The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 1,001-2,000 of 99,458 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
1011615-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone101Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1014175-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione172Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
2985-HT1ACORTEXPIG3H-8-OH-DPATICS 205-930>10000HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
5545-HT1ACORTEXPIG3H-8-OH-DPATSUMATRIPTAN741SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
668585-HT1ACLONEDHUMAN3H-WAY100635N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide52Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
683945-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) piperid-1-yl] 6-nitroindan-1-010.74131Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33705-HT1ACLONEDHUMAN3H-8-OH-DPATNOREPINEPHRINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
704425-HT1ACLONEDHUMAN3H-WAY100635MRP50676.7Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
765865-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
113065-HT1ACLONEDHUMAN3H-8-OH-DPATPIPAMPERONE2770Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123305-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATBMY 73781.99Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788905-HT1ACLONEDHUMAN3H-WAY100635cis-2a2.3Ray TS 2010 Jan 15, 2025Jan 15, 2025
5555-HT1ACORTEXRAT3H-8-OH-DPATSUMATRIPTAN741SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
683955-HT1ACLONEDHUMAN3H-8-OH-DPATS 155350.794328Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33715-HT1ACLONEDHUMAN3H-8-OH-DPATPHENTOLAMINE2151TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
719795-HT1Atesttest[3H] Way1006351-(Benzo[d]thiazol-2-yl)-5-(4-(bis(4-fluorophenyl) methyl)piperazin-1-yl)pentan-1-one dihydrochloride>10000Etukala JR et al 2016Jan 15, 2025Jan 15, 2025
755635-HT1ACLONEDHUMAN3H-WAY1006353-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
113075-HT1ACLONEDHUMAN3H-8-OH-DPATFLUSPIRILENE56Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123315-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATNAN-1900.7Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788915-HT1ACLONEDHUMAN3H-WAY100635R,R-2b5.2Ray TS 2010 Jan 15, 2025Jan 15, 2025
858035-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-22145Luethi D et al 2019Jan 15, 2025Jan 15, 2025
256435-HT1ACLONEDHUMAN3H-8-OH-DPATCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
333235-HT1ACLONEDHUMAN3H-8-OH-DPATPiroxicam>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
5565-HT1ACELLSC0S-73H-8-OH-DPATTFMPP32.1RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
33725-HT1ACLONEDHUMAN3H-8-OH-DPATPIMOZIDE650TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
732605-HT1Atesttest[3H] Way100635N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
735165-HT1Atesttest[3H] Way100635N-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
113085-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE140Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123325-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATALPRENOLOL,(-)19.95Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788925-HT1ACLONEDHUMAN3H-WAY100635S,S-2c0.4Ray TS 2010 Jan 15, 2025Jan 15, 2025
804285-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((1H-indol-3-yl)methylene)-2-amino-1-methyl-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
835005-HT1AHEK293 cellsHUMAN3H-8-OH-DPATMBDB>10000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
870845-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one31.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
312765-HT1ACLONEDHUMAN3H-8-OH-DPATMDL 100907>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
330685-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATNOMIFENSINE>10000Andersen PH, et al., 1989Jan 15, 2025Jan 15, 2025
1011645-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone142Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
5575-HT1ACORTEXRAT3H-8-OH-DPATTFMPP75SCHLEGEL & PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
33735-HT1ACLONEDHUMAN3H-8-OH-DPATPPP, S(-)-34174TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113095-HT1ACLONEDHUMAN3H-8-OH-DPATZOTEPINE330Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123335-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATTERTATOLOL(-)8.31Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788935-HT1ACLONEDHUMAN3H-WAY1006355-MeO-TMT200Ray TS 2010 Jan 15, 2025Jan 15, 2025
909255-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane43.6516Franchini S et al 2014Jan 15, 2025Jan 15, 2025
1011655-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone302Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
5585-HT1ACORTEXRAT3H-8-OH-DPATTFMPP130PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
678865-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole111Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33745-HT1ACLONEDHUMAN3H-8-OH-DPATPROPRANOLOL272TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113105-HT1ACLONEDHUMAN3H-8-OH-DPATOLANZAPINE2720Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123345-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATWAY 100,13532.35Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788945-HT1ACLONEDHUMAN3H-WAY100635EMDT170Ray TS 2010 Jan 15, 2025Jan 15, 2025
858065-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-3158Luethi D et al 2019Jan 15, 2025Jan 15, 2025
896465-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone389.045Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
1014225-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione373Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
5595-HT1AHIPPOCAMPUSBOVINE3H-8-OH-DPATTFMPP148.15PEROUTKA, 1985Jan 15, 2025Jan 15, 2025
33755-HT1ACLONEDHUMAN3H-8-OH-DPATQUINPIROLE1713TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
730075-HT1ACLONEDHUMAN3H-WAY1006352-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline1,3-dione499Ofori E et al 2016Jan 15, 2025Jan 15, 2025
113115-HT1ACLONEDHUMAN3H-8-OH-DPATQuetiapine320Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123355-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSPIPERONE114.81Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788955-HT1ACLONEDHUMAN3H-WAY100635IBOGAINE>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
817115-HT1ACLONEDHUMAN3H-WAY100635psammopemmin A>10000Lebar MD et al 2011Jan 15, 2025Jan 15, 2025
870875-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one12Cao X et al 2018Jan 15, 2025Jan 15, 2025
896475-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone0.524807Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
282075-HT1ACLONEDHUMAN3H-8-OH-DPATNorfenfluramine (+)1950PDSP Certified DataJan 15, 2025Jan 15, 2025
988635-HT1ACLONEDHUMAN3H-WAY1006353-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane1297Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
5605-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATTFMPP173TITELER ET AL., 1987Jan 15, 2025Jan 15, 2025
671205-HT1ACLONEDHUMAN3H-WAY100635{2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
33765-HT1ACLONEDHUMAN3H-8-OH-DPATQUIPAZINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
724965-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-1-(5-fluoro-4-(1-(3-fluorophenyl)ethoxy)pyrimidin-2-yl)-1,4-diazepane578Kim J et al 2019Jan 15, 2025Jan 15, 2025
113125-HT1ACLONEDHUMAN3H-8-OH-DPATORG-522210Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123365-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSDZ 216,5251.58Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788965-HT1ACLONEDHUMAN3H-WAY100635Salvinorin A>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
817125-HT1ACLONEDHUMAN3H-WAY100635meridianin A684Lebar MD et al 2011Jan 15, 2025Jan 15, 2025
893925-HT1ACLONEDHUMAN3H-8-OH-DPAT4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide163Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
1011685-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone15.2Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
602085-HT1ACLONEDHUMAN3H-WAY100635MRS56987600Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
5615-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATTFMPP175GLENNON ET AL., 1988Jan 15, 2025Jan 15, 2025
33775-HT1ACLONEDHUMAN3H-8-OH-DPATRESERPINE1832TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
719855-HT1Atesttest[3H] Way1006351-(3-(Benzo[d]thiazol-2-yl)propyl)-4-(4-chlorophenyl) piperidin-4-ol hydrochloride34Etukala JR et al 2016Jan 15, 2025Jan 15, 2025
724975-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-1-(5-fluoro-4-(1-(4-fluorophenyl)ethoxy)pyrimidin-2-yl)-1,4-diazepane1066Kim J et al 2019Jan 15, 2025Jan 15, 2025
113135-HT1ACLONEDHUMAN3H-8-OH-DPATSERTINDOLE280Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
817135-HT1ACLONEDHUMAN3H-WAY1006354-methoxymeridianin A1354Lebar MD et al 2011Jan 15, 2025Jan 15, 2025
858095-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-4204Luethi D et al 2019Jan 15, 2025Jan 15, 2025
909295-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane60.256Franchini S et al 2014Jan 15, 2025Jan 15, 2025
932335-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine65Lober S et al 2012Jan 15, 2025Jan 15, 2025
1011695-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(4-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
5625-HT1AHIPPOCAMPUSRAT125I-BH-8-MeO-N-PATFMPP218.4GOZLAN ET AL., 1988Jan 15, 2025Jan 15, 2025
33785-HT1ACLONEDHUMAN3H-8-OH-DPATRITANSERIN2919TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
724985-HT1ACLONEDHUMAN3H-8-OH-DPAT5-fluoro-4-[(4-fluorophenyl)methoxy]-2-[(2R)-2methylpiperazin-1-yl]pyrimidine271Kim J et al 2019Jan 15, 2025Jan 15, 2025
113145-HT1ACLONEDHUMAN3H-8-OH-DPATZiprasidone12Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
817145-HT1ACLONEDHUMAN3H-WAY1006352-debromo-2-chloro-psammopemmin A>10000Lebar MD et al 2011Jan 15, 2025Jan 15, 2025
870905-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT7-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one25.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
896505-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone35.4813Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
589305-HT1ACLONEDHUMAN3H-WAY100635(-)-SYA 09832Ablordeppey S, et al., 2006Jan 15, 2025Jan 15, 2025
5635-HT1ABRAINRAT3H-8-OH-DPATTFMPP230ARNT & HYTTEL,1989Jan 15, 2025Jan 15, 2025
678915-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole120Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
684035-HT1ACLONEDHUMAN[11C[R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1478Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
33795-HT1ACLONEDHUMAN3H-8-OH-DPATSCH 23390,R(+)661TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
704515-HT1ACLONEDHUMAN3H-WAY100635MRP42706Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
753155-HT1ACLONEDHUMAN3H-WAY100635ethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
812035-HT1ACLONEDHUMAN3H-8-OH-DPATN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
817155-HT1ACLONEDHUMAN3H-WAY100635Methsergide49Lebar MD et al 2011Jan 15, 2025Jan 15, 2025
184835-HT1ABRAINpigeon3H-8-OH-DPATDU1255300.7Mos J et al., 1997Jan 15, 2025Jan 15, 2025
893955-HT1ACLONEDHUMAN3H-8-OH-DPAT4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide105Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
896515-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone208.93Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
1014275-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one19Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
497155-HT1ACLONEDHUMAN3H-8-OH-DPATPramipexole6514PDSP Certified DataJan 15, 2025Jan 15, 2025
661005-HT1ACLONEDHUMAN3H-WAY100635ARIPIPRAZOLE1.7Hirose, Tsuyoshi. et. al, 2005Jan 15, 2025Jan 15, 2025
33805-HT1ACLONEDHUMAN3H-8-OH-DPAT5-Hydroxy Tryptamine1.3TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
704525-HT1ACLONEDHUMAN3H-WAY100635MRP32006.2Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
806925-HT1ACLONEDHUMAN3H-8-OH-DPAT(5E)-5-((5-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one2513Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
822285-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one1.5Besnard J et al 2012Jan 15, 2025Jan 15, 2025
202765-HT1ACORTEXRAT3H-8-OH-DPATHMA>10000Garritsen A et al., 1991Jan 15, 2025Jan 15, 2025
858125-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-51246Luethi D et al 2019Jan 15, 2025Jan 15, 2025
1011725-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(2-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
3095-HT1ACORTEXRAT3H-8-OH-DPATICYANOPINDOLOL2.33HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
5655-HT1ACORTEXPIG3H-8-OH-DPATTFMPP288SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
33815-HT1ACLONEDHUMAN3H-8-OH-DPATSKF 383933096TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
763415-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
786455-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
870935-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one19.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
251415-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE427PDSP Certified DataJan 15, 2025Jan 15, 2025
909335-HT1AHeLaHUMAN3H-8-OH-DPAT8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane144.544Franchini S et al 2014Jan 15, 2025Jan 15, 2025
261655-HT1ACLONEDHUMAN3H-8-OH-DPATPseudonorephedrine, (-) [cathine, (-)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1011735-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(4-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
594455-HT1ACLONEDHUMAN3H-WAY100635DESIPRAMINE>10000Deupree, J. et. al., 2007Jan 15, 2025Jan 15, 2025
3105-HT1ACORTEXPIG3H-8-OH-DPATICYANOPINDOLOL5.39HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
5665-HT1ACORTEXPIG3H-8-OH-DPATTFMPP288SCHOEFFTER ET AL., 1989Jan 15, 2025Jan 15, 2025
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858155-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-7479Luethi D et al 2019Jan 15, 2025Jan 15, 2025
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678965-HT1ACLONEDHUMAN3H-8-OH-DPATS)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole25Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
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571445-HT1AUNDEFINEDUNDEFINEDUNDEFINEDBUSPIRONE20Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
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617535-HT1ACLONEDHUMAN3H-WAY100635(+)-Cimbi-775192Herth, Matthis et. al. 2015Jan 15, 2025Jan 15, 2025
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1016925-HT1ACLONEDHUMAN[3H]8-OH-DPATQuetiapine267PDSP Certified DataMar 21, 2025Jul 28, 2026
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571485-HT1AUNDEFINEDUNDEFINEDUNDEFINED2-Methoxy-10-allyl-11-hydroxy-N-methylaporphine144Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
617565-HT1ACLONEDHUMAN3H-WAY100635(-)-Cimbi-772633Herth, Matthis et. al. 2015Jan 15, 2025Jan 15, 2025
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750695-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
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617575-HT1ACLONEDHUMAN3H-WAY100635(+)-Cimbi-772787Herth, Matthis et. al. 2015Jan 15, 2025Jan 15, 2025
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33905-HT1ACLONEDHUMAN3H-8-OH-DPATBUTACLAMOL,(+)528TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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597105-HT1ACLONEDHUMAN3H-WAY1006354-(3- f 4-[2-(2-Fluoroethoxy)-phenyl]-piperazin-1-yl g -propoxy)-4- aza-tricyclo[5.2.1.02,6]dec-8-ene-3,5-dion4.2Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
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279675-HT1ACLONEDHUMAN3H-8-OH-DPATDMT,2-Me-5-methoxy200Glennon RA, et.al., 2000Jan 15, 2025Jan 15, 2025
940155-HT1ACORTEXPIG[3H]WAY 6001352-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one68Ortega R et al 2011Jan 15, 2025Jan 15, 2025
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1006715-HT1ACLONEDHUMAN3H-WAY100635Pizotyline270Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
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528105-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide4.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538345-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole14.9Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
558825-HT1AUNDEFINEDRATUNDEFINEDN-[4-(1,2,3,4-Tetrahydro-5-methoxy--carbolin-2-yl)butyl]isoquinoline-3-carboxamide118Butini S et al., 2009Jan 15, 2025Jan 15, 2025
571625-HT1AUNDEFINEDUNDEFINEDUNDEFINED(R)-11-(allyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline279Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
584425-HT1ACLONEDHUMAN3H-WAY100635MRS5202>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
684275-HT1ACLONEDHUMAN[11C]R107474mirtazapine3334Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
95475-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDESIPRAMINE2272Owens MJ, et al, 1997Jan 15, 2025Jan 15, 2025
873715-HT1ACLONEDHUMAN3H-WAY1006351-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
236275-HT1ACLONEDHUMAN3H-8-OH-DPATCyamemazine517Hameg A. et al., 2003Jan 15, 2025Jan 15, 2025
894195-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide149Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
922355-HT1ACLONEDHUMAN3H-8-OH-DPAT9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
932595-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine91Lober S et al 2012Jan 15, 2025Jan 15, 2025
983795-HT1ACLONEDHUMAN[3H]-Way1006352-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole111Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001715-HT1ACLONEDHUMAN3H-WAY100635Perospirone0.7PDSP Certified DataJan 15, 2025Jan 15, 2025
528115-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide66.7Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538355-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole2.5Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
571635-HT1AUNDEFINEDUNDEFINEDUNDEFINED2-Methoxy-11-hydroxyaporphine258Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
584435-HT1ACLONEDHUMAN3H-WAY100635MRS5923>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
663805-HT1ACLONEDHUMAN3H-WAY100635N-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
679165-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole14Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
720125-HT1ACLONEDHUMAN3H-WAY1006351-methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g] quinoxalin-2(6H)-one HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
95485-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATPAROXETINE>10000Owens MJ, et al, 1997Jan 15, 2025Jan 15, 2025
807165-HT1ACLONEDHUMAN3H-8-OH-DPAT(5E)-5-((7-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
825085-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-(Indolin-1-yl)ethyl)-2-((pyridin-3-yloxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
899325-HT1ACLONEDHUMAN3H-WAY1006353-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
983805-HT1ACLONEDHUMAN[3H]-Way1006352-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline65Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001725-HT1ACLONEDHUMAN3H-WAY100635Ziprasidone1.5PDSP Certified DataJan 15, 2025Jan 15, 2025
528125-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide56Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538365-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole1.6Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
571645-HT1AUNDEFINEDUNDEFINEDUNDEFINED(R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol49Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
584445-HT1ACLONEDHUMAN3H-WAY100635MRS5930>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
594685-HT1ACLONEDHUMAN3H-WAY100635Desmethylcitalopram6760Deupree, J. et. al., 2007Jan 15, 2025Jan 15, 2025
622845-HT1ACLONEDHUMANWAY100635Diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
661255-HT1ACLONEDHUMAN3H-WAY100635RISPERIDONE210Hirose, Tsuyoshi. et. al, 2005Jan 15, 2025Jan 15, 2025
727815-HT1ACLONEDHUMAN3H-WAY100635epigallocatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
730375-HT1ACLONEDHUMAN3H-WAY1006352-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline1689Ofori E et al 2016Jan 15, 2025Jan 15, 2025
95495-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSERTRALINE3663Owens MJ, et al, 1997Jan 15, 2025Jan 15, 2025
871175-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one12Cao X et al 2018Jan 15, 2025Jan 15, 2025
983815-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride15Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001735-HT1ACLONEDHUMAN3H-WAY100635Asenapine4.7PDSP Certified DataJan 15, 2025Jan 15, 2025
528135-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide28.1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538375-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole0.78Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
571655-HT1AUNDEFINEDUNDEFINEDUNDEFINED11-Hydroxy-N-propylnoraporphine45Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
584455-HT1ACLONEDHUMAN3H-WAY100635MRS5474>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
622855-HT1ACLONEDHUMANWAY1006352-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
666385-HT1ACLONEDHUMAN3H-WAY1006353-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
95505-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATFLUOXETINE8313Owens MJ, et al, 1997Jan 15, 2025Jan 15, 2025
771345-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
894225-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide74Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
983825-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride42Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001745-HT1ACLONEDHUMAN3H-WAY100635NEMONAPRIDE5.8PDSP Certified DataJan 15, 2025Jan 15, 2025
528145-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide41.8Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538385-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]benzoxazole14.1Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
571665-HT1AUNDEFINEDUNDEFINEDUNDEFINED8-OH-DPAT1.2Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
622865-HT1ACLONEDHUMANWAY1006353-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
49435-HT1ACORTEXRAT3H-8-OH-DPATRS-102221>10000BONHAUS DW, ET AL., 1997Jan 15, 2025Jan 15, 2025
95515-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATVenlafaxine>10000Owens MJ, et al, 1997Jan 15, 2025Jan 15, 2025
812315-HT1Atesttest3H-8-OH-DPAT5’-Iodo-HEAT HCl5.6Petrie EC et al 2012Jan 15, 2025Jan 15, 2025
983835-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride11Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001755-HT1ACLONEDHUMAN3H-WAY100635ARIPIPRAZOLE13PDSP Certified DataJan 15, 2025Jan 15, 2025
528155-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide12Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538395-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]benzothiazole9.6Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561435-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide3775Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571675-HT1AUNDEFINEDUNDEFINEDUNDEFINED11-(1-Methylallyloxy)-N-methylaporphine>10000Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
622875-HT1ACLONEDHUMANWAY1006354-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
95525-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT5-Hydroxy Tryptamine0.12Owens MJ, et al, 1997Jan 15, 2025Jan 15, 2025
804645-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-2-amino-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
983845-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride9.9Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001765-HT1ACLONEDHUMAN3H-WAY100635ILOPERIDONE27PDSP Certified DataJan 15, 2025Jan 15, 2025
528165-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide12Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538405-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]1H-benzimidazole16.6Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561445-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)benzamide>10000Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571685-HT1AUNDEFINEDUNDEFINEDUNDEFINED(E/Z)-11-(2-butenyloxy)-N-propylnoraporphine11Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
622885-HT1ACLONEDHUMANWAY1006352-Cl-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
679215-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole16Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
827695-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
876335-HT1ACLONEDHUMAN3H-WAY1006353-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
983855-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline1109Ofon E et al 2016Jan 15, 2025Jan 15, 2025
333615-HT1ACLONEDHUMAN3H-8-OH-DPATibuprofen solid, (S)-(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1001775-HT1ACLONEDHUMAN3H-WAY100635Lurasidone HCl53PDSP Certified DataJan 15, 2025Jan 15, 2025
528175-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide5.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538415-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzoxazole0.55Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561455-HT1AUNDEFINEDRATUNDEFINEDN-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide7586Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571695-HT1AUNDEFINEDUNDEFINEDUNDEFINEDN-Methyl-2-hydroxy-2'-methyl-2',3'-dihydrofuro[m]aporphine12Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
597295-HT1ACLONEDHUMAN3H-WAY1006354-(3- f 4-[2-(4-Fluoroethoxy)-phenyl]-piperazin-1-yl g -propoxy)-4- aza-tricyclo[5.2.1.02,6]dec-8-ene-3,5-dion>10000Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
768825-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
118585-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATBUSPIRONE12.58Millan MJ, et al., 2000Jan 15, 2025Jan 15, 2025
983865-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline138Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001785-HT1ACLONEDHUMAN3H-WAY100635CLOZAPINE104PDSP Certified DataJan 15, 2025Jan 15, 2025
528185-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538425-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzothiazole0.29Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561465-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide7440Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571705-HT1AUNDEFINEDUNDEFINEDUNDEFINED8-(1-Buten-3-yl)-11-hydroxy-N-propylnoraporphine626Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
766275-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
118595-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATYOHIMBINE125.89Millan MJ, et al., 2000Jan 15, 2025Jan 15, 2025
835395-HT1AHEK293 cellsHUMAN3H-8-OH-DPATmephedrone>10000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
983875-HT1ACLONEDHUMAN[3H]-Way1006352-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001795-HT1ACLONEDHUMAN3H-WAY100635ZOTEPINE131PDSP Certified DataJan 15, 2025Jan 15, 2025
528195-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide7.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538435-HT1AUNDEFINEDRATUNDEFINED2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]1H-benzimidazole1Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561475-HT1AUNDEFINEDRATUNDEFINED2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide497Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571715-HT1AUNDEFINEDUNDEFINEDUNDEFINEDN-Propyl-2',3'-bismethyl-2',3'-dihydrofuro[m]noraporphine90Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
725325-HT1ACLONEDHUMAN3H-WAY100635Amentoflavone>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
745805-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
756045-HT1ACLONEDHUMAN3H-WAY1006352-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
118605-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATFluparoxan630.95Millan MJ, et al., 2000Jan 15, 2025Jan 15, 2025
861005-HT1ACLONEDHUMAN3H-WAY1006354-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
983885-HT1ACLONEDHUMAN[3H]-Way1006351-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001805-HT1ACLONEDHUMAN3H-WAY100635RISPERIDONE158PDSP Certified DataJan 15, 2025Jan 15, 2025
528205-HT1AUNDEFINEDHUMANUNDEFINED6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-amine2Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538445-HT1AUNDEFINEDRATUNDEFINED2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]benzoxazole326Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561485-HT1AUNDEFINEDRATUNDEFINEDAdamantane-1-carboxylic acid ((S)-1-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-2,5-dioxo-pyrrolidin-3-yl)-amide579Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571725-HT1AUNDEFINEDUNDEFINEDUNDEFINEDN-Propyl-2'-methyl-2',3'-dihydrofuro[m]noraporphine340Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
118615-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT3.16Millan MJ, et al., 2000Jan 15, 2025Jan 15, 2025
894295-HT1ACLONEDHUMAN3H-8-OH-DPATN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide771Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
983895-HT1ACLONEDHUMAN[3H]-Way1006351-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione339Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001815-HT1ACLONEDHUMAN3H-WAY100635SERTINDOLE236PDSP Certified DataJan 15, 2025Jan 15, 2025
528215-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide4.9Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538455-HT1AUNDEFINEDRATUNDEFINED2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]benzothiazole1702Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561495-HT1AUNDEFINEDRATUNDEFINED(S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide8518Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
571735-HT1AUNDEFINEDUNDEFINEDUNDEFINED10-(2-Butenyl)-11-hydroxy-N-propylnoraporphine>10000Liu Z et al., 2010Jan 15, 2025Jan 15, 2025
589655-HT1ACLONEDHUMAN3H-WAY100635CLOZAPINE140Ablordeppey S, et al., 2006Jan 15, 2025Jan 15, 2025
669025-HT1ACLONEDHUMAN3H-WAY100635N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
679265-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole179Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
118625-HT1ACLONEDHUMAN3H-8-OH-DPATYOHIMBINE50.11Millan MJ, et al., 2000Jan 15, 2025Jan 15, 2025
246625-HT1ACLONEDHUMANUNDEFINEDSR 144528>10000Rinaldi-Carmona, M et al., 1998Jan 15, 2025Jan 15, 2025
983905-HT1ACLONEDHUMAN[3H]-Way1006354-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one19.5Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001825-HT1ACLONEDHUMAN3H-WAY100635Paliperidone404PDSP Certified DataJan 15, 2025Jan 15, 2025
528225-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
538465-HT1AUNDEFINEDRATUNDEFINED2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]1H-benzimidazole95.2Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561505-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide1001Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3435-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATLISURIDE2.59HALL ET AL., 1985Jan 15, 2025Jan 15, 2025
730475-HT1ACLONEDHUMAN3H-WAY1006352-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4- tetrahydroisoquinoline hydrochloride193Ofori E et al 2016Jan 15, 2025Jan 15, 2025
733035-HT1Atesttest[3H] Way100635N-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
118635-HT1ACLONEDHUMAN3H-8-OH-DPATFluparoxan158.48Millan MJ, et al., 2000Jan 15, 2025Jan 15, 2025
983915-HT1ACLONEDHUMAN[3H]-Way1006351-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 8.3Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001835-HT1ACLONEDHUMAN3H-WAY100635OLANZAPINE1114PDSP Certified DataJan 15, 2025Jan 15, 2025
538475-HT1AUNDEFINEDRATUNDEFINED2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]benzoxazole67.2Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561515-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide1507Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3445-HT1AHIPPO:LESIONEDRAT3H-WB4101LISURIDE2.68MORROW ET AL., 1985Jan 15, 2025Jan 15, 2025
735605-HT1Atesttest[3H] Way1006353-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
807285-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-5-((1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
894325-HT1ACLONEDHUMAN3H-8-OH-DPATN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide2870Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
932725-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine100Lober S et al 2012Jan 15, 2025Jan 15, 2025
983925-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001845-HT1ACLONEDHUMAN3H-WAY100635Blonanserin1215PDSP Certified DataJan 15, 2025Jan 15, 2025
538485-HT1AUNDEFINEDRATUNDEFINED2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]benzothiazole31.2Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561525-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide1950Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3455-HT1ACORTEXHUMAN3H-8-OH-DPATLOXAPINE2900WANDER ET AL., 1987Jan 15, 2025Jan 15, 2025
159615-HT1ACLONEDRAT125I-LSD5-CT11Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
983935-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001855-HT1ACLONEDHUMAN3H-WAY100635Melperone HCl1328PDSP Certified DataJan 15, 2025Jan 15, 2025
535935-HT1AUNDEFINEDHUMANUNDEFINEDCyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide0.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561535-HT1AUNDEFINEDRATUNDEFINED(S)-1-acetyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide6600Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
661385-HT1ACLONEDHUMAN3H-WAY100635OLANZAPINE2100Hirose, Tsuyoshi. et. al, 2005Jan 15, 2025Jan 15, 2025
110985-HT1ACLONEDHUMAN3H-8-OH-DPATP88-8991426.57CINP 2000 PROCEEDINGJan 15, 2025Jan 15, 2025
159625-HT1ACLONEDRAT125I-LSDMETHIOTHEPIN8.7Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
966025-HT1ACLONEDHUMAN[3H]-Way1006351,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
983945-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride1712Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001865-HT1ACLONEDHUMAN3H-WAY100635Remoxapride2989PDSP Certified DataJan 15, 2025Jan 15, 2025
535945-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-trans)-4-[4-(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine7.8Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561545-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide3553Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
671635-HT1ACLONEDHUMAN3H-WAY100635{2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
679315-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole96Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
710035-HT1ACLONEDHUMAN3H-WAY100635N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide245Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
110995-HT1ACLONEDHUMAN3H-8-OH-DPATP95-12113>10000CINP 2000 PROCEEDINGJan 15, 2025Jan 15, 2025
159635-HT1ACLONEDRAT125I-LSD5-Hydroxy Tryptamine134Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
868755-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione27Zareba P et al 2020Jan 15, 2025Jan 15, 2025
249235-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL1202PDSP Certified DataJan 15, 2025Jan 15, 2025
940435-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-methylthiophenethylamine1035Luethi D et al 2018Jan 15, 2025Jan 15, 2025
983955-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid214Ofon E et al 2016Jan 15, 2025Jan 15, 2025
1001875-HT1ACLONEDHUMAN3H-WAY100635RS-(+/-)-Sulpriride7610PDSP Certified DataJan 15, 2025Jan 15, 2025
535955-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-cis)-4-[(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine15.8Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561555-HT1AUNDEFINEDRATUNDEFINED(S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-amide350Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3485-HT1ACORTEXPIG3H-8-OH-DPATLSD2.57ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
712605-HT1ACLONEDHUMANWAY100635N,N-diallyltryptamine100Klein LM et al 2018Jan 15, 2025Jan 15, 2025
753565-HT1ACLONEDHUMAN3H-WAY100635Ethyl(1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
111005-HT1ACLONEDHUMAN3H-8-OH-DPATILOPERIDONE93.32CINP 2000 PROCEEDINGJan 15, 2025Jan 15, 2025
116125-HT1ABRAINHUMAN3H-8-OH-DPATAdinazolam>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
804765-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-2-amino-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one7269Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
159645-HT1ACLONEDRAT125I-LSDMESULERGINE545Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
822685-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one0.9Besnard J et al 2012Jan 15, 2025Jan 15, 2025
256925-HT1ACLONEDHUMAN3H-8-OH-DPATEphedrine,(-)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
940445-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-dimethoxy-4-(b-methallyl)thio-phenethylamine812Luethi D et al 2018Jan 15, 2025Jan 15, 2025
983965-HT1ACLONEDHUMAN[3H]-Way1006355-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,122Ofon E et al 2016Jan 15, 2025Jan 15, 2025
994205-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide26Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
1019805-HT1ACLONEDHUMAN[3H]8-OH-DPATRS-(+/-)-Sulpriride7610PDSP Certified DataMar 24, 2025Jul 28, 2026
535965-HT1AUNDEFINEDHUMANUNDEFINED5-Fluoro-3-[(1,4-trans)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole42.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561565-HT1AUNDEFINEDRATUNDEFINED(S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclopentanecarbonyl)pyrrolidine-2-carboxamide2013Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
684455-HT1ACLONEDHUMAN3H-WAY100635N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
763815-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
116135-HT1ABRAINHUMAN3H-8-OH-DPATAMITRIPTYLINE450Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159655-HT1ACLONEDRAT125I-LSDMETERGOLINE273Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
940455-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-isopropylthiophenethylamine916Luethi D et al 2018Jan 15, 2025Jan 15, 2025
983975-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,19Ofon E et al 2016Jan 15, 2025Jan 15, 2025
994215-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide12Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
535975-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-trans)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile9.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561575-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide360Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
116145-HT1ABRAINHUMAN3H-8-OH-DPATBUPROPION>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159665-HT1ACLONEDRAT125I-LSDMETHYSERGIDE545Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
940465-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-propylthiophenethylamine878Luethi D et al 2018Jan 15, 2025Jan 15, 2025
983985-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride48.3Ofon E et al 2016Jan 15, 2025Jan 15, 2025
994225-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide21Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
535985-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-cis)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile156.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561585-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide480Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3515-HT1ACORTEXRAT3H-8-OH-DPATLSD1.2SCHLEGEL & PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
116155-HT1ABRAINHUMAN3H-8-OH-DPATDESIPRAMINE6400Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
786875-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-butyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
159675-HT1ACLONEDRAT125I-LSDERGOTAMINE3Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
886715-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol102Sampson D et al 2014Jan 15, 2025Jan 15, 2025
894395-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide147Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
940475-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-allylthiophenethylamine660Luethi D et al 2018Jan 15, 2025Jan 15, 2025
983995-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride16Ofon E et al 2016Jan 15, 2025Jan 15, 2025
336315-HT1ACLONEDHUMAN3H-8-OH-DPATPARECOXIB>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
994235-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide84Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
1017275-HT1ACLONEDHUMAN[3H]8-OH-DPATRemoxapride2989PDSP Certified DataMar 24, 2025Jul 28, 2026
535995-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-trans)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile2.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561595-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide230Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3525-HT1AHIPPOCAMPUSBOVINE3H-IPSAPIRONELSD0.31DOMPERT ET AL., 1985Jan 15, 2025Jan 15, 2025
679365-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole86Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
730565-HT1ACLONEDHUMAN3H-WAY1006352-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride141Ofori E et al 2016Jan 15, 2025Jan 15, 2025
738245-HT1Atesttest[3H] Way100635{2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
116165-HT1ABRAINHUMAN3H-8-OH-DPATDesmethylsertraline>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159685-HT1ACLONEDRAT125I-LSDRITANSERIN545Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
825285-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-(Indolin-1-yl)ethyl)-2-((pyridin-3-yloxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
868805-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione12Zareba P et al 2020Jan 15, 2025Jan 15, 2025
940485-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-n-butylthiophenethylamine1019Luethi D et al 2018Jan 15, 2025Jan 15, 2025
994245-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide58Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
536005-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-cis)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile43.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
538565-HT1AUNDEFINEDRATUNDEFINED3-amino-6-ethyl-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propylthio)thieno[2,3-d]pyrimidin-4(3H,4aH,7aH)-one7.4Siracusa MA et al., 2008Jan 15, 2025Jan 15, 2025
561605-HT1AUNDEFINEDRATUNDEFINED2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide40Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3535-HT1ACORTEXHUMAN3H-WB4101LSD0.64WANDER ET AL., 1987Jan 15, 2025Jan 15, 2025
704975-HT1ACLONEDHUMAN3H-WAY100635MRP32015.7Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
116175-HT1ABRAINHUMAN3H-8-OH-DPATDOXEPIN276Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159695-HT1ACLONEDRAT125I-LSD8-OH-DPAT27Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
835535-HT1AHEK293 cellsHUMAN3H-8-OH-DPATNaphyrone6000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
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994255-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide54Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
408015-HT1ACLONEDHUMAN3H-8-OH-DPATRWAY,(-)0.6PDSP Certified DataJan 15, 2025Jan 15, 2025
536015-HT1AUNDEFINEDHUMANUNDEFINED8-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline6.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
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561615-HT1AUNDEFINEDRATUNDEFINEDN-[(3S)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide63Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3545-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATLSD2.05HALL ET AL., 1985Jan 15, 2025Jan 15, 2025
116185-HT1ABRAINHUMAN3H-8-OH-DPATEtoperidone85Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
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164825-HT1ACLONEDHUMAN3H-8-OH-DPATFluorocarazolol,(S)34Roth BL, et al., 2001Jan 15, 2025Jan 15, 2025
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994265-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide91Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
536025-HT1AUNDEFINEDHUMANUNDEFINED8-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline69.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
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561625-HT1AUNDEFINEDRATUNDEFINED(S)-N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide1730Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
707555-HT1Atesttest3H-8-OH-DPAT1-Butanoyl-d-lysergic acid diethylamide345Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
715235-HT1ACLONEDHUMANWAY1006355-methoxy-2-fluoro-N,N-diallyltryptamine318Klein LM et al 2018Jan 15, 2025Jan 15, 2025
116195-HT1ABRAINHUMAN3H-8-OH-DPATFemoxetine2285Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
784355-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-cyclohexyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
159715-HT1ACLONEDRAT125I-LSDBUSPIRONE68.7Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
940515-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-isobutylthiophenethylamine1036Luethi D et al 2018Jan 15, 2025Jan 15, 2025
994275-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide19Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
456675-HT1ACLONEDHUMAN3H-8-OH-DPAT(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536035-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-trans)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile6.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
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561635-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-5-oxopyrrolidine-2-carboxamide390Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
574435-HT1AUNDEFINEDUNDEFINEDUNDEFINED[125I]1-(2-iodophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxylate93.5Donohue SR et al., 2009Jan 15, 2025Jan 15, 2025
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159725-HT1ACLONEDRAT125I-LSDPINDOLOL,(+/-)31Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
940525-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-benzylthiophenethylamine,1166Luethi D et al 2018Jan 15, 2025Jan 15, 2025
994285-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(4-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide327Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
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456685-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536045-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-cis)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile58.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561645-HT1AUNDEFINEDRATUNDEFINED(S)-1-acetyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)pyrrolidine-2-carboxamide580Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
3575-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATLSD0.43TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
679415-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
116215-HT1ABRAINHUMAN3H-8-OH-DPATIMIPRAMINE5800Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159735-HT1ACLONEDRAT125I-LSDNOREPINEPHRINE545Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
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282615-HT1ACLONEDHUMAN3H-8-OH-DPATNorfenfluramine1600PDSP Certified DataJan 15, 2025Jan 15, 2025
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994295-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide156Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
456695-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-0161760Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536055-HT1AUNDEFINEDHUMANUNDEFINED5-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline8.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561655-HT1AUNDEFINEDRATUNDEFINEDN-((S)-1-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-3-yl)cyclohexanecarboxamide26Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
630775-HT1ACLONEDHUMAN3H-WAY100635Mitragynine3708PDSP Certified DataJan 15, 2025Jan 15, 2025
3585-HT1ACORTEXPIG3H-8-OH-DPATLSD2.57MARKSTEIN ET AL, 1986Jan 15, 2025Jan 15, 2025
707585-HT1Atesttest3H-8-OH-DPAT1-propionyl-lysergic acid diethylamide637Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
751105-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
116225-HT1ABRAINHUMAN3H-8-OH-DPATLofepramine4600Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159745-HT1ACLONEDRAT125I-LSDDOPAMINE545Lovenberg TW, et al., 1993aJan 15, 2025Jan 15, 2025
853505-HT1ArecombinantHUMAN3H-8-OH-DPATTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
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1012225-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-([1,1'-biphenyl]-2-yl)piperazin-1-yl)-1-(3,4-dichlorophenyl)ethanol hydrochloride 2.4Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
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536065-HT1AUNDEFINEDHUMANUNDEFINED5-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline97.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561665-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)benzamide41Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
661515-HT1ACLONEDHUMAN3H-WAY100635Quetiapine230Hirose, Tsuyoshi. et. al, 2005Jan 15, 2025Jan 15, 2025
116235-HT1ABRAINHUMAN3H-8-OH-DPATNefazodone80Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159755-HT1ACLONEDHUMAN3H-8-OH-DPATBUSPIRONE21.1Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
853515-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
868875-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione18Zareba P et al 2020Jan 15, 2025Jan 15, 2025
231435-HT1ACLONEDHUMAN3H-8-OH-DPATDL-homocysteine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
246795-HT1AFR. CORTEXRAT3H-8-OH-DPATBIMT 1719.0546Borsini F, et al., 1995Jan 15, 2025Jan 15, 2025
940555-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine1063Luethi D et al 2018Jan 15, 2025Jan 15, 2025
994315-HT1ACLONEDHUMANUNDEFINED2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide20Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
456715-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-0252150Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536075-HT1AUNDEFINEDHUMANUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole3.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561675-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide69Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
600075-HT1ACLONEDHUMAN3H-WAY1006352-{4-[4-(3-Methoxyphenyl)-1-piperazinyl]butyl}-4-methyl-1,2,4-triazine-3,5(2H,4H)-dione1.1Prabhakaran, J. et. al, 2006Jan 15, 2025Jan 15, 2025
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3605-HT1ACORTEXRAT3H-8-OH-DPATLSD3.9PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
116245-HT1ABRAINHUMAN3H-8-OH-DPATNORFLUOXETINE>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
781845-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
804885-HT1ACLONEDHUMAN3H-8-OH-DPAT(E)-5-((1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
159765-HT1ACLONEDHUMAN3H-8-OH-DPAT5-CT0.53Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
231445-HT1ACLONEDHUMAN3H-8-OH-DPATL-cysteine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
267285-HT1ACLONEDHUMAN3H-8-OH-DPATPseudohypericin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938005-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione6.3Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
940565-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine1411Luethi D et al 2018Jan 15, 2025Jan 15, 2025
994325-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide9Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
1012245-HT1ACLONEDHUMAN3H-8-OH-DPAT1-([1,1'-biphenyl]-2-yl)-4-(3,4-dichlorophenethyl)piperazine hydrochloride 6.3Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
456725-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-048-45000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536085-HT1AUNDEFINEDHUMANUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole16.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
561685-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide19Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
1055-HT1ACORTEXPIG3H-8-OH-DPAT1-NP38.9SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
3615-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATLSD4.1HALL ET AL., 1986Jan 15, 2025Jan 15, 2025
707615-HT1Atesttest3H-8-OH-DPAT1-Acetyl-D-lysergic acid diethylamide1054Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
761375-HT1ACLONEDHUMAN3H-WAY1006352S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
116255-HT1ABRAINHUMAN3H-8-OH-DPATNORTRYPTYLINE294Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159775-HT1ACLONEDHUMAN3H-8-OH-DPATIPSAPIRONE3.85Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
231455-HT1ACLONEDHUMAN3H-8-OH-DPATD-homocysteine thiolactone>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
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267295-HT1ACLONEDHUMAN3H-8-OH-DPATHypericin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938015-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione4.9Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
940575-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-Bromo-2,5-dimethoxyphenethylamine311Luethi D et al 2018Jan 15, 2025Jan 15, 2025
994335-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide4Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
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561695-HT1AUNDEFINEDRATUNDEFINED2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide9Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
1065-HT1ACORTEXPIG3H-8-OH-DPAT1-NP38.9SCHOEFFTER ET AL., 1989Jan 15, 2025Jan 15, 2025
3625-HT1ACORTEXHUMAN3H-8-OH-DPATLSD4.92PIERCE & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
679465-HT1ACLONEDHUMAN3H-8-OH-DPATS)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline18Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
116265-HT1ABRAINHUMAN3H-8-OH-DPATPAROXETINE>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
159785-HT1ACLONEDHUMAN3H-8-OH-DPATLISURIDE0.41Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
868905-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione55Zareba P et al 2020Jan 15, 2025Jan 15, 2025
231465-HT1ACLONEDHUMAN3H-8-OH-DPATL-homocysteine thiolactone>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
267305-HT1ACLONEDHUMAN3H-8-OH-DPATHyperforin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938025-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion2.3Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
940585-HT1ACLONEDHUMAN[3H]-8-OH-DPATLSD1.5Luethi D et al 2018Jan 15, 2025Jan 15, 2025
331305-HT1ACLONEDHUMAN3H-8-OH-DPATvaleryl salicylate>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
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1012265-HT1ACLONEDHUMAN3H-8-OH-DPATVortioxetine9.5Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
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561705-HT1AUNDEFINEDRATUNDEFINEDN-[(3S)-1-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide4Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
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456755-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid2790Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
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193085-HT1AHIPPOCAMPUSRAT35S-GTPGammaSRec 15/30790.7Leonardi A et al., 2001Jan 15, 2025Jan 15, 2025
231485-HT1ACLONEDHUMAN3H-8-OH-DPATL-homocysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
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267325-HT1ACLONEDHUMAN3H-8-OH-DPATHyperoside>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938045-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione246Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
961085-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
994365-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide23Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
1012285-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one3755Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
372285-HT1ACORTEXRAT3H-8-OH-DPATAMITRIPTYLINE>10000Sanchez C, et al., 1999Jan 15, 2025Jan 15, 2025
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482365-HT1ACLONEDHUMAN3H-8-OH-DPATstepholidine143.4PDSP Certified DataJan 15, 2025Jan 15, 2025
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561725-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-oxopyrrolidine-2-carboxamide17Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
1095-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT1-PP1410GLENNON ET AL., 1988Jan 15, 2025Jan 15, 2025
111175-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT9-OH-risperidone380Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
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159815-HT1ACLONEDHUMAN3H-8-OH-DPATBUTACLAMOL,(+)680Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
193095-HT1ACLONEDHUMAN35S-GTPGammaSRec 15/30790.2Leonardi A et al., 2001Jan 15, 2025Jan 15, 2025
231495-HT1ACLONEDHUMAN3H-8-OH-DPATL-cysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
267335-HT1ACLONEDHUMAN3H-8-OH-DPATRutin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938055-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion68.7Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
961095-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
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456775-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
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116305-HT1ABRAINHUMAN3H-8-OH-DPATVenlafaxine>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
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267345-HT1ACLONEDHUMAN3H-8-OH-DPATQuercetin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938065-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione48.7Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
961105-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
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456785-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
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597585-HT1ACLONEDHUMAN3H-WAY1006354-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)-1-butanone27.7Ablordeppey S, et al., 2006Jan 15, 2025Jan 15, 2025
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3675-HT1ACORTEXRAT3H-8-OH-DPATMETERGOLINE3.45HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
679515-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)10Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
748635-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
111195-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATPIPAMPERONE2600Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
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231515-HT1ACLONEDHUMAN3H-8-OH-DPATD-homocysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
246875-HT1AFR. CORTEXRAT3H-8-OH-DPAT8-OH-DPAT6.16595Borsini F, et al., 1995Jan 15, 2025Jan 15, 2025
267355-HT1ACLONEDHUMAN3H-8-OH-DPATQuercitrin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938075-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione222Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
961115-HT1ACLONEDHUMAN3H-WAY1006354-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
372315-HT1ACORTEXRAT3H-8-OH-DPATFLUOXETINE>10000Sanchez C, et al., 1999Jan 15, 2025Jan 15, 2025
456795-HT1ACLONEDHUMAN3H-8-OH-DPATN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide2546Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
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561755-HT1AUNDEFINEDRATUNDEFINED(2S)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}pyrrolidine-2-carboxamide3Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
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3685-HT1ACORTEXRAT3H-8-OH-DPATMETERGOLINE3.7SCHLEGEL & PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
111205-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATFLUSPIRILENE110Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
776805-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
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822885-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one0.7Besnard J et al 2012Jan 15, 2025Jan 15, 2025
231525-HT1ACLONEDHUMAN3H-8-OH-DPATL-homocysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
886885-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol123Sampson D et al 2014Jan 15, 2025Jan 15, 2025
267365-HT1ACLONEDHUMAN3H-8-OH-DPATAmentoflavone>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
938085-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione240Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
961125-HT1ACLONEDHUMAN3H-WAY1006354′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
1012325-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 2891Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
372325-HT1ACORTEXRAT3H-8-OH-DPATPAROXETINE>10000Sanchez C, et al., 1999Jan 15, 2025Jan 15, 2025
456805-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3275Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536165-HT1AUNDEFINEDHUMANUNDEFINED5-Chloro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole325.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
548965-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine10.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
561765-HT1AUNDEFINEDRATUNDEFINEDBUSPIRONE36Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
618085-HT1ACLONEDHUMAN3H-WAY100635FECIMBI-361433Prabhakaran, Jaya et. al. 2015Jan 15, 2025Jan 15, 2025
1135-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDMA1131TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
3695-HT1ACORTEXHUMAN3H-8-OH-DPATMETERGOLINE4.34HOYER ET AL., 1986Jan 15, 2025Jan 15, 2025
111215-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATCLOZAPINE180Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
159855-HT1ACLONEDHUMAN3H-8-OH-DPATSPIPERONE411Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
868975-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione32Zareba P et al 2020Jan 15, 2025Jan 15, 2025
231535-HT1ACLONEDHUMAN3H-8-OH-DPATL-cysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
252015-HT1ACLONEDHUMAN3H-8-OH-DPATTHIORIDAZINE108PDSP Certified DataJan 15, 2025Jan 15, 2025
938095-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione13Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
961135-HT1ACLONEDHUMAN3H-WAY1006354′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
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899775-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-methyl) ethanamine440Rickli A et al 2015Jan 15, 2025Jan 15, 2025
933055-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATEthyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-butyric acid457Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
938175-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione5000Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
966335-HT1ACLONEDHUMAN[3H]-Way1006351,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
968895-HT1ACLONEDPIG[3H]WAY100635ARIPIPRAZOLE88Mannel B et al 2017Jan 15, 2025Jan 15, 2025
456895-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536255-HT1AUNDEFINEDHUMANUNDEFINED3-{4-[(1,4-trans)-4-(1H-indol-4-yl)-pipera-zinyl-1-yl]cyclohexyl}-1H-indole-5-carbonitrile3.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
549055-HT1AUNDEFINEDHUMANUNDEFINED8-OH-DPAT3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
1225-HT1ACORTEXPIG3H-8-OH-DPAT5,7-DHT>10000ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
3785-HT1ACORTEXRAT3H-8-OH-DPATMETERGOLINE13PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
666825-HT1ACLONEDHUMAN3H-WAY100635ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate894Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
723145-HT1ACLONEDHUMAN3H-8-OH-DPAT2-Aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 15, 2025
728265-HT1ACLONEDHUMAN3H-WAY100635isoginkgetin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
159945-HT1ACLONEDHUMAN3H-SPIPERONEMETHIOTHEPIN24.6Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
871625-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one78Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
899785-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane360Rickli A et al 2015Jan 15, 2025Jan 15, 2025
933065-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-Phenyl-1-piperazinyl)-propyl]-3-phenylpyrrolidine-2,5-dione dihydrochloride1069Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
938185-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione122Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
968905-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde14Mannel B et al 2017Jan 15, 2025Jan 15, 2025
380105-HT1ArecombinantHUMAN3H-8-OH-DPATK376>10000Mimura H, et al., 2005Jan 15, 2025Jan 15, 2025
456905-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536265-HT1AUNDEFINEDHUMANUNDEFINED3-{4-[(1,4-cis)-4-(1H-Indol-4-yl)-pipera-zinyl-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile69.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
549065-HT1AUNDEFINEDHUMANUNDEFINEDrac-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine15.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
587465-HT1ACLONEDHUMAN3H-8-OH-DPATN-[2-(4-Phenylpiperazin-1-yl)ethyl]-2-quinoxaline Carboxamide28Graulich A, et al., 2010Jan 15, 2025Jan 15, 2025
1235-HT1ACORTEXPIG3H-8-OH-DPAT5-CT0.16HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
3795-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATMETERGOLINE26.99GOZLAN ET AL., 1983Jan 15, 2025Jan 15, 2025
159955-HT1ACLONEDHUMAN3H-SPIPERONEPINDOLOL,(+/-)61.1Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
835795-HT1AHEK293 cellsHUMAN3H-8-OH-DPATCOCAINE>10000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
869075-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione4Zareba P et al 2020Jan 15, 2025Jan 15, 2025
871635-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one55Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
899795-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxyphenethylamine70Rickli A et al 2015Jan 15, 2025Jan 15, 2025
933075-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride177Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
938195-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[3-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione183Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
968915-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde21Mannel B et al 2017Jan 15, 2025Jan 15, 2025
380115-HT1ArecombinantHUMAN3H-8-OH-DPATK117>10000Mimura H, et al., 2005Jan 15, 2025Jan 15, 2025
456915-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione165.3Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
536275-HT1AUNDEFINEDHUMANUNDEFINED4-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole22.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
549075-HT1AUNDEFINEDHUMANUNDEFINED(3R)-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-3,4-dihydro-2H-chromen-2.14Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
587475-HT1ACLONEDHUMAN3H-8-OH-DPATN-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide13Graulich A, et al., 2010Jan 15, 2025Jan 15, 2025
1245-HT1ACORTEXPIG3H-8-OH-DPAT5-CT0.21ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
3805-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATMETERGOLINE42.8HALL ET AL., 1986Jan 15, 2025Jan 15, 2025
769245-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one8590Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
807645-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
159965-HT1ACLONEDHUMAN3H-SPIPERONESPIPERONE17.2Sundaram H, et al., 1993Jan 15, 2025Jan 15, 2025
820445-HT1ACLONEDHUMAN3H-WAY1006351-(1,3-Benzodioxol-4-ylmethyl)-4-[4-(trifluoromethyl)phenyl]piperazine1000DeRuiter J et al 2018Jan 15, 2025Jan 15, 2025
244445-HT1AHippocampalGUINEA PIG3H-Cyclic AMPSPIPERONE16Bockaert J, et al., 1990Jan 15, 2025Jan 15, 2025
899805-HT1ACLONEDHUMAN3H-8-OH-DPAT4-iodo-2,5-dimethoxyphenethylamine180Rickli A et al 2015Jan 15, 2025Jan 15, 2025
933085-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-chlorophenyl)-pyrrolidine-2,5-dione dihydrochloride258Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025