50947 MOR UNDEFINED HUMAN UNDEFINED Naltrexone 0.23 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51459 Alpha1A UNDEFINED HUMAN UNDEFINED 3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 11 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51971 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1.72 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52227 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(adamantan-1-ylamino)-3-(1H-indol-5-yloxy)-propan-2-ol 833 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52483 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 106 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52995 CB2 UNDEFINED HUMAN UNDEFINED 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide 6000 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53251 D2 UNDEFINED HUMAN UNDEFINED 1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 4.7 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53763 H1 UNDEFINED HUMAN UNDEFINED RISPERIDONE 19 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54275 SLC6A4 UNDEFINED HUMAN UNDEFINED 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 73.7 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54531 A3 UNDEFINED HUMAN UNDEFINED N-(4-cyanophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 570 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54787 D2 UNDEFINED HUMAN UNDEFINED N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine 210 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55043 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 8.2 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55299 DOR UNDEFINED HUMAN UNDEFINED 8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 538 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
56323 A1 UNDEFINED HUMAN UNDEFINED 2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 1410 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56579 DOR UNDEFINED HUMAN UNDEFINED 4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 807 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56835 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-(N-tert-Butylamino)propiophenone 5700 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57091 D2 UNDEFINED HUMAN UNDEFINED Bifeprunox 0.04 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
57347 A1 UNDEFINED HUMAN UNDEFINED (E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-propenone 0.49 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57603 SST3 UNDEFINED HUMAN UNDEFINED N-(3-((3-ethoxy-4-methoxyphenylamino)methyl)phenyl)benzo[d]thiazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57859 MOR UNDEFINED HUMAN UNDEFINED (-)-1-[(1R,2S,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo-[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone 1000 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58115 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 25.1 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58371 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5678 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58627 hERG CLONED HUMAN 3H-N-Me-Dofetilide MRS5698 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58883 nAChR CLONED HUMAN 3H-Epibatidine Nicotine 4.4 Harris A, et al., 2015 Jan 15, 2025 Jan 15, 2025
59139 5-HT1A CLONED HUMAN 3H-WAY100635 CHLORPROMAZINE 3000 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59395 D2 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-2'-formyl-4-biphenylcarboxamide 3100 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59907 5-HT7 CLONED HUMAN 3H-LSD 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60163 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60419 GABAA CLONED HUMAN FNZ CM-A-87 1000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60675 GABAA CLONED HUMAN FNZ SPH-38 5.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60931 GABAA CLONED HUMAN FNZ 3 EBC 6.43 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61187 GABAA CLONED HUMAN FNZ CM-A58 1012 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61443 GABAA CLONED HUMAN FNZ JYI-03 185.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61699 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine 200 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62211 NET CLONED HUMAN [3H] Nisoxetine 6-APB 574 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62467 M3 CLONED HUMAN 3H-QNB 4-methoxy-diphenidine 2397 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63235 GCCR CLONED HUMAN 125I-Glucagon Benzoxacole N-methylation 5000 Madsen, P et al., 1998 Jan 15, 2025 Jan 15, 2025
63491 D2 CLONED HUMAN 3H-N-Methylspiperone RISPERIDONE 1.9 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64003 5-HT6 CLONED HUMAN 3H-LSD 2-[5-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-diethyl-2-oxoacetamide 224.4 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64259 5-HT2A CLONED HUMAN 3H-KETANSERIN PROCHLORPERAZINE 7.24436 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64515 D2 CLONED HUMAN 3H-N-Methylspiperone MOLINDONE 63.0957 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65027 H1 FR. CORTEX HUMAN 3H-MEPYRAMINE HALOPERIDOL 2500 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
65283 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073A (R Enriched) 15 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65540 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-1788 0.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65796 GABAA CLONED HUMAN [3H] Flunitrazepam RY-053 15 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66308 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Finazine 5.7 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66564 Alpha1B CLONED HUMAN 3H-PRAZOSIN 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66820 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67076 5-HT1A CLONED HUMAN 3H-WAY100635 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67332 DOR CLONED HUMAN 3H-DADLE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 29, 2025
67588 5-HT2C KIDNEY HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol 298 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67844 5-HT7 CLONED HUMAN 3H-5CT (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 349 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
2564 5-HT2A CORTEX HUMAN 3H-SPIPERONE TIMOLOL >10000 PEROUTKA, 1988 Jan 15, 2025 Jan 15, 2025
68356 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 307.1 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
3332 D3 CLONED HUMAN 3H-YM 09151-2 YOHIMBINE 2489 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68868 SST1 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 19.9526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69124 H4 CLONED HUMAN 3H-Histamine VUF4614 25.1189 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 427 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4100 KOR CLONED HUMAN 3H-U69,593 DPDPE-OH >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69636 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4356 5-HT6 CLONED HUMAN 3H-LSD SUMATRIPTAN 2600 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69892 D1 CLONED HUMAN 3H-SCH23390 4-[1-(4-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4612 SLC6A3 CLONED HUMAN 3H-DA UPTAKE MAZINDOL 60 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4868 5-HT2B CLONED HUMAN 3H-5HT RAUWOLSCINE 14.3 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70404 5-HT1A CLONED HUMAN 3H-WAY100635 MRP5063 5.7 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5124 5-HT2B CLONED HUMAN 3H-5HT DOF 227 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70660 M2 CLONED HUMAN 3H-QNB MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5380 5-HT2B CLONED HUMAN 3H-5HT SPIPERONE 1584.89 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
71172 D4 CLONED HUMAN 3H-Methylspiperone HALOPERIDOL 30.3 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5892 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE p-AMINOCLONIDINE 4.5 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71428 5-HT1E CLONED HUMAN 3H-5HT 4-acetoxy-N,N-diallyltryptamine 467 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6660 5-HT1E CLONED HUMAN 3H-5HT PINDOLOL,(+/-) >10000 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72196 D5 CLONED HUMAN 3H-SCH23390 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6916 5-HT2A CLONED HUMAN 3H-KETANSERIN HALOPERIDOL 25 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72708 Alpha1B CLONED HUMAN 3H-PRAZOSIN naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7428 MOR CLONED HUMAN 3H-DAMGO Naloxonazine 0.05 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72964 5-HT6 CLONED HUMAN 3H-LSD catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7684 GABAA CLONED HUMAN 3H-MUSCIMOL Muscimol 5.75 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7940 GABAA CLONED HUMAN 3H-RO-15-1788 CGS 8216, 1 17 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8196 GABAA CLONED HUMAN 3H-RO-15-1788 44 3000 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
8452 SST5 CLONED HUMAN 125I-Tyr3-octreotide CST17 0.14 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8708 SST2 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.09 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8964 SST1 CLONED HUMAN 125I-SRIF-28 MK 678 1000 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74500 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74756 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75012 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9732 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl 0.2 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75268 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75524 5-HT2B CLONED HUMAN 3H-LSD propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75780 Alpha1B CLONED HUMAN 3H-PRAZOSIN 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76036 D5 CLONED HUMAN 3H-SCH23390 Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76292 M4 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76548 5-HT1E CLONED HUMAN 3H-5-HT (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76804 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77060 5-HT7 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11780 H1 FR. CORTEX HUMAN 3H-doxepin PROCHLORPERAZINE 19 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77316 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77572 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77828 D2 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12548 Neutrophil HUMAN 3H-LTB4 CGS 23130 8 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78084 H1 CLONED HUMAN 3H-PYRILAMINE (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78340 M1 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78596 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78852 DOR CLONED HUMAN 3H-DADLE (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79108 5-HT5A CLONED HUMAN 3H-LSD (±)-2,5-Dimethoxy-4-methylamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79364 Alpha1A CLONED HUMAN 3H-PRAZOSIN LYSERGIC ACID 1127.7 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14084 CLONED HUMAN 3H-LTD4 Montelukast >10000 Heise CE, et al., 2000 Jan 15, 2025 Jan 15, 2025
79620 NET CLONED HUMAN 3H-Nisoxetine EMDT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14340 5-HT2B CLONED HUMAN 3H-LSD Nor-d-fenfluramine 27 FITZGERALD LW, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
79876 M5 CLONED HUMAN 3H-QNB (±)-3,4-Methylenedioxyamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80132 CLONED HUMAN 3H-VASOPRESSIN LYSERGIC ACID >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14852 TP Washed Platelets HUMAN 3H-SQ 29548 U44069 4.4 Hedberg, A, et al., 1988 Jan 15, 2025 Jan 15, 2025
80388 5-HT4 CLONED HUMAN 3H-GR113808 (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15108 CLONED HUMAN 3H-PGE2 AGN 191088 >10000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80644 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80900 5-HT2A CLONED HUMAN 3H-KETANSERIN (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 3593 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15876 5-HT7 CLONED HUMAN 3H-5HT SPIPERONE 109.64 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81412 H1 CLONED HUMAN 3H-PYRILAMINE methyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate 2758 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16132 D1 CLONED HUMAN 3H-SCH23390 PERGOLIDE 1363 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81924 DAT CLONED HUMAN 3H-WIN 35,428 (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 15, 2025
16644 Y4 CLONED HUMAN 125I-hPP Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26, Pro34]-NPY 31.4 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
82180 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 35.8 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82436 5-HT4 CLONED HUMAN 3H-GR113808 (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17156 5-HT2A BRAIN HUMAN 3H-KETANSERIN Quetiapine 31 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82692 5-HT1E CLONED HUMAN 3H-5-HT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82948 A3 CHO cells HUMAN 3H-PSB-11 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
17668 CLONED HUMAN 125I-VIP VIP [D-Ser2] 1.9 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83204 5-HT2A CLONED HUMAN 125I-DOI DMT 210 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83460 M3 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.891251 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83716 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 8396 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83972 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 4300 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84228 MOR CLONED HUMAN 3H-DAMGO (±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 1783 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84484 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84740 KOR CLONED HUMAN 3H-U69593 (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19460 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Gly10 3.3 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84996 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85252 GPR8 recombinant HUMAN 125I-NPW-23 Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 15, 2025
86020 DAT CLONED HUMAN 3H-WIN 35,428 (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
86276 Sigma 2 CLONED HUMAN 3H-DTG JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
87556 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
22276 A3 CLONED HUMAN 125I-Aba 6 90.3 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87812 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€3,4â€difluoroâ€Nâ€(2â€phenylethyl)aniline 114 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22532 5-HT2C CLONED HUMAN 3H-MESULERGINE SL650155 4780 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
22788 H2 CLONED HUMAN 3H-TIOTIDINE D-homocysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88580 M1 CLONED HUMAN 3H-QNB 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88836 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23556 H3 CLONED HUMAN 3H-NAMH A-317920 93.3254 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
89092 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 17.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
24068 5-HT2A CLONED HUMAN UNDEFINED OLANZAPINE 3 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89604 M1 CLONED HUMAN 3H-NMS 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89860 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 631 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90116 D1 CLONED HUMAN 3H-SCH23390 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24836 D4 CLONED HUMAN 3H-NMSP CLOZAPINE 39 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25092 Alpha1B CLONED HUMAN 125I-HEAT Quetiapine 39 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90628 A2A CLONED HUMAN 3H-MSX-2 N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 82.5 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25348 M3 CLONED HUMAN 3H-QNB ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90884 Alpha1D CHO cells HUMAN 3H-PRAZOSIN 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 28.1838 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
25604 5-HT7 CLONED HUMAN 3H-LSD Methcathinone, (-) 1000 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
91140 A2A H9 HUMAN 3H-NECA Ethyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
25860 Alpha2C CLONED HUMAN 3H-CLONIDINE Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91396 CB1 CLONED HUMAN 3H-CP55940 O-6212 86 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26116 M4 CLONED HUMAN 3H-QNB Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91652 A3 CLONED HUMAN 3H-PSB-11 N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide 8.23 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26372 Alpha2C CLONED HUMAN 3H-CLONIDINE Hyperoside >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91908 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3,4-dichloro-phenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26628 MOR CLONED HUMAN 3H-Diprenorphine Pseudohypericin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92164 5-HT6 CLONED HUMAN 3H-LSD N-{1-[2-(3-Fluorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 1779 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26884 M1 CLONED HUMAN 3H-QNB xanomeline 79.4328 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92420 DOR CLONED HUMAN 3H-DADLE (8S,9R,10S)-15,16-epoxy-9α-hydroxylabda-5,13(16),14-trien-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27140 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92676 M5 CLONED HUMAN 3H-QNB 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27396 Beta1 CLONED HUMAN 3H-CGP-12177 Ropinirole >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92932 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27652 D4 CLONED HUMAN 3H-NMSP MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93188 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 60 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
27908 5-HT2A CLONED HUMAN 3H-KETANSERIN DMT,5-OH 145 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28164 D1 CLONED HUMAN 3H-SCH23390 METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93700 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 5.62 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28420 nAChR CLONED HUMAN 3H-Epibatidine ERGOTAMINE >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
94212 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29188 SST2 CLONED HUMAN UNDEFINED L-779,976 0.05 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94724 5-HT2A CLONED HUMAN 3H-KETANSERIN 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94980 D2 CLONED HUMAN 3H-N-Methylspiperone 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29700 D4 CLONED HUMAN UNDEFINED HALOPERIDOL 6.5 Liao Y, et.al., 1999 Jan 15, 2025 Jan 27, 2025
29956 H4 CLONED HUMAN 3H-Histamine (7-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 7 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95748 5-HT7 CLONED HUMAN 3H-LSD Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96004 DAT CLONED HUMAN 3H-WIN 35,428 N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96260 Alpha1D CLONED HUMAN 3H-PRAZOSIN 3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96516 5-HT4 CLONED HUMAN [3H]GR113808 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31236 D4 CLONED HUMAN 3H-NMSP MDL 100907 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96772 D1 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31492 Alpha1B CLONED HUMAN UNDEFINED (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 3162.28 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97028 Beta1 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97284 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 2.33 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97540 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 449.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97796 H1 Sf9 HUMAN 3H-MEPYRAMINE UR-AK59 6000 Xie, S. et. al., 2006 Jan 15, 2025 Jan 15, 2025
98052 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide 780 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98308 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline 915 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98564 5-HT2B CLONED HUMAN [3H]-LSD 2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 1166 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98820 5-HT1D CLONED HUMAN 125I-aminopotentidine 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine 871 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33540 5-HT5A CLONED HUMAN 3H-LSD Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99076 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99332 D2 CLONED HUMAN [3H]N-methylspiperone 1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(quinolin-6-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol 424 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34052 P2X3 CLONED HUMAN 3H-A-317491 AP2A >10000 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99588 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthin 0.499 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99844 Alpha1A CLONED HUMAN [125I] HEAT (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 4600 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100100 D2 CLONED HUMAN 3H-N-Methylspiperone Cariprazine 18 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100356 5-HT7 CLONED HUMAN 3H-LSD Melperone HCl 346 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100868 nAChR CLONED HUMAN Functional Decamethonium >10000 Kuo YP, et al., 2005 Jan 15, 2025 Jan 29, 2025
35588 CLONED HUMAN 3H-SQ 29548 LATANOPROST (Free Acid) >10000 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35844 SLC6A4 CLONED HUMAN 3H-PAROXETINE 5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 16 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101380 5-HT7 CLONED HUMAN 3H-5-CT 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 119 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36100 COX-2 whole blood assay (WBA) HUMAN Functional Meloxicam sodium 2100 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101636 5-HT3 CLONED HUMAN [3H]GR65630 Perospirone >10000 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101892 D4 CLONED HUMAN [3H]-N-methylspiperone Ziprasidone 39 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36612 D2 CLONED HUMAN 3H-SPIPERONE OLANZAPINE 78 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102148 NET CLONED HUMAN [3H]Nisoxetine NEMONAPRIDE 473 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37892 MPP-2 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-trimethylsilyl-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 1500 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38660 UNDEFINED HUMAN 3H-hypoxanthine N-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-2-hydroxy-3-[2-(3-methoxy-phenyl)-ethylcarbamoyl]-propyl}-2,4,6-trifluoro-benzamide 308 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39172 D4 CLONED HUMAN R-SAT OLANZAPINE 31 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39428 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39684 5-HT2B CLONED HUMAN 3H-5HT mCPP 40.738 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39940 5-HT2C CLONED HUMAN Functional BW-723C86 501.187 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
40708 mGluR5 CLONED HUMAN Functional 3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one 816 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41220 CLONED HUMAN 125I-Chemokine 5-(4-(3,4-Dichlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41988 M1 CLONED HUMAN 3H-QNB BUPROPION >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42244 CLONED HUMAN 125I-[Ile]Motilin [Bpa5,Ile13]Motilin 50 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
43012 FRK CLONED HUMAN 3H-Staurosporine ZD-6474 480 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43268 CDK5 CLONED HUMAN 3H-Staurosporine Roscovitine 2000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43524 FGFR2 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
43780 TEK CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44036 STK16 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44292 STK6 CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44548 FGFR3 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44804 PKMYT1 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45060 PDGFRB CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45316 CLONED HUMAN Functional Indirubin-3monoxime 190 Bain J, et al., 2003 Jan 15, 2025 Jan 15, 2025
45572 NET CLONED HUMAN 3H-Nisoxetine Desmethylsertraline 390 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45828 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46084 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46596 SLC6A3 CLONED HUMAN 3H-WIN 35,428 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46852 M5 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47364 GRIA4 CLONED HUMAN 3H-AMPA LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47620 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 0.8 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47876 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
48132 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48644 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49668 SST2 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50180 mGluR3 CLONED HUMAN Functional L-CCG-I 380 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50436 SLC6A4 CLONED HUMAN 3H-CITALOPRAM 4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenylthio)benzylamine 13 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
50948 MOR UNDEFINED HUMAN UNDEFINED Nalbuphine 0.89 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51460 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide 1 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51972 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1.85 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52228 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-5-yloxy)-3-(cyclohexylamino)propan-2-ol 3000 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52484 SLC6A3 UNDEFINED HUMAN UNDEFINED 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline 46 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52996 CB2 UNDEFINED HUMAN UNDEFINED N-cyclohexyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide >10000 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53252 D2 UNDEFINED HUMAN UNDEFINED 1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 55 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53764 H1 UNDEFINED HUMAN UNDEFINED 4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one 1014 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54276 SLC6A4 UNDEFINED HUMAN UNDEFINED 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 4.1 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54532 A3 UNDEFINED HUMAN UNDEFINED N-(2-hydroxyethyl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 422 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54788 D2 UNDEFINED HUMAN UNDEFINED N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine 610 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55044 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide 13 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55300 DOR UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 1790 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
56324 A1 UNDEFINED HUMAN UNDEFINED 2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 379 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56580 DOR UNDEFINED HUMAN UNDEFINED 4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 443 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56836 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-(N-tert-Butylamino)-3',4'-dichloropropiophenone 5400 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57092 D2 UNDEFINED HUMAN UNDEFINED OPC-14597 2.8 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
57348 A1 UNDEFINED HUMAN UNDEFINED 8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-methyl-1-propyl-3,7-dihydro-purine-2,6-dione 0.295 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57604 SST3 UNDEFINED HUMAN UNDEFINED 6-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]thiazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57860 DOR UNDEFINED HUMAN UNDEFINED (+)-1-{(1S,2S,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one 1000 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58116 5-HT2A CLONED HUMAN 125I-DOI N-(2-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 2.34 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58372 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5697 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58628 hERG CLONED HUMAN 3H-N-Me-Dofetilide MRS5678 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58884 nAChR CLONED HUMAN 3H-Epibatidine Camel Snus extract 3.8 Harris A, et al., 2015 Jan 15, 2025 Jan 15, 2025
59140 5-HT2A CLONED HUMAN 3H-KETANSERIN CYPROHEPTADINE 1.67 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59396 D4 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4'-formyl-4-biphenylcarboxamide 70 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59908 D1 CLONED HUMAN 3H-SCH23390 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60164 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2S,3R,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiazol-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60420 GABAA CLONED HUMAN FNZ WY-S-2 4000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60676 GABAA CLONED HUMAN FNZ SPH-38 2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60932 GABAA CLONED HUMAN FNZ 3 EBC 25.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61188 GABAA CLONED HUMAN FNZ QH-II-067a 3000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61444 GABAA CLONED HUMAN FNZ RY-054 126 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61700 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(4-methoxyphenyl)propan-1-amine 267 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62212 SLC6A3 CLONED HUMAN [3H] WIN35428 6-APB 565 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62468 M3 CLONED HUMAN 3H-QNB 2-Cl-diphenidine 615 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63236 GCCR CLONED HUMAN 125I-Glucagon 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethanone >10000 Madsen, P et al., 1998 Jan 15, 2025 Jan 15, 2025
63492 D3 CLONED HUMAN 3H-N-Methylspiperone RISPERIDONE 13 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64004 5-HT6 CLONED HUMAN 3H-LSD N,N-Diethyl-2-[5-(naphthalene-1-sulfonylamino)-1H-indol-3-yl]-2-oxoacetamide 1000 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64260 5-HT2A CLONED HUMAN 3H-KETANSERIN Quetiapine 218.776 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64516 D2 CLONED HUMAN 3H-N-Methylspiperone OLANZAPINE 20.4174 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65284 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073A (R Enriched) 1.18 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65541 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-1788 148 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65797 GABAA CLONED HUMAN [3H] Flunitrazepam RY-053 1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66053 CLONED HUMAN 3H-VASOPRESSIN Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
66309 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Finazine 2.2 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66565 Alpha1D CLONED HUMAN 3H-PRAZOSIN 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66821 5-HT3 CLONED HUMAN 3H-GR113808 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67077 5-HT1B CLONED HUMAN 3H-5-CT 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67589 A1 KIDNEY HUMAN 3H-N6 -phenylisopropyladenosine (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol 298 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67845 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
3333 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Amphetamine,(+) 6606 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68869 SST2 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 19.9526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69125 H4 CLONED HUMAN 3H-Histamine VUF4616 12.5893 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 105 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4101 KOR CLONED HUMAN 3H-U69,593 DSLET-OH >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69637 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 3-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4357 5-HT6 CLONED HUMAN 3H-LSD KETANSERIN 2800 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69893 D1 CLONED HUMAN 3H-SCH23390 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4613 SLC6A3 CLONED HUMAN 3H-DA UPTAKE Amphetamine,(+) 116 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4869 5-HT2B CLONED HUMAN 3H-5HT RITANSERIN 1.64 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70405 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) MRP5063 7.9 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5125 5-HT2B CLONED HUMAN 3H-5HT DOC 31.8 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70661 M3 CLONED HUMAN 3H-QNB MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5381 5-HT2B CLONED HUMAN 3H-5HT KETANSERIN 630.95 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
71173 D4 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 54 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5893 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE CLONIDINE 7.2 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71429 5-HT2A CLONED HUMAN 125I-DOI 4-acetoxy-N,N-diallyltryptamine 565 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6661 5-HT1E CLONED HUMAN 3H-5HT ZACOPRIDE >10000 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72197 D2 CLONED HUMAN 3H-N-Methylspiperone 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6917 5-HT2A CLONED HUMAN 3H-KETANSERIN ISOCLOZAPINE 1.45 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72709 Alpha1D CLONED HUMAN 3H-PRAZOSIN naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7429 MOR CLONED HUMAN 3H-DAMGO ETORPHINE - HCI 0.23 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72965 5-HT7 CLONED HUMAN 3H-LSD catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7685 GABAA CLONED HUMAN 3H-MUSCIMOL Thiomuscimol 37.15 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7941 GABAA CLONED HUMAN 3H-RO-15-1788 2 4 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8197 GABAA CLONED HUMAN 3H-RO-15-1788 45 1000 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
8453 SST5 CLONED HUMAN 125I-Tyr3-octreotide CST14 0.45 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8709 SST2 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.1 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8965 SST1 CLONED HUMAN 125I-SRIF-28 RC 160 158.48 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74501 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74757 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75013 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9733 MT2 CLONED HUMAN 125I-Iodomelatonin Luzindole,5-Methoxy 0.25 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75269 Sigma 2 CLONED HUMAN 3H-DTG ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75525 5-HT2C CLONED HUMAN 3H-MESULERGINE propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75781 Alpha1D CLONED HUMAN 3H-PRAZOSIN 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76037 D2 CLONED HUMAN 3H-N-Methylspiperone Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76293 M5 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76549 5-HT2A CLONED HUMAN 3H-KETANSERIN (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76805 5-HT3 CLONED HUMAN 3H-GR-65630 (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11525 CLONED HUMAN 3H-SUBSTANCE P Substance P 0.1 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
77061 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
11781 H1 FR. CORTEX HUMAN 3H-doxepin FLUPHENAZINE 21 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77317 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77573 Beta 2 CLONED HUMAN 3H-CGP-12177 (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77829 D3 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12549 Neutrophil HUMAN 3H-LTB4 CGS 23131 15 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78085 5-HT1D CLONED HUMAN 3H-Cimetidine (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78341 M2 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78597 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2420 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78853 KOR CLONED HUMAN 3H-U69593 (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 100 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79109 5-HT5A CLONED HUMAN 3H-LSD (±)-3,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79365 Alpha1A CLONED HUMAN 3H-PRAZOSIN cis-2a 528.8 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14085 CLONED HUMAN 3H-LTD4 LTB4 >10000 Heise CE, et al., 2000 Jan 15, 2025 Jan 15, 2025
79621 CLONED HUMAN 3H-CLONIDINE (±)-2,5-Dimethoxy-4-bromoamphetamine 1596.1 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14341 5-HT2B CLONED HUMAN 3H-LSD l-norfenfluramine 65 FITZGERALD LW, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
79877 M5 CLONED HUMAN 3H-QNB (±)-3,4-Methylenedioxymethamphetamine 6330 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80133 CLONED HUMAN 3H-VASOPRESSIN cis-2a >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14853 TP Washed Platelets HUMAN 3H-SQ 29548 U46619 3.6 Hedberg, A, et al., 1988 Jan 15, 2025 Jan 15, 2025
80389 5-HT5A CLONED HUMAN 3H-LSD (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15109 CLONED HUMAN 3H-PGE2 PGF2Alpha,17-phenyl 168 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80645 5-HT1B CLONED HUMAN 3H-5-CT (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15365 5-HT1B CLONED HUMAN 3H-5HT LYSERGOL 1.2 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80901 5-HT2B CLONED HUMAN 3H-LSD (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 353 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81157 H1 CLONED HUMAN 3H-PYRILAMINE N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
15877 5-HT7 CLONED HUMAN 3H-5HT DHE 9.12 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81413 H1 CLONED HUMAN 3H-PYRILAMINE 4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole 3265 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16133 D1 CLONED HUMAN 3H-SCH23390 N-0437 2172 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81925 DOR CLONED HUMAN 3H-DADLE (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16645 M1 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.035 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82181 Alpha1B CLONED HUMAN 3H-PRAZOSIN 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 152.5 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82437 5-HT5A CLONED HUMAN 3H-LSD (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17157 5-HT2A BRAIN HUMAN 3H-KETANSERIN RISPERIDONE 0.15 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82693 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17669 CLONED HUMAN 125I-VIP VIP [D-Asp3] 1.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83205 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DMT 450 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83461 M4 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.676083 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83717 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2284 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83973 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 194 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84229 5-HT2B CLONED HUMAN 3H-LSD (±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 8306 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
84485 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19205 SLC6A4 Platelets HUMAN 3H-5HT LY248685 0.35 Wong DT et al., 1993 Jan 15, 2025 Jan 15, 2025
84741 DOR CLONED HUMAN 3H-DADLE methyl (±)-(S)-2-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)-2-phenylacetate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19461 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Arg11 0.55 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84997 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86021 D1 CLONED HUMAN 3H-SCH23390 (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
87557 Alpha1B CLONED HUMAN 3H-PRAZOSIN 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
22277 A3 CLONED HUMAN 125I-Aba 8 30 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87813 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€3,4â€difluoroâ€Nâ€(2â€phenylethyl)aniline 79 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22533 5-HT1B CLONED HUMAN 3H-GR-125743 SL650155 5500 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
88069 A1 CLONED HUMAN 3H-CCPA H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22789 H2 CLONED HUMAN 3H-TIOTIDINE L-homocysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23045 nAChR CLONED HUMAN 3H-Epibatidine DL-homocysteine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88581 5-HT7 CLONED HUMAN 3H-LSD 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 90 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88837 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89093 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 3345 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
24069 5-HT2A CLONED HUMAN UNDEFINED RACLOPRIDE 4000 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89605 M1 CLONED HUMAN 3H-NMS 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89861 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 953 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90117 D1 CLONED HUMAN 3H-SCH23390 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24837 5-HT1B CLONED HUMAN 3H-GR-125743 CLOZAPINE 398 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90629 A2B CLONED HUMAN 3H-PSB-603 Preladenant (SCH420814) 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25349 M2 CLONED HUMAN 3H-QNB ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90885 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 42.658 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
25605 Alpha2C CLONED HUMAN 3H-CLONIDINE PRAZOSIN 14.5 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
91141 A3 CHO cells HUMAN 3H-HEMADO Ethyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate 1300 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
25861 nAChR CLONED HUMAN 3H-Epibatidine Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
91397 CB1 CLONED HUMAN 3H-SR144528 O-6212 41 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26117 D1 CLONED HUMAN 3H-SCH23390 Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91653 A3 CLONED HUMAN 3H-PSB-11 N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 83.3 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26373 Alpha2C CLONED HUMAN 3H-CLONIDINE Miquelianin 4063 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91909 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3-trifluoromethylphenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26629 MOR CLONED HUMAN 3H-Diprenorphine Hypericin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92165 5-HT6 CLONED HUMAN 3H-LSD 5-Chloro-N-{1-[2-(2,3-dichlorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 91 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26885 M2 CLONED HUMAN 3H-QNB xanomeline 125.893 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92421 DOR CLONED HUMAN 3H-DADLE 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27141 5-HT1A CLONED HUMAN 3H-8-OH-DPAT AL-37350A >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92677 M5 CLONED HUMAN 3H-QNB 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27397 Beta2 CLONED HUMAN 3H-CGP-12177 Roxindole 933.254 Millan MJ, et al., 2002 Jan 15, 2025 Jan 28, 2025
92933 A3 CLONED HUMAN 125I-AB-MECA 2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
93189 D3 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 370 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
27909 5-HT2A CLONED HUMAN 3H-DOB DMT,5-OH 15 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28165 D2 CLONED HUMAN 3H-NMSP METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93701 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 6.05 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28677 5-HT5A CLONED HUMAN 3H-LSD ARIPIPRAZOLE 1240 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94213 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29189 SST2 CLONED HUMAN UNDEFINED L-797,591 1875 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94725 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94981 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29957 H4 CLONED HUMAN 3H-Histamine (5,7- Dichloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 11 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95749 5-HT5A CLONED HUMAN 3H-LSD Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96005 DAT CLONED HUMAN 3H-WIN 35,428 tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96261 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30981 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96517 5-HT5A CLONED HUMAN [3H]-LSD 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31237 Alpha2A CLONED HUMAN 3H-CLONIDINE MDL 100907 1900 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96773 D1 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31493 D2 CLONED HUMAN 125I-IODOSULPRIDE (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 1584.89 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97029 Beta2 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97285 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 171 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97541 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 517.1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98053 CB2 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide 6000 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
32773 NK1 CLONED HUMAN 3H-Sar9,Met(O2)11-Substance P SCH 206272 1.3 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98309 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 272 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98565 5-HT2B CLONED HUMAN [3H]-LSD 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one 614 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33285 CB2 CLONED HUMAN 3H-CP-55940 nimesulide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98821 H3 CLONED HUMAN 3H-Alpha-methylhistamine 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
99077 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99333 D2 CLONED HUMAN [3H]N-methylspiperone 1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(naphtha-len-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol >10000 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34053 P2X3 CLONED HUMAN 3H-A-317491 A-317491 10.8 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99589 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine 3.99 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99845 Alpha1A CLONED HUMAN [125I] HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100101 5-HT1A CLONED HUMAN 3H-WAY100635 Quetiapine 267 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100357 5-HT7 CLONED HUMAN 3H-LSD Blonanserin 1010 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100869 nAChR CLONED HUMAN Functional Pancuronium >10000 Kuo YP, et al., 2005 Jan 15, 2025 Jan 29, 2025
35589 CLONED HUMAN 3H-SQ 29548 Latanoprost (Isopropyl Ester) >10000 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35845 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide 20 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101381 D2 CLONED HUMAN 3H-RACLOPRIDE 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 30 Zareba P, et al., 2019 Jan 15, 2025 Jan 28, 2025
36101 COX-2 whole blood assay (WBA) HUMAN Functional nimesulide 1900 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101637 D1 CLONED HUMAN [3H]SCH23390 Perospirone 65 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101893 D5 CLONED HUMAN [3H]SCH23390 Ziprasidone 136 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36613 D2 CLONED HUMAN 3H-SPIPERONE RISPERIDONE 6.4 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102149 DAT CLONED HUMAN [3H]WIN35428 NEMONAPRIDE 2368 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37893 MPP-9 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-trimethylsilyl-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 550 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38661 UNDEFINED HUMAN 3H-hypoxanthine N-{(1S,2S)-2-Hydroxy-3-[2-(3-methoxy-phenyl)-ethylcarbamoyl]-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl}-2,4,6-trifluoro-benzamide 693 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39173 D4 CLONED HUMAN R-SAT L 745,870 1.8 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39429 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39685 5-HT2B CLONED HUMAN 3H-5HT METHYLERGONOVINE 0.457088 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40709 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one 44 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41221 CLONED HUMAN 125I-Chemokine 5-(4-Hydroxy-4-p-tolylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41989 M1 CLONED HUMAN 3H-QNB DESIPRAMINE 110 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42245 CLONED HUMAN 125I-[Ile]Motilin Motilin 2.3 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
43013 FRK CLONED HUMAN 3H-Staurosporine CI-1033 8100 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43269 CDK5 CLONED HUMAN 3H-Staurosporine Flavopiridol 43 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43525 FGFR3 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43781 KIAA0551 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44037 STK18 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44293 AURKC CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44549 FGR CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44805 MAPK14 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45061 PHKG1 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45317 LCK CLONED HUMAN Functional Indirubin-3monoxime 300 Bain J, et al., 2003 Jan 15, 2025 Jan 15, 2025
45573 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Desmethylsertraline 129 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45829 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46085 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46597 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46853 M5 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47365 GRIA4 CLONED HUMAN 3H-AMPA LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47621 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-(4-fluorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 26 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47877 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 0.7 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
48133 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 29 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48645 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 9.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49669 SST3 CLONED HUMAN 125I-LTT-SST-28 L-796,778 127 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50181 mGluR3 CLONED HUMAN Functional 1S, 3R-ACPD 5400 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50437 SLC6A4 CLONED HUMAN 3H-CITALOPRAM MADAM 1.65 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
50949 KOR UNDEFINED HUMAN UNDEFINED 17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol 0.079 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51461 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide 4.3 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51717 NR3C1 UNDEFINED HUMAN UNDEFINED dexamethasone 2.1 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51973 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 3.11 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52229 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-4-yloxy)-4-(cyclohexylamino)butan-2-ol 125 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52485 SLC6A3 UNDEFINED HUMAN UNDEFINED (S)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline 102 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52997 CB2 UNDEFINED HUMAN UNDEFINED N-butyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide 9400 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53253 D2 UNDEFINED HUMAN UNDEFINED 1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 54 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53765 H1 UNDEFINED HUMAN UNDEFINED 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one 188.6 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54277 SLC6A4 UNDEFINED HUMAN UNDEFINED 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 90.7 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54533 A3 UNDEFINED HUMAN UNDEFINED 8-(4-(1-(4-(5-chlorobenzo[d]thiazol-2-yl)piperazin-1-yl)-2-methyl-1-oxopropan-2-yloxy)phenyl)-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione 1000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54789 D2 UNDEFINED HUMAN UNDEFINED N-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine 4100 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55045 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide 139 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55301 DOR UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one 3103 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
56325 A1 UNDEFINED HUMAN UNDEFINED 2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione >10000 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56581 DOR UNDEFINED HUMAN UNDEFINED 4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 75 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56837 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-(N-tert-Butylamino)-3'-chloro-4'-methylpropiophenone 5100 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57093 D2 UNDEFINED HUMAN UNDEFINED (S)-3-(3-Methanesulfonyl-phenyl)-1-propyl-piperidine 755 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
57349 A1 UNDEFINED HUMAN UNDEFINED (4-(furan-2-yl)-2-(2-(thiophen-2-yl)ethylamino)thiazol-5-yl)(phenyl)methanone 6700 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57605 SST3 UNDEFINED HUMAN UNDEFINED N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)thiazolo[5,4-b]pyridin-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57861 DOR UNDEFINED HUMAN UNDEFINED (-)-1-{(1R,2R,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one 1000 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58117 5-HT2A CLONED HUMAN 125I-DOI N-(3-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 1.48 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58373 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS3558 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58629 hERG CLONED HUMAN 3H-N-Me-Dofetilide MRS5697 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58885 nAChR CLONED HUMAN 3H-Epibatidine Kodiak extract 3.9 Harris A, et al., 2015 Jan 15, 2025 Jan 15, 2025
59141 5-HT1A CLONED HUMAN 3H-WAY100635 CYPROHEPTADINE 50 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59397 D2 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4'-formyl-4-biphenylcarboxamide 3700 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59909 D2 CLONED HUMAN 3H-NMSP 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60165 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-4-(2-((Ferrocen-yl)ethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60421 GABAA CLONED HUMAN FNZ WY-S-2 300 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60677 GABAA CLONED HUMAN FNZ XHE-I-093 2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60933 GABAA CLONED HUMAN FNZ 3 EBC 28.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61189 GABAA CLONED HUMAN FNZ QH-II-067a 199 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61445 GABAA CLONED HUMAN FNZ RY-054 1.3 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61701 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2,5-dimethoxyphenyl)propan-1-amine 919 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62213 Serotonin CLONED HUMAN [3H] Citalopram 6-APB 4046 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62469 M4 CLONED HUMAN 3H-QNB 2-Cl-diphenidine 828 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63493 5-HT1A CLONED HUMAN 3H-WAY100635 RISPERIDONE 420 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64005 5-HT6 CLONED HUMAN 3H-LSD N,N-Diethyl-2-oxo-2-[5-(quinoline-8-sulfonylamino)-1H-indol-3-yl]-acetamide 1000 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64261 5-HT2A CLONED HUMAN 3H-KETANSERIN REMOXIPRIDE 5248.07 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64517 D2 CLONED HUMAN 3H-N-Methylspiperone PERPHENAZINE 0.977237 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65285 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073A (R Enriched) 140 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65542 GABAA CLONED HUMAN [3H] Flunitrazepam MLT-I-70 1.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65798 GABAA CLONED HUMAN [3H] Flunitrazepam RY-053 46 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66054 V1B CLONED HUMAN 3H-VASOPRESSIN Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
66310 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Finazine 4.4 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66566 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 367 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66822 5-HT5A CLONED HUMAN 3H-LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67078 5-HT1D CLONED HUMAN 3H-5-CT 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67590 A2A KIDNEY HUMAN 3H-2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol 2690 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2310 5-HT3 AMYGDALA HUMAN 3H-ZACOPRIDE FLUPHENAZINE >10000 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67846 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3334 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SKF 82958 1781 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68870 SST3 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 25.1189 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69126 H4 CLONED HUMAN 3H-Histamine VUF4617 12.5893 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT OLANZAPINE 2063 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4102 KOR CLONED HUMAN 3H-U69,593 DADLE-OH >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69638 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-MXP 1909 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4358 5-HT6 CLONED HUMAN 3H-LSD QUIPAZINE 3600 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69894 D1 CLONED HUMAN 3H-SCH23390 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4614 SLC6A3 CLONED HUMAN 3H-DA UPTAKE DICLOFENSINE,(-) 606 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4870 5-HT2B CLONED HUMAN 3H-5HT SPIPERONE 592 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70406 Sigma 2 CLONED HUMAN 3H-DTG MRP5063 6.5 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5126 5-HT2B CLONED HUMAN 3H-5HT DOB 26.9 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70662 M4 CLONED HUMAN 3H-QNB MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5382 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 7.94 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
71174 D4 CLONED HUMAN 3H-N-Methylspiperone SYA013 60.6 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5894 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE WB 4101 17 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71430 5-HT2B CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 63 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6662 5-HT1E CLONED HUMAN 3H-5HT PAPP >10000 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72198 D3 CLONED HUMAN 3H-N-Methylspiperone 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6918 5-HT2A CLONED HUMAN 3H-KETANSERIN LOXAPINE 10.2 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72710 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7430 MOR CLONED HUMAN 3H-DAMGO LEVORPHANOL-tartarate 0.08 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72966 Alpha1A CLONED HUMAN 3H-PRAZOSIN catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7686 GABAA CLONED HUMAN 3H-MUSCIMOL THIP 165.95 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7942 GABAA CLONED HUMAN 3H-RO-15-1788 3 100 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8198 SST5 CLONED HUMAN 125I-LTT-SST-28 somatostatin-28 0.19 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
8454 SST5 CLONED HUMAN 125I-Tyr3-octreotide CST14-Tyr10 0.22 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8710 SST2 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.15 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8966 SST1 CLONED HUMAN 125I-SRIF-28 RC 160II 100 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74502 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74758 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75014 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9734 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Hydroxy 5.5 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75270 SERT CLONED HUMAN 3H-CITALOPRAM ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75526 5-HT3 CLONED HUMAN 3H-GR-65630 propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75782 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76038 D3 CLONED HUMAN 3H-N-Methylspiperone Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76294 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76550 5-HT2B CLONED HUMAN 3H-LSD (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76806 5-HT5A CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77062 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
11782 H1 FR. CORTEX HUMAN 3H-doxepin TRIFLUOPERAZINE 62 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77318 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77574 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77830 D4 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12550 Neutrophil HUMAN 3H-LTB4 CGS 23356 116 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78086 H3 CLONED HUMAN 3H-Alpha-methylhistamine (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78342 M3 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78598 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78854 MOR CLONED HUMAN 3H-DAMGO (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79110 5-HT5A CLONED HUMAN 3H-LSD (±)-2,5-Dimethoxy-4-ethylamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79366 Alpha1A CLONED HUMAN 3H-PRAZOSIN R,R-2b 5187 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79622 CLONED HUMAN 3H-CLONIDINE (±)-3,4-Methylenedioxyamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79878 M5 CLONED HUMAN 3H-QNB 3,4,5-Trimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80134 CLONED HUMAN 3H-VASOPRESSIN R,R-2b >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80390 5-HT6 CLONED HUMAN 3H-LSD (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15110 CLONED HUMAN 3H-PGE2 PGF2 Alpha, 1-isopropyl ester 5000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80646 5-HT1D CLONED HUMAN 3H-5-CT (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15366 5-HT1B CLONED HUMAN 3H-5HT 5-CT 1.58 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80902 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 678 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81158 5-HT1D CLONED HUMAN 3H-Cimetidine N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81414 D2 CLONED HUMAN 3H-N-Methylspiperone 4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16134 D1 CLONED HUMAN 3H-SCH23390 NPA 1816 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81670 D1 CLONED HUMAN 3H-SCH23390 (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
16646 M1 CLONED HUMAN 3H-QNB BENZTROPINE 0.231 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82182 Alpha1D CLONED HUMAN 3H-PRAZOSIN 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 72.2 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82438 5-HT6 CLONED HUMAN 3H-LSD (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17158 5-HT2A BRAIN HUMAN 3H-KETANSERIN 9-OH-risperidone 1.21 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82694 5-HT2B CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine 3169 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17670 CLONED HUMAN 125I-VIP VIP [D-Ala4] 1.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83206 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOM >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83462 M5 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.660693 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83718 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2961 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83974 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2825 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84486 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19206 SLC6A4 Platelets HUMAN 3H-5HT LY248686 0.2 Wong DT et al., 1993 Jan 15, 2025 Jan 15, 2025
84742 MOR CLONED HUMAN 3H-DAMGO methyl (±)-(S)-2-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)-2-phenylacetate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19462 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Arg14 330 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84998 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86022 D5 CLONED HUMAN 3H-SCH23390 (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86534 A1 CLONED HUMAN 3H-CCPA 1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 124 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87558 Alpha1D CLONED HUMAN 3H-PRAZOSIN 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
22278 A3 CLONED HUMAN 125I-Aba 9 922 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87814 5-HT2A CLONED HUMAN 3H-KETANSERIN 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 295 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22534 5-HT2B CLONED HUMAN 3H-LSD SL650155 1560 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
88070 A1 CLONED HUMAN 3H-CCPA 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22790 H2 CLONED HUMAN 3H-TIOTIDINE L-cysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23046 nAChR CLONED HUMAN 3H-Epibatidine L-cysteine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88582 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 308.2 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88838 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89094 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89350 D2 CLONED HUMAN 3H-RACLOPRIDE N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 4346 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
24070 5-HT2A CLONED HUMAN UNDEFINED REMOXIPRIDE 5200 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89606 M2 CLONED HUMAN 3H-NMS 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89862 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 9520 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90118 D1 CLONED HUMAN 3H-SCH23390 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24838 M1 CLONED HUMAN 3H-QNB CLOZAPINE 14 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25094 M4 CLONED HUMAN 3H-QNB Quetiapine 542 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90630 A2B CLONED HUMAN 3H-PSB-603 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 365 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25350 nAChR CLONED HUMAN 3H-Epibatidine ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
90886 Alpha1A CHO cells HUMAN 3H-PRAZOSIN 8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 30.903 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
91142 A1 CHO cells HUMAN 3H-CCPA Ethyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
91398 CB1 CLONED HUMAN 3H-SR144528 O-6617 43 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26118 D4 CLONED HUMAN 3H-NMSP Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91654 A3 CLONED HUMAN 3H-PSB-11 N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide 25.4 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
91910 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (4-methylphenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26630 MOR CLONED HUMAN 3H-Diprenorphine Hyperforin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92166 5-HT6 CLONED HUMAN 3H-LSD 5-Chloro-N-{1-[2-(2,5-dichlorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 225 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26886 M3 CLONED HUMAN 3H-QNB xanomeline 39.8107 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92422 DOR CLONED HUMAN 3H-DADLE 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27142 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOI,(-) 3843 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92678 M4 CLONED HUMAN 3H-QNB 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27398 Beta1 CLONED HUMAN 3H-CGP-12177 Roxindole 2691.53 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92934 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27654 D2 CLONED HUMAN 3H-NMSP MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93190 D4 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 19 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
27910 5-HT2A CLONED HUMAN 3H-KETANSERIN DOM 306 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93702 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 32 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28422 nAChR CLONED HUMAN 3H-Epibatidine ERGOTAMINE >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
28678 5-HT6 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 570 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94214 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-isopropoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29190 SST2 CLONED HUMAN UNDEFINED CH275 1000 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94726 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94982 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29958 H4 CLONED HUMAN 3H-Histamine (5,7-Dimethyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 31 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95750 5-HT6 CLONED HUMAN 3H-LSD Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96006 DAT CLONED HUMAN 3H-WIN 35,428 4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96262 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96518 5-HT6 CLONED HUMAN [3H]-LSD 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31238 Alpha2B CLONED HUMAN 3H-CLONIDINE MDL 100907 270.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96774 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31494 D3 CLONED HUMAN 125I-IODOSULPRIDE (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 1258.93 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97030 Beta3 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97286 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 370 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97542 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 49.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98054 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide 3 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
32774 NK1 CLONED HUMAN 3H-Sar9,Met(O2)11-Substance P CP 99994 0.27 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98310 D2 CLONED HUMAN [3H]-N-methylspiperone 5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 138 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98566 5-HT2B CLONED HUMAN [3H]-LSD 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one 273 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98822 H4 CLONED HUMAN 3H-Histamine 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33542 Alpha1A CLONED HUMAN 3H-PRAZOSIN Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99078 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99334 D2 CLONED HUMAN [3H]N-methylspiperone 4-(4-([1,1’-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol >10000 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34054 P2X3 CLONED HUMAN 3H-A-317491 ATP,TNP 7.5 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99590 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine 1.68 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99846 Alpha2A CLONED HUMAN [125I] iodoclonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 4700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100102 5-HT2A CLONED HUMAN 3H-KETANSERIN Quetiapine 352 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100358 5-HT7 CLONED HUMAN 3H-LSD RS-(+/-)-Sulpriride 1085 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100870 5-HT1A CLONED HUMAN 3H-WAY100635 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1) 85.7 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 15, 2025
35590 CLONED HUMAN 3H-SQ 29548 ILOPROST 6487 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35846 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide 2.7 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 48 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36102 COX-2 whole blood assay (WBA) HUMAN Functional ROFECOXIB 840 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101638 D2 CLONED HUMAN [3H]-N-methylspiperone Perospirone 14 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101894 SERT CLONED HUMAN [3H] Citalopram Ziprasidone 165 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36614 D2 CLONED HUMAN 3H-SPIPERONE mirtazepine 5454 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102150 MOR CLONED HUMAN [3H]DAMGO NEMONAPRIDE 3698 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37894 MPP-2 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 12 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38662 UNDEFINED HUMAN 3H-hypoxanthine N-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-cyclohexylcarbamoyl-2-hydroxypropyl]-2,4,6-trifluorobenzamide 230 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39174 D4 CLONED HUMAN R-SAT ARIPIPRAZOLE 1000 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39430 V1A CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39686 5-HT2B CLONED HUMAN 3H-5HT MK 212 616.595 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39942 5-HT2A CLONED HUMAN Functional BW-723C86 100 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
40710 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one 344 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41222 CLONED HUMAN 125I-Chemokine 5-(4-Benzyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41990 M1 CLONED HUMAN 3H-QNB Desmethylsertraline 1650 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42246 CLONED HUMAN 125I-[Ile]Motilin [D-Bpa5,Ile13]Motilin 420 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
43014 FYN CLONED HUMAN 3H-Staurosporine Staurosporine 51 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43270 CLK1 CLONED HUMAN 3H-Staurosporine EKB-569 1000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43526 FGR CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43782 TTK CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44038 STK3 mouse CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44294 BMX CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44550 FLT3 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44806 MAPK P38 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45062 PRKACA CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45318 CLONED HUMAN Functional Indirubin-3monoxime 380 Bain J, et al., 2003 Jan 15, 2025 Jan 15, 2025
45574 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Dothiepin 8.6 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45830 5-HT2B CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46086 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46598 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46854 M5 CLONED HUMAN 3H-QNB PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47366 GRIA4 CLONED HUMAN 3H-AMPA LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47622 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.2 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
48134 Y2 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 0.03 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48646 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49670 SST4 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50182 mGluR3 CLONED HUMAN Functional Quisqualate >10000 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50438 SLC6A4 CLONED HUMAN 3H-CITALOPRAM 4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 7 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
50950 KOR UNDEFINED HUMAN UNDEFINED (5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate 0.13 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51462 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide 25 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51718 NR3C1 UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline 4.4 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51974 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1.64 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52230 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(adamantan-1-ylamino)-4-(1H-indol-4-yloxy)-butan-2-ol 551 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52486 SLC6A3 UNDEFINED HUMAN UNDEFINED 2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 29 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52998 CB2 UNDEFINED HUMAN UNDEFINED N-cyclopentyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide 7400 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53254 D2 UNDEFINED HUMAN UNDEFINED 1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 127 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53766 H1 UNDEFINED HUMAN UNDEFINED 1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one 911.8 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54278 SLC6A4 UNDEFINED HUMAN UNDEFINED 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 189 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54534 A3 UNDEFINED HUMAN UNDEFINED 8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-3-ethyl-1-propyl-1H-purine-2,6(3H,7H)-dione 1070 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54790 D2 UNDEFINED HUMAN UNDEFINED N-(4-Propylaminobutyl)-4-biphenylcarboxamide >10000 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55046 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide 161 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55302 DOR UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 795 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
56326 A3 UNDEFINED HUMAN UNDEFINED NECA 20 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56582 DOR UNDEFINED HUMAN UNDEFINED (4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol 1350 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56838 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-Piperidino-3'-chloropropiophenone 4760 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57350 A1 UNDEFINED HUMAN UNDEFINED N-[5-pyridin-4-yl-4-(3,4,5-trimethoxyphenyl)thiazol-2-yl]acetamide >10000 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57606 SST3 UNDEFINED HUMAN UNDEFINED N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57862 DOR UNDEFINED HUMAN UNDEFINED (+)-1-{(1S,2R,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one 1000 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58118 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(3-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 6.76 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58374 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5676 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58630 hERG CLONED HUMAN 3H-N-Me-Dofetilide MRS3558 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
59142 5-HT1A CLONED HUMAN 3H-WAY100635 HALOPERIDOL 3500 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59398 D4 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4-(2-thienyl)benzamide 3 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59910 D3 CLONED HUMAN 3H-NMSP 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60166 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-4-(2-(Cyclopropylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60422 GABAA CLONED HUMAN FNZ WY-S-2 300 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60678 GABAA CLONED HUMAN FNZ XHE-I-093 7.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60934 GABAA CLONED HUMAN FNZ 3 EBC 826 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61190 GABAA CLONED HUMAN FNZ QH-II-067a 52 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61446 GABAA CLONED HUMAN FNZ RY-054 27 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61702 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine 146 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62214 NET CLONED HUMAN [3H] Nisoxetine Desoxypipradol 281 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62470 M4 CLONED HUMAN 3H-QNB Diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63494 5-HT2A CLONED HUMAN 3H-Ketaserin RISPERIDONE 0.22 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64006 5-HT6 CLONED HUMAN 3H-LSD N-[3-(3-Diethylaminopropyl)-1H-indol-5-yl]naphthalene-2-sulfonamide 163 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64262 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.436516 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64518 D2 CLONED HUMAN 3H-N-Methylspiperone PIMOZIDE 6.76083 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65030 H1 FR. CORTEX HUMAN 3H-MEPYRAMINE THIORIDAZINE 22 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
65286 GABAA CLONED HUMAN [3H] Flunitrazepam SH-I-030 14.42 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65543 GABAA CLONED HUMAN [3H] Flunitrazepam MLT-I-70 1.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65799 GABAA CLONED HUMAN [3H] Flunitrazepam YT-6 15.31 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66055 V2 CLONED HUMAN 3H-VASOPRESSIN Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
66311 Beta1 CLONED HUMAN I-125-Pindolol Finazine 1254 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66567 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 363 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66823 5-HT6 CLONED HUMAN 3H-LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67079 5-HT1E CLONED HUMAN 3H-5-HT 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67591 A3 KIDNEY HUMAN I-125-N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamide (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol 3240 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2311 5-HT3 HIPPOCAMPUS HUMAN 3H-ZACOPRIDE FLUPHENAZINE >10000 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67847 5-HT7 CLONED HUMAN 3H-5-CT S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 142 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
2567 5-HT2A CORTEX HUMAN 3H-KETANSERIN TMA,3,4,5- >10000 SADZOT ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3335 5-HT1A CLONED HUMAN 3H-8-OH-DPAT APOMORPHINE 4929 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68871 SST4 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 1.99526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69127 H4 CLONED HUMAN 3H-Histamine VUF4742 125.893 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Quetiapine 431 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4103 KOR CLONED HUMAN 3H-U69,593 DELTORPHIN-II >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69639 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4359 5-HT6 CLONED HUMAN 3H-LSD MESULERGINE 3800 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69895 D2 CLONED HUMAN 3H-N-Methylspiperone 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4615 SLC6A3 CLONED HUMAN 3H-DA UPTAKE COCAINE 743 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4871 5-HT2B CLONED HUMAN 3H-5HT SPIROXATRINE 475 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70407 Sigma 2 CLONED HUMAN 3H-DTG MRP4268 6.5 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5127 5-HT2B CLONED HUMAN 3H-5HT DOI 20 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70663 M5 CLONED HUMAN 3H-QNB MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5383 5-HT2B CLONED HUMAN 3H-5HT RITANSERIN 5.01 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
70919 5-HT2B CLONED HUMAN 3H-LSD 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 742 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
71175 D4 CLONED HUMAN 3H-N-Methylspiperone SYA16263 30.5 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5895 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE PRAZOSIN 23 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71431 5-HT2C CLONED HUMAN UNKNOWN 4-acetoxy-N,N-diallyltryptamine 1515 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6663 5-HT1E CLONED HUMAN 3H-5HT 5-CT,DP >10000 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72199 D4 CLONED HUMAN 3H-N-Methylspiperone 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6919 5-HT2A CLONED HUMAN 3H-KETANSERIN MELPERONE 280 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72711 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7431 MOR CLONED HUMAN 3H-DAMGO Methadone 0.72 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72967 Alpha1B CLONED HUMAN 3H-PRAZOSIN catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7687 GABAA CLONED HUMAN 3H-MUSCIMOL P4S 107.15 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7943 GABAA CLONED HUMAN 3H-RO-15-1788 5 40 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8199 SST5 CLONED HUMAN 125I-LTT-SST-28 LTT-SST-28 0.11 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
8455 SST5 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.06 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8711 SST2 CLONED HUMAN 125I-Tyr3-octreotide BIM 23014 0.28 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8967 SST1 CLONED HUMAN 125I-SRIF-28 L-362,855 100 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74503 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74759 Beta2 CLONED HUMAN 3H-CGP12177 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75015 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9735 MT2 CLONED HUMAN 125I-Iodomelatonin 8-M-ADOT 4.1 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75271 NET CLONED HUMAN 3H-Nisoxetine ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75527 5-HT5A CLONED HUMAN 3H-LSD propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75783 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76039 D4 CLONED HUMAN 3H-N-Methylspiperone Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76295 Sigma 2 CLONED HUMAN 3H-DTG (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76551 5-HT2C CLONED HUMAN 3H-MESULERGINE (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76807 5-HT6 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77063 Alpha1D CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
11783 H1 FR. CORTEX HUMAN 3H-doxepin d-Butaclamol 390 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77319 Beta 1 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77575 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77831 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
12551 Neutrophil HUMAN 3H-LTB4 CGS 24115 131 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78087 H4 CLONED HUMAN 3H-Histamine (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78343 M4 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78599 Sigma 2 CLONED HUMAN 3H-DTG (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78855 MOR CLONED HUMAN 3H-DAMGO (±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79111 5-HT5A CLONED HUMAN 3H-LSD 2,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79367 Alpha1A CLONED HUMAN 3H-PRAZOSIN S,S-2c 850.2 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79623 CLONED HUMAN 3H-CLONIDINE (±)-3,4-Methylenedioxymethamphetamine 219.7 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79879 M5 CLONED HUMAN 3H-QNB 4-Bromo-2,5-dimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80135 CLONED HUMAN 3H-VASOPRESSIN S,S-2c >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80391 5-HT7 CLONED HUMAN 3H-LSD (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 799 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15111 PTGFR CLONED HUMAN 3H-PGF2Alpha PGF2Alpha 48 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80647 5-HT1E CLONED HUMAN 3H-5-HT (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15367 5-HT1B CLONED HUMAN 3H-5HT 5-Methoxytryptamine 33.88 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80903 5-HT3 CLONED HUMAN 3H-GR-65630 (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81159 H3 CLONED HUMAN 3H-Alpha-methylhistamine N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81415 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 15, 2025
16135 D1 CLONED HUMAN 3H-SCH23390 5-Hydroxy Tryptamine 9690 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81671 D5 CLONED HUMAN 3H-SCH23390 (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81927 H1 CLONED HUMAN 3H-PYRILAMINE (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16647 M1 CLONED HUMAN 3H-QNB Biperidine 0.48 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82183 D1 CLONED HUMAN 3H-SCH23390 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82439 5-HT7 CLONED HUMAN 3H-LSD (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17159 5-HT2A BRAIN HUMAN 3H-KETANSERIN SERTINDOLE 0.14 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82695 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82951 A2B CHO cells HUMAN 3H-PSB-603 (R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
17671 CLONED HUMAN 125I-VIP VIP [D-Val5] 6.2 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83207 5-HT2A CLONED HUMAN 125I-DOI DOM 4.3 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83463 M5 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 20.893 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83719 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83975 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-N-(3-bromobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3275 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84231 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 9747 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84487 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84743 MOR CLONED HUMAN 3H-DAMGO benzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19463 GPR145 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH hMCH 2.9 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84999 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86023 D2 CLONED HUMAN 3H-Alpha-methylhistamine (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86535 A2A CLONED HUMAN 3H-MSX-2 1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 542 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87559 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
87815 5-HT7 CLONED HUMAN 3H-5-CT 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 19 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22535 5-HT2A CLONED HUMAN 3H-KETANSERIN SL650155 1320 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
88071 A1 CLONED HUMAN 3H-CCPA 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22791 H2 CLONED HUMAN 3H-TIOTIDINE D-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23047 nAChR CLONED HUMAN 3H-Epibatidine D-homocysteine thiolactone >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88583 5-HT7 CLONED HUMAN 3H-LSD 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 291 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88839 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89095 A3 HeLa HUMAN 3H-NECA N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 3.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89351 5-HT6 CLONED HUMAN 3H-LSD N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 3441 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24071 5-HT2A CLONED HUMAN UNDEFINED Quetiapine 110 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89607 M3 CLONED HUMAN 3H-NMS 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89863 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 59.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90119 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24839 Alpha1A CLONED HUMAN 125I-HEAT CLOZAPINE 1.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25095 SLC6A3 CLONED HUMAN 3H-GBR 12935 Quetiapine >10000 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90631 A2B CLONED HUMAN 3H-PSB-603 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 225 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25351 5-HT5A CLONED HUMAN 3H-LSD ZOTEPINE 29 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90887 Alpha1B CHO cells HUMAN 3H-PRAZOSIN 8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 109.648 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
25607 5-HT5A CLONED HUMAN 3H-LSD COCAINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91143 A2A CHO cells HUMAN 3H-NECA Ethyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
25863 5-HT1B CLONED HUMAN 3H-GR-125743 Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91399 CB1 CLONED HUMAN 3H-CP55940 O-6617 85 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26119 nAChR CLONED HUMAN 3H-Epibatidine Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
91655 A3 CLONED HUMAN 3H-PSB-11 N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide 1000 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
91911 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (4-chlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26631 MOR CLONED HUMAN 3H-Diprenorphine Miquelianin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92167 5-HT6 CLONED HUMAN 3H-LSD 5-Chloro-N-{1-[2-(phenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 957 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26887 M4 CLONED HUMAN 3H-QNB xanomeline 19.9526 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92423 KOR CLONED HUMAN 3H-U69593 (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92679 M3 CLONED HUMAN 3H-QNB 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27399 Beta1 CLONED HUMAN 3H-CGP-12177 Talipexole >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92935 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine 110 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27655 D1 CLONED HUMAN 3H-SCH23390 MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27911 5-HT2A CLONED HUMAN 3H-DOB DOM 21 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93703 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 348 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28423 CLONED HUMAN 3H-Quisqualate Quisqualate 10 Mutel V, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93959 D2 CLONED HUMAN 3H-SPIPERONE compound 42 21 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
28679 5-HT7 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 10.3 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94215 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,4,5-trimethoxyamphetamine >10000 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29191 SST2 CLONED HUMAN UNDEFINED BIM 23197 0.19 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94727 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94983 D3 CLONED HUMAN 3H-N-Methylspiperone 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29959 H4 CLONED HUMAN 3H-Histamine (5,7-Difluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 14 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95751 5-HT7 CLONED HUMAN 3H-LSD Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96007 DAT CLONED HUMAN 3H-WIN 35,428 2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96263 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96519 5-HT7 CLONED HUMAN [3H]-LSD 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 29, 2025
31239 Alpha2C CLONED HUMAN 3H-CLONIDINE MDL 100907 1442 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96775 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31495 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) 1584.89 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97031 D1 CLONED HUMAN [3H]SCH23390 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97287 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 235 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97543 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 31.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98055 CB2 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide 420 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
32775 NK1 CLONED HUMAN 3H-Sar9,Met(O2)11-Substance P SR 142801 291 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98311 D2 CLONED HUMAN [3H]-N-methylspiperone 5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 853 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98567 5-HT2B CLONED HUMAN [3H]-LSD 4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile 152 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33287 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98823 MOR CLONED HUMAN 3H-DAMGO 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33543 Alpha1B CLONED HUMAN 3H-PRAZOSIN Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99079 Beta1 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99335 D2 CLONED HUMAN [3H]N-methylspiperone 4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 789 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34055 P2X3 CLONED HUMAN 3H-A-317491 A-317344 1220 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99591 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine 0.683 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99847 Alpha2C CLONED HUMAN [125I] iodoclonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 240 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100103 5-HT2B CLONED HUMAN 3H-LSD Quetiapine 86 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100359 DAT CLONED HUMAN 3H-WIN 35,428 Cariprazine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100615 CGRP CLONED HUMAN Functional N2-(3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100871 Beta2 CLONED HUMAN 3H-CGP-12177 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1) 2 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 28, 2025
35591 CLONED HUMAN 3H-SQ 29548 CICAPROST 1340 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35847 SLC6A4 CLONED HUMAN 3H-PAROXETINE 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide 23 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101383 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 578 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36103 COX-2 whole blood assay (WBA) HUMAN Functional valeryl salicylate 2300 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101639 D3 CLONED HUMAN [3H]-N-methylspiperone Perospirone 7.7 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101895 NET CLONED HUMAN [3H]Nisoxetine Ziprasidone 69 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36615 D2 CLONED HUMAN 3H-SPIPERONE MIANSERIN 2197 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102151 DOR CLONED HUMAN [3H]DADLE NEMONAPRIDE >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37895 MPP-9 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 19 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38663 UNDEFINED HUMAN 3H-hypoxanthine N-[(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-cyclohexylcarbamoyl-2-hydroxy-propyl]-2,4,6-trifluoro-benzamide 214 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39175 D4 CLONED HUMAN R-SAT N-DESMETHYLCLOZAPINE 70 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39431 V2 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39687 5-HT2B CLONED HUMAN 3H-5HT ORG-12962 91.2011 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40711 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one 84 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41223 CLONED HUMAN 125I-Chemokine 5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41991 M1 CLONED HUMAN 3H-QNB Dothiepin 18 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42247 CLONED HUMAN 125I-[Ile]Motilin [L-Bpa5,Ile13]Motilin 50 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
43015 FYN CLONED HUMAN 3H-Staurosporine Gleevec 5500 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43271 CLK1 CLONED HUMAN 3H-Staurosporine SU11248 100 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43527 FLT3 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43783 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44039 STK36 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44295 CaMK CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44551 FLT4 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44807 MAPK12 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45063 PTK2 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45319 CDK2 CLONED HUMAN Functional kenpaullone 670 Bain J, et al., 2003 Jan 15, 2025 Jan 28, 2025
45575 NET CLONED HUMAN 3H-Nisoxetine Dothiepin 46 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45831 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46087 Alpha2A CLONED HUMAN 3H-CLONIDINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46599 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46855 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47367 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
47623 ADK recombinant HUMAN Functional 4-N-(4-Chlorophenyl)amino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2.7 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
48135 Y2 CLONED HUMAN 3H-Propionyl-NPY PP, human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48647 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49671 SST5 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50183 mGluR3 CLONED HUMAN Functional L-CCG-I 2100 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50439 SLC6A4 CLONED HUMAN 3H-CITALOPRAM 5-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 8 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
50951 KOR UNDEFINED HUMAN UNDEFINED 17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate 0.12 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51463 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide 36 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51719 NR3C1 UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline 1.1 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51975 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1.82 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52231 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(1H-indol-4-yloxy)-1-(cyclohexylamino)butan-2-ol 872 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52487 Alpha2A UNDEFINED HUMAN UNDEFINED IDAZOXAN 8 Hagihara K et al., 2007 Jan 15, 2025 Jan 15, 2025
52999 CB2 UNDEFINED HUMAN UNDEFINED N-(4-fluorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide 4000 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53255 D2 UNDEFINED HUMAN UNDEFINED 1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 2.4 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53767 H1 UNDEFINED HUMAN UNDEFINED 4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 259.6 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54279 SLC6A4 UNDEFINED HUMAN UNDEFINED 2-(2-Dimethylaminomethyl-phenylsulfanyl)-5-methyl-phenylamine 2.03 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54535 A3 UNDEFINED HUMAN UNDEFINED 8-[4-(4-benzylpiperazide-1-sulfonyl)phenyl]-1-propylxanthine 1000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54791 D2 UNDEFINED HUMAN UNDEFINED N-(4-Dipropylaminobutyl)-4-biphenylcarboxamide 9700 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55047 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-methylthiophenyl)-1-piperazinehexanamide 12 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55303 DOR UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 2639 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
56071 CB1 UNDEFINED HUMAN UNDEFINED HU-210 1.5 Fan H et al., 2009 Jan 15, 2025 Jan 15, 2025
56327 A3 UNDEFINED HUMAN UNDEFINED 2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione 209 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56583 KOR UNDEFINED HUMAN UNDEFINED 4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 9500 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56839 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-(N-tert-Butylamino)-4'-bromo-5'-methylpropiophenone 4600 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025