarbamoyl)HyPro-Phg-D-Trp-Lys-Tyr(Bzl)-Phe] 0.125893 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
31356 5-HT7 BRAIN RAT 3H-MESULERGINE 5-Hydroxy Tryptamine 0.125893 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
31437 5-HT7 CLONED RAT 3H-5HT 5-CT 0.125893 Eglen RM et al., 1997 Jan 15, 2025 Jan 27, 2025
64734 H1 CLONED HUMAN 3H-PYRILAMINE Doxepine 0.125893 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
68859 SST2 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Ala-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 0.125893 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
99650 A2A CLONED HUMAN 3H-NECA 8-[{3-(2-(Diethylaminoethylamino)-2-oxoethoxy)-4-meth-oxy}phenyl]-1,3-dimethylxanthine 0.126 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99630 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine 0.128 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
32357 M4 LUNG RABBIT 3H-NMS Ipratropium 0.128825 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
16997 M1 CLONED HUMAN 3H-NMS NNC 11-1585 0.129 Christopoulos A, et al., 2001 Jan 15, 2025 Jan 15, 2025
8449 SST5 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.13 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
50950 KOR UNDEFINED HUMAN UNDEFINED (5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate 0.13 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
32009 D2 Striatal Membranes RAT 125I-Spectramide Spectramide 0.13 Sanchez-Roa, P.M., et al., 1989 Jan 15, 2025 Jan 15, 2025
48658 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.13 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
53012 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)phenylacetamido]morphinan 0.13 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
87324 Alpha1B placeholder HUMAN Placeholder Tamsulosin 0.13 Rak A et al 2016 Jan 15, 2025 Jan 28, 2025
6690 D2 CLONED HUMAN 3H-NEMONAPRIDE SPIPERONE 0.13 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
86818 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide 0.13 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
56354 CHRNA4 UNDEFINED RAT UNDEFINED 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine 0.13 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
53028 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan 0.13 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
5926 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE RAUWOLSCINE 0.13 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
23595 Spinal cord RAT 125I-1DMe-Y8Fa NPFF 0.13 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
5932 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE SPIROXATRINE 0.13 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
68397 Alpha2A CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 0.13 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
13363 D4 CLONED HUMAN 35S-GTPGammaS SPIPERONE 0.13 Newman-Tancredi A, et al., 1997 Jan 15, 2025 Jan 27, 2025
4153 5-HT1D CLONED HUMAN 3H-5HT DHE 0.13 HAMBLIN AND METCALF, 1991 Jan 15, 2025 Jan 15, 2025
8506 SST3 CLONED HUMAN 125I-CGP23996 CST17 0.13 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
19773 D3 CLONED HUMAN UNDEFINED PERPHENAZINE 0.13 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
20285 HEART RAT 3H-Nitrendipine NIFEDIPINE 0.13 Ehlert FJ et al., 1982 Jan 15, 2025 Jan 15, 2025
60477 GABAA CLONED HUMAN FNZ CGS8216 0.13 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
45634 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE PAROXETINE 0.13 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
47682 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Indatraline 0.13 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
38983 SPLEEN BOVINE 3H-DPCPX 4-amino-2-decylpyrazolo[3,4-d]pyrimidine 0.13 Da Settimo F, et al., 2005 Jan 15, 2025 Jan 15, 2025
8776 SST5 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.13 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
7241 ETA CLONED HUMAN 125I-ENDOTHELIN SB 234551 0.13 Ohlstein EH, et al., 1998 Jan 15, 2025 Jan 15, 2025
23889 D2 CLONED HUMAN 3H-RACLOPRIDE PIMOZIDE 0.13 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
30052 SST2 CLONED MOUSE 125I-SOMATOSTATIN MK 678 0.13 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
29285 KOR Placenta Membranes HUMAN 3H-U69,593 dihydroetorphine 0.13 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
41836 H3 CLONED HUMAN 3H-Alpha-Me-histamine 4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile 0.13 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
47741 Y1 CLONED RAT [125I] - Peptide YY PYY, porcine 0.13 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
11143 5-HT2A FR. CORTEX RAT 3H-KETANSERIN ORG-5222 0.13 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
23951 D3 CLONED HUMAN UNDEFINED PERPHENAZINE 0.13 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
34975 nAChR CLONED UNDEFINED 3H-Epibatidine 2-exo-(5-(6-Hydroxy-1-hexynyl)-3-pyridyl)-7-azabicyclo[2.2.1]heptane 0.13 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
37543 D3 CLONED RAT 3H-SPIROPERIDOL N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-7-methoxy-2-benzofurancarboxamide 0.13 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
53956 D3 UNDEFINED HUMAN UNDEFINED N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-7-methoxybenzofuran-2-carboxamide 0.13 Leopoldo M et al., 2009 Jan 15, 2025 Jan 15, 2025
15301 5-HT1D CLONED HUMAN 3H-5HT DHE 0.13 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
51673 5-HT7 UNDEFINED RAT UNDEFINED 4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 0.13 Leopoldo M et al., 2007 Jan 15, 2025 Jan 15, 2025
9949 M2 CLONED HUMAN 3H-MQNB(-) IMIPRAMINE 0.13 Kovacs, Yamamura, Waite, Varga, Roeske, 1998 Jan 15, 2025 Jan 15, 2025
7392 KOR CLONED HUMAN 3H-U69,593 ETORPHINE - HCI 0.13 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
58101 5-HT2C CLONED HUMAN 125I-DOI N-(3-Methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 0.13 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
8695 SST5 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.13 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
11518 MOR FOREBRAIN RAT 3H-Sufentanil Dextromoramide 0.13 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
60460 GABAA CLONED HUMAN FNZ JYI-57 0.131 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
87875 A2B test MOUSE 3H-PSB-603 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.131 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
65469 nAChR CLONED HUMAN [3H] Flunitrazepam JYI-57 0.131 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
27354 Alpha2B CLONED HUMAN 3H-RX821002 LISURIDE 0.134896 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
55671 AChE UNDEFINED HUMAN UNDEFINED 1,4-bis[3-(1,2,3,4-Tetrahydroacridin-9-yl)aminopropyl]piperazine 0.1359 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
50236 Y2 CLONED GUINEA PIG 125I-PYY NPY22-36, porcine 0.136 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
98285 KOR CEREBELLUM GUINEA PIG 3H-U69593 N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide 0.136 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
87873 A2B test HUMAN 3H-PSB-603 8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.137 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
16520 Beta2 CLONED HUMAN 125I-Pindolol Fluorocarazolol,(R) 0.138 Roth BL, et al., 2001 Jan 15, 2025 Jan 28, 2025
24746 Y1 CLONED HUMAN 125I-PYY PYY, porcine 0.138038 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
32475 NOP CLONED HUMAN 35S-GTPGammaS OFQ/N 0.138038 Carra' G., et.al., 2004 Jan 15, 2025 Jan 15, 2025
8452 SST5 CLONED HUMAN 125I-Tyr3-octreotide CST17 0.14 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
63748 nAChR BRAIN MICE 3H-NICOTINE Cytisine 0.14 Damaj, MI et al., 1998 Jan 15, 2025 Jan 15, 2025
17159 5-HT2A BRAIN HUMAN 3H-KETANSERIN SERTINDOLE 0.14 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
6925 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.14 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
19726 D2 CLONED HUMAN UNDEFINED FLUPENTHIXOL, Alpha 0.14 Seeman P et al,1997b Jan 15, 2025 Jan 15, 2025
9744 retina RABBIT 125I-Iodomelatonin S 20098 0.14 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
5649 Alpha2C CELLS OK 3H-RAUWOLSCINE L-654,284 0.14 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
64017 D3 CLONED MOUSE 3H-SPIPERONE (+)-Butaclamol 0.14 Fishburn CS, et al., 1993 Jan 15, 2025 Jan 15, 2025
8469 SST3 CLONED HUMAN 125I-LTT-SRIF28 LTT-SRIF28 0.14 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
6679 D2 ANTERIOR PITUITARY PIG 3H-NEMONAPRIDE NEMONAPRIDE 0.14 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
33815 D1 BRAIN RAT 3H-SCH23390 SCH 23390 0.14 Karlsson P, et al., 1993 Jan 15, 2025 Jan 15, 2025
14618 H4 CORTEX GUINEA PIG 3H-Histamine HISTAMINE 0.14 Zhu, Yand, et al., 2001 Jan 15, 2025 Jan 15, 2025
65577 GABAA CLONED HUMAN [3H] Flunitrazepam SPH-121 0.14 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
56106 DOR UNDEFINED HUMAN UNDEFINED NALTRINDOLE 0.14 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
15405 5-HT1B CLONED HUMAN 3H-5HT 5-CT 0.14 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
55853 D3 UNDEFINED UNDEFINED UNDEFINED 3-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyloxy]isoquinoline 0.14 Butini S et al., 2009 Jan 15, 2025 Jan 15, 2025
17967 CCK2 BRAIN RAT 125I-CCK-8 14i 0.14 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
22324 A1 BRAIN HAMSTER 3H-DPCPX DPCPX 0.14 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
33849 D1 FR. CORTEX RAT 3H-SCH23390 SCH 23390 0.14 Andersen PH, et al., 1985 Jan 15, 2025 Jan 15, 2025
54077 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-pyridyl)acetamido]morphinan 0.14 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
3391 5-HT3 CORTEX RAT 3H-LY 278584 ZACOPRIDE,RS 0.14 WONG ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67905 D2 CLONED HUMAN 3H-R-ZACOPRIDE (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 0.14 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
8002 GABAA CLONED HUMAN 3H-RO-15-1788 26 0.14 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
15939 CB1 CEREBELLUM RAT 3H-CP-55940 WIN 55212-2 0.14 Iwamura H, et al., 2000 Jan 15, 2025 Jan 15, 2025
47683 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE CLOMIPRAMINE 0.14 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
60483 GABAA CLONED HUMAN FNZ SPH-121 0.14 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
19786 5-HT2A CLONED HUMAN UNDEFINED MDL 100907 0.14 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
35150 5-HT2A CORTEX RAT 3H-KETANSERIN OCTOCLOTHEPIN-S 0.14 Campiani G, et al., 2002 Jan 15, 2025 Jan 15, 2025
37458 D3 Sf9 RAT 3H-SPIPERONE butylamide benzthiophene 0.14 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
29269 DOR BRAIN RAT 3H-[Ile5,6]deltorphin II 14-phenylpropoxymetopon 0.14 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
26970 PKCα CLONED HUMAN 3H-PDBU 12-Deoxyphorbol 13-phenylacetate 0.14 Wang QJ, et.al.,2003 Jan 15, 2025 Jan 28, 2025
34650 5-HT2A CORTEX RAT 3H-KETANSERIN OCTOCLOTHEPIN-S 0.14 Campiani G, et al., 2004 Jan 15, 2025 Jan 15, 2025
99935 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 0.14 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
51553 Alpha1D UNDEFINED HUMAN UNDEFINED 5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 0.14 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
32610 D1 Striatal Membranes RAT 3H-SCH23390 SCH 23390 0.14 Andersen PH, et al., 1992 Jan 15, 2025 Jan 15, 2025
40550 GABAA CLONED HUMAN 3H-RO-15-1788 7-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.14 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
4466 SLC6A4 BRAIN RAT 3H-IMIPRAMINE CLOMIPRAMINE 0.14 PALVIMAKI EP, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
35442 EP3 CLONED HUMAN 3H-PGE2 M&B-28767 0.14 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
6004 M4 ATRIA RAT 3H-QNB SCOPOLAMINE 0.14 CHELALA JL, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
32894 D1 BRAIN MOUSE 3H-SCH23390 SCH 23390 0.14 Andersen PH, et al., 1988 Jan 15, 2025 Jan 15, 2025
1669 5-HT2A CORTEX RAT 3H-KETANSERIN ALTANSERIN 0.14 LEYSEN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
16773 SLC6A4 CLONED HUMAN 3H-PAROXETINE CLOMIPRAMINE 0.14 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
41867 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(3-nitropyridin-2-yl)amine 0.14 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
6814 Y1 CLONED HUMAN 125I-PYY PYY, porcine 0.14 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
6817 Y1 CLONED HUMAN 125I-PYY P34-PYY,human 0.14 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
37542 D3 CLONED RAT 3H-SPIROPERIDOL N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide 0.14 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
18860 CB2 CLONED HUMAN 3H-BAY 38-7271 HU-210 0.14 Mauler F et al., 2002 Jan 15, 2025 Jan 15, 2025
30892 BRAIN RAT 3H-Cytisine 3-(2(R)-Pyrrolidinylmethoxy)pyridine Dihydrochloride 0.14 Abreo MA, et al., 1996 Jan 15, 2025 Jan 15, 2025
47794 MOR CLONED HUMAN 3H-DAMGO MCL-135 0.14 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
14259 D3 CLONED RAT 3H-SPIPERONE ETICLOPRIDE 0.14 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 15, 2025
30389 5-HT1B CLONED HUMAN 3H-5HT GR 127935 0.14 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
93645 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 0.14 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
5843 Alpha2B LUNG NEONATAL RAT 3H-RAUWOLSCINE BDF6143 0.14 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
60633 GABAA CLONED HUMAN FNZ DM-239 0.14 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
47071 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-03I 0.14 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47072 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-03I 0.14 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
65505 GABAA CLONED HUMAN [3H] Flunitrazepam DM-239 0.14 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
9442 MT1 CLONED HUMAN 125I-Iodomelatonin GR 196429 0.14 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
6116 Alpha1B CLONED HAMSTER 125I-HEAT PRAZOSIN 0.14 HORIE K, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
56041 MOR UNDEFINED UNDEFINED UNDEFINED (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-2-carboxylate 0.14 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
14315 SLC6A3 STRIATUM RAT 125I-RTI-55 Binding WF-23 0.14 Letchworth SR, et al., 2000 Jan 15, 2025 Jan 15, 2025
9454 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl 0.14 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
51950 MOR UNDEFINED HUMAN UNDEFINED 7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 0.14 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
34545 nAChR CLONED RAT 3H-Epibatidine A-85380 0.14 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
68083 Y1 CLONED HUMAN [125I] - Peptide YY PYY, human 0.14 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
63736 nAChR BRAIN MICE 3H-NICOTINE NMCC 0.14 Damaj, MI et al., 1998 Jan 15, 2025 Jan 15, 2025
27041 MOR ILEUM GUINEA PIG 3H-DAMGO [Dmt1]DALDA 0.143 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
27092 MOR BRAIN MOUSE 3H-DAMGO [Dmt1]DALDA 0.143 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
24749 Y1 CLONED HUMAN 125I-PYY PYY Pro34, Human 0.144544 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
50373 Y1 CLONED HUMAN 125I-PYY PYY Pro34, Human 0.144544 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
54959 Beta2 UNDEFINED HUMAN UNDEFINED GNF-Pf-1694 0.145 Sabio M et al., 2008 Jan 15, 2025 Jan 28, 2025
27087 MOR BRAIN MOUSE 3H-[Dmt1]DALDA Dmt-d-Arg-Phe-A2pr-NH2 0.145 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
34086 KOR CLONED HUMAN 35S-GTPGammaS FE200041 0.146 Vanderah TW et. al., 2004 Jan 15, 2025 Jan 15, 2025
60505 GABAA CLONED HUMAN FNZ JYI-42 0.146 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65486 nAChR CLONED HUMAN [3H] Flunitrazepam JYI-42 0.146 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
27408 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LISURIDE 0.147911 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
87846 A2B test HUMAN 3H-PSB-603 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.148 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
7425 MOR CLONED HUMAN 3H-DAMGO Sufentanyl 0.15 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
16385 Y2 CLONED RAT [125I] - Peptide YY NPY, C2 0.15 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
12036 H3 Striatal Membranes RAT 125I-Iodoproxyfan Imetit 0.15 Ligneau X, et al., 1994 Jan 15, 2025 Jan 15, 2025
17157 5-HT2A BRAIN HUMAN 3H-KETANSERIN RISPERIDONE 0.15 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
8710 SST2 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.15 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
11531 SLC6A4 Platelets HUMAN 3H-PAROXETINE IMIPRAMINE 0.15 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
2318 5-HT3 AREA POSTREMA RAT 3H-GR-65630 GRANISETRON 0.15 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
50711 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 0.15 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
18201 CCK2 PANCREAS RAT 125I-BH-CCK-8 30m 0.15 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
65820 GABAA CLONED HUMAN [3H] Flunitrazepam CM-D45 C19H21N3O4 0.15 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
9501 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Phenyl 0.15 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
14621 H4 myenteric plexus GUINEA PIG 3H-Histamine R-alpha-methylhistamine 0.15 Zhu, Yand, et al., 2001 Jan 15, 2025 Jan 15, 2025
9247 SST2 CLONED MOUSE 125I-MK-678 BIM 23068 0.15 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
47648 GABAA CLONED HUMAN 3H-RO-15-1788 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.15 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
8738 SST2 CLONED HUMAN 125I-CGP23996 seglitide 0.15 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8486 SST3 CLONED HUMAN 125I-Tyr10-CST14 somatostatin-28 0.15 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
5415 5-HT4 CLONED HUMAN 3H-GR-113808 GR 125487 0.15 Van den Wyngaert I, et al., 1997 Jan 15, 2025 Jan 15, 2025
53287 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(4-fluorophenyl)deschloroepibatidine 0.15 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
38956 T47D HUMAN Functional 5-(4,4-Dimethyl-2-thioxo-1,4-dihydro-2H-3, 1-benzoxazin-6-yl)-1H-pyrrole-2-carbonitrile 0.15 Fensome A, et al., 2005 Jan 15, 2025 Jan 15, 2025
38957 T47D HUMAN Functional Tanaproget 0.15 Fensome A, et al., 2005 Jan 15, 2025 Jan 15, 2025
52782 5-HT2A UNDEFINED HUMAN UNDEFINED N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide 0.15 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
68399 Alpha2C CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 0.15 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
5428 5-HT4 BRAIN HUMAN 3H-GR-113808 GR 113808 0.15 Van den Wyngaert I, et al., 1997 Jan 15, 2025 Jan 15, 2025
48692 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride 0.15 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
38969 nAChR BRAIN RAT 3H-Cytisine A-84543 0.15 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
9530 SLC6A4 CLONED HUMAN 3H-CITALOPRAM SERTRALINE 0.15 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
57403 CB1 UNDEFINED HUMAN UNDEFINED N-Cyclohexyl-4-[(2,4-dichlorophenyl)(p-tolyl)methyl]piperazine-1-carboxamide 0.15 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
35132 BRAIN RAT 3H-Cytisine 6-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 0.15 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
54078 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-pyridyl)acetamido]morphinan 0.15 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
23364 A1 BRAIN PIG 3H-DPCPX CCPA 0.15 Klotz KN et al., 1991 Jan 15, 2025 Jan 27, 2025
52299 MOR UNDEFINED HUMAN UNDEFINED 3-((3R,4R)-1-((S)-3-cyclohexyl-3-hydroxypropyl)-3,4-dimethylpiperidin-4-yl)phenol 0.15 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
23372 A1 BRAIN BOVINE 3H-DPCPX CCPA 0.15 Klotz KN et al., 1991 Jan 15, 2025 Jan 27, 2025
4175 5-HT1B CLONED HUMAN 3H-5HT 5-CT 0.15 HAMBLIN MW, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
31059 BRAIN RAT 3H-Cytisine A-84543 0.15 Abreo MA, et al., 1996 Jan 15, 2025 Jan 15, 2025
13396 D3 CLONED HUMAN 3H-thymidine Quinerolane 0.15 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
33117 NET BRAIN RAT UNDEFINED DESIPRAMINE 0.15 Muth, EA et al., 1986 Jan 15, 2025 Jan 15, 2025
55903 MOR UNDEFINED HUMAN UNDEFINED (1S,9R,10S)-17-(cyclobutylmethyl)-10-hydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-triene-4-carboxamide 0.15 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
29288 MOR BRAIN RAT 3H-DAMGO 14-methoxymetopon 0.15 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
8810 SST5 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.15 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
36971 MOR BRAIN RAT 3H-DAMGO 14-methoxymetopon 0.15 Spetea M.,et.al.,2003 Jan 15, 2025 Jan 15, 2025
50040 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-COOH, [Aib15] 0.15 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
56186 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane 0.15 Sippy KB et al., 2009 Jan 15, 2025 Jan 15, 2025
2429 5-HT3 AREA POSTREMA RAT 3H-GR-65630 METOCLOPRAMIDE 0.15 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
7295 ETA Coronary artery HUMAN 125I-ENDOTHELIN PD156707 0.15 Maguire JJ, et al., 1996 Jan 15, 2025 Jan 15, 2025
100751 MT2 C.H.O. HUMAN 125I-Iodomelatonin MELATONIN 0.15 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
47248 CLONED HUMAN Functional Motilin 0.15 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
52120 MOR UNDEFINED HUMAN UNDEFINED 4-(4-((phenethylamino)methyl)phenoxy)benzamide 0.15 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
20385 PANCREAS RAT 3H-CCK8 Guanylyl imidodiphosphate 0.15 Van Dijk A et al., 1984 Jan 15, 2025 Jan 15, 2025
52646 CB2 UNDEFINED HUMAN UNDEFINED HU-210 0.15 Manera C et al., 2007 Jan 15, 2025 Jan 15, 2025
8873 GABAA CLONED HUMAN 3H-15-4513 CGS 20625 0.15 Scholze P, et al., 1996 Jan 15, 2025 Jan 27, 2025
43177 STK3 mouse CLONED HUMAN 3H-Staurosporine Staurosporine 0.15 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
8365 SST2 CLONED HUMAN 125I-CGP23996 seglitide 0.15 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
68277 CCK1 CEREBRAL CORTEX RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester 0.15 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68279 CCK2 PANCREAS RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester 0.15 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
10681 M3 CLONED HUMAN 3H-NMS ATR 0.15 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
8383 SST2 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.15 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
11972 H3 CORTEX RAT 3H-GR168320 GR 168320 0.15 Brown JD, et al., 1996 Jan 15, 2025 Jan 15, 2025
34502 nAChR CLONED RAT 3H-Epibatidine Epibatidine-I,(+/-) 0.15 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
52170 MOR UNDEFINED HUMAN UNDEFINED 3-((3R,4R)-1-((S)-3-cyclohexyl-3-hydroxypropyl)-3,4-dimethylpiperidin-4-yl)phenol 0.15 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
11981 H3 CORTEX RAT 3H-NAMH VUF9153 0.15 Brown JD, et al., 1996 Jan 15, 2025 Jan 15, 2025
15823 5-HT7 CLONED RAT 3H-5HT 5-CT 0.15 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
61398 GABAA CLONED HUMAN FNZ CM-D45 0.15 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
36062 MOR Membranes RAT 3H-DAMGO 14-methoxymetopon 0.15 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
40160 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.15 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
51939 MOR UNDEFINED HUMAN UNDEFINED 14beta-(2'-chlorocinnamoylamino)-7,8-dihydromorphinone 0.15 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
8679 SST2 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.15 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
4840 5-HT4 CAUDATE HUMAN 3H-GR-113808 GR 113808 0.15 ANSANAY H, ET AL.,1996 Jan 15, 2025 Jan 15, 2025
2284 5-HT3 AREA POSTREMA RAT 3H-GR-65630 COCAINE 0.15 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
34541 nAChR CLONED RAT 3H-Epibatidine Epibatidine-I,(+/-) 0.15 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
8431 SST5 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.15 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
18159 SLC6A3 FOREBRAIN RAT 3H-beta-CIT GBR-12909 0.15 Davids E et al., 2002 Jan 15, 2025 Jan 15, 2025
14580 H3 CLONED HUMAN 3H-RAMHA R-alpha-methylhistamine 0.15 Zhu, Yand, et al., 2001 Jan 15, 2025 Jan 15, 2025
48628 GNRHR CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.15 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
34554 nAChR CLONED RAT 3H-Epibatidine Epibatidine-I,(+/-) 0.15 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
51196 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane 0.15 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
36351 MOR BRAIN RAT 3H-DAMGO 14-methoxymetopon 0.15 Spetea M, et al., 2004 Jan 15, 2025 Jan 15, 2025
27042 MOR ILEUM GUINEA PIG 3H-DAMGO H-Dmt-D-Arg-Phe-Orn-NH2 0.151 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
27084 MOR BRAIN MOUSE 3H-DAMGO Dmt-d-Arg-Phe-Orn-NH2 0.151 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
67556 nAChR FOREBRAIN RAT 3H-Epibatidine (1R)-2-(2-Chloropyrimidin-5-yl)-9-azabicyclo[4/2/1]non-2-ene Hydrochloride 0.151 Gohlke, H et al., 2003 Jan 15, 2025 Jan 15, 2025
69263 H3 CLONED HUMAN 3H-Alpha-Me-histamine Clobenpropit 0.151356 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
87849 A2B test HUMAN 3H-PSB-603 8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.153 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
86725 5-HT2C FR. CORTEX RAT 3H-MESULERGINE N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide 0.156 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
54592 A2B UNDEFINED HUMAN UNDEFINED 1-Ethyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 0.157 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
28926 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.157 Wei ZL, et. al., 2003 Jan 15, 2025 Jan 27, 2025
59272 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-methyl-7-azabicyclo[2.2.1]heptane 0.158 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
68898 SST1 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ala-Cys}-NH2 0.158489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
86607 5-HT4 CLONED HUMAN 3H-GR113808 N-[[1-(2-Cyclohexylethyl)-4-piperidinyl]methyl]-1-isopropyl-1Hindazole-3-carboxamide 0.158489 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
28766 SST3 CLONED HUMAN 125I-Tyr10-CST14 somatostatin-28 0.158489 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
86623 5-HT4 CLONED HUMAN 3H-GR-113808 piboserod 0.158489 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
100475 D3 CLONED HUMAN [3H]spiperone F17464 0.158489 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
17316 Alpha1B CEREBRAL CORTEX PIG 3H-PRAZOSIN PRAZOSIN 0.158489 Wikberg-Matsson A, et al., 1998 Jan 15, 2025 Jan 15, 2025
17375 Alpha1A CLONED HUMAN 3H-PRAZOSIN Fiduxosin 0.158489 Hancock A, et al., 2001 Jan 15, 2025 Jan 15, 2025
68849 SST2 CLONED HUMAN 125I-SRIF H-Ala-Ala-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 0.158489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
22002 LHRH Pituitary RAT UNDEFINED 10 0.158489 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
68862 SST5 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Ala-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 0.158489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
27585 CORTEX RAT 3H-RX821002 S18616 0.1585 Millan MJ, et al., 2000a Jan 15, 2025 Jan 15, 2025
87872 A2B test HUMAN 3H-PSB-603 8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 0.159 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
19456 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH hAc-MCH(6-16)-NH2 0.16 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
18959 H1 CLONED GUINEA PIG 3H-trans-H2-PAT,(-) DOXEPIN 0.16 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
53011 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzylacetamido)morphinan 0.16 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
9496 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Phenyl 0.16 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
53273 CHRNA4 UNDEFINED RAT UNDEFINED rac-3-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride 0.16 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
9499 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Bromo 0.16 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
56095 MOR UNDEFINED HUMAN UNDEFINED (1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide 0.16 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
35616 5-HT2A CLONED RAT 125I-LSD RISPERIDONE 0.16 Phillips ST, et. al., 1995 Jan 15, 2025 Jan 15, 2025
19746 D2 CLONED HUMAN UNDEFINED PERPHENAZINE 0.16 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
53027 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3'-methoxy)benzamido]morphinan 0.16 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
56361 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.16 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
2355 5-HT3 CORTEX RAT 3H-QICS 205-930 ICS 205-930, Q 0.16 WATLING ET AL., 1988 Jan 15, 2025 Jan 15, 2025
17973 CCK2 BRAIN RAT 125I-CCK-8 14c 0.16 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
23866 D2 CLONED HUMAN UNDEFINED PERPHENAZINE 0.16 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
2375 5-HT3 CORTEX RAT 3H-QICS 205-930 mCPP 0.16 WATLING ET AL., 1988 Jan 15, 2025 Jan 15, 2025
63048 MC4 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Oic-DNal(2') Arg-Trp-Lys]-NH2 0.16 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
47178 H1 CLONED HUMAN 3H-MEPYRAMINE DOXEPIN 0.16 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42573 Alpha1A CLONED UNDEFINED UNDEFINED WB 4101 0.16 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
10831 D3 CLONED HUMAN 125I-IODOSULPRIDE PHNO 0.16 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
55631 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(5-Phenylpyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bistrifluoroacetate 0.16 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
55892 MOR UNDEFINED HUMAN UNDEFINED Cyclazocine 0.16 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
29013 SST3 CLONED HUMAN 125I-LTT-SST-28 Leu8, D-Trp22, Tyr25 SST-28 0.16 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
53082 KOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan 0.16 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
23390 NK3 BRAIN CORTEX Gerbil 125I-Iodohistidyl [MePhe7]NKB NKB [MePhe7] 0.16 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
12138 D2 BRAIN HUMAN UNDEFINED SPIPERONE 0.16 Richelson E., 1988 Jan 15, 2025 Jan 15, 2025
8811 SST5 CLONED HUMAN 125I-CGP23996 Tyr10-cortistatin 0.16 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
29295 AT1 CLONED HUMAN 125I-Angiotensin II Angiotensin II 0.16 Inada Y, et al., 2002 Jan 15, 2025 Jan 28, 2025
12408 D3 CLONED RAT 125I-NCQ 298 125I-NCQ 298 0.16 Boundy VA, et al., 1993 Jan 15, 2025 Jan 15, 2025
100985 SERT CLONED HUMAN 125I-RTI-55 (S)-N-((1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-yl)methyl)-4-(4-(prop-2-yn-1-yloxy)benzoyl)benzamide 0.16 Yarravarapu N, et. al., 2018 Jan 15, 2025 Jan 28, 2025
123 5-HT1A CORTEX PIG 3H-8-OH-DPAT 5-CT 0.16 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
11134 5-HT2A FR. CORTEX RAT 3H-KETANSERIN RISPERIDONE 0.16 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
10881 D3 CLONED RAT 3H-SPIPERONE ETICLOPRIDE 0.16 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
14991 5-HT2A FR. CORTEX RAT 3H-Risperidone RISPERIDONE 0.16 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
62869 D2 Brain caudate nucleus HUMAN 3H-SPIROPERIDOL SPIPERONE 0.16 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 28, 2025
100246 5-HT2A CLONED HUMAN 3H-KETANSERIN Asenapine 0.16 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
9879 BRAIN RAT 5-125I-Iodo-A-85380 Cytisine-(-) 0.16 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
6811 Y1 CLONED HUMAN 125I-PYY L31,P34-NPY,human 0.16 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
34977 nAChR CLONED UNDEFINED 3H-Epibatidine Epibatidine 0.16 Wei ZL, et al., 2005 Jan 15, 2025 Jan 27, 2025
30891 BRAIN RAT 3H-Cytisine 3-(2-(S)-Pyrrolidinylmethoxy)pyridine Fumarate 0.16 Abreo MA, et al., 1996 Jan 15, 2025 Jan 15, 2025
39852 AT1 LIVER RAT 125I-Angiotensin II Ang II Sar1 0.16 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47797 MOR CLONED HUMAN 3H-DAMGO MCL-139 0.16 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
2240 5-HT3 CORTEX RAT 3H-QICS 205-930 5-HT,2-Me 0.16 WATLING ET AL., 1988 Jan 15, 2025 Jan 15, 2025
64966 D2 Ovary HAMSTER 125I-7-OH-PIPAT TERGURIDE 0.16 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
64975 D2 Ovary HAMSTER 3H-SPIPERONE BUTACLAMOL 0.16 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
64976 D2 Ovary HAMSTER 3H-SPIPERONE HALOPERIDOL 0.16 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
17619 CLONED RAT 125I-VIP VIP Ala9 0.16 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
11734 D2 CAUDATE NUCLEUS HUMAN 3H-SPIPERONE SPIPERONE 0.16 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
2523 5-HT3 CELLS N1E-115 3H-ICS 205-930 SDZ 206-830 0.16 HOYER & NEIJT, 1988 Jan 15, 2025 Jan 15, 2025
4316 5-HT7 CLONED RAT 3H-5HT 5-CT 0.16 SHEN Y, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
36060 MOR Membranes RAT 3H-DAMGO 14-ethoxy-3-hydroxy-5-methyl- 17-(2-phenylethyl)morphinan-6-one 0.16 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
11486 H1 CLONED HUMAN 3H-PYRILAMINE ORG-5222 0.16 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
32745 5-HT2C CLONED RAT 3H-MESULERGINE 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+) 0.16 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
9451 MT2 CLONED HUMAN 125I-Iodomelatonin GR 196429 0.16 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
38126 CLONED RAT 3H-dexamethasone C54H76NO6 0.16 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
50414 H1 BRAIN RODENT 3H-MEPYRAMINE DOXEPIN 0.16 Bucholtz E., et.al.1999 Jan 15, 2025 Jan 15, 2025
58094 5-HT2A CLONED HUMAN 125I-DOI N-(2-Methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 0.16 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
40176 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 0.16 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
8436 SST5 CLONED HUMAN 125I-CGP23996 CST14-Tyr10 0.16 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
34553 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.16 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
27083 MOR BRAIN MOUSE 3H-[Dmt1]DALDA Dmt-d-Arg-Phe-Orn-NH2 0.161 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
55673 AChE UNDEFINED HUMAN UNDEFINED N-Ethyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine 0.162 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
42511 CLONED HUMAN UNDEFINED Motilin 0.162181 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
100472 5-HT1A CLONED HUMAN [3H]8-OH-DPAT F17464 0.162181 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
69266 H3 CORTEX HUMAN 3H-Alpha-Me-histamine Imetit 0.162181 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
24743 Y1 CLONED HUMAN 125I-PYY NPY [Leu31, Pro34], human 0.162181 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
50368 Y1 CLONED HUMAN 125I-PYY PP,SALMON 0.162181 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
50378 Y1 CLONED HUMAN 125I-PYY NPY [Leu31, Pro34], human 0.162181 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
99631 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine 0.163 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
27076 MOR BRAIN MOUSE 3H-[Dmt1]DALDA [Dmt1]DALDA 0.163 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
97352 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 0.169 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
24745 Y1 CLONED HUMAN 125I-PYY PYY, human 0.169824 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
50370 Y1 CLONED HUMAN 125I-PYY PYY, human 0.169824 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
19457 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH hMCH 0.17 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
51212 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-chloro-5-hydroxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane 0.17 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
72466 5-HT1A test test [3H] Way100635 ERGOTAMINE 0.17 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
11541 H1 BRAIN HUMAN 3H-PYRILAMINE DOXEPIN 0.17 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
33814 D1 BRAIN RAT 3H-SCH23390 NNC-756 0.17 Karlsson P, et al., 1993 Jan 15, 2025 Jan 15, 2025
51224 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-fluoro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.17 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
99618 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]xanthine 0.17 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
53284 CHRNA4 UNDEFINED RAT UNDEFINED rac-3'-(3-nitrophenyl)deschloroepibatidine dihydrochloride 0.17 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
60454 GABAA CLONED HUMAN FNZ QH-II-092 0.17 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
53288 CHRNA4 UNDEFINED RAT UNDEFINED rac-3'-(3-chlorophenyl)deschloroepibatidine dihydrochloride 0.17 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
17966 CCK2 BRAIN RAT 125I-CCK-8 14j 0.17 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
28487 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.17 Kroeze WK, et.al., 2003 Jan 15, 2025 Jan 15, 2025
52300 MOR UNDEFINED HUMAN UNDEFINED 6-(4-((phenethylamino)methyl)phenoxy)nicotinamide 0.17 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
60498 GABAA CLONED HUMAN FNZ PWZ-0071 0.17 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
32609 D1 Striatal Membranes RAT 3H-SCH23390 NNC-756 0.17 Andersen PH, et al., 1992 Jan 15, 2025 Jan 15, 2025
40548 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.17 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
29293 AT1 CLONED HUMAN 125I-Angiotensin II CANDESARTAN 0.17 Inada Y, et al., 2002 Jan 15, 2025 Jan 28, 2025
57716 NR3C1 UNDEFINED HUMAN UNDEFINED CP-409069 0.17 Onnis V et al., 2010 Jan 15, 2025 Jan 15, 2025
9594 H1 BRAIN GUINEA PIG 3H-PYRILAMINE AMITRIPTYLINE 0.17 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
7293 BRAIN GUINEA PIG 3H-SR 48692 SR 142948A 0.17 Gully D, et al., 1996 Jan 15, 2025 Jan 15, 2025
6794 Y2 CLONED HUMAN 125I-PYY PYY, human 0.17 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
57746 H3 UNDEFINED HUMAN UNDEFINED 2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole 0.17 Ishikawa M et al., 2010 Jan 15, 2025 Jan 15, 2025
11155 5-HT2C Choroid Plexus PIG 3H-MESULERGINE ORG-5222 0.17 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
97686 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-propoxycarbonyl-4-quinolone 0.17 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
37529 D3 CLONED RAT 3H-SPIROPERIDOL N-[4-[4-(2,3-Dimethylphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 0.17 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
23962 D3 CLONED HUMAN 3H-RACLOPRIDE FLUPHENAZINE 0.17 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
6813 Y1 CLONED HUMAN 125I-PYY PYY, human 0.17 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
16285 mGluR5 CLONED HUMAN 125I-SCH 23982 SCH 23390 0.17 Tiberi M, et al., 1991 Jan 15, 2025 Jan 27, 2025
65438 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-092 0.17 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7850 GABAA CLONED HUMAN 3H-RO-15-1788 16 0.17 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
17583 CLONED HUMAN 125I-VIP VIP Ala8 0.17 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
65463 nAChR CLONED HUMAN [3H] Flunitrazepam PWZ-0071 0.17 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
9406 MT2 CLONED HUMAN 125I-Mel Melatonin,2-Iodo 0.17 Reppert, Godson, Mahle, Weaver, Slaugenhaupt, 1995 Jan 15, 2025 Jan 15, 2025
85183 MT2 NIH-3T3 HUMAN 125I-Iodomelatonin Tasimelteon 0.17 Lavedan C et al 2015 Jan 15, 2025 Jan 29, 2025
52160 MOR UNDEFINED HUMAN UNDEFINED 6-(4-((phenethylamino)methyl)phenoxy)nicotinamide 0.17 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
17612 CLONED RAT 125I-VIP VIP Ala2 0.17 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
28369 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ERGOTAMINE 0.17 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
17120 BRAIN HUMAN 3H-QNB Quinuclidinyl benzilate 0.17 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
7911 GABAA CLONED HUMAN 3H-RO-15-1788 7 0.17 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
47848 KOR CLONED HUMAN 3H-U69,593 MCL-143 0.17 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
38125 CLONED RAT 3H-dexamethasone C54H80NO8 0.17 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
63731 nAChR BRAIN RAT 3H-NICOTINE UB-165 0.17 Wright, E et al., 1997 Jan 15, 2025 Jan 15, 2025
11508 CORTEX RAT 3H-PRAZOSIN Aceperone 0.17 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
63476 Alpha1B CLONED HUMAN 3H-PRAZOSIN Brexpiprazole 0.17 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
17404 NOP BRAIN MOUSE 125I-Tyr14-OFQ OFQ/N 0.17 Mogil JS, Pasternak GW., 2001 Jan 15, 2025 Jan 15, 2025
59278 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.171 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
27093 MOR CLONED HUMAN 3H-[Dmt1]DALDA [Dmt1]DALDA 0.172 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
60554 GABAA CLONED HUMAN FNZ SH-I-048A 0.1723 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65496 nAChR CLONED HUMAN [3H] Flunitrazepam SH-I-048A 0.1723 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
27080 MOR BRAIN MOUSE 3H-DAMGO Dmt-d-Ala-Phe-Phe-NH2 0.173 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
97858 5-HT2A CELLS HUMAN [3H]-ketanserin MDL 100907 0.17378 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
27079 MOR BRAIN MOUSE 3H-[Dmt1]DALDA Dmt-d-Ala-Phe-Phe-NH2 0.174 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
23549 H3 CLONED RAT 3H-NAMH Clobenpropit 0.177828 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
99625 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthin 0.178 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
98274 KOR CEREBELLUM GUINEA PIG 3H-U69593 Nalfurafine 0.178 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
99632 A2A CLONED HUMAN 3H-NECA 8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine 0.179 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
7426 MOR CLONED HUMAN 3H-DAMGO CTOP 0.18 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
9224 SST2 CLONED MOUSE 125I-MK-678 MK 678 0.18 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
69386 H1 CLONED HUMAN 3H-PYRILAMINE CHLORPROMAZINE 0.18 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
5650 Alpha2C CELLS OK 3H-RAUWOLSCINE YOHIMBINE 0.18 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
53026 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan 0.18 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
55845 D3 UNDEFINED UNDEFINED UNDEFINED 1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 0.18 Butini S et al., 2009 Jan 15, 2025 Jan 15, 2025
60467 GABAA CLONED HUMAN FNZ XHE-II-024 0.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
22325 A1 BRAIN RAT 3H-DPCPX DPCPX 0.18 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
13369 D2 CLONED HUMAN 3H-thymidine LISURIDE 0.18 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
60733 GABAA CLONED HUMAN FNZ TG-4-29 0.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
10308 MOR CLONED HUMAN 3H-DAMGO ETORPHINE - HCI 0.18 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
60484 GABAA CLONED HUMAN FNZ QH-II-075 0.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
68677 DOR BRAIN RAT 3H-DPDPE DPI-3290 0.18 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
64582 D3 CLONED HUMAN 3H-SPIPERONE SSR181507 0.18 Claustre Y, et.al., 2003 Jan 15, 2025 Jan 15, 2025
10313 MOR CLONED HUMAN 3H-DAMGO Diprenorphine 0.18 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
9043 SST4 CLONED RAT 125I-CGP23996 BIM 23023 0.18 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
29012 SST2 CLONED HUMAN 125I-LTT-SST-28 Leu8, D-Trp22, Tyr25 SST-28 0.18 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
32606 D1 Striatal Membranes RAT 3H-SCH23390 NNC-112 0.18 Andersen PH, et al., 1992 Jan 15, 2025 Jan 15, 2025
8547 SST4 CLONED RAT 125I-Tyr11-SRIF SMS 201-995 0.18 O'Carroll AM, et al., 1993 Jan 15, 2025 Jan 15, 2025
29284 KOR Placenta Membranes HUMAN 3H-U69,593 Etorphine 0.18 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
65125 GABAA CLONED HUMAN [3H] Flunitrazepam TG-4-29 0.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
30568 NOP CLONED HUMAN 3H-Nociceptin Nociceptin 0.18 Valenzano KJ et. al., 2004 Jan 15, 2025 Jan 28, 2025
4969 5-HT2A CLONED RAT 3H-KETANSERIN METERGOLINE 0.18 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
14699 LUNG RABBIT 3H-PZ ATR 0.18 Bloom JW, et al., 1987 Jan 15, 2025 Jan 15, 2025
7806 GABAA CLONED HUMAN 3H-RO-15-1788 5 0.18 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
47743 Y1 CLONED RAT [125I] - Peptide YY PYY, zebrafish 0.18 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
8589 SST2 CLONED MOUSE 125I-Tyr11-SRIF MK 678 0.18 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
52629 CB1 UNDEFINED HUMAN UNDEFINED HU-210 0.18 Manera C et al., 2007 Jan 15, 2025 Jan 15, 2025
30363 KOR CLONED RAT 3H-Diprenorphine 17-Cyclopropylmethyl-6,7-didehydro-4,5-alpha-epoxy-5'-guanidinyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 0.18 Stevens WC, et al., 2000 Jan 15, 2025 Jan 15, 2025
63644 KOR CLONED HUMAN 3H-U69,593 GNTI 0.18 Thomas JB, et al., 2003 Jan 15, 2025 Jan 28, 2025
67487 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE YOHIMBINE 0.18 Song, Gang et., al. 2017 Jan 15, 2025 Jan 15, 2025
12707 DOR BE(2)-C HUMAN 3H-DPDPE DADLE 0.18 Standifer KM, et al., 1994 Jan 15, 2025 Jan 15, 2025
37541 D3 CLONED RAT 3H-SPIROPERIDOL N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indazole-3-carboxamide 0.18 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
9897 nAChR BRAIN RAT 3H-Epibatidine Cytisine-(-) 0.18 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
6827 Y4 CLONED HUMAN 125I-PYY PP, rat 0.18 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
7854 GABAA CLONED HUMAN 3H-RO-15-1788 20 0.18 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
30384 KOR CLONED HUMAN 3H-U69,593 5'-guanidinonaltrindole 0.18 Jones RM, et al., 2000 Jan 15, 2025 Jan 15, 2025
39860 AT2 Uterus PIG 125I-Angiotensin II Ang II Sar1 0.18 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
18869 KOR BRAIN GUINEA PIG 3H-U69,593 Cyclazocine 0.18 Bidlack JM et al., 2002 Jan 15, 2025 Jan 15, 2025
13495 CLONED OPOSSUM 3H-Yohimbine YOHIMBINE 0.18 Murphy TJ, et al., 1988 Jan 15, 2025 Jan 15, 2025
13504 CLONED OPOSSUM 3H-RAUWOLSCINE YOHIMBINE 0.18 Murphy TJ, et al., 1988 Jan 15, 2025 Jan 15, 2025
24773 H1 CLONED HUMAN 3H-PYRILAMINE CHLORPROMAZINE 0.18 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
65480 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-075 0.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
17614 CLONED RAT 125I-VIP Vasoactive intestinal polypeptide 0.18 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
47058 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S,25R)-DLAM-1P 0.18 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
65490 nAChR CLONED HUMAN [3H] Flunitrazepam XHE-II-024 0.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
34515 nAChR CLONED RAT 3H-Epibatidine Epibatidine-I,(+/-) 0.18 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
30677 DOR CLONED HUMAN 3H-Diprenorphine Leu-ENKEPHALIN 0.18 Lecoq I et. al., 2004 Jan 15, 2025 Jan 15, 2025
36057 MOR Membranes RAT 3H-DAMGO 14-Benzyloxymetopon 0.18 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
8666 SST5 CLONED RAT 125I-Tyr11-SRIF BIM 23023 0.18 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
36058 MOR Membranes RAT 3H-DAMGO 14-O-(1-naphthylmethyl)oxymorphone 0.18 Lattanzi R, et al., 2005 Jan 15, 2025 Jan 15, 2025
5087 5-HT2C CLONED HUMAN 3H-MESULERGINE METERGOLINE 0.18 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
47851 CLONED HUMAN 1251-CGRP h-alpha-CGRP 0.18 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
51947 MOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 0.18 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
87021 5-HT2A CEREBRAL CORTEX RAT 3H-KETANSERIN RISPERIDONE 0.18 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
68082 Y1 CLONED HUMAN [125I] - Peptide YY NPY, human 0.18 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
9727 MT2 CLONED HUMAN 125I-Iodomelatonin MELATONIN 0.18 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
50239 Y2 CLONED GUINEA PIG 125I-PYY NPY5-24, Ahx 0.181 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
32308 M3 Submandibular gland RAT 3H-NMS SCOPOLAMINE 0.18197 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
47260 Beta1 CEREBRAL CORTEX RAT 125I-ICYP Arotinolol 0.18197 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
98266 DOR BRAIN MOUSE 3H-DPDPE (E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide 0.182 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
61432 GABAA CLONED HUMAN FNZ SH-I-75 0.1825 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
85695 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide 0.183 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
21993 LHRH Pituitary RAT UNDEFINED 1 0.186209 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
32252 M1 CORTEX RAT 3H-PIRENZEPINE SCOPOLAMINE 0.186209 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
10753 D2 CLONED RAT 3H-LSD TRIFLUOPERAZINE 0.19 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
8198 SST5 CLONED HUMAN 125I-LTT-SST-28 somatostatin-28 0.19 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
29191 SST2 CLONED HUMAN UNDEFINED BIM 23197 0.19 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
24584 5-HT4 STRIATUM RAT 3H-GR-113808 BIMU 1 0.19 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
8969 SST2 CLONED HUMAN 125I-SRIF-28 Somatostatin-14 0.19 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
8971 SST2 CLONED HUMAN 125I-SRIF-28 somatostatin-28 0.19 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
7441 BB2 CLONED MOUSE 125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14) DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14) 0.19 Katsuno T, et al., 1999 Jan 15, 2025 Jan 15, 2025
9493 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.19 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
5920 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE SPIROXATRINE 0.19 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
9504 BRAIN Chick 125I-Iodomelatonin 5-MeOT-N-butanyl 0.19 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
53024 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan 0.19 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
6689 D2 ANTERIOR PITUITARY PIG 3H-NEMONAPRIDE SPIPERONE 0.19 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
53025 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-nitro)benzamido]morphinan 0.19 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
24101 5-HT2A CLONED HUMAN 3H-SPIPERONE RISPERIDONE 0.19 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
5422 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 GR 125487 0.19 Van den Wyngaert I, et al., 1997 Jan 15, 2025 Jan 15, 2025
15409 5-HT1B CLONED HUMAN 3H-5HT METHIOTHEPIN 0.19 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
8503 SST3 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.19 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
9015 SST5 CLONED HUMAN 125I-SRIF-28 SS-25 0.19 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
49467 KOR CLONED GUINEA PIG 3H-Diprenorphine [D-Ala8] Dyn A-(1-11)NH2 0.19 Bennet MA, et al., 2002 Jan 15, 2025 Jan 15, 2025
56125 KOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.19 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
25150 5-HT2A CLONED RAT 3H-KETANSERIN RISPERIDONE 0.19 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
5952 Alpha2C CELLS OK 3H-RAUWOLSCINE YOHIMBINE 0.19 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
63041 MC3 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Pro-DNal(2'Arg-Trp-Lys]-NH2 0.19 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
8519 SST3 CLONED HUMAN 125I-CGP23996 BIM 23052 0.19 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
37200 SLC6A4 BRAIN RAT 3H-5-HT Uptake SERTRALINE 0.19 Sanchez C, et al., 1999 Jan 15, 2025 Jan 15, 2025
41811 CLONED HUMAN 3H-Estradiol 1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.19 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
55891 MOR UNDEFINED HUMAN UNDEFINED Nalorphine 0.19 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
9045 SST4 CLONED RAT 125I-CGP23996 BIM 23034 0.19 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
16223 D2 CLONED MOUSE 3H-SPIPERONE PIMOZIDE 0.19 Neve KA, 1990 Jan 15, 2025 Jan 15, 2025
29281 MOR CEREBELLUM Gerbil 3H-DAMGO dihydroetorphine 0.19 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
33122 SLC6A4 BRAIN RAT UNDEFINED WY-45651 0.19 Muth, EA et al., 1986 Jan 15, 2025 Jan 15, 2025
55906 MOR UNDEFINED HUMAN UNDEFINED Naltrexone-6-beta-ol 0.19 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
41833 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitrothiazol-2-yl)amine 0.19 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
8812 SST5 CLONED HUMAN 125I-CGP23996 SRIF28-Leu8,D-Trp22,Tyr25 0.19 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
9838 BRAIN Chick 125I-Iodomelatonin 5-MeOT-N-butanyl 0.19 Teh MT, Sugden D, 1998 Jan 15, 2025 Jan 15, 2025
12911 CELLS OPOSSUM 3H-RX821002 RAUWOLSCINE 0.19 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
34927 CCR5 CLONED UNDEFINED 3H-Epibatidine 2-exo-(5-(6-Hydroxy-1-hexynyl)-3-pyridyl)-7-azabicyclo[2.2.1]heptane 0.19 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
51062 Alpha1A UNDEFINED HUMAN UNDEFINED Tamsulosin 0.19 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
2430 5-HT3 VAGUS NERVE RAT 3H-GR-65630 METOCLOPRAMIDE 0.19 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
8325 SST2 CLONED HUMAN 125I-LTT-SRIF28 LTT-SRIF28 0.19 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
68747 5-HT4 CAUDATE PIG 3H-GR-113808 GR 125487 0.19 Schiavi, GB et al., 1994 Jan 15, 2025 Jan 15, 2025
55952 KOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.19 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
53172 Alpha1A UNDEFINED HUMAN UNDEFINED Tamsulosin 0.19 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
55999 CB1 UNDEFINED HUMAN UNDEFINED Rimonabant 0.19 Griffith DA et al., 2009 Jan 15, 2025 Jan 15, 2025
2241 5-HT3 VAGUS NERVE RABBIT 3H-GR-65630 5-HT,2-Me 0.19 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
70090 5-HT3 CORTICAL MEMBRANES RAT 3H-GR-65630 0-[(2-Methyl-lH-imidazol-l-yl)methyl]-5,6,8,9,10,llhexahydro-4H-pyrido[3^,l-ji]carbazol-1l-oneHydrochloride 0.19 Van Wijingaarden, I. et, al. 1993 Jan 15, 2025 Jan 15, 2025
70091 5-HT3 CORTICAL MEMBRANES RAT 3H-GR-65630 l-(2,3-Dihydropyrrolo[l,2,3-de][l,4]benzothiazin-6-yl)-3-(5-methylimidazol-4-yl)propan-l-one Hydrochloride 0.19 Van Wijingaarden, I. et, al. 1993 Jan 15, 2025 Jan 15, 2025
49613 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 BIM 23197 0.19 Shimon I, et.al., 1997 Jan 15, 2025 Jan 15, 2025
11982 H3 CORTEX RAT 3H-NAMH GR 168320 0.19 Brown JD, et al., 1996 Jan 15, 2025 Jan 15, 2025
17618 CLONED RAT 125I-VIP VIP Ala8 0.19 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
47061 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-3P 0.19 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47062 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-2P 0.19 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
38369 D1 BRAIN RAT 3H-SCH23390 MCL-203 0.19 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
70118 5-HT3 CORTICAL MEMBRANES RAT 3H-GR-65630 cilansetron 0.19 Van Wijingaarden, I. et, al. 1993 Jan 15, 2025 Jan 15, 2025
9450 MT2 CLONED HUMAN 125I-Iodomelatonin MELATONIN 0.19 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
51946 MOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 0.19 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
2285 5-HT3 VAGUS NERVE RAT 3H-GR-65630 COCAINE 0.19 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
51437 Alpha1A UNDEFINED HUMAN UNDEFINED Tamsulosin 0.19 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
8433 SST5 CLONED HUMAN 125I-CGP23996 LTT-SRIF28 0.19 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
36088 COS-1 whole blood assay (WBA) HUMAN Functional Ketorolac tris salt 0.19 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
27044 MOR ILEUM GUINEA PIG 3H-DAMGO Tmt-D-Arg-Phe-Lys-NH2 0.192 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
99628 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthine 0.193 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
69255 H3 CORTEX RAT 3H-Alpha-Me-histamine GT 2331 0.194984 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
98251 MOR BRAIN MOUSE 3H-DAMGO N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide 0.197 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
68624 UT CLONED HUMAN I125-urotensin II H-P5U-Asp-C[Pen-Phe-Trp-Lys-Tyr-Cys]Val-OH 0.199526 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
35120 NOP CLONED HUMAN Functional OFQ/N 0.199526 Kapusta DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
97860 5-HT2A CELLS HUMAN [3H]-ketanserin ACP-103 0.199526 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
18779 M1 CLONED RAT 3H-PIRENZEPINE NMS,(-) 0.199526 Hulme EC et al., 1990 Jan 15, 2025 Jan 15, 2025
86619 5-HT4 CLONED HUMAN 3H-GR113808 N-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide 0.199526 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
39844 5-HT2B CLONED HUMAN 3H-MESULERGINE LY 266097 0.199526 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
66215 D2 STRIATUM RAT 3H-SPIPERONE methiothepine 0.199526 Campiani G, et al., 1998 Jan 15, 2025 Jan 28, 2025
31412 5-HT7 CLONED HUMAN 3H-5CT 5-CT 0.199526 Eglen RM et al., 1997 Jan 15, 2025 Jan 27, 2025
37056 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Rec 15/3079 0.199526 Corradetti R, et al., 2005 Jan 15, 2025 Jan 15, 2025
68814 SST2 CLONED HUMAN 125I-SRIF Somatostatin-14 0.199526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
31458 5-HT7 CLONED GUINEA PIG 3H-5CT 5-CT 0.199526 Eglen RM et al., 1997 Jan 15, 2025 Jan 27, 2025
68844 SST2 CLONED HUMAN 125I-SRIF L-363,301 HyPro 0.199526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
50156 SST2 CLONED HUMAN 125I-SOMATOSTATIN 14 Somatostatin-14 0.199526 Weckbecker G, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68848 SST1 CLONED HUMAN 125I-SRIF H-Ala-Ala-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 0.199526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
68851 SST4 CLONED HUMAN 125I-SRIF H-Ala-Ala-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 0.199526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
68861 SST4 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Ala-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 0.199526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
3329 D3 CLONED HUMAN 3H-YM 09151-2 SPIPERONE 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
3331 D3 CLONED HUMAN 3H-YM 09151-2 YM-09151-2 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
9732 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl 0.2 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
19206 SLC6A4 Platelets HUMAN 3H-5HT LY248686 0.2 Wong DT et al., 1993 Jan 15, 2025 Jan 15, 2025
12039 H3 Striatal Membranes RAT 125I-Iodoproxyfan Iodoproxyfan 0.2 Ligneau X, et al., 1994 Jan 15, 2025 Jan 15, 2025
98056 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3-dimethylbutanamide 0.2 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
48649 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
27147 5-HT2A BRAIN RAT 125I-DOI 1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride 0.2 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
51723 NR3C1 UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline 0.2 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
59148 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.2 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
27149 5-HT2A BRAIN RAT 125I-DOI AL-37350A 0.2 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
4110 KOR CLONED HUMAN 3H-U69,593 U50,488H 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
24592 D1 STRIATUM RAT 3H-SCH23390 SCH 23390 0.2 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
29200 SST2 CLONED HUMAN UNDEFINED somatostatin-28 0.2 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
31760 5-HT2C CORTEX HUMAN 3H-MESULERGINE ORG-5222 0.2 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
4113 KOR CLONED HUMAN 3H-U69,593 ETORPHINE - HCI 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
24593 D2 STRIATUM RAT 3H-SPIROPERIDOL HALOPERIDOL 0.2 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
29201 SST2 CLONED HUMAN UNDEFINED Somatostatin-14 0.2 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
4115 KOR CLONED HUMAN 3H-U69,593 NOR-BNI (HCI)2 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
19475 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH Salmon MCH 0.2 Sailer AW et al., 2001 Jan 15, 2025 Jan 15, 2025
4116 KOR CLONED HUMAN 3H-U69,593 DYNORPHIN(1-8)-OH 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
4117 KOR CLONED HUMAN 3H-U69,593 DYNORPHIN(1-11)-OH 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
29205 SST3 CLONED HUMAN UNDEFINED rCST-29 0.2 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
24086 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.2 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
9495 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Chloro 0.2 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
100632 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.2 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
64537 CLONED HUMAN 3H-Estradiol 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoic Acid 0.2 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
55579 MOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.2 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
4124 KOR CLONED HUMAN 3H-U69,593 WIN 44,441(-) 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
1054 5-HT2C Choroid Plexus RAT 3H-MIANSERIN RITANSERIN 0.2 Sanders-Bush E, Breeding M., 1988 Jan 15, 2025 Jan 15, 2025
71199 5-HT1A CLONED HUMAN WAY100635 FEMPT 0.2 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
54815 D3 UNDEFINED HUMAN UNDEFINED Biphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 0.2 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
2336 5-HT3 CORTEX RAT 3H-LY 278584 ICS 205-930 0.2 WONG ET AL., 1989 Jan 15, 2025 Jan 15, 2025
14881 5-HT2A CLONED RAT UNDEFINED SERTINDOLE 0.2 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
30756 5-HT2A CLONED HUMAN 3H-KETANSERIN AC-90179 0.2 Vanover, KE et.al., 2004 Jan 15, 2025 Jan 15, 2025
53286 CHRNA4 UNDEFINED RAT UNDEFINED rac-3'-(3-fluorophenyl)deschloroepibatidine dihydrochloride 0.2 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
11047 H3 CLONED RAT 3H-methylhistamine Imetit 0.2 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
4137 KOR BRAIN GUINEA PIG 3H-U69,593 U50,488H 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
17962 CCK2 BRAIN RAT 125I-CCK-8 15d 0.2 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
100907 AChE BRAIN HUMAN Functional N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-2-(1H-indol-3-yl)acetamide 0.2 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
23596 Spinal cord RAT 125I-1DMe-Y8Fa 1DMe-Y8Fa 0.2 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
34349 nAChR CORTEX RAT 3H-NICOTINE Cytisine-(-) 0.2 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 15, 2025
42800 CLONED HUMAN 125I-ghrelin 6-[(Benzyloxy)methyl]-5-{4-[(4-nitrobenzyl)amino]phenyl}pyrimidine-2,4-diamine 0.2 Serby MD, et al., 2006 Jan 15, 2025 Jan 15, 2025
85554 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate 0.2 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
35890 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 7-Hydroxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
48690 GNRHR CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
20531 A1 myocardial membranes BOVINE 125I-HPIA XAC 0.2 Lohse MJ et al., 1987 Jan 15, 2025 Jan 15, 2025
37171 Y5 BRAIN RAT 125I-hPP PP, human 0.2 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
29236 SST5 CLONED HUMAN UNDEFINED Somatostatin-14 0.2 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
14389 gastrointestinal tract RAT 125I-BH Substance P Substance P 0.2 Burcher E, et al., 1986 Jan 15, 2025 Jan 15, 2025
85558 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate 0.2 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
6711 D4 CLONED HUMAN 3H-SPIPERONE NEMONAPRIDE 0.2 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
37175 Y5 BRAIN RAT 125I-hPP NPY [hPP(1-17), Ala31,Aib32], human 0.2 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
4152 KOR BRAIN GUINEA PIG 3H-U69,593 WIN 44,441(-) 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
57400 CB1 UNDEFINED HUMAN UNDEFINED N-Cyclohexyl-4-[(2,4-dichlorophenyl)(phenyl)methyl]-piperazine-1-carbothioamide 0.2 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
35897 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7-[2-(2-Ethoxyethoxy)ethoxy]-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
60473 GABAA CLONED HUMAN FNZ PWZ-007A 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
24125 VPAC1 CLONED HUMAN 125I-VIP Vasoactive intestinal polypeptide 0.2 Igarashi H, et al., 2002 Jan 15, 2025 Jan 15, 2025
35906 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Acetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
85572 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate 0.2 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
3397 MOR CLONED HUMAN 3H-DAMGO ETONITAZENE 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
35909 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
23366 A1 BRAIN RABBIT 3H-DPCPX CCPA 0.2 Klotz KN et al., 1991 Jan 15, 2025 Jan 27, 2025
42567 Alpha1A CLONED UNDEFINED UNDEFINED PRAZOSIN 0.2 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
35912 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Methoxyacetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
60491 GABAA CLONED HUMAN FNZ PZII-028 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60492 GABAA CLONED HUMAN FNZ PZII-028 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
81997 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-fluoroethyl)-cyclopropyl]pyridine trifluoroacetate 0.2 Zhang HK et al 2012 Jan 15, 2025 Jan 29, 2025
4176 5-HT1B CLONED HUMAN 3H-5HT METHIOTHEPIN 0.2 HAMBLIN MW, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
55632 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(6-Chloro-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Hydrochloride 0.2 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
29268 MOR BRAIN RAT 3H-DAMGO 14-phenylpropoxymetopon 0.2 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
10069 MOR BRAIN MOUSE 125I-Endomorphin-1 NALBzoH 0.2 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
38747 CLONED RAT 3H-dexamethasone (5-(4-(((2,4-Difluorobenzyl)(2-methyl-3-((methylsulfonyl)amino)phenyl)amino)methyl)phenoxy)-2-fluorophenoxy)acetic Acid 0.2 Link JT, et al., 2005 Jan 15, 2025 Jan 15, 2025
39004 D2 CLONED HUMAN R-SAT FLUSPIRILENE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
55900 MOR UNDEFINED HUMAN UNDEFINED Phenazocine 0.2 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
39006 D2 CLONED HUMAN R-SAT PROCHLORPERAZINE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
51551 Alpha1D UNDEFINED HUMAN UNDEFINED Tamsulosin 0.2 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
39008 D2 CLONED HUMAN R-SAT TRIFLUORPERIDOL 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39009 D2 CLONED HUMAN R-SAT FLUPENTHIXOL, Alpha 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
29282 DOR FOREBRAIN GUINEA PIG 3H-DPDPE-Cl dihydroetorphine 0.2 Schutz J, et al., 2003 Jan 15, 2025 Jan 15, 2025
39014 D2 CLONED HUMAN R-SAT FLUPHENAZINE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
40553 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine 0.2 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
60521 GABAA CLONED HUMAN FNZ Bretazenil 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
18796 M1 CLONED HUMAN 3H-NMS MT-7 0.2 Adem A and Karlsson E. 1997 Jan 15, 2025 Jan 15, 2025
19309 5-HT1A CLONED HUMAN 35S-GTPGammaS Rec 15/3079 0.2 Leonardi A et al., 2001 Jan 15, 2025 Jan 15, 2025
39028 D2 CLONED HUMAN R-SAT sulforidazine 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39030 D2 CLONED HUMAN R-SAT THIOTHIXENE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
31863 M1 CLONED HUMAN 3H-QNB ATR 0.2 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
39032 D2 CLONED HUMAN R-SAT OCTOCLOTHEPIN 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
3705 MOR BRAIN GUINEA PIG 3H-DAMGO DIPRENORPHINE-HCl 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
31865 M3 CLONED HUMAN 3H-QNB ATR 0.2 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
39035 D2 CLONED HUMAN R-SAT FLUSPIRILENE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
3708 KOR CLONED HUMAN 3H-U69,593 DIPRENORPHINE-HCl 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18556 CCK1 PANCREAS RAT 125I-BH-CCK-8 5 0.2 Pierson ME et al., 1997 Jan 15, 2025 Jan 15, 2025
18045 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 CCK-8 0.2 Pendley CE et al., 1995 Jan 15, 2025 Jan 15, 2025
85629 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 0.2 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
97664 SST4 CLONED HUMAN Functional L-803,087 0.2 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
7814 GABAA CLONED HUMAN 3H-RO-15-1788 13 0.2 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
4492 D2 BRAIN RAT 3H-SPIPERONE TRIFLUOPERAZINE 0.2 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
3726 MOR CLONED HUMAN 3H-DAMGO NALTREXONE-HCl 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
100755 PDE4a CLONED HUMAN Functional Roflumilast 0.2 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
3988 5-HT4 CLONED MOUSE 3H-GR-113808 GR 113808 0.2 CLAEYSEN S, ET AL., 1996 Jan 15, 2025 Jan 27, 2025
85653 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 0.2 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
34199 D2 Striatal Membranes RAT 125I-IABN DOMPERIDONE 0.2 Luedtke RR, et al., 2000 Jan 15, 2025 Jan 27, 2025
3736 KOR CLONED HUMAN 3H-U69,593 b-FNA-HCl 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
63643 KOR CLONED HUMAN 3H-U69,593 Nor-BNI 0.2 Thomas JB, et al., 2003 Jan 15, 2025 Jan 28, 2025
26271 5-HT1B CLONED HUMAN 3H-5HT 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-o-xylylpiperazin-1-yl)ethanone 0.2 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
39075 D3 CLONED HUMAN R-SAT SPIPERONE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
5797 Alpha2A CELLS HT29 3H-RAUWOLSCINE RX 811033 0.2 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
8869 GABAA CLONED HUMAN 3H-15-4513 Abecarnil 0.2 Scholze P, et al., 1996 Jan 15, 2025 Jan 27, 2025
39077 D3 CLONED HUMAN R-SAT PIMOZIDE 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
70054 D3 CLONED HUMAN 3H-SPIPERONE (S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)5,6,7,8-tetrahydronaphthalen-1-ol 0.2 Ghosh, B. et, al 2010 Jan 15, 2025 Jan 28, 2025
4775 5-HT1A test test 3H-DPAT NN-DIPROP-5-CT 0.2 HAMON M, ET AL., 1990 Jan 15, 2025 Jan 15, 2025
3753 MOR CLONED HUMAN 3H-DAMGO BREMAZOCINE(-) 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
17577 CLONED HUMAN 125I-VIP Vasoactive intestinal polypeptide 0.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
23978 D3 CLONED HUMAN 3H-SPIPERONE FLUPHENAZINE 0.2 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
35754 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
65451 nAChR CLONED HUMAN [3H] Flunitrazepam PWZ-007A 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
11693 D2 CLONED HUMAN 125I-IODOSULPRIDE Pipotiazine 0.2 Sokoloff P, et al., 1992 Jan 15, 2025 Jan 15, 2025
32943 SST2 CLONED HUMAN 125I-Tyr11-SRIF Somatostatin-14 0.2 Ankersen M, et. al.,1998 Jan 15, 2025 Jan 15, 2025
43185 STK4 CLONED HUMAN 3H-Staurosporine Staurosporine 0.2 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39859 AT2 Uterus PIG 125I-Angiotensin II Angiotensin II 0.2 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
4789 5-HT1A test test 3H-DPAT S 20499 0.2 HAMON M, ET AL., 1990 Jan 15, 2025 Jan 15, 2025
4790 5-HT1A test test 3H-DPAT 5-CT 0.2 HAMON M, ET AL., 1990 Jan 15, 2025 Jan 15, 2025
51127 Alpha1D UNDEFINED HUMAN UNDEFINED Tamsulosin 0.2 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
47803 MOR CLONED HUMAN 3H-DAMGO MCL-145 0.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
66237 Ghrelin CLONED HUMAN 125I-ghrelin 6-[(Benzyloxy)methyl]-5-{4-[(4-nitrobenzyl)amino]phenyl}pyrimidine-2,4-diamine 0.2 Serby MD, et al., 2006 Jan 15, 2025 Jan 15, 2025
3773 MOR BRAIN GUINEA PIG 3H-DAMGO NALTRINDOLE 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11968 H2 CORTICAL MEMBRANES GUINEA PIG 3H-Histamine Alpha-Dimethylhistane-alpha 0.2 Hill JA., 1992 Jan 15, 2025 Jan 15, 2025
39104 D3 CLONED HUMAN R-SAT BROMPERIDOL 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
11969 H2 CORTICAL MEMBRANES GUINEA PIG 3H-Histamine S-Beta-Dimethylhistamine-R-alpha 0.2 Hill JA., 1992 Jan 15, 2025 Jan 15, 2025
65473 nAChR CLONED HUMAN [3H] Flunitrazepam Bretazenil 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
39108 D3 CLONED HUMAN R-SAT HALOPERIDOL 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
65476 GABAA CLONED HUMAN [3H] Flunitrazepam PZII-028 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65477 nAChR CLONED HUMAN [3H] Flunitrazepam PZII-028 0.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
48070 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
7882 GABAA CLONED HUMAN 3H-RO-15-1788 13 0.2 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
48074 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
15051 gastrointestinal tract GUINEA PIG 125I-BH Substance P Substance P 0.2 Burcher E, et al., 1986 Jan 15, 2025 Jan 15, 2025
48075 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
3789 MOR BRAIN GUINEA PIG 3H-DAMGO NALBzoH 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
48593 CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48595 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
62677 SST5 Ovary HAMSTER UNKNOWN Somatostatin-14 0.2 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
4055 DOR CLONED HUMAN 3H-DPDPE-Cl NALTRINDOLE 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
39134 D3 CLONED HUMAN R-SAT OCTOCLOTHEPIN 0.2 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
19169 NB-OK-1 HUMAN 125I-PACAP(1-27) PACAP 0.2 Gourlet P et al., 1991 Jan 15, 2025 Jan 15, 2025
51937 MOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.2 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
48866 KOR BRAIN RAT 3H-EKC CAM 0.2 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
8932 SST1 CLONED RAT 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
13797 NK1 CLONED HUMAN 125I-Bolton Hunter Substance P 0.2 Kudlacz EM, et al., 1996 Jan 15, 2025 Jan 15, 2025
16613 Y1 CLONED HUMAN [125I] - Peptide YY Des-AA10-17[Cys7,21, Pro34]-NPY 0.2 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
17637 CLONED RAT 125I-VIP VIP Ala28 0.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
53222 Alpha1D UNDEFINED HUMAN UNDEFINED Tamsulosin 0.2 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
4583 5-HT2A BRAIN RAT 3H-KETANSERIN RISPERIDONE 0.2 ROTH BL, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
16615 Y1 CLONED HUMAN [125I] - Peptide YY Des-AA11-18[Cys7,21,D-Lys9 (Ac), Pro34]-NPY 0.2 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
29160 SST4 CLONED HUMAN 125I-Tyr11-SRIF SMS 201-995 0.2 Reisine T, et.al., 1995 Jan 15, 2025 Jan 15, 2025
63976 5-HT6 CLONED HUMAN 3H-LSD N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-5-chloronaphthalene-2-sulfonamide 0.2 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
8937 SST2 CLONED RAT 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
8938 SST2 CLONED RAT 125I-Tyr11-somatostatin-14 H2N-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2 0.2 Bass RT, et al, 1996 Jan 15, 2025 Jan 15, 2025
48618 GNRHR CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
7916 GABAA CLONED HUMAN 3H-RO-15-1788 12 0.2 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
69361 D3 CLONED RAT 3H-NMSP FLUPHENAZINE 0.2 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
35828 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.2 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
48630 CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
51192 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-chloro-3-pyridinyl)-5,5-dimethyl-2,5-diazabicyclo-[2.2.1]heptanium iodide 0.2 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
69372 5-HT2A CLONED HUMAN 125I-DOI RISPERIDONE 0.2 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
17151 5-HT2A BRAIN HUMAN 3H-KETANSERIN ILOPERIDONE 0.2 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
100607 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.2 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
50234 Y2 CLONED GUINEA PIG 125I-PYY NPY13-36, porcine 0.201 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
98283 KOR CEREBELLUM GUINEA PIG 3H-U69593 (E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide 0.204 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
64939 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.205 Ishibashi, Tadashi. et. al, 2010 Jan 15, 2025 Jan 15, 2025
22008 LHRH Pituitary RAT UNDEFINED 16 0.20893 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
99634 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine 0.209 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
24072 5-HT2A CLONED HUMAN UNDEFINED RISPERIDONE 0.21 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
54807 D3 UNDEFINED HUMAN UNDEFINED N-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide 0.21 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
53022 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan 0.21 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
53023 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan 0.21 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
8485 SST3 CLONED HUMAN 125I-Tyr10-CST14 Somatostatin-14 0.21 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
93989 D3 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 0.21 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
16166 D2 CLONED RAT 125I-IODOSULPRIDE Thioproperazine 0.21 Sokoloff P, et al., 1990 Jan 15, 2025 Jan 15, 2025
53289 CHRNA4 UNDEFINED RAT UNDEFINED 3-(4-chlorophenyl)deschloroepibatidine 0.21 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
32814 D2 CLONED RAT 3H-SPIPERONE Thioproperazine 0.21 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
8751 SST2 CORTEX HUMAN 125I-Tyr3-octreotide somatostatin-28 0.21 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
17968 CCK2 BRAIN RAT 125I-CCK-8 14h 0.21 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
22326 A1 BRAIN RABBIT 3H-DPCPX DPCPX 0.21 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
54070 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-quinolyl)acetamido]morphinan 0.21 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
20284 HEART RAT 3H-Nitrendipine NITRENDIPINE 0.21 Ehlert FJ et al., 1982 Jan 15, 2025 Jan 15, 2025
8765 SST2 CLONED HUMAN 125I-Tyr3-octreotide BIM 23014 0.21 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
63044 MC3 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Hyp-DNal(2')Arg-Trp-Lys]-NH2 0.21 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
60485 GABAA CLONED HUMAN FNZ QH-II-075 0.21 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60493 GABAA CLONED HUMAN FNZ CGS9895 0.21 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
55889 MOR UNDEFINED HUMAN UNDEFINED BUPRENORPHINE 0.21 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
19795 5-HT2A CORTEX RAT UNDEFINED RISPERIDONE 0.21 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
10839 D3 CLONED HUMAN 125I-IODOSULPRIDE R(-)NPA 0.21 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
16225 D2 CLONED MOUSE 3H-SPIPERONE BUTACLAMOL,(+) 0.21 Neve KA, 1990 Jan 15, 2025 Jan 15, 2025
33123 SLC6A4 BRAIN RAT UNDEFINED WY-45030 0.21 Muth, EA et al., 1986 Jan 15, 2025 Jan 15, 2025
55908 MOR UNDEFINED HUMAN UNDEFINED Naltrexone-6-alpha-ol 0.21 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
5993 M4 LUNG PORCINE 3H-QNB SCOPOLAMINE 0.21 CHELALA JL, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
29304 AT1 CLONED RAT 125I-Angiotensin II Angiotensin II 0.21 Inada Y, et al., 2002 Jan 15, 2025 Jan 28, 2025
124 5-HT1A CORTEX PIG 3H-8-OH-DPAT 5-CT 0.21 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
43396 PDGFRB CLONED HUMAN 3H-Staurosporine SU11248 0.21 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
36752 5-HT2C CLONED HUMAN 3H-MESULERGINE (-)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 0.21 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
14228 D2 CLONED RAT 3H-Methylspiperone DM 1451 0.21 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 27, 2025
7317 PTH1 CLONED HUMAN 125I-[Nle8,18,Tyr34]bPTH(3-34) High hPTH(1-34) 0.21 Hoare SR, et al., 1999 Jan 15, 2025 Jan 15, 2025
14230 D2 CLONED RAT 3H-Methylspiperone SULPIRIDE 0.21 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 27, 2025
65944 GABAA CLONED HUMAN [3H] Flunitrazepam CGS9895 0.21 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7841 GABAA CLONED HUMAN 3H-RO-15-1788 5 0.21 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
30629 5-HT3 CLONED MOUSE 3H-GRANISETRON GR 65630 0.21 Green, T et. al., 1995 Jan 15, 2025 Jan 15, 2025
100262 5-HT2B CLONED HUMAN 3H-LSD Asenapine 0.21 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
10664 M1 CEREBRAL CORTEX RAT 3H-NMS ATR 0.21 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
47789 MOR CLONED HUMAN 3H-DAMGO Levorphanol 0.21 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
31150 NK3 CLONED HUMAN 125I-Iodohistidyl [MePhe7]NKB SR 142801 0.21 Oury-Donat F, et.al.,1995 Jan 15, 2025 Jan 15, 2025
37555 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[2-[4-(1-Naphthalenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.21 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
70842 5-HT2A test test 3H- Ketanserin 2-(4-bromo-2,5-dimethoxyphenyl)ethanamine 0.21 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
31166 NK3 CLONED HUMAN 125I-Iodohistidyl [MePhe7]NKB SR 142801 0.21 Emonds-Alt X., et.al., 1995 Jan 15, 2025 Jan 15, 2025
9415 MT1 CLONED HUMAN 125I-Mel Melatonin,2-Phenyl 0.21 Reppert, Godson, Mahle, Weaver, Slaugenhaupt, 1995 Jan 15, 2025 Jan 15, 2025
10696 M5 CLONED HUMAN 3H-NMS ATR 0.21 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
65481 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-075 0.21 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
34519 nAChR CLONED RAT 3H-Epibatidine A-85380 0.21 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
32744 5-HT2C CLONED RAT 3H-MESULERGINE 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+/-) 0.21 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
38124 CLONED RAT 3H-dexamethasone C56H80NO8 0.21 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
16366 Y2 jejunal crypt cells RAT [125I] - Peptide YY PYY, N-alpha-Ac, 25-36 0.21 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
6128 Alpha1C CLONED HUMAN 125I-HEAT PRAZOSIN 0.21 HIRASAWA A, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
34376 MOR FOREBRAIN RAT 3H-DAMGO Levallorphan 0.213 Codd EE et al, 1995 Jan 15, 2025 Jan 15, 2025
48907 Y1 CLONED Chicken [125I] - Peptide YY NPY, porcine 0.213796 Holmberg, SK et al., 2002 Jan 15, 2025 Jan 15, 2025
48925 Y5 CLONED Chicken [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.213796 Holmberg, SK et al., 2002 Jan 15, 2025 Jan 15, 2025
28760 SST3 CLONED HUMAN 125I-Tyr10-CST14 Somatostatin-14 0.213796 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
32356 M4 HEART Chick 3H-NMS Ipratropium 0.213796 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
30362 KOR CLONED RAT 3H-Diprenorphine 5'-Amidinomethyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 0.214 Stevens WC, et al., 2000 Jan 15, 2025 Jan 15, 2025
32000 D2 BRAIN RAT 3H-SPIPERONE Spectramide 0.215 Sanchez-Roa, P.M., et al., 1989 Jan 15, 2025 Jan 15, 2025
54584 A2B UNDEFINED HUMAN UNDEFINED 8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1-ethyl-1H-purine-2,6(3H,7H)-dione 0.215 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
87923 A2B test HUMAN 3H-PSB-603 8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.215 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
8454 SST5 CLONED HUMAN 125I-Tyr3-octreotide CST14-Tyr10 0.22 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
63494 5-HT2A CLONED HUMAN 3H-Ketaserin RISPERIDONE 0.22 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
8468 SST3 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 0.22 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
48662 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.22 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
9500 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Chloro 0.22 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
8777 SST5 CLONED HUMAN 125I-Tyr3-octreotide Tyr10-cortistatin 0.22 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
37714 DOR CLONED HUMAN 3H-Diprenorphine HS595 0.22 Tryoen-Toth P, et al., 2005 Jan 15, 2025 Jan 15, 2025
26976 PKCα CLONED HUMAN 3H-PDBU Thymeleatoxin (low PS) 0.22 Wang QJ, et.al.,2003 Jan 15, 2025 Jan 28, 2025
23403 MOR CLONED HUMAN 3H-DAMGO Cyclazocine 0.22 Gharagozlou P, et al., 2003 Jan 15, 2025 Jan 15, 2025
6271 5-HT7 CLONED GUINEA PIG 3H-5CT 5-CT 0.22 TO ZP, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
41859 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(2-nitrophenyl)amine 0.22 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
6533 5-HT7B CLONED HUMAN 3H-5CT 5-CT 0.22 JASPER JR,ET AL., Jan 15, 2025 Jan 15, 2025
17546 CLONED HUMAN 125I-VIP VIP Ala11 0.22 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
55960 KOR UNDEFINED HUMAN UNDEFINED Butorphanol 0.22 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
14252 D2 CLONED RAT 3H-SPIPERONE ETICLOPRIDE 0.22 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 27, 2025
93616 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 0.22 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
51382 M3 UNDEFINED HUMAN UNDEFINED 7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 0.22 Sonda S et al., 2007 Jan 15, 2025 Jan 15, 2025
8655 SST5 CLONED RAT 125I-Tyr11-SRIF somatostatin-28 0.22 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
36580 5-HT2A FR. CORTEX RAT 3H-KETANSERIN 9-OH-risperidone 0.22 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
51941 MOR UNDEFINED HUMAN UNDEFINED 1'-(o-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 0.22 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
21482 nAChR CLONED Xenopus 3H-Epibatidine NBEP 0.22 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
68075 Y1 CLONED Rhesus Monkey [125I] - Peptide YY PYY, human 0.22 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
38123 CLONED RAT 3H-dexamethasone C55H78NO7 0.22 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
38127 CLONED RAT 3H-dexamethasone C54H76NO5 0.22 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
8696 SST5 CLONED HUMAN 125I-Tyr3-octreotide Tyr10-cortistatin 0.22 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
48633 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 0.22 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
9725 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.22 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
99582 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine 0.22 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
27045 MOR ILEUM GUINEA PIG 3H-DAMGO H-Mmt-D-Arg-Phe-Lys-NH2 0.222 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
55675 AChE UNDEFINED HUMAN UNDEFINED N-{4-[(1,2,3,4-Tetrahydroacridin-9-yl)amino]butyl}-N{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}acetamide 0.223 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
28763 SST3 CLONED HUMAN 125I-LTT-SRIF28 somatostatin-28 0.223872 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
32369 M4 LUNG RABBIT 3H-NMS SCOPOLAMINE 0.223872 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
23546 H3 BRAIN CORTEX GUINEA PIG 3H-NAMH Clobenpropit 0.223872 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
30360 KOR CLONED RAT 3H-Diprenorphine Nor-BNI 0.224 Stevens WC, et al., 2000 Jan 15, 2025 Jan 15, 2025
23719 MC3 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH alpha-MSH, [Nle4, D-Phe7] 0.224 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
22499 MC3 CLONED HUMAN 125I-NDP-MSH NDP-MSH 0.224 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
99635 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 0.226 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
30365 KOR CLONED RAT 3H-Diprenorphine 5'-N-Biguanidino-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 0.226 Stevens WC, et al., 2000 Jan 15, 2025 Jan 15, 2025
86799 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide 0.228 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
54137 TRPV1 UNDEFINED RAT UNDEFINED [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1,10}.0^{2,6}.0^{11,15}]octadeca-3,8-dien-8-yl]methyl 2-(4-methanesulfonamido-3-methoxyphenyl)acetate 0.228 Choi HK et al., 2009 Jan 15, 2025 Jan 15, 2025
98250 MOR BRAIN MOUSE 3H-DAMGO N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide 0.229 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
48921 Y5 CLONED Chicken [125I] - Peptide YY NPY, porcine 0.229087 Holmberg, SK et al., 2002 Jan 15, 2025 Jan 15, 2025
9730 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6,7 di-cl-2-Me 0.23 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
11522 CORTEX RAT 3H-Nitrendipine NIFEDIPINE 0.23 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
50947 MOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.23 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
7429 MOR CLONED HUMAN 3H-DAMGO ETORPHINE - HCI 0.23 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
62730 SST2 COLON RAT UNKNOWN Somatostatin-14 0.23 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
69389 H1 CLONED HUMAN 3H-PYRILAMINE CLOZAPINE 0.23 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
65822 GABAA CLONED HUMAN [3H] Flunitrazepam CM-D45 C19H21N3O4 0.23 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7202 NK2 CLONED HUMAN 125I-[MePhe7]-NKB SR 48968 0.23 Sarau HM, et al., 1997 Jan 15, 2025 Jan 15, 2025
22327 A1 BRAIN PIG 3H-DPCPX DPCPX 0.23 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
57402 CB1 UNDEFINED HUMAN UNDEFINED 4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-cyclohexylpiperazine-1-carboxamide 0.23 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
8768 SST2 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 0.23 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
63045 MC4 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Hyp-DNal(2')Arg-Trp-Lys]-NH2 0.23 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
9030 SST4 CLONED RAT 125I-CGP23996 somatostatin-28 0.23 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
23368 A1 BRAIN RAT 3H-DPCPX CCPA 0.23 Klotz KN et al., 1991 Jan 15, 2025 Jan 27, 2025
101193 MOR CLONED HUMAN 3H-Diprenorphine (S)-1-((3-((3,4-Dihydroisoquinolin-2(1H)-yl)methyl)benzyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate 0.23 Henry S,et al., 2021 Jan 15, 2025 Jan 28, 2025
35148 5-HT2A CORTEX RAT 3H-KETANSERIN OCTOCLOTHEPIN 0.23 Campiani G, et al., 2002 Jan 15, 2025 Jan 15, 2025
56142 KOR UNDEFINED HUMAN UNDEFINED CCDC 710249, HCl salt 0.23 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
9807 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl 0.23 Nonno,Pannacci,Lucini, Angeloni,Fraschini,Stankov Jan 15, 2025 Jan 15, 2025
29009 SST4 CLONED HUMAN 125I-LTT-SST-28 D-Trp8 SST-14 0.23 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
13394 D3 CLONED HUMAN 3H-thymidine Pramipexole 0.23 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
60499 GABAA CLONED HUMAN FNZ PWZ-0071 0.23 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
23382 NK1 ILEUM GUINEA PIG 125I-Bolton Hunter SSR240600 0.23 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
49500 KOR CLONED HUMAN 3H-Diprenorphine Dynorphin A(1-13)-OH 0.23 Schlechtingen, G et al., 2003 Jan 15, 2025 Jan 15, 2025
63068 MC3 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-His-DNal(2')Arg-Trp-Lys]-NH2 0.23 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
30049 SST2 CLONED MOUSE 125I-SOMATOSTATIN Somatostatin-14 0.23 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
7266 V1B Pituitary RAT 3H-AVP AVP 0.23 Tahara A, et al., 1997 Jan 15, 2025 Jan 15, 2025
40546 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.23 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
9831 CLONED HUMAN 125I-Iodomelatonin MELATONIN 0.23 Reppert SM, Weaver DR, Ebisawa, 1994 Jan 15, 2025 Jan 15, 2025
12409 D3 CLONED RAT 125I-NCQ 298 ETICLOPRIDE 0.23 Boundy VA, et al., 1993 Jan 15, 2025 Jan 15, 2025
56954 KOR UNDEFINED UNDEFINED UNDEFINED 4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-yl]benzamide; oxalic acid 0.23 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
15233 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IPSAPIRONE 0.23 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
34951 nAChR CLONED UNDEFINED 3H-Epibatidine 2-exo-(5-(6-Hydroxy-1-hexynyl)-3-pyridyl)-7-azabicyclo[2.2.1]heptane 0.23 Wei ZL, et al., 2005 Jan 15, 2025 Jan 27, 2025
7817 GABAA CLONED HUMAN 3H-RO-15-1788 16 0.23 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8347 SST2 CLONED HUMAN 125I-Tyr10-CST14 seglitide 0.23 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
23967 D3 CLONED HUMAN 3H-RACLOPRIDE PERPHENAZINE 0.23 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
48799 D3 CLONED HUMAN 3H-SPIPERONE N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide 0.23 Bettinetti L, et al., 2002 Jan 15, 2025 Jan 15, 2025
49573 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.23 Shimon I, et.al., 1997 Jan 15, 2025 Jan 15, 2025
9126 SST1 CLONED HUMAN 125I-CGP23996 SRIF-D-Trp8 0.23 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
10918 D4 CLONED HUMAN 3H-SPIPERONE QUINPIROLE 0.23 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
47788 MOR CLONED HUMAN 3H-DAMGO MCL-101 0.23 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
10419 nAChR CLONED RAT 125I-Alpha-bgt Bungarotoxin,Alpha 0.23 Quik M, Choremis, Komourian, Lukas, Puchacz, 1996 Jan 15, 2025 Jan 27, 2025
47796 MOR CLONED HUMAN 3H-DAMGO MCL-176 0.23 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
65462 GABAA CLONED HUMAN [3H] Flunitrazepam PWZ-0071 0.23 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7358 DOR CLONED HUMAN 3H-Naltrindole DIPRENORPHINE-HCl 0.23 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
9408 MT2 CLONED HUMAN 125I-Mel S 20098 0.23 Reppert, Godson, Mahle, Weaver, Slaugenhaupt, 1995 Jan 15, 2025 Jan 15, 2025
30401 MOR thalamus CALF 3H-DADL DIHYDROMORPHINE 0.23 Gilbert AK et al., 2004 Jan 15, 2025 Jan 15, 2025
53955 D3 UNDEFINED HUMAN UNDEFINED N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide 0.23 Leopoldo M et al., 2009 Jan 15, 2025 Jan 15, 2025
43473 KDR CLONED HUMAN 3H-Staurosporine SU11248 0.23 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
61396 GABAA CLONED HUMAN FNZ CM-D45 0.23 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
17878 CCK1 Gallbladder GUINEA PIG 125I-CCK-8 CCK-8 0.23 Ito H et al., 1993 Jan 15, 2025 Jan 15, 2025
11482 H1 CLONED HUMAN 3H-PYRILAMINE CLOZAPINE 0.23 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
98275 KOR CEREBELLUM GUINEA PIG 3H-U69593 (E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-3-yl)-N-methylacrylamide 0.23 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
51948 MOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 0.23 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
6129 Alpha1C CLONED HUMAN 125I-HEAT WB 4101 0.23 HIRASAWA A, ET AL., 1993 Jan 15, 2025 Jan 15, 2025