The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 1,001-2,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
50947MORUNDEFINEDHUMANUNDEFINEDNaltrexone0.23Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51459Alpha1AUNDEFINEDHUMANUNDEFINED3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51971KORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine1.72Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522275-HT1AUNDEFINEDHUMANUNDEFINED1-(adamantan-1-ylamino)-3-(1H-indol-5-yloxy)-propan-2-ol833Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52483SLC6A2UNDEFINEDHUMANUNDEFINED2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline106Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52995CB2UNDEFINEDHUMANUNDEFINED5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide6000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53251D2UNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea4.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53763H1UNDEFINEDHUMANUNDEFINEDRISPERIDONE19Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54275SLC6A4UNDEFINEDHUMANUNDEFINED3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile73.7Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54531A3UNDEFINEDHUMANUNDEFINEDN-(4-cyanophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide570Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54787D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine210Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550435-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide8.2Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55299DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one538Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
56323A1UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione1410Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56579DORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol807Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56835SLC6A2UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)propiophenone5700Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57091D2UNDEFINEDHUMANUNDEFINEDBifeprunox0.04Pettersson F et al., 2010Jan 15, 2025Jan 15, 2025
57347A1UNDEFINEDHUMANUNDEFINED(E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-propenone0.49Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57603SST3UNDEFINEDHUMANUNDEFINEDN-(3-((3-ethoxy-4-methoxyphenylamino)methyl)phenyl)benzo[d]thiazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57859MORUNDEFINEDHUMANUNDEFINED(-)-1-[(1R,2S,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo-[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone1000Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581155-HT2ACLONEDHUMAN3H-KETANSERINN-(2-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate25.1Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58371H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5678>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58627hERGCLONEDHUMAN3H-N-Me-DofetilideMRS5698>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58883nAChRCLONEDHUMAN3H-EpibatidineNicotine4.4Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
591395-HT1ACLONEDHUMAN3H-WAY100635CHLORPROMAZINE3000Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59395D2CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-2'-formyl-4-biphenylcarboxamide3100Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
599075-HT7CLONEDHUMAN3H-LSD4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60163A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60419GABAACLONEDHUMANFNZCM-A-871000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60675GABAACLONEDHUMANFNZSPH-385.4Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60931GABAACLONEDHUMANFNZ3 EBC6.43Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61187GABAACLONEDHUMANFNZCM-A581012Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61443GABAACLONEDHUMANFNZJYI-03185.4Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
616995-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine200Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62211NETCLONEDHUMAN[3H] Nisoxetine6-APB574Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62467M3CLONEDHUMAN3H-QNB4-methoxy-diphenidine2397Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
63235GCCRCLONEDHUMAN125I-GlucagonBenzoxacole N-methylation5000Madsen, P et al., 1998Jan 15, 2025Jan 15, 2025
63491D2CLONEDHUMAN3H-N-MethylspiperoneRISPERIDONE1.9Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640035-HT6CLONEDHUMAN3H-LSD2-[5-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-diethyl-2-oxoacetamide224.4Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642595-HT2ACLONEDHUMAN3H-KETANSERINPROCHLORPERAZINE7.24436Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64515D2CLONEDHUMAN3H-N-MethylspiperoneMOLINDONE63.0957Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65027H1FR. CORTEXHUMAN3H-MEPYRAMINEHALOPERIDOL2500Chang, R et., 1978Jan 15, 2025Jan 15, 2025
65283GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-073A (R Enriched)15Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65540GABAACLONEDHUMAN[3H] FlunitrazepamRo15-17880.6Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65796GABAACLONEDHUMAN[3H] FlunitrazepamRY-05315Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66308Alpha2ACLONEDHUMAN3H-RAUWOLSCINEFinazine5.7Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66564Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
668205-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
670765-HT1ACLONEDHUMAN3H-WAY1006351-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67332DORCLONEDHUMAN3H-DADLE1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 29, 2025
675885-HT2CKIDNEYHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol298Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
678445-HT7CLONEDHUMAN3H-5CT(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline349Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
25645-HT2ACORTEXHUMAN3H-SPIPERONETIMOLOL>10000PEROUTKA, 1988Jan 15, 2025Jan 15, 2025
68356nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid307.1Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
3332D3CLONEDHUMAN3H-YM 09151-2YOHIMBINE2489TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68868SST1CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH219.9526Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69124H4CLONEDHUMAN3H-HistamineVUF461425.1189Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693805-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE427Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4100KORCLONEDHUMAN3H-U69,593DPDPE-OH>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69636Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43565-HT6CLONEDHUMAN3H-LSDSUMATRIPTAN2600KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69892D1CLONEDHUMAN3H-SCH233904-[1-(4-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4612SLC6A3CLONEDHUMAN3H-DA UPTAKEMAZINDOL60PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48685-HT2BCLONEDHUMAN3H-5HTRAUWOLSCINE14.3WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704045-HT1ACLONEDHUMAN3H-WAY100635MRP50635.7Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51245-HT2BCLONEDHUMAN3H-5HTDOF227NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70660M2CLONEDHUMAN3H-QNBMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
53805-HT2BCLONEDHUMAN3H-5HTSPIPERONE1584.89BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
71172D4CLONEDHUMAN3H-MethylspiperoneHALOPERIDOL30.3Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5892Alpha2BCLONEDHUMAN3H-RAUWOLSCINEp-AMINOCLONIDINE4.5WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714285-HT1ECLONEDHUMAN3H-5HT4-acetoxy-N,N-diallyltryptamine467Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66605-HT1ECLONEDHUMAN3H-5HTPINDOLOL,(+/-)>10000ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72196D5CLONEDHUMAN3H-SCH233902-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69165-HT2ACLONEDHUMAN3H-KETANSERINHALOPERIDOL25SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72708Alpha1BCLONEDHUMAN3H-PRAZOSINnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7428MORCLONEDHUMAN3H-DAMGONaloxonazine0.05Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
729645-HT6CLONEDHUMAN3H-LSDcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7684GABAACLONEDHUMAN3H-MUSCIMOLMuscimol5.75Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7940GABAACLONEDHUMAN3H-RO-15-1788CGS 8216, 117He X, et al., 1999Jan 15, 2025Jan 27, 2025
8196GABAACLONEDHUMAN3H-RO-15-1788443000Huang Q, et al., 1999Jan 15, 2025Jan 27, 2025
8452SST5CLONEDHUMAN125I-Tyr3-octreotideCST170.14Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8708SST2CLONEDHUMAN125I-Tyr3-octreotideSomatostatin-140.09Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8964SST1CLONEDHUMAN125I-SRIF-28MK 6781000Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
745005-HT2BCLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74756Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75012D4CLONEDHUMAN3H-N-Methylspiperone(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9732MT2CLONEDHUMAN125I-IodomelatoninMelatonin,6-Cl0.2Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75268Sigma 1CLONEDHUMAN3H-Pentazocine(+)ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
755245-HT2BCLONEDHUMAN3H-LSDpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75780Alpha1BCLONEDHUMAN3H-PRAZOSIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76036D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76292M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765485-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768045-HT2CCLONEDHUMAN3H-MESULERGINE(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
770605-HT7CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11780H1FR. CORTEXHUMAN3H-doxepinPROCHLORPERAZINE19Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77316Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77572Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77828D2CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12548NeutrophilHUMAN3H-LTB4CGS 231308Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78084H1CLONEDHUMAN3H-PYRILAMINE(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78340M1CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78596NETCLONEDHUMAN3H-Nisoxetine(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78852DORCLONEDHUMAN3H-DADLE(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791085-HT5ACLONEDHUMAN3H-LSD(±)-2,5-Dimethoxy-4-methylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79364Alpha1ACLONEDHUMAN3H-PRAZOSINLYSERGIC ACID1127.7Ray TS 2010 Jan 15, 2025Jan 28, 2025
14084CLONEDHUMAN3H-LTD4Montelukast>10000Heise CE, et al., 2000Jan 15, 2025Jan 15, 2025
79620NETCLONEDHUMAN3H-NisoxetineEMDT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
143405-HT2BCLONEDHUMAN3H-LSDNor-d-fenfluramine27FITZGERALD LW, ET AL., 1999Jan 15, 2025Jan 15, 2025
79876M5CLONEDHUMAN3H-QNB(±)-3,4-Methylenedioxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80132CLONEDHUMAN3H-VASOPRESSINLYSERGIC ACID>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14852TPWashed PlateletsHUMAN3H-SQ 29548U440694.4Hedberg, A, et al., 1988Jan 15, 2025Jan 15, 2025
803885-HT4CLONEDHUMAN3H-GR113808(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15108CLONEDHUMAN3H-PGE2AGN 191088>10000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806445-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
809005-HT2ACLONEDHUMAN3H-KETANSERIN(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one3593Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
158765-HT7CLONEDHUMAN3H-5HTSPIPERONE109.64BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81412H1CLONEDHUMAN3H-PYRILAMINEmethyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate2758Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16132D1CLONEDHUMAN3H-SCH23390PERGOLIDE1363Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81924DATCLONEDHUMAN3H-WIN 35,428(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 15, 2025
16644Y4CLONEDHUMAN125I-hPPDes-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26, Pro34]-NPY31.4Mullins D et al., 2001Jan 15, 2025Jan 15, 2025
82180Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one35.8Besnard J et al 2012Jan 15, 2025Jan 28, 2025
824365-HT4CLONEDHUMAN3H-GR113808(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171565-HT2ABRAINHUMAN3H-KETANSERINQuetiapine31Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826925-HT1ECLONEDHUMAN3H-5-HT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82948A3CHO cellsHUMAN3H-PSB-111,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione>10000Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
17668CLONEDHUMAN125I-VIPVIP [D-Ser2]1.9Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832045-HT2ACLONEDHUMAN125I-DOIDMT210Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83460M3CLONEDHUMAN3H-NMS1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide0.891251Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83716NETCLONEDHUMAN3H-Nisoxetine(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide8396PDSP Certified DataJan 15, 2025Jan 15, 2025
83972KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide4300PDSP Certified DataJan 15, 2025Jan 28, 2025
84228MORCLONEDHUMAN3H-DAMGO(±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide1783PDSP Certified DataJan 15, 2025Jan 28, 2025
84484MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84740KORCLONEDHUMAN3H-U69593(±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19460GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Gly103.3Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84996KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85252GPR8recombinantHUMAN125I-NPW-23Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
86020DATCLONEDHUMAN3H-WIN 35,428(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86276Sigma 2CLONEDHUMAN3H-DTGJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
87556Alpha1ACLONEDHUMAN3H-PRAZOSIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
22276A3CLONEDHUMAN125I-Aba690.3Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878125-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline114Staron J et al 2016Jan 15, 2025Jan 15, 2025
225325-HT2CCLONEDHUMAN3H-MESULERGINESL6501554780Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
22788H2CLONEDHUMAN3H-TIOTIDINED-homocysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88580M1CLONEDHUMAN3H-QNB1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88836A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23556H3CLONEDHUMAN3H-NAMHA-31792093.3254Esbenshade TA, et al., 2003Jan 15, 2025Jan 15, 2025
89092A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide17.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
240685-HT2ACLONEDHUMANUNDEFINEDOLANZAPINE3Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89604M1CLONEDHUMAN3H-NMS3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89860nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride631Liu J et al 2010Jan 15, 2025Jan 29, 2025
90116D1CLONEDHUMAN3H-SCH233902-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24836D4CLONEDHUMAN3H-NMSPCLOZAPINE39PDSP Certified DataJan 15, 2025Jan 15, 2025
25092Alpha1BCLONEDHUMAN125I-HEATQuetiapine39Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90628A2ACLONEDHUMAN3H-MSX-2N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide82.5 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25348M3CLONEDHUMAN3H-QNBZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
90884Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane28.1838Franchini S et al 2014Jan 15, 2025Jan 28, 2025
256045-HT7CLONEDHUMAN3H-LSDMethcathinone, (-)1000Rothman RB, et al., 2003aJan 15, 2025Jan 15, 2025
91140A2AH9HUMAN3H-NECAEthyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
25860Alpha2CCLONEDHUMAN3H-CLONIDINEPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91396CB1CLONEDHUMAN3H-CP55940O-621286Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26116M4CLONEDHUMAN3H-QNBPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91652A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide8.23Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26372Alpha2CCLONEDHUMAN3H-CLONIDINEHyperoside>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91908A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3,4-dichloro-phenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26628MORCLONEDHUMAN3H-DiprenorphinePseudohypericin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921645-HT6CLONEDHUMAN3H-LSDN-{1-[2-(3-Fluorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide1779Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
26884M1CLONEDHUMAN3H-QNBxanomeline79.4328Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92420DORCLONEDHUMAN3H-DADLE(8S,9R,10S)-15,16-epoxy-9α-hydroxylabda-5,13(16),14-trien-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271405-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92676M5CLONEDHUMAN3H-QNB15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27396Beta1CLONEDHUMAN3H-CGP-12177Ropinirole>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
92932A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
27652D4CLONEDHUMAN3H-NMSPMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93188D2CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine60Lober S et al 2012Jan 15, 2025Jan 29, 2025
279085-HT2ACLONEDHUMAN3H-KETANSERINDMT,5-OH145Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28164D1CLONEDHUMAN3H-SCH23390METHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93700A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester5.62Federico S et al 2018Jan 15, 2025Jan 15, 2025
28420nAChRCLONEDHUMAN3H-EpibatidineERGOTAMINE>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
942125-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29188SST2CLONEDHUMANUNDEFINEDL-779,9760.05Patel YC, 1999Jan 15, 2025Jan 15, 2025
947245-HT2ACLONEDHUMAN3H-KETANSERIN5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94980D2CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29700D4CLONEDHUMANUNDEFINEDHALOPERIDOL6.5Liao Y, et.al., 1999Jan 15, 2025Jan 27, 2025
29956H4CLONEDHUMAN3H-Histamine(7-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone7Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957485-HT7CLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96004DATCLONEDHUMAN3H-WIN 35,428N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96260Alpha1DCLONEDHUMAN3H-PRAZOSIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
965165-HT4CLONEDHUMAN[3H]GR1138086-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31236D4CLONEDHUMAN3H-NMSPMDL 100907>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
96772D1CLONEDHUMAN[3H]SCH233904-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
31492Alpha1BCLONEDHUMANUNDEFINED(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)3162.28Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97028Beta1CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97284MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol2.33Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97540A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate449.3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97796H1Sf9HUMAN3H-MEPYRAMINEUR-AK596000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
98052CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide780Amato G et al 2019Jan 15, 2025Jan 28, 2025
98308D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline915Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985645-HT2BCLONEDHUMAN[3H]-LSD2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride1166Ofon E et al 2016aJan 15, 2025Jan 15, 2025
988205-HT1DCLONEDHUMAN125I-aminopotentidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine871Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
335405-HT5ACLONEDHUMAN3H-LSDNaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99076Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99332D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(quinolin-6-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol424Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34052P2X3CLONEDHUMAN3H-A-317491AP2A>10000Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99588A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthin0.499Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99844Alpha1ACLONEDHUMAN[125I] HEAT(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide4600Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
100100D2CLONEDHUMAN3H-N-MethylspiperoneCariprazine18PDSP Certified DataJan 15, 2025Jan 28, 2025
1003565-HT7CLONEDHUMAN3H-LSDMelperone HCl346PDSP Certified DataJan 15, 2025Jan 15, 2025
100868nAChRCLONEDHUMANFunctionalDecamethonium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
35588CLONEDHUMAN3H-SQ 29548LATANOPROST (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35844SLC6A4CLONEDHUMAN3H-PAROXETINE5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole16Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013805-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one119Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36100COX-2whole blood assay (WBA)HUMANFunctionalMeloxicam sodium2100Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
1016365-HT3CLONEDHUMAN[3H]GR65630Perospirone>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
101892D4CLONEDHUMAN[3H]-N-methylspiperoneZiprasidone39PDSP Certified DataMar 24, 2025Jul 28, 2026
36612D2CLONEDHUMAN3H-SPIPERONEOLANZAPINE78Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102148NETCLONEDHUMAN[3H]NisoxetineNEMONAPRIDE473PDSP Certified DataMar 25, 2025Jul 28, 2026
37892MPP-2CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-trimethylsilyl-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione1500Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38660UNDEFINEDHUMAN3H-hypoxanthineN-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-2-hydroxy-3-[2-(3-methoxy-phenyl)-ethylcarbamoyl]-propyl}-2,4,6-trifluoro-benzamide308Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39172D4CLONEDHUMANR-SATOLANZAPINE31Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39428CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396845-HT2BCLONEDHUMAN3H-5HTmCPP40.738Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
399405-HT2CCLONEDHUMANFunctionalBW-723C86501.187Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
40708mGluR5CLONEDHUMANFunctional3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one816Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41220CLONEDHUMAN125I-Chemokine5-(4-(3,4-Dichlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41988M1CLONEDHUMAN3H-QNBBUPROPION>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42244CLONEDHUMAN125I-[Ile]Motilin[Bpa5,Ile13]Motilin50Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
43012FRKCLONEDHUMAN3H-StaurosporineZD-6474480Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43268CDK5CLONEDHUMAN3H-StaurosporineRoscovitine2000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43524FGFR2CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
43780TEKCLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44036STK16CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44292STK6CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44548FGFR3CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44804PKMYT1CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45060PDGFRBCLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45316CLONEDHUMANFunctionalIndirubin-3monoxime190Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45572NETCLONEDHUMAN3H-NisoxetineDesmethylsertraline390Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458285-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46084Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46596SLC6A3CLONEDHUMAN3H-WIN 35,428N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46852M5CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47364GRIA4CLONEDHUMAN3H-AMPALY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47620ADKrecombinantHUMANFunctional4-N-Phenylamino-5-phenyl-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine0.8Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47876CLONEDHUMAN3H-propionyl-K24-CGRP 8-37[(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37>10000Lang M, et al., 2006Jan 15, 2025Jan 15, 2025
48132Y1CLONEDHUMAN3H-Propionyl-NPYNPY D-Trp32, human, rat1000Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48644CLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.3Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49668SST2CLONEDHUMAN125I-LTT-SST-28L-796,778>10000Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50180mGluR3CLONEDHUMANFunctionalL-CCG-I380Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50436SLC6A4CLONEDHUMAN3H-CITALOPRAM4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenylthio)benzylamine13Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
50948MORUNDEFINEDHUMANUNDEFINEDNalbuphine0.89Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51460Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51972KORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine1.85Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522285-HT1AUNDEFINEDHUMANUNDEFINED1-(1H-indol-5-yloxy)-3-(cyclohexylamino)propan-2-ol3000Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52484SLC6A3UNDEFINEDHUMANUNDEFINED7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline46Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52996CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide>10000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53252D2UNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea55Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53764H1UNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one1014Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54276SLC6A4UNDEFINEDHUMANUNDEFINED3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile4.1Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54532A3UNDEFINEDHUMANUNDEFINEDN-(2-hydroxyethyl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide422Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54788D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine610Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550445-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide13Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55300DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one1790Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
56324A1UNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione379Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56580DORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol443Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56836SLC6A2UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3',4'-dichloropropiophenone5400Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57092D2UNDEFINEDHUMANUNDEFINEDOPC-145972.8Pettersson F et al., 2010Jan 15, 2025Jan 15, 2025
57348A1UNDEFINEDHUMANUNDEFINED8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-methyl-1-propyl-3,7-dihydro-purine-2,6-dione0.295Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57604SST3UNDEFINEDHUMANUNDEFINED6-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]thiazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57860DORUNDEFINEDHUMANUNDEFINED(+)-1-{(1S,2S,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one1000Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581165-HT2ACLONEDHUMAN125I-DOIN-(2-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate2.34Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58372H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5697>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58628hERGCLONEDHUMAN3H-N-Me-DofetilideMRS5678>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58884nAChRCLONEDHUMAN3H-EpibatidineCamel Snus extract3.8Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
591405-HT2ACLONEDHUMAN3H-KETANSERINCYPROHEPTADINE1.67Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59396D4CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4'-formyl-4-biphenylcarboxamide70Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59908D1CLONEDHUMAN3H-SCH233904-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60164A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2S,3R,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiazol-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60420GABAACLONEDHUMANFNZWY-S-24000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60676GABAACLONEDHUMANFNZSPH-382Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60932GABAACLONEDHUMANFNZ3 EBC25.1Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61188GABAACLONEDHUMANFNZQH-II-067a3000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61444GABAACLONEDHUMANFNZRY-054126Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617005-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(4-methoxyphenyl)propan-1-amine267Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62212SLC6A3CLONEDHUMAN[3H] WIN354286-APB565Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62468M3CLONEDHUMAN3H-QNB2-Cl-diphenidine615Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
63236GCCRCLONEDHUMAN125I-Glucagon2-(1H-benzimidazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethanone>10000Madsen, P et al., 1998Jan 15, 2025Jan 15, 2025
63492D3CLONEDHUMAN3H-N-MethylspiperoneRISPERIDONE13Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640045-HT6CLONEDHUMAN3H-LSDN,N-Diethyl-2-[5-(naphthalene-1-sulfonylamino)-1H-indol-3-yl]-2-oxoacetamide1000Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642605-HT2ACLONEDHUMAN3H-KETANSERINQuetiapine218.776Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64516D2CLONEDHUMAN3H-N-MethylspiperoneOLANZAPINE20.4174Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65284GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-073A (R Enriched)1.18Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65541GABAACLONEDHUMAN[3H] FlunitrazepamRo15-1788148Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65797GABAACLONEDHUMAN[3H] FlunitrazepamRY-0531Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66053CLONEDHUMAN3H-VASOPRESSINOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
66309Alpha2BCLONEDHUMAN3H-RAUWOLSCINEFinazine2.2Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66565Alpha1DCLONEDHUMAN3H-PRAZOSIN3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
668215-HT3CLONEDHUMAN3H-GR113808N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
670775-HT1BCLONEDHUMAN3H-5-CT1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67589A1KIDNEYHUMAN3H-N6 -phenylisopropyladenosine(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol298Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
67845D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
33335-HT1ACLONEDHUMAN3H-8-OH-DPATAmphetamine,(+)6606TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68869SST2CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH219.9526Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69125H4CLONEDHUMAN3H-HistamineVUF461612.5893Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693815-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE105Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4101KORCLONEDHUMAN3H-U69,593DSLET-OH>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69637Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43575-HT6CLONEDHUMAN3H-LSDKETANSERIN2800KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69893D1CLONEDHUMAN3H-SCH233904-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4613SLC6A3CLONEDHUMAN3H-DA UPTAKEAmphetamine,(+)116PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48695-HT2BCLONEDHUMAN3H-5HTRITANSERIN1.64WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70405Sigma 1CLONEDHUMAN3H-Pentazocine(+)MRP50637.9Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51255-HT2BCLONEDHUMAN3H-5HTDOC31.8NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70661M3CLONEDHUMAN3H-QNBMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
53815-HT2BCLONEDHUMAN3H-5HTKETANSERIN630.95BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
71173D4CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE54Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5893Alpha2BCLONEDHUMAN3H-RAUWOLSCINECLONIDINE7.2WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714295-HT2ACLONEDHUMAN125I-DOI4-acetoxy-N,N-diallyltryptamine565Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66615-HT1ECLONEDHUMAN3H-5HTZACOPRIDE>10000ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72197D2CLONEDHUMAN3H-N-Methylspiperone2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69175-HT2ACLONEDHUMAN3H-KETANSERINISOCLOZAPINE1.45SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72709Alpha1DCLONEDHUMAN3H-PRAZOSINnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7429MORCLONEDHUMAN3H-DAMGOETORPHINE - HCI0.23Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
729655-HT7CLONEDHUMAN3H-LSDcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7685GABAACLONEDHUMAN3H-MUSCIMOLThiomuscimol37.15Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7941GABAACLONEDHUMAN3H-RO-15-178824He X, et al., 1999Jan 15, 2025Jan 27, 2025
8197GABAACLONEDHUMAN3H-RO-15-1788451000Huang Q, et al., 1999Jan 15, 2025Jan 27, 2025
8453SST5CLONEDHUMAN125I-Tyr3-octreotideCST140.45Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8709SST2CLONEDHUMAN125I-Tyr3-octreotidesomatostatin-280.1Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8965SST1CLONEDHUMAN125I-SRIF-28RC 160158.48Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
745015-HT2CCLONEDHUMAN3H-MESULERGINE(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74757Beta 1CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75013DORCLONEDHUMAN3H-DADLE(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9733MT2CLONEDHUMAN125I-IodomelatoninLuzindole,5-Methoxy0.25Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75269Sigma 2CLONEDHUMAN3H-DTGethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
755255-HT2CCLONEDHUMAN3H-MESULERGINEpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75781Alpha1DCLONEDHUMAN3H-PRAZOSIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76037D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76293M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765495-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768055-HT3CLONEDHUMAN3H-GR-65630(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11525CLONEDHUMAN3H-SUBSTANCE PSubstance P0.1Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
77061Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
11781H1FR. CORTEXHUMAN3H-doxepinFLUPHENAZINE21Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77317Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77573Beta 2CLONEDHUMAN3H-CGP-12177(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77829D3CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12549NeutrophilHUMAN3H-LTB4CGS 2313115Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
780855-HT1DCLONEDHUMAN3H-Cimetidine(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78341M2CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78597SERTCLONEDHUMAN3H-CITALOPRAM(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide2420Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78853KORCLONEDHUMAN3H-U69593(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide100Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791095-HT5ACLONEDHUMAN3H-LSD(±)-3,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79365Alpha1ACLONEDHUMAN3H-PRAZOSINcis-2a528.8Ray TS 2010 Jan 15, 2025Jan 28, 2025
14085CLONEDHUMAN3H-LTD4LTB4>10000Heise CE, et al., 2000Jan 15, 2025Jan 15, 2025
79621CLONEDHUMAN3H-CLONIDINE(±)-2,5-Dimethoxy-4-bromoamphetamine1596.1Ray TS 2010 Jan 15, 2025Jan 15, 2025
143415-HT2BCLONEDHUMAN3H-LSDl-norfenfluramine65FITZGERALD LW, ET AL., 1999Jan 15, 2025Jan 15, 2025
79877M5CLONEDHUMAN3H-QNB(±)-3,4-Methylenedioxymethamphetamine6330Ray TS 2010 Jan 15, 2025Jan 15, 2025
80133CLONEDHUMAN3H-VASOPRESSINcis-2a>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14853TPWashed PlateletsHUMAN3H-SQ 29548U466193.6Hedberg, A, et al., 1988Jan 15, 2025Jan 15, 2025
803895-HT5ACLONEDHUMAN3H-LSD(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15109CLONEDHUMAN3H-PGE2PGF2Alpha,17-phenyl168Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806455-HT1BCLONEDHUMAN3H-5-CT(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153655-HT1BCLONEDHUMAN3H-5HTLYSERGOL1.2BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809015-HT2BCLONEDHUMAN3H-LSD(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one353Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
81157H1CLONEDHUMAN3H-PYRILAMINEN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
158775-HT7CLONEDHUMAN3H-5HTDHE9.12BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81413H1CLONEDHUMAN3H-PYRILAMINE4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole3265Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16133D1CLONEDHUMAN3H-SCH23390N-04372172Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81925DORCLONEDHUMAN3H-DADLE(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16645M1CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.035Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82181Alpha1BCLONEDHUMAN3H-PRAZOSIN2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one152.5Besnard J et al 2012Jan 15, 2025Jan 28, 2025
824375-HT5ACLONEDHUMAN3H-LSD(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171575-HT2ABRAINHUMAN3H-KETANSERINRISPERIDONE0.15Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826935-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17669CLONEDHUMAN125I-VIPVIP [D-Asp3]1.1Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832055-HT1ACLONEDHUMAN3H-8-OH-DPATDMT450Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83461M4CLONEDHUMAN3H-NMS1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide0.676083Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83717SERTCLONEDHUMAN3H-CITALOPRAM(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide2284PDSP Certified DataJan 15, 2025Jan 28, 2025
83973KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide194PDSP Certified DataJan 15, 2025Jan 28, 2025
842295-HT2BCLONEDHUMAN3H-LSD(±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide8306PDSP Certified DataJan 15, 2025Jan 15, 2025
84485DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19205SLC6A4PlateletsHUMAN3H-5HTLY2486850.35Wong DT et al., 1993Jan 15, 2025Jan 15, 2025
84741DORCLONEDHUMAN3H-DADLEmethyl (±)-(S)-2-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)-2-phenylacetate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19461GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Arg110.55Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84997KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
86021D1CLONEDHUMAN3H-SCH23390(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
87557Alpha1BCLONEDHUMAN3H-PRAZOSIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
22277A3CLONEDHUMAN125I-Aba830Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878135-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline79Staron J et al 2016Jan 15, 2025Jan 15, 2025
225335-HT1BCLONEDHUMAN3H-GR-125743SL6501555500Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
88069A1CLONEDHUMAN3H-CCPAH2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22789H2CLONEDHUMAN3H-TIOTIDINEL-homocysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23045nAChRCLONEDHUMAN3H-EpibatidineDL-homocysteine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
885815-HT7CLONEDHUMAN3H-LSD1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine90Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88837A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89093A2AHeLaHUMAN3H-ZM241385N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide3345Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
240695-HT2ACLONEDHUMANUNDEFINEDRACLOPRIDE4000Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89605M1CLONEDHUMAN3H-NMS3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89861nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride953Liu J et al 2010Jan 15, 2025Jan 29, 2025
90117D1CLONEDHUMAN3H-SCH233902-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
248375-HT1BCLONEDHUMAN3H-GR-125743CLOZAPINE398PDSP Certified DataJan 15, 2025Jan 15, 2025
90629A2BCLONEDHUMAN3H-PSB-603Preladenant (SCH420814)1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25349M2CLONEDHUMAN3H-QNBZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
908855-HT1AHeLaHUMAN3H-8-OH-DPAT8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane42.658Franchini S et al 2014Jan 15, 2025Jan 15, 2025
25605Alpha2CCLONEDHUMAN3H-CLONIDINEPRAZOSIN14.5Rothman RB, et al., 2003aJan 15, 2025Jan 15, 2025
91141A3CHO cellsHUMAN3H-HEMADOEthyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate1300Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
25861nAChRCLONEDHUMAN3H-EpibatidinePseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 27, 2025
91397CB1CLONEDHUMAN3H-SR144528O-621241Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26117D1CLONEDHUMAN3H-SCH23390Pseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91653A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide83.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26373Alpha2CCLONEDHUMAN3H-CLONIDINEMiquelianin4063Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91909A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3-trifluoromethylphenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26629MORCLONEDHUMAN3H-DiprenorphineHypericin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921655-HT6CLONEDHUMAN3H-LSD5-Chloro-N-{1-[2-(2,3-dichlorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide91Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
26885M2CLONEDHUMAN3H-QNBxanomeline125.893Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92421DORCLONEDHUMAN3H-DADLE15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271415-HT1ACLONEDHUMAN3H-8-OH-DPATAL-37350A>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92677M5CLONEDHUMAN3H-QNB9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27397Beta2CLONEDHUMAN3H-CGP-12177Roxindole933.254Millan MJ, et al., 2002Jan 15, 2025Jan 28, 2025
92933A3CLONEDHUMAN125I-AB-MECA2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
93189D3CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine370Lober S et al 2012Jan 15, 2025Jan 28, 2025
279095-HT2ACLONEDHUMAN3H-DOBDMT,5-OH15Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28165D2CLONEDHUMAN3H-NMSPMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93701A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester6.05Federico S et al 2018Jan 15, 2025Jan 15, 2025
286775-HT5ACLONEDHUMAN3H-LSDARIPIPRAZOLE1240Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942135-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29189SST2CLONEDHUMANUNDEFINEDL-797,5911875Patel YC, 1999Jan 15, 2025Jan 15, 2025
947255-HT2ACLONEDHUMAN3H-KETANSERIN4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94981D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29957H4CLONEDHUMAN3H-Histamine(5,7- Dichloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone11Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957495-HT5ACLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96005DATCLONEDHUMAN3H-WIN 35,428tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96261Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30981CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
965175-HT5ACLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31237Alpha2ACLONEDHUMAN3H-CLONIDINEMDL 1009071900PDSP Certified DataJan 15, 2025Jan 15, 2025
96773D1CLONEDHUMAN[3H]SCH233904-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA6000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
31493D2CLONEDHUMAN125I-IODOSULPRIDE(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)1584.89Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97029Beta2CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97285MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol171Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97541A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate517.1Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98053CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide6000Amato G et al 2019Jan 15, 2025Jan 28, 2025
32773NK1CLONEDHUMAN3H-Sar9,Met(O2)11-Substance PSCH 2062721.3Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98309D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride272Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985655-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one614Ofon E et al 2016aJan 15, 2025Jan 15, 2025
33285CB2CLONEDHUMAN3H-CP-55940nimesulide>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98821H3CLONEDHUMAN3H-Alpha-methylhistamine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
99077Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99333D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(naphtha-len-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34053P2X3CLONEDHUMAN3H-A-317491A-31749110.8Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99589A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine3.99Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99845Alpha1ACLONEDHUMAN[125I] HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
1001015-HT1ACLONEDHUMAN3H-WAY100635Quetiapine267PDSP Certified DataJan 15, 2025Jan 15, 2025
1003575-HT7CLONEDHUMAN3H-LSDBlonanserin1010PDSP Certified DataJan 15, 2025Jan 15, 2025
100869nAChRCLONEDHUMANFunctionalPancuronium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
35589CLONEDHUMAN3H-SQ 29548Latanoprost (Isopropyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35845Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide20Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
101381D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione30Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
36101COX-2whole blood assay (WBA)HUMANFunctionalnimesulide1900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
101637D1CLONEDHUMAN[3H]SCH23390Perospirone65PDSP Certified DataMar 21, 2025Jul 28, 2026
101893D5CLONEDHUMAN[3H]SCH23390Ziprasidone136PDSP Certified DataMar 24, 2025Jul 28, 2026
36613D2CLONEDHUMAN3H-SPIPERONERISPERIDONE6.4Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102149DATCLONEDHUMAN[3H]WIN35428NEMONAPRIDE2368PDSP Certified DataMar 25, 2025Jul 28, 2026
37893MPP-9CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-trimethylsilyl-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione550Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38661UNDEFINEDHUMAN3H-hypoxanthineN-{(1S,2S)-2-Hydroxy-3-[2-(3-methoxy-phenyl)-ethylcarbamoyl]-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl}-2,4,6-trifluoro-benzamide693Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39173D4CLONEDHUMANR-SATL 745,8701.8Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39429CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396855-HT2BCLONEDHUMAN3H-5HTMETHYLERGONOVINE0.457088Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40709mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one44Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41221CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-p-tolylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41989M1CLONEDHUMAN3H-QNBDESIPRAMINE110Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42245CLONEDHUMAN125I-[Ile]MotilinMotilin2.3Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
43013FRKCLONEDHUMAN3H-StaurosporineCI-10338100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43269CDK5CLONEDHUMAN3H-StaurosporineFlavopiridol43Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43525FGFR3CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43781KIAA0551CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44037STK18CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44293AURKCCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44549FGRCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44805MAPK14CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45061PHKG1CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45317LCKCLONEDHUMANFunctionalIndirubin-3monoxime300Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45573SLC6A3CLONEDHUMAN3H-WIN 35,428Desmethylsertraline129Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458295-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46085Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46597SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46853M5CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47365GRIA4CLONEDHUMAN3H-AMPALY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47621ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-(4-fluorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 26Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47877CLONEDHUMAN3H-propionyl-K24-CGRP 8-37[(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-370.7Lang M, et al., 2006Jan 15, 2025Jan 15, 2025
48133Y2CLONEDHUMAN3H-Propionyl-NPYNPY D-Trp32, human, rat29Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48645CLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride9.4Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49669SST3CLONEDHUMAN125I-LTT-SST-28L-796,778127Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50181mGluR3CLONEDHUMANFunctional1S, 3R-ACPD5400Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50437SLC6A4CLONEDHUMAN3H-CITALOPRAMMADAM1.65Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
50949KORUNDEFINEDHUMANUNDEFINED17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol0.079Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51461Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide4.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51717NR3C1UNDEFINEDHUMANUNDEFINEDdexamethasone2.1Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51973KORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine3.11Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522295-HT1AUNDEFINEDHUMANUNDEFINED1-(1H-indol-4-yloxy)-4-(cyclohexylamino)butan-2-ol125Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52485SLC6A3UNDEFINEDHUMANUNDEFINED(S)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline102Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52997CB2UNDEFINEDHUMANUNDEFINEDN-butyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide9400Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53253D2UNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea54Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53765H1UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one188.6Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54277SLC6A4UNDEFINEDHUMANUNDEFINED3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile90.7Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54533A3UNDEFINEDHUMANUNDEFINED8-(4-(1-(4-(5-chlorobenzo[d]thiazol-2-yl)piperazin-1-yl)-2-methyl-1-oxopropan-2-yloxy)phenyl)-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione1000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54789D2UNDEFINEDHUMANUNDEFINEDN-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine4100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550455-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide139Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55301DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one3103Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
56325A1UNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione>10000Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56581DORUNDEFINEDHUMANUNDEFINED4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol75Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56837SLC6A2UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chloro-4'-methylpropiophenone5100Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57093D2UNDEFINEDHUMANUNDEFINED(S)-3-(3-Methanesulfonyl-phenyl)-1-propyl-piperidine755Pettersson F et al., 2010Jan 15, 2025Jan 15, 2025
57349A1UNDEFINEDHUMANUNDEFINED(4-(furan-2-yl)-2-(2-(thiophen-2-yl)ethylamino)thiazol-5-yl)(phenyl)methanone6700Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57605SST3UNDEFINEDHUMANUNDEFINEDN-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)thiazolo[5,4-b]pyridin-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57861DORUNDEFINEDHUMANUNDEFINED(-)-1-{(1R,2R,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one1000Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581175-HT2ACLONEDHUMAN125I-DOIN-(3-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate1.48Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58373H3CLONEDHUMAN3H-Alpha-Me-histamineMRS3558>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58629hERGCLONEDHUMAN3H-N-Me-DofetilideMRS5697>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58885nAChRCLONEDHUMAN3H-EpibatidineKodiak extract3.9Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
591415-HT1ACLONEDHUMAN3H-WAY100635CYPROHEPTADINE50Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59397D2CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4'-formyl-4-biphenylcarboxamide3700Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59909D2CLONEDHUMAN3H-NMSP4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60165A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-4-(2-((Ferrocen-yl)ethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60421GABAACLONEDHUMANFNZWY-S-2300Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60677GABAACLONEDHUMANFNZXHE-I-0932Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60933GABAACLONEDHUMANFNZ3 EBC28.2Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61189GABAACLONEDHUMANFNZQH-II-067a199Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61445GABAACLONEDHUMANFNZRY-0541.3Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617015-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2,5-dimethoxyphenyl)propan-1-amine919Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62213SerotoninCLONEDHUMAN[3H] Citalopram6-APB4046Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62469M4CLONEDHUMAN3H-QNB2-Cl-diphenidine828Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
634935-HT1ACLONEDHUMAN3H-WAY100635RISPERIDONE420Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640055-HT6CLONEDHUMAN3H-LSDN,N-Diethyl-2-oxo-2-[5-(quinoline-8-sulfonylamino)-1H-indol-3-yl]-acetamide1000Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642615-HT2ACLONEDHUMAN3H-KETANSERINREMOXIPRIDE5248.07Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64517D2CLONEDHUMAN3H-N-MethylspiperonePERPHENAZINE0.977237Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65285GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-073A (R Enriched)140Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65542GABAACLONEDHUMAN[3H] FlunitrazepamMLT-I-701.1Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65798GABAACLONEDHUMAN[3H] FlunitrazepamRY-05346Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66054V1BCLONEDHUMAN3H-VASOPRESSINOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
66310Alpha2CCLONEDHUMAN3H-RAUWOLSCINEFinazine4.4Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66566Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride367Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
668225-HT5ACLONEDHUMAN3H-LSDN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
670785-HT1DCLONEDHUMAN3H-5-CT1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67590A2AKIDNEYHUMAN3H-2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol2690Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
23105-HT3AMYGDALAHUMAN3H-ZACOPRIDEFLUPHENAZINE>10000BARNES ET AL., 1989Jan 15, 2025Jan 15, 2025
678465-HT1ACLONEDHUMAN3H-8-OH-DPATS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33345-HT1ACLONEDHUMAN3H-8-OH-DPATSKF 829581781TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68870SST3CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH225.1189Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69126H4CLONEDHUMAN3H-HistamineVUF461712.5893Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693825-HT1ACLONEDHUMAN3H-8-OH-DPATOLANZAPINE2063Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4102KORCLONEDHUMAN3H-U69,593DADLE-OH>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69638Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-MXP1909Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43585-HT6CLONEDHUMAN3H-LSDQUIPAZINE3600KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69894D1CLONEDHUMAN3H-SCH233904-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4614SLC6A3CLONEDHUMAN3H-DA UPTAKEDICLOFENSINE,(-)606PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48705-HT2BCLONEDHUMAN3H-5HTSPIPERONE592WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70406Sigma 2CLONEDHUMAN3H-DTGMRP50636.5Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51265-HT2BCLONEDHUMAN3H-5HTDOB26.9NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70662M4CLONEDHUMAN3H-QNBMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
53825-HT2BCLONEDHUMAN3H-5HTMETHYSERGIDE7.94BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
71174D4CLONEDHUMAN3H-N-MethylspiperoneSYA01360.6Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5894Alpha2BCLONEDHUMAN3H-RAUWOLSCINEWB 410117WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714305-HT2BCLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine63Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66625-HT1ECLONEDHUMAN3H-5HTPAPP>10000ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72198D3CLONEDHUMAN3H-N-Methylspiperone2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69185-HT2ACLONEDHUMAN3H-KETANSERINLOXAPINE10.2SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72710Alpha2ACLONEDHUMAN3H-RAUWOLSCINEnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7430MORCLONEDHUMAN3H-DAMGOLEVORPHANOL-tartarate0.08Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
72966Alpha1ACLONEDHUMAN3H-PRAZOSINcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7686GABAACLONEDHUMAN3H-MUSCIMOLTHIP165.95Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7942GABAACLONEDHUMAN3H-RO-15-17883100He X, et al., 1999Jan 15, 2025Jan 27, 2025
8198SST5CLONEDHUMAN125I-LTT-SST-28somatostatin-280.19Panetta R, et al., 1993Jan 15, 2025Jan 15, 2025
8454SST5CLONEDHUMAN125I-Tyr3-octreotideCST14-Tyr100.22Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8710SST2CLONEDHUMAN125I-Tyr3-octreotideseglitide0.15Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8966SST1CLONEDHUMAN125I-SRIF-28RC 160II100Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
745025-HT3CLONEDHUMAN3H-GR-65630(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74758Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75014KORCLONEDHUMAN3H-U69593(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9734MT2CLONEDHUMAN125I-IodomelatoninMelatonin,6-Hydroxy5.5Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75270SERTCLONEDHUMAN3H-CITALOPRAMethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
755265-HT3CLONEDHUMAN3H-GR-65630propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75782Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76038D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76294Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
765505-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768065-HT5ACLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77062Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
11782H1FR. CORTEXHUMAN3H-doxepinTRIFLUOPERAZINE62Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77318Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77574D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77830D4CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12550NeutrophilHUMAN3H-LTB4CGS 23356116Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78086H3CLONEDHUMAN3H-Alpha-methylhistamine(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78342M3CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78598Sigma 1CLONEDHUMAN3H-Pentazocine(+)(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78854MORCLONEDHUMAN3H-DAMGO(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791105-HT5ACLONEDHUMAN3H-LSD(±)-2,5-Dimethoxy-4-ethylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79366Alpha1ACLONEDHUMAN3H-PRAZOSINR,R-2b5187Ray TS 2010 Jan 15, 2025Jan 28, 2025
79622CLONEDHUMAN3H-CLONIDINE(±)-3,4-Methylenedioxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79878M5CLONEDHUMAN3H-QNB3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80134CLONEDHUMAN3H-VASOPRESSINR,R-2b>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
803905-HT6CLONEDHUMAN3H-LSD(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15110CLONEDHUMAN3H-PGE2PGF2 Alpha, 1-isopropyl ester5000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806465-HT1DCLONEDHUMAN3H-5-CT(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153665-HT1BCLONEDHUMAN3H-5HT5-CT1.58BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809025-HT2CCLONEDHUMAN3H-MESULERGINE(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one678Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
811585-HT1DCLONEDHUMAN3H-CimetidineN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
81414D2CLONEDHUMAN3H-N-Methylspiperone4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16134D1CLONEDHUMAN3H-SCH23390NPA1816Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81670D1CLONEDHUMAN3H-SCH23390(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
16646M1CLONEDHUMAN3H-QNBBENZTROPINE0.231Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82182Alpha1DCLONEDHUMAN3H-PRAZOSIN2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one72.2Besnard J et al 2012Jan 15, 2025Jan 28, 2025
824385-HT6CLONEDHUMAN3H-LSD(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171585-HT2ABRAINHUMAN3H-KETANSERIN9-OH-risperidone1.21Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826945-HT2BCLONEDHUMAN3H-LSD(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine3169Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17670CLONEDHUMAN125I-VIPVIP [D-Ala4]1.1Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832065-HT1ACLONEDHUMAN3H-8-OH-DPATDOM>10000Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83462M5CLONEDHUMAN3H-NMS1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide0.660693Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83718DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide2961PDSP Certified DataJan 15, 2025Jan 28, 2025
83974MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide2825PDSP Certified DataJan 15, 2025Jan 28, 2025
84486DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19206SLC6A4PlateletsHUMAN3H-5HTLY2486860.2Wong DT et al., 1993Jan 15, 2025Jan 15, 2025
84742MORCLONEDHUMAN3H-DAMGOmethyl (±)-(S)-2-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)-2-phenylacetate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19462GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Arg14330Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84998MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
86022D5CLONEDHUMAN3H-SCH23390(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86534A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione124Koch P et al 2018Jan 15, 2025Jan 15, 2025
87558Alpha1DCLONEDHUMAN3H-PRAZOSIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
22278A3CLONEDHUMAN125I-Aba9922Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878145-HT2ACLONEDHUMAN3H-KETANSERIN4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline295Staron J et al 2016Jan 15, 2025Jan 15, 2025
225345-HT2BCLONEDHUMAN3H-LSDSL6501551560Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
88070A1CLONEDHUMAN3H-CCPA1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22790H2CLONEDHUMAN3H-TIOTIDINEL-cysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23046nAChRCLONEDHUMAN3H-EpibatidineL-cysteine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
88582Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine308.2Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88838A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89094A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89350D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide4346Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
240705-HT2ACLONEDHUMANUNDEFINEDREMOXIPRIDE5200Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89606M2CLONEDHUMAN3H-NMS3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89862nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride9520Liu J et al 2010Jan 15, 2025Jan 29, 2025
90118D1CLONEDHUMAN3H-SCH233902-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24838M1CLONEDHUMAN3H-QNBCLOZAPINE14PDSP Certified DataJan 15, 2025Jan 15, 2025
25094M4CLONEDHUMAN3H-QNBQuetiapine542Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90630A2BCLONEDHUMAN3H-PSB-603N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide365 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25350nAChRCLONEDHUMAN3H-EpibatidineZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 27, 2025
90886Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane30.903Franchini S et al 2014Jan 15, 2025Jan 28, 2025
91142A1CHO cellsHUMAN3H-CCPAEthyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91398CB1CLONEDHUMAN3H-SR144528O-661743Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26118D4CLONEDHUMAN3H-NMSPPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91654A3CLONEDHUMAN3H-PSB-11N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide25.4Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91910A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (4-methylphenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26630MORCLONEDHUMAN3H-DiprenorphineHyperforin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921665-HT6CLONEDHUMAN3H-LSD5-Chloro-N-{1-[2-(2,5-dichlorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide225Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
26886M3CLONEDHUMAN3H-QNBxanomeline39.8107Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92422DORCLONEDHUMAN3H-DADLE9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271425-HT1ACLONEDHUMAN3H-8-OH-DPATDOI,(-)3843May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92678M4CLONEDHUMAN3H-QNB9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27398Beta1CLONEDHUMAN3H-CGP-12177Roxindole2691.53Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
92934A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
27654D2CLONEDHUMAN3H-NMSPMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93190D4CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine19Lober S et al 2012Jan 15, 2025Jan 29, 2025
279105-HT2ACLONEDHUMAN3H-KETANSERINDOM306Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
93702A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester32Federico S et al 2018Jan 15, 2025Jan 15, 2025
28422nAChRCLONEDHUMAN3H-EpibatidineERGOTAMINE>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
286785-HT6CLONEDHUMAN3H-LSDARIPIPRAZOLE570Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942145-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-isopropoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29190SST2CLONEDHUMANUNDEFINEDCH2751000Patel YC, 1999Jan 15, 2025Jan 15, 2025
947265-HT2ACLONEDHUMAN3H-KETANSERIN4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94982D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29958H4CLONEDHUMAN3H-Histamine(5,7-Dimethyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone31Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957505-HT6CLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96006DATCLONEDHUMAN3H-WIN 35,4284-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96262Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
965185-HT6CLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31238Alpha2BCLONEDHUMAN3H-CLONIDINEMDL 100907270.6PDSP Certified DataJan 15, 2025Jan 15, 2025
96774D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
31494D3CLONEDHUMAN125I-IODOSULPRIDE(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)1258.93Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97030Beta3CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97286MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol370Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97542A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate49.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98054CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide3Amato G et al 2019Jan 15, 2025Jan 28, 2025
32774NK1CLONEDHUMAN3H-Sar9,Met(O2)11-Substance PCP 999940.27Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98310D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride138Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985665-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one273Ofon E et al 2016aJan 15, 2025Jan 15, 2025
98822H4CLONEDHUMAN3H-Histamine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33542Alpha1ACLONEDHUMAN3H-PRAZOSINNaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99078Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99334D2CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,1’-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34054P2X3CLONEDHUMAN3H-A-317491ATP,TNP7.5Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99590A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine1.68Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99846Alpha2ACLONEDHUMAN[125I] iodoclonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide4700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
1001025-HT2ACLONEDHUMAN3H-KETANSERINQuetiapine352PDSP Certified DataJan 15, 2025Jan 15, 2025
1003585-HT7CLONEDHUMAN3H-LSDRS-(+/-)-Sulpriride1085PDSP Certified DataJan 15, 2025Jan 15, 2025
1008705-HT1ACLONEDHUMAN3H-WAY1006351-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1)85.7Stephenson, K. et. al., 2008Jan 15, 2025Jan 15, 2025
35590CLONEDHUMAN3H-SQ 29548ILOPROST6487Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35846Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide2.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013825-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione48Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36102COX-2whole blood assay (WBA)HUMANFunctionalROFECOXIB840Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
101638D2CLONEDHUMAN[3H]-N-methylspiperonePerospirone14PDSP Certified DataMar 21, 2025Jul 28, 2026
101894SERTCLONEDHUMAN[3H] CitalopramZiprasidone165PDSP Certified DataMar 24, 2025Jul 28, 2026
36614D2CLONEDHUMAN3H-SPIPERONEmirtazepine5454Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102150MORCLONEDHUMAN[3H]DAMGONEMONAPRIDE3698PDSP Certified DataMar 25, 2025Jul 28, 2026
37894MPP-2CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione12Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38662UNDEFINEDHUMAN3H-hypoxanthineN-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-cyclohexylcarbamoyl-2-hydroxypropyl]-2,4,6-trifluorobenzamide230Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39174D4CLONEDHUMANR-SATARIPIPRAZOLE1000Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39430V1ACLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396865-HT2BCLONEDHUMAN3H-5HTMK 212616.595Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
399425-HT2ACLONEDHUMANFunctionalBW-723C86100Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
40710mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one344Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41222CLONEDHUMAN125I-Chemokine5-(4-Benzyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41990M1CLONEDHUMAN3H-QNBDesmethylsertraline1650Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42246CLONEDHUMAN125I-[Ile]Motilin[D-Bpa5,Ile13]Motilin420Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
43014FYNCLONEDHUMAN3H-StaurosporineStaurosporine51Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43270CLK1CLONEDHUMAN3H-StaurosporineEKB-5691000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43526FGRCLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43782TTKCLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44038STK3 mouseCLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44294BMXCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44550FLT3CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44806MAPK P38CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45062PRKACACLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45318CLONEDHUMANFunctionalIndirubin-3monoxime380Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45574SLC6A4CLONEDHUMAN3H-IMIPRAMINEDothiepin8.6Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458305-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46086Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46598SLC6A3CLONEDHUMAN3H-WIN 35,428PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46854M5CLONEDHUMAN3H-QNBPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47366GRIA4CLONEDHUMAN3H-AMPALY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47622ADKrecombinantHUMANFunctional4-N-Phenylamino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine1.2Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
48134Y2CLONEDHUMAN3H-Propionyl-NPYPYY 3-360.03Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48646CLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.7Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49670SST4CLONEDHUMAN125I-LTT-SST-28L-796,778>10000Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50182mGluR3CLONEDHUMANFunctionalQuisqualate>10000Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50438SLC6A4CLONEDHUMAN3H-CITALOPRAM4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine7Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
50950KORUNDEFINEDHUMANUNDEFINED(5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate0.13Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51462Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide25Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51718NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline4.4Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51974KORUNDEFINEDHUMANUNDEFINED7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine1.64Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522305-HT1AUNDEFINEDHUMANUNDEFINED1-(adamantan-1-ylamino)-4-(1H-indol-4-yloxy)-butan-2-ol551Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52486SLC6A3UNDEFINEDHUMANUNDEFINED2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline29Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52998CB2UNDEFINEDHUMANUNDEFINEDN-cyclopentyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide7400Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53254D2UNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea127Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53766H1UNDEFINEDHUMANUNDEFINED1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one911.8Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54278SLC6A4UNDEFINEDHUMANUNDEFINED3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile189Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54534A3UNDEFINEDHUMANUNDEFINED8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-3-ethyl-1-propyl-1H-purine-2,6(3H,7H)-dione1070Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54790D2UNDEFINEDHUMANUNDEFINEDN-(4-Propylaminobutyl)-4-biphenylcarboxamide>10000Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550465-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide161Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55302DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one795Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
56326A3UNDEFINEDHUMANUNDEFINEDNECA20Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56582DORUNDEFINEDHUMANUNDEFINED(4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol1350Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56838SLC6A2UNDEFINEDHUMANUNDEFINED2-Piperidino-3'-chloropropiophenone4760Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57350A1UNDEFINEDHUMANUNDEFINEDN-[5-pyridin-4-yl-4-(3,4,5-trimethoxyphenyl)thiazol-2-yl]acetamide>10000Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57606SST3UNDEFINEDHUMANUNDEFINEDN-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57862DORUNDEFINEDHUMANUNDEFINED(+)-1-{(1S,2R,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one1000Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581185-HT2ACLONEDHUMAN3H-KETANSERINN-(3-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate6.76Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58374H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5676>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58630hERGCLONEDHUMAN3H-N-Me-DofetilideMRS3558>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
591425-HT1ACLONEDHUMAN3H-WAY100635HALOPERIDOL3500Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59398D4CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4-(2-thienyl)benzamide3Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59910D3CLONEDHUMAN3H-NMSP4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60166A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-4-(2-(Cyclopropylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60422GABAACLONEDHUMANFNZWY-S-2300Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60678GABAACLONEDHUMANFNZXHE-I-0937.1Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60934GABAACLONEDHUMANFNZ3 EBC826Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61190GABAACLONEDHUMANFNZQH-II-067a52Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61446GABAACLONEDHUMANFNZRY-05427Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617025-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine146Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62214NETCLONEDHUMAN[3H] NisoxetineDesoxypipradol281Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62470M4CLONEDHUMAN3H-QNBDiphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
634945-HT2ACLONEDHUMAN3H-KetaserinRISPERIDONE0.22Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640065-HT6CLONEDHUMAN3H-LSDN-[3-(3-Diethylaminopropyl)-1H-indol-5-yl]naphthalene-2-sulfonamide163Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642625-HT2ACLONEDHUMAN3H-KETANSERINRISPERIDONE0.436516Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64518D2CLONEDHUMAN3H-N-MethylspiperonePIMOZIDE6.76083Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65030H1FR. CORTEXHUMAN3H-MEPYRAMINETHIORIDAZINE22Chang, R et., 1978Jan 15, 2025Jan 15, 2025
65286GABAACLONEDHUMAN[3H] FlunitrazepamSH-I-03014.42Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65543GABAACLONEDHUMAN[3H] FlunitrazepamMLT-I-701.2Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65799GABAACLONEDHUMAN[3H] FlunitrazepamYT-615.31Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66055V2CLONEDHUMAN3H-VASOPRESSINOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
66311Beta1CLONEDHUMANI-125-PindololFinazine1254Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66567Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride363Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
668235-HT6CLONEDHUMAN3H-LSDN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
670795-HT1ECLONEDHUMAN3H-5-HT1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67591A3KIDNEYHUMANI-125-N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamide(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol3240Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
23115-HT3HIPPOCAMPUSHUMAN3H-ZACOPRIDEFLUPHENAZINE>10000BARNES ET AL., 1989Jan 15, 2025Jan 15, 2025
678475-HT7CLONEDHUMAN3H-5-CTS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline142Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
25675-HT2ACORTEXHUMAN3H-KETANSERINTMA,3,4,5->10000SADZOT ET AL., 1989Jan 15, 2025Jan 15, 2025
33355-HT1ACLONEDHUMAN3H-8-OH-DPATAPOMORPHINE4929TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68871SST4CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH21.99526Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69127H4CLONEDHUMAN3H-HistamineVUF4742125.893Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693835-HT1ACLONEDHUMAN3H-8-OH-DPATQuetiapine431Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4103KORCLONEDHUMAN3H-U69,593DELTORPHIN-II>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69639Alpha2ACLONEDHUMAN3H-RAUWOLSCINEDPH>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43595-HT6CLONEDHUMAN3H-LSDMESULERGINE3800KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69895D2CLONEDHUMAN3H-N-Methylspiperone4-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4615SLC6A3CLONEDHUMAN3H-DA UPTAKECOCAINE743PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48715-HT2BCLONEDHUMAN3H-5HTSPIROXATRINE475WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70407Sigma 2CLONEDHUMAN3H-DTGMRP42686.5Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51275-HT2BCLONEDHUMAN3H-5HTDOI20NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70663M5CLONEDHUMAN3H-QNBMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
53835-HT2BCLONEDHUMAN3H-5HTRITANSERIN5.01BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
709195-HT2BCLONEDHUMAN3H-LSD4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione742Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
71175D4CLONEDHUMAN3H-N-MethylspiperoneSYA1626330.5Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5895Alpha2BCLONEDHUMAN3H-RAUWOLSCINEPRAZOSIN23WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714315-HT2CCLONEDHUMANUNKNOWN4-acetoxy-N,N-diallyltryptamine1515Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66635-HT1ECLONEDHUMAN3H-5HT5-CT,DP>10000ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72199D4CLONEDHUMAN3H-N-Methylspiperone2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69195-HT2ACLONEDHUMAN3H-KETANSERINMELPERONE280SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72711Alpha2BCLONEDHUMAN3H-RAUWOLSCINEnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7431MORCLONEDHUMAN3H-DAMGOMethadone0.72Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
72967Alpha1BCLONEDHUMAN3H-PRAZOSINcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7687GABAACLONEDHUMAN3H-MUSCIMOLP4S107.15Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7943GABAACLONEDHUMAN3H-RO-15-1788540He X, et al., 1999Jan 15, 2025Jan 27, 2025
8199SST5CLONEDHUMAN125I-LTT-SST-28LTT-SST-280.11Panetta R, et al., 1993Jan 15, 2025Jan 15, 2025
8455SST5CLONEDHUMAN125I-Tyr3-octreotideseglitide0.06Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8711SST2CLONEDHUMAN125I-Tyr3-octreotideBIM 230140.28Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8967SST1CLONEDHUMAN125I-SRIF-28L-362,855100Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
745035-HT5ACLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74759Beta2CLONEDHUMAN3H-CGP12177(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75015MORCLONEDHUMAN3H-DAMGO(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9735MT2CLONEDHUMAN125I-Iodomelatonin8-M-ADOT4.1Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75271NETCLONEDHUMAN3H-Nisoxetineethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
755275-HT5ACLONEDHUMAN3H-LSDpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75783Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76039D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76295Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
765515-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768075-HT6CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77063Alpha1DCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
11783H1FR. CORTEXHUMAN3H-doxepind-Butaclamol390Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77319Beta 1CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77575D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77831DATCLONEDHUMAN3H-WIN 35,428(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
12551NeutrophilHUMAN3H-LTB4CGS 24115131Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78087H4CLONEDHUMAN3H-Histamine(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78343M4CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78599Sigma 2CLONEDHUMAN3H-DTG(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78855MORCLONEDHUMAN3H-DAMGO(±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791115-HT5ACLONEDHUMAN3H-LSD2,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79367Alpha1ACLONEDHUMAN3H-PRAZOSINS,S-2c850.2Ray TS 2010 Jan 15, 2025Jan 28, 2025
79623CLONEDHUMAN3H-CLONIDINE(±)-3,4-Methylenedioxymethamphetamine219.7Ray TS 2010 Jan 15, 2025Jan 15, 2025
79879M5CLONEDHUMAN3H-QNB4-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80135CLONEDHUMAN3H-VASOPRESSINS,S-2c>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
803915-HT7CLONEDHUMAN3H-LSD(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one799Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15111PTGFRCLONEDHUMAN3H-PGF2AlphaPGF2Alpha48Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806475-HT1ECLONEDHUMAN3H-5-HT(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153675-HT1BCLONEDHUMAN3H-5HT5-Methoxytryptamine33.88BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809035-HT3CLONEDHUMAN3H-GR-65630(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
81159H3CLONEDHUMAN3H-Alpha-methylhistamineN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
814155-HT2ACLONEDHUMAN3H-KETANSERIN4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole>10000Weiss DR et al 2018Jan 15, 2025Jan 15, 2025
16135D1CLONEDHUMAN3H-SCH233905-Hydroxy Tryptamine9690Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81671D5CLONEDHUMAN3H-SCH23390(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
81927H1CLONEDHUMAN3H-PYRILAMINE(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16647M1CLONEDHUMAN3H-QNBBiperidine0.48Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82183D1CLONEDHUMAN3H-SCH233902-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
824395-HT7CLONEDHUMAN3H-LSD(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171595-HT2ABRAINHUMAN3H-KETANSERINSERTINDOLE0.14Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826955-HT2CCLONEDHUMAN3H-MESULERGINE(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82951A2BCHO cellsHUMAN3H-PSB-603(R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
17671CLONEDHUMAN125I-VIPVIP [D-Val5]6.2Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832075-HT2ACLONEDHUMAN125I-DOIDOM4.3Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83463M5CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+)20.893Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83719DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
83975MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(3-bromobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide3275PDSP Certified DataJan 15, 2025Jan 28, 2025
84231Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide9747PDSP Certified DataJan 15, 2025Jan 28, 2025
84487MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84743MORCLONEDHUMAN3H-DAMGObenzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19463GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHhMCH2.9Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84999DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
86023D2CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86535A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione542Koch P et al 2018Jan 15, 2025Jan 15, 2025
87559Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
878155-HT7CLONEDHUMAN3H-5-CT4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline19Staron J et al 2016Jan 15, 2025Jan 15, 2025
225355-HT2ACLONEDHUMAN3H-KETANSERINSL6501551320Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
88071A1CLONEDHUMAN3H-CCPA9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22791H2CLONEDHUMAN3H-TIOTIDINED-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23047nAChRCLONEDHUMAN3H-EpibatidineD-homocysteine thiolactone>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
885835-HT7CLONEDHUMAN3H-LSD1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine291Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88839A3HeLaHUMAN3H-NECAN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89095A3HeLaHUMAN3H-NECAN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide3.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893515-HT6CLONEDHUMAN3H-LSDN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide3441Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240715-HT2ACLONEDHUMANUNDEFINEDQuetiapine110Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89607M3CLONEDHUMAN3H-NMS3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89863nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride59.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
90119D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24839Alpha1ACLONEDHUMAN125I-HEATCLOZAPINE1.6PDSP Certified DataJan 15, 2025Jan 15, 2025
25095SLC6A3CLONEDHUMAN3H-GBR 12935Quetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90631A2BCLONEDHUMAN3H-PSB-6033-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide225 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
253515-HT5ACLONEDHUMAN3H-LSDZOTEPINE29PDSP Certified DataJan 15, 2025Jan 15, 2025
90887Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane109.648Franchini S et al 2014Jan 15, 2025Jan 28, 2025
256075-HT5ACLONEDHUMAN3H-LSDCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91143A2ACHO cellsHUMAN3H-NECAEthyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
258635-HT1BCLONEDHUMAN3H-GR-125743Pseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91399CB1CLONEDHUMAN3H-CP55940O-661785Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26119nAChRCLONEDHUMAN3H-EpibatidinePseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 27, 2025
91655A3CLONEDHUMAN3H-PSB-11N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91911A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (4-chlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26631MORCLONEDHUMAN3H-DiprenorphineMiquelianin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921675-HT6CLONEDHUMAN3H-LSD5-Chloro-N-{1-[2-(phenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide957Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
26887M4CLONEDHUMAN3H-QNBxanomeline19.9526Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92423KORCLONEDHUMAN3H-U69593(5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92679M3CLONEDHUMAN3H-QNB9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27399Beta1CLONEDHUMAN3H-CGP-12177Talipexole>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
92935A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine110Varano F et al 2015Jan 15, 2025Jan 15, 2025
27655D1CLONEDHUMAN3H-SCH23390MDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279115-HT2ACLONEDHUMAN3H-DOBDOM21Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
93703A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester348Federico S et al 2018Jan 15, 2025Jan 15, 2025
28423CLONEDHUMAN3H-QuisqualateQuisqualate10Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93959D2CLONEDHUMAN3H-SPIPERONEcompound 4221Ortega R et al 2011Jan 15, 2025Jan 28, 2025
286795-HT7CLONEDHUMAN3H-LSDARIPIPRAZOLE10.3Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942155-HT1ACLONEDHUMAN3H-8-OH-DPAT2,4,5-trimethoxyamphetamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29191SST2CLONEDHUMANUNDEFINEDBIM 231970.19Patel YC, 1999Jan 15, 2025Jan 15, 2025
947275-HT2ACLONEDHUMAN3H-KETANSERIN4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94983D3CLONEDHUMAN3H-N-Methylspiperone4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29959H4CLONEDHUMAN3H-Histamine(5,7-Difluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone14Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957515-HT7CLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96007DATCLONEDHUMAN3H-WIN 35,4282-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96263Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
965195-HT7CLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
31239Alpha2CCLONEDHUMAN3H-CLONIDINEMDL 1009071442PDSP Certified DataJan 15, 2025Jan 15, 2025
96775D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314955-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)1584.89Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97031D1CLONEDHUMAN[3H]SCH23390Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97287MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o235Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97543A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate31.3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98055CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide420Amato G et al 2019Jan 15, 2025Jan 28, 2025
32775NK1CLONEDHUMAN3H-Sar9,Met(O2)11-Substance PSR 142801291Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98311D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride853Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985675-HT2BCLONEDHUMAN[3H]-LSD4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile152Ofon E et al 2016aJan 15, 2025Jan 15, 2025
332875-HT1ACLONEDHUMAN3H-8-OH-DPATAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98823MORCLONEDHUMAN3H-DAMGO1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33543Alpha1BCLONEDHUMAN3H-PRAZOSINNaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99079Beta1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99335D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol789Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34055P2X3CLONEDHUMAN3H-A-317491A-3173441220Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99591A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine0.683Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99847Alpha2CCLONEDHUMAN[125I] iodoclonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide240Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
1001035-HT2BCLONEDHUMAN3H-LSDQuetiapine86PDSP Certified DataJan 15, 2025Jan 15, 2025
100359DATCLONEDHUMAN3H-WIN 35,428Cariprazine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100615CGRPCLONEDHUMANFunctionalN2-(3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100871Beta2CLONEDHUMAN3H-CGP-121771-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)2Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
35591CLONEDHUMAN3H-SQ 29548CICAPROST1340Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35847SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide23Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013835-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione578Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36103COX-2whole blood assay (WBA)HUMANFunctionalvaleryl salicylate2300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
101639D3CLONEDHUMAN[3H]-N-methylspiperonePerospirone7.7PDSP Certified DataMar 21, 2025Jul 28, 2026
101895NETCLONEDHUMAN[3H]NisoxetineZiprasidone69PDSP Certified DataMar 24, 2025Jul 28, 2026
36615D2CLONEDHUMAN3H-SPIPERONEMIANSERIN2197Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102151DORCLONEDHUMAN[3H]DADLENEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
37895MPP-9CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione19Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38663UNDEFINEDHUMAN3H-hypoxanthineN-[(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-cyclohexylcarbamoyl-2-hydroxy-propyl]-2,4,6-trifluoro-benzamide214Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39175D4CLONEDHUMANR-SATN-DESMETHYLCLOZAPINE70Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39431V2CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396875-HT2BCLONEDHUMAN3H-5HTORG-1296291.2011Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40711mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one84Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41223CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41991M1CLONEDHUMAN3H-QNBDothiepin18Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42247CLONEDHUMAN125I-[Ile]Motilin[L-Bpa5,Ile13]Motilin50Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
43015FYNCLONEDHUMAN3H-StaurosporineGleevec5500Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43271CLK1CLONEDHUMAN3H-StaurosporineSU11248100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43527FLT3CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43783CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44039STK36CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44295CaMKCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44551FLT4CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44807MAPK12CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45063PTK2CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45319CDK2CLONEDHUMANFunctionalkenpaullone670Bain J, et al., 2003Jan 15, 2025Jan 28, 2025
45575NETCLONEDHUMAN3H-NisoxetineDothiepin46Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458315-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46087Alpha2ACLONEDHUMAN3H-CLONIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46599SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46855M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47367Kainate receptorCLONEDHUMAN3H-Kainic acidLY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
47623ADKrecombinantHUMANFunctional4-N-(4-Chlorophenyl)amino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine2.7Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
48135Y2CLONEDHUMAN3H-Propionyl-NPYPP, human1000Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48647GNRHRCLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
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50183mGluR3CLONEDHUMANFunctionalL-CCG-I2100Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
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50951KORUNDEFINEDHUMANUNDEFINED17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate0.12Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51463Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide36Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51719NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline1.1Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51975KORUNDEFINEDHUMANUNDEFINED7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine1.82Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522315-HT1AUNDEFINEDHUMANUNDEFINED4-(1H-indol-4-yloxy)-1-(cyclohexylamino)butan-2-ol872Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52487Alpha2AUNDEFINEDHUMANUNDEFINEDIDAZOXAN8Hagihara K et al., 2007Jan 15, 2025Jan 15, 2025
52999CB2UNDEFINEDHUMANUNDEFINEDN-(4-fluorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide4000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
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54279SLC6A4UNDEFINEDHUMANUNDEFINED2-(2-Dimethylaminomethyl-phenylsulfanyl)-5-methyl-phenylamine2.03Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54535A3UNDEFINEDHUMANUNDEFINED8-[4-(4-benzylpiperazide-1-sulfonyl)phenyl]-1-propylxanthine1000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54791D2UNDEFINEDHUMANUNDEFINEDN-(4-Dipropylaminobutyl)-4-biphenylcarboxamide9700Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
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55303DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2639Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
56071CB1UNDEFINEDHUMANUNDEFINEDHU-2101.5Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56327A3UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione209Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56583KORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol9500Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56839SLC6A2UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-4'-bromo-5'-methylpropiophenone4600Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025