22739 D1 CLONED HUMAN 3H-SCH23390 L-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
33491 D5 CLONED HUMAN 3H-SCH23390 Meloxicam sodium >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41683 D5 CLONED HUMAN 3H-SCH23390 ORG-5222 22.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
42451 D1 CLONED HUMAN 3H-SCH23390 3-methoxy-dibenz[d,g]azecine 28.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46547 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
71892 D1 test test 3H-SCH23390 10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
78036 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79316 D5 CLONED HUMAN 3H-SCH23390 4-Bromo-2,5-dimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
82644 D1 CLONED HUMAN 3H-SCH23390 (S)-1-(Indolin-1-yl)-2-(2-((3-methoxyphenoxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
83668 D1 HEK293 cells HUMAN 3H-SCH23390 Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
84180 D1 CLONED HUMAN 3H-SCH23390 (±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 2465 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
22740 D1 CLONED HUMAN 3H-SCH23390 D-methionine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
39636 D1 STRIATUM RAT 3H-SCH23390 SCH 39166 3.6 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
46548 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid 1824 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70357 D1 CLONED HUMAN 3H-SCH23390 N-Octyl-3-(3-hydroxyphenyl)pyrrolidine 170 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
70613 D1 CLONED HUMAN 3H-SCH23390 MRP3172 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
71381 D5 CLONED HUMAN 3H-SCH23390 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
78037 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79317 D5 CLONED HUMAN 3H-SCH23390 DMT >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
81109 D1 CLONED HUMAN 3H-SCH23390 N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
82645 D5 CLONED HUMAN 3H-SCH23390 (S)-1-(Indolin-1-yl)-2-(2-((3-methoxyphenoxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
22741 D1 CLONED HUMAN 3H-SCH23390 L-methionine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
25301 D5 CLONED HUMAN 3H-SCH23390 Ziprasidone 152 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
26837 D1 BRAIN HUMAN 3H-SCH23390 mCPP 7000 Hamik A, et. al., 1989 Jan 15, 2025 Jan 15, 2025
28117 D5 CLONED HUMAN 3H-SCH23390 Fenfluramine (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
39637 D1 STRIATUM RAT 3H-SCH23390 SCH 23390 0.4 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
46549 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70358 D5 CLONED HUMAN 3H-SCH23390 N-Octyl-3-(3-hydroxyphenyl)pyrrolidine 286 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
70614 D5 CLONED HUMAN 3H-SCH23390 MRP3172 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
71894 D5 test test 3H-SCH23390 10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
79318 D5 CLONED HUMAN 3H-SCH23390 4-Hydroxy-N,N-dimethyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
81110 D5 CLONED HUMAN 3H-SCH23390 N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
25558 D1 CLONED HUMAN 3H-SCH23390 pdspTestCompound3 628 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25814 D5 CLONED HUMAN 3H-SCH23390 Pseudoephedrine, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
39638 D1 STRIATUM RAT 3H-SCH23390 HALOPERIDOL 781 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
42454 D1 CLONED HUMAN 3H-SCH23390 4-chloro-3-hydroxy-dibenz[d,g]azecine 0.83 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46550 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
74967 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
79319 D5 CLONED HUMAN 3H-SCH23390 DMT,5-MeO >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
46551 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
74968 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77784 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79320 D5 CLONED HUMAN 3H-SCH23390 N,N-Diisopropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
24792 D5 CLONED HUMAN 3H-SCH23390 CHLORPROMAZINE 133 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
46552 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
58072 D1 CLONED HUMAN 3H-SCH23390 Memantine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
71897 D5 test test 3H-SCH23390 6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
77785 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79321 D5 CLONED HUMAN 3H-SCH23390 5-Methoxy-N,N-diisopropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
42457 D5 CLONED HUMAN 3H-SCH23390 4-chloro-3-hydroxy-dibenz[d,g]azecine 0.057 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46553 D5 CLONED HUMAN 3H-SCH23390 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
71898 D1 test test 3H-SCH23390 6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
75994 D1 CLONED HUMAN 3H-SCH23390 Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
79322 D5 CLONED HUMAN 3H-SCH23390 N,N-Dipropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
42458 D1 CLONED HUMAN 3H-SCH23390 2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine 3.2 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46554 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
59866 D1 CLONED HUMAN 3H-SCH23390 4-(2-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
71899 D5 test test 3H-SCH23390 6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
75995 D5 CLONED HUMAN 3H-SCH23390 Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
79323 D5 CLONED HUMAN 3H-SCH23390 4-Ethylthio-2,5-dimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
84187 D1 CLONED HUMAN 3H-SCH23390 (±)-4-bromo-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 3135 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
38875 D1 CLONED HUMAN 3H-SCH23390 MDL 11,939 327.2 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
46555 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
71900 D1 test test 3H-SCH23390 N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
77532 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79324 D5 CLONED HUMAN 3H-SCH23390 6-Fluoro-N,N-dimethyltryptamine 6291 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
84188 D5 CLONED HUMAN 3H-SCH23390 (±)-4-bromo-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 8550 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
25820 D1 CLONED HUMAN 3H-SCH23390 Pseudoephedrine, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
28380 D1 CLONED HUMAN 3H-SCH23390 ERGOTAMINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33756 D1 CLONED HUMAN 3H-SCH23390 N-(4-Acetamidophenyl)indomethacinamide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
38876 D1 CLONED HUMAN 3H-SCH23390 SR 46349B >10000 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
42460 D1 CLONED HUMAN 3H-SCH23390 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 9.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46556 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
58076 D5 CLONED HUMAN 3H-SCH23390 Memantine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
70365 D1 CLONED HUMAN 3H-SCH23390 N-Nonyl-3-(3-Hydroxyphenyl)Pyrrolidine 174 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71901 D2 test test 3H-SCH23390 N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
77533 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79325 D5 CLONED HUMAN 3H-SCH23390 LISURIDE 77 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
38877 D1 CLONED HUMAN 3H-SCH23390 MDL 100907 2964 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
46557 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70366 D5 CLONED HUMAN 3H-SCH23390 N-Nonyl-3-(3-Hydroxyphenyl)Pyrrolidine 101 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71902 D5 test test 3H-SCH23390 N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
79326 D5 CLONED HUMAN 3H-SCH23390 (±)-2,5-Dimethoxy-4-iodoamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
94942 D1 CLONED HUMAN 3H-SCH23390 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid 520 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
42462 D5 CLONED HUMAN 3H-SCH23390 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 226.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46558 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
59870 D5 CLONED HUMAN 3H-SCH23390 4-(2-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
79327 D5 CLONED HUMAN 3H-SCH23390 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16095 D5 CLONED HUMAN 3H-SCH23390 SKF-82526, (+) 15 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82143 D1 CLONED HUMAN 3H-SCH23390 6-methoxy-2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)isoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
94943 D1 CLONED HUMAN 3H-SCH23390 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
33759 D5 CLONED HUMAN 3H-SCH23390 N-(4-Acetamidophenyl)indomethacinamide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
38367 D1 BRAIN RAT 3H-SCH23390 MCL-204 0.11 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42463 D1 CLONED HUMAN 3H-SCH23390 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 8.9 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46559 D5 CLONED HUMAN 3H-SCH23390 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
69344 D1 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 83 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
71904 D1 test test 3H-SCH23390 N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
77280 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79328 D5 CLONED HUMAN 3H-SCH23390 (±)-2,5-Dimethoxy-4-methylamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16096 D5 CLONED HUMAN 3H-SCH23390 SKF 38393 100 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82144 D5 CLONED HUMAN 3H-SCH23390 6-methoxy-2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)isoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
94944 D1 CLONED HUMAN 3H-SCH23390 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38368 D1 BRAIN RAT 3H-SCH23390 SCH 23390 0.12 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46560 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
69345 D1 CLONED HUMAN 3H-SCH23390 FLUPHENAZINE 24 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
70369 D1 CLONED HUMAN 3H-SCH23390 N-Decyl-3-(3-hydroxyphenyl)pyrrolidine 128 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
72673 D1 CLONED HUMAN 3H-SCH23390 2,3-dihydrohinokiflavone >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
77281 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79329 D5 CLONED HUMAN 3H-SCH23390 (±)-3,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16097 D5 CLONED HUMAN 3H-SCH23390 Ergocryptine, beta 113 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
87521 D1 CLONED HUMAN 3H-SCH23390 1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
94945 D1 CLONED HUMAN 3H-SCH23390 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31713 D1 STRIATUM RAT 3H-SCH23390 OLANZAPINE 31 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
38369 D1 BRAIN RAT 3H-SCH23390 MCL-203 0.19 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46561 D5 CLONED HUMAN 3H-SCH23390 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
69346 D1 CLONED HUMAN 3H-SCH23390 CHLORPROMAZINE 112 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
70370 D5 CLONED HUMAN 3H-SCH23390 N-Decyl-3-(3-hydroxyphenyl)pyrrolidine 143 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71906 D5 test test 3H-SCH23390 N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
72674 D5 CLONED HUMAN 3H-SCH23390 2,3-dihydrohinokiflavone >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
79330 D5 CLONED HUMAN 3H-SCH23390 (±)-2,5-Dimethoxy-4-ethylamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16098 D5 CLONED HUMAN 3H-SCH23390 APOMORPHINE 363 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
83682 D1 HEK293 cells HUMAN 3H-SCH23390 pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
87522 D5 CLONED HUMAN 3H-SCH23390 1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
94946 D1 CLONED HUMAN 3H-SCH23390 4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31714 D1 STRIATUM RAT 3H-SCH23390 CLOZAPINE 85 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
38370 D1 BRAIN RAT 3H-SCH23390 MCL-207 0.46 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42466 D5 CLONED HUMAN 3H-SCH23390 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 42.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46562 D5 CLONED HUMAN 3H-SCH23390 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
69347 D1 CLONED HUMAN 3H-SCH23390 RACLOPRIDE >10000 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
71907 D5 test test 3H-SCH23390 2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-1-ol >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
79331 D5 CLONED HUMAN 3H-SCH23390 (±)-2,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16099 D5 CLONED HUMAN 3H-SCH23390 BROMOCRIPTINE 454 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82403 D1 CLONED HUMAN 3H-SCH23390 (R)-1-(Indolin-1-yl)-2-(2-(((4-methylpyridin-2-yl)oxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
26083 D1 CLONED HUMAN 3H-SCH23390 Methcathinone, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
28387 D5 CLONED HUMAN 3H-SCH23390 ERGOTAMINE 170 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94947 D1 CLONED HUMAN 3H-SCH23390 4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31715 D1 STRIATUM RAT 3H-SCH23390 REMOXIPRIDE >10000 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
38371 D1 BRAIN RAT 3H-SCH23390 MCL-202 0.49 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
38883 D5 CLONED HUMAN 3H-SCH23390 MDL 11,939 2869 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
42467 D1 CLONED HUMAN 3H-SCH23390 2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 82 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46563 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47331 D1 CLONED HUMAN 3H-SCH23390 WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
69348 D1 CLONED HUMAN 3H-SCH23390 RISPERIDONE 267 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
71908 D5 test test 3H-SCH23390 1,2-dimethoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
72420 D1 CLONED HUMAN 3H-SCH23390 5,6-methylenedioxy-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 28, 2025
72932 D1 CLONED HUMAN 3H-SCH23390 vicenin-2 >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
75748 D1 CLONED HUMAN 3H-SCH23390 3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77028 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79332 D5 CLONED HUMAN 3H-SCH23390 LYSERGIC ACID 344.4 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16100 D5 CLONED HUMAN 3H-SCH23390 SKF-76783 530 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82404 D5 CLONED HUMAN 3H-SCH23390 (R)-1-(Indolin-1-yl)-2-(2-(((4-methylpyridin-2-yl)oxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
25060 D5 CLONED HUMAN 3H-SCH23390 OLANZAPINE 90 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94948 D1 CLONED HUMAN 3H-SCH23390 4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31716 D1 STRIATUM RAT 3H-SCH23390 Quetiapine 455 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
38372 D1 BRAIN RAT 3H-SCH23390 MCL-210 0.52 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
38884 D5 CLONED HUMAN 3H-SCH23390 MDL 100907 >10000 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
46564 D5 CLONED HUMAN 3H-SCH23390 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
69349 D1 CLONED HUMAN 3H-SCH23390 CLOZAPINE 189 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
72933 D5 CLONED HUMAN 3H-SCH23390 vicenin-2 >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
75749 D5 CLONED HUMAN 3H-SCH23390 3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77029 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79333 D5 CLONED HUMAN 3H-SCH23390 cis-2a 1013 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16101 D5 CLONED HUMAN 3H-SCH23390 SKF-82526, (-) 800 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
86245 D1 CLONED HUMAN 3H-SCH23390 JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
94949 D1 CLONED HUMAN 3H-SCH23390 4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31717 D1 STRIATUM RAT 3H-SCH23390 ORG-5222 5 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
38373 D1 BRAIN RAT 3H-SCH23390 MCL-209 0.6 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46565 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
69350 D1 CLONED HUMAN 3H-SCH23390 OLANZAPINE 58 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
71910 D1 test test 3H-SCH23390 1-(cyclopropylmethoxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
74726 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
79334 D5 CLONED HUMAN 3H-SCH23390 R,R-2b 591.9 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16102 D5 CLONED HUMAN 3H-SCH23390 ADTN, (+) 909 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
86246 D5 CLONED HUMAN 3H-SCH23390 JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
24806 D1 CLONED HUMAN 3H-SCH23390 CHLORPROMAZINE 112 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94950 D1 CLONED HUMAN 3H-SCH23390 4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31718 D1 STRIATUM RAT 3H-SCH23390 HALOPERIDOL 25 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
38374 D1 BRAIN RAT 3H-SCH23390 MCL-214 1.1 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42470 D1 CLONED HUMAN 3H-SCH23390 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 25.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46566 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
59110 D1 CLONED HUMAN 3H-SCH23390 Beta-LT >10000 Buhler A, et al., 2007 Jan 15, 2025 Jan 15, 2025
69351 D1 CLONED HUMAN 3H-SCH23390 Quetiapine 712 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
74727 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
79335 D5 CLONED HUMAN 3H-SCH23390 S,S-2c 402.2 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16103 D5 CLONED HUMAN 3H-SCH23390 PERGOLIDE 918 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
84199 D5 CLONED HUMAN 3H-SCH23390 (±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 6789 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
94951 D1 CLONED HUMAN 3H-SCH23390 4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38375 D1 BRAIN RAT 3H-SCH23390 SKF-83959 1.18 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46567 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47335 D5 CLONED HUMAN 3H-SCH23390 WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
72424 D5 CLONED HUMAN 3H-SCH23390 5,6-methylenedioxy-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 28, 2025
76776 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79336 D5 CLONED HUMAN 3H-SCH23390 5-MeO-TMT >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16104 D5 CLONED HUMAN 3H-SCH23390 N-0437 986 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82664 D1 CLONED HUMAN 3H-SCH23390 (R)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
84200 D1 CLONED HUMAN 3H-SCH23390 (±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 2703 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
25320 D1 CLONED HUMAN 3H-SCH23390 Ziprasidone 30 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94952 D1 CLONED HUMAN 3H-SCH23390 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38376 D1 BRAIN RAT 3H-SCH23390 MCL-216 1.81 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46568 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70377 D1 CLONED HUMAN 3H-SCH23390 (-)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine 181 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
73193 D1 test test 3H-SCH23390 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
76777 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79337 D5 CLONED HUMAN 3H-SCH23390 EMDT >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16105 D5 CLONED HUMAN 3H-SCH23390 NPA 1136 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82665 D5 CLONED HUMAN 3H-SCH23390 (R)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
25065 D1 CLONED HUMAN 3H-SCH23390 OLANZAPINE 58 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94953 D1 CLONED HUMAN 3H-SCH23390 2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38377 D1 BRAIN RAT 3H-SCH23390 SKF 81297 1.9 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42473 D1 CLONED HUMAN 3H-SCH23390 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 0.46 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46569 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70378 D5 CLONED HUMAN 3H-SCH23390 (-)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine 227 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71914 D1 test test 3H-SCH23390 1-(allyloxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
73194 D5 test test 3H-SCH23390 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74474 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
79338 D5 CLONED HUMAN 3H-SCH23390 Salvinorin A >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
16106 D5 CLONED HUMAN 3H-SCH23390 5-Hydroxy Tryptamine 3000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
94954 D1 CLONED HUMAN 3H-SCH23390 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
33258 D1 CLONED HUMAN 3H-SCH23390 nimesulide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
38378 D1 BRAIN RAT 3H-SCH23390 MCL-206 1.93 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46570 D5 CLONED HUMAN 3H-SCH23390 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
73451 D1 test test 3H-SCH23390 N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74475 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75499 D1 CLONED HUMAN 3H-SCH23390 propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
16107 D5 CLONED HUMAN 3H-SCH23390 NOREPINEPHRINE >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
94955 D5 CLONED HUMAN 3H-SCH23390 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid 1440 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38379 D1 BRAIN RAT 3H-SCH23390 (R)(+)-BrAPB 2.29 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46571 D5 CLONED HUMAN 3H-SCH23390 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
59627 D1 CLONED HUMAN 3H-SCH23390 RU 24213 >10000 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
66028 D1 CLONED HUMAN 3H-SCH23390 Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
71916 D5 test test 3H-SCH23390 1-(allyloxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
75500 D5 CLONED HUMAN 3H-SCH23390 propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
16108 D5 CLONED HUMAN 3H-SCH23390 LY-171555 >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
94956 D5 CLONED HUMAN 3H-SCH23390 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38380 D1 BRAIN RAT 3H-SCH23390 MCL-205 4.41 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42476 D5 CLONED HUMAN 3H-SCH23390 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 0.98 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46572 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70381 D1 CLONED HUMAN 3H-SCH23390 (+)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine >10000 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
76525 D1 CLONED HUMAN 3H-SCH23390 (1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
11501 D1 STRIATUM RAT 3H-SCH23390 Pifluthixol 0.63 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
16109 D5 CLONED HUMAN 3H-SCH23390 SCH 23390 0.3 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
21741 D1 STRIATUM RAT 3H-SCH23390 Amisulpride >10000 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
94957 D5 CLONED HUMAN 3H-SCH23390 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38381 D1 BRAIN RAT 3H-SCH23390 SKF 82958 4.56 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42477 D1 CLONED HUMAN 3H-SCH23390 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3.1 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
46573 D5 CLONED HUMAN 3H-SCH23390 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
70382 D5 CLONED HUMAN 3H-SCH23390 (+)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine 639 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71918 D5 test test 3H-SCH23390 2-methoxy-6-methyl-10-nitro-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
76526 D5 CLONED HUMAN 3H-SCH23390 (1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
16110 D5 CLONED HUMAN 3H-SCH23390 SKF 83566 0.4 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
21742 D1 STRIATUM RAT 3H-SCH23390 HALOPERIDOL 250 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
94958 D5 CLONED HUMAN 3H-SCH23390 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
33262 D5 CLONED HUMAN 3H-SCH23390 nimesulide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
38382 D1 BRAIN RAT 3H-SCH23390 MCL-211 8.66 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
46574 D5 CLONED HUMAN 3H-SCH23390 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
73455 D5 test test 3H-SCH23390 N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
16111 D5 CLONED HUMAN 3H-SCH23390 FLUPENTHIXOL, Alpha 8 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
21743 D1 STRIATUM RAT 3H-SCH23390 CLOZAPINE 590 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
94959 D5 CLONED HUMAN 3H-SCH23390 4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38383 D1 BRAIN RAT 3H-SCH23390 SKF 77434 10.5 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
59631 D5 CLONED HUMAN 3H-SCH23390 RU 24213 >10000 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
59887 D1 CLONED HUMAN 3H-SCH23390 4-(4-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
66032 D5 CLONED HUMAN 3H-SCH23390 Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
71920 D5 test test 3H-SCH23390 1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
12528 D1 Choroid Plexus CANINE 3H-SCH23390 5-Hydroxy Tryptamine >10000 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
16112 D5 CLONED HUMAN 3H-SCH23390 BUTACLAMOL,(+) 27 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
83696 D1 HEK293 cells HUMAN 3H-SCH23390 MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
94960 D5 CLONED HUMAN 3H-SCH23390 4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38384 D1 BRAIN RAT 3H-SCH23390 MCL-212 19.3 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42480 D5 CLONED HUMAN 3H-SCH23390 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 4.9 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
12529 D1 Choroid Plexus CANINE 3H-SCH23390 MIANSERIN 161 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
78833 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
16113 D5 CLONED HUMAN 3H-SCH23390 SCH 23388 35 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
94961 D5 CLONED HUMAN 3H-SCH23390 4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38385 D1 BRAIN RAT 3H-SCH23390 MCL-201 21.3 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42481 D1 CLONED HUMAN 3H-SCH23390 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 8.7 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
67314 D1 CLONED HUMAN 3H-SCH23390 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
71410 D1 CLONED HUMAN 3H-SCH23390 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71922 D5 test test 3H-SCH23390 1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
12530 D1 Choroid Plexus CANINE 3H-SCH23390 KETANSERIN 166 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
78834 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
16114 D5 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 48 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
94962 D5 CLONED HUMAN 3H-SCH23390 4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38386 D1 BRAIN RAT 3H-SCH23390 SKF 38393 26.6 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
73715 D1 test test 3H-SCH23390 [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
12531 D1 Choroid Plexus CANINE 3H-SCH23390 DOPAMINE >10000 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
16115 D5 CLONED HUMAN 3H-SCH23390 CHLORPROMAZINE 133 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82163 D1 CLONED HUMAN 3H-SCH23390 5-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one 2734 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
84211 D1 CLONED HUMAN 3H-SCH23390 (±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 2100 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
90099 D1 CLONED HUMAN 3H-SCH23390 4-Bromo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
25331 D5 CLONED HUMAN 3H-SCH23390 ZOTEPINE 248 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94963 D5 CLONED HUMAN 3H-SCH23390 4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
31731 D1 STRIATUM RAT 3H-SCH23390 RISPERIDONE 75 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
98803 D1 CLONED HUMAN 3H-SCH23390 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
38387 D1 BRAIN RAT 3H-SCH23390 MCL-215 37.1 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
59635 D1 CLONED HUMAN 3H-SCH23390 SK&F 83822 3.2 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
59891 D5 CLONED HUMAN 3H-SCH23390 4-(4-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
71156 D1 CLONED HUMAN 3H-SCH23390 ARIPIPRAZOLE 1960 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71924 D5 test test 3H-SCH23390 1-(allyloxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
73972 D1 test test 3H-SCH23390 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
12532 D1 Choroid Plexus CANINE 3H-SCH23390 FLUPENTHIXOL, Alpha 30 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
16116 D5 CLONED HUMAN 3H-SCH23390 CLOZAPINE 250 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82164 D5 CLONED HUMAN 3H-SCH23390 5-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
84212 D5 CLONED HUMAN 3H-SCH23390 (±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 7178 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
90100 D1 CLONED HUMAN 3H-SCH23390 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
25332 D1 CLONED HUMAN 3H-SCH23390 ZOTEPINE 71 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
94964 D5 CLONED HUMAN 3H-SCH23390 4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
98804 D5 CLONED HUMAN 3H-SCH23390 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine 3016 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
38388 D1 BRAIN RAT 3H-SCH23390 MCL-213 128 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42484 D1 CLONED HUMAN 3H-SCH23390 4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 7.6 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
67317 D5 CLONED HUMAN 3H-SCH23390 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
70389 D1 CLONED HUMAN 3H-SCH23390 (Rac)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 831 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71157 D1 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 120 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71925 D5 test test 3H-SCH23390 2-methoxy-6-methyl-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
73973 D5 test test 3H-SCH23390 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
12533 D1 Choroid Plexus CANINE 3H-SCH23390 BUTACLAMOL,(+) 3.7 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
78581 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
16117 D5 CLONED HUMAN 3H-SCH23390 THIORIDAZINE 300 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
85237 D1 recombinant HUMAN 3H-SCH23390 Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 28, 2025
90101 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
94965 D5 CLONED HUMAN 3H-SCH23390 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
38389 D1 BRAIN RAT 3H-SCH23390 MCL-218 1238 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
70390 D5 CLONED HUMAN 3H-SCH23390 (Rac)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 312 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
70902 D1 test test 3H-SCH23390 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 5.7 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
71158 D1 CLONED HUMAN 3H-SCH23390 CLOZAPINE 290 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71414 D5 CLONED HUMAN 3H-SCH23390 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
75254 D1 CLONED HUMAN 3H-SCH23390 ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
12534 D1 Choroid Plexus CANINE 3H-SCH23390 BUTACLAMOL, (-) >10000 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
78582 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
16118 D5 CLONED HUMAN 3H-SCH23390 KETANSERIN 2500 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
90102 D1 CLONED HUMAN 3H-SCH23390 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
94966 D5 CLONED HUMAN 3H-SCH23390 2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate 3010 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
34294 D1 STRIATUM RAT 3H-SCH23390 Dihydrexidine, DHX 10 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
38390 D1 BRAIN RAT 3H-SCH23390 MCL-230A >10000 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
70903 D5 test test 3H-SCH23390 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6.7 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
71159 D1 CLONED HUMAN 3H-SCH23390 SYA013 163 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
73719 D5 test test 3H-SCH23390 [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
75255 D5 CLONED HUMAN 3H-SCH23390 ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
16119 D5 CLONED HUMAN 3H-SCH23390 SPIPERONE 4500 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82423 D1 CLONED HUMAN 3H-SCH23390 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((4-methylpyridin-2-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
90103 D1 CLONED HUMAN 3H-SCH23390 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
94967 D5 CLONED HUMAN 3H-SCH23390 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
33527 D1 CLONED HUMAN 3H-SCH23390 Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34295 D1 STRIATUM RAT 3H-SCH23390 Dihydrexidine, DHX 9.7 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
36599 D1 STRIATUM RAT 3H-SCH23390 RISPERIDONE >10000 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
38391 D1 BRAIN RAT 3H-SCH23390 MCL-217 >10000 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
42487 D1 CLONED HUMAN 3H-SCH23390 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 2 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
59639 D5 CLONED HUMAN 3H-SCH23390 RU 24213 3.1 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
70904 D1 test test 3H-SCH23390 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione 10 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
71160 D1 CLONED HUMAN 3H-SCH23390 SYA16263 238 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71928 D5 test test 3H-SCH23390 N-(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl) >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
76280 D1 CLONED HUMAN 3H-SCH23390 (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
16120 D5 CLONED HUMAN 3H-SCH23390 ETICLOPRIDE >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82424 D5 CLONED HUMAN 3H-SCH23390 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((4-methylpyridin-2-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
90104 D1 CLONED HUMAN 3H-SCH23390 4-iodo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
34296 D1 STRIATUM HUMAN 3H-SCH23390 Dihydrexidine, DHX 35.7 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
36600 D1 STRIATUM RAT 3H-SCH23390 9-OH-risperidone 510 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
3833 D1 CLONED RAT 3H-SCH23390 LY 344864 >10000 PHEBUS LA, ET AL, 1997 Jan 15, 2025 Jan 15, 2025
70649 D1 CLONED HUMAN 3H-SCH23390 MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
70905 D5 test test 3H-SCH23390 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione 15 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
76281 D5 CLONED HUMAN 3H-SCH23390 (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
16121 D5 CLONED HUMAN 3H-SCH23390 SULPIRIDE,(+) >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
90105 D1 CLONED HUMAN 3H-SCH23390 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
25849 D1 CLONED HUMAN 3H-SCH23390 Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
26361 D1 CLONED HUMAN 3H-SCH23390 Hyperforin 595.8 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
34297 D1 STRIATUM RAT 3H-SCH23390 Dihydrexidine, DHX 2.3 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
70650 D5 CLONED HUMAN 3H-SCH23390 MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
78330 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
81402 D1 CLONED HUMAN 3H-SCH23390 [1-(1-phenoxypropan-2-yl)piperidin-3-yl]-pyridin-3-ylmethanone >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16122 D5 CLONED HUMAN 3H-SCH23390 SULPIRIDE,(-) >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
85242 D5 recombinant HUMAN 3H-SCH23390 Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 28, 2025
90106 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 8400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
26106 D5 CLONED HUMAN 3H-SCH23390 Methcathinone, (-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34298 D1 STRIATUM RAT 3H-SCH23390 Dihydrexidine, DHX 4.59 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
42490 D5 CLONED HUMAN 3H-SCH23390 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1.68 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
70907 D1 test test 3H-SCH23390 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 70 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
71931 D5 test test 3H-SCH23390 N-(1-(allyloxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
78331 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
16123 D1 CLONED HUMAN 3H-SCH23390 SKF-82526, (+) 28 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
90107 D1 CLONED HUMAN 3H-SCH23390 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
93947 D1 STRIATUM PIG 3H-SCH23390 compound 42 2500 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
33531 D5 CLONED HUMAN 3H-SCH23390 Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34299 D1 STRIATUM RAT 3H-SCH23390 Dihydrexidine, DHX 6.2 Salmi P, et al., 2004 Jan 15, 2025 Jan 15, 2025
36603 D1 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 359 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
42491 D1 CLONED HUMAN 3H-SCH23390 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 9.4 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
59643 D1 CLONED HUMAN 3H-SCH23390 SK&F 83959 0.5 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
70396 D1 CLONED HUMAN 3H-SCH23390 (-)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 4589 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
70908 D5 test test 3H-SCH23390 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 171 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
74236 D1 test test 3H-SCH23390 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
16124 D1 CLONED HUMAN 3H-SCH23390 SKF 38393 150 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
82684 D1 CLONED HUMAN 3H-SCH23390 (S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine 8366 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
90108 D1 CLONED HUMAN 3H-SCH23390 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
93948 D1 STRIATUM PIG 3H-SCH23390 compound 43 2900 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
36604 D1 CLONED HUMAN 3H-SCH23390 CLOZAPINE 539 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
70397 D5 CLONED HUMAN 3H-SCH23390 (-)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 955 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
71933 D5 test test 3H-SCH23390 N-(2-methoxy-6-methyl-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide >10000 Karki A et al., 2020 Jan 15, 2025 Jan 28, 2025
74237 D5 test test 3H-SCH23390 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
82685 D5 CLONED HUMAN 3H-SCH23390 (S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine 8525 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
90109 D1 CLONED HUMAN 3H-SCH23390 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
93949 D1 STRIATUM PIG 3H-SCH23390 3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 2100 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
36605 D1 CLONED HUMAN 3H-SCH23390 OLANZAPINE 118 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
3838 D1 CLONED RAT 3H-SCH23390 ILOPERIDONE 546 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
70398 D5 CLONED HUMAN 3H-SCH23390 (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide >10000 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
78078 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
81150 D1 CLONED HUMAN 3H-SCH23390 N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
16126 D1 CLONED HUMAN 3H-SCH23390 DOPAMINE 2340 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81918 D1 CLONED HUMAN 3H-SCH23390 (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
90110 D1 CLONED HUMAN 3H-SCH23390 MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
93950 D1 STRIATUM PIG 3H-SCH23390 7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one 2300 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
36606 D1 CLONED HUMAN 3H-SCH23390 RISPERIDONE 147 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
42494 D5 CLONED HUMAN 3H-SCH23390 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 12.6 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
3839 D1 CLONED RAT 3H-SCH23390 RISPERIDONE 550 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
70399 D1 CLONED HUMAN 3H-SCH23390 (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide >10000 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
70911 D1 test test 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 93 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
78079 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
81151 D5 CLONED HUMAN 3H-SCH23390 N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
16127 D1 CLONED HUMAN 3H-SCH23390 APOMORPHINE 680 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81919 D5 CLONED HUMAN 3H-SCH23390 (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
90111 D1 CLONED HUMAN 3H-SCH23390 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 9300 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
93951 D1 STRIATUM PIG 3H-SCH23390 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one 640 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
36607 D1 CLONED HUMAN 3H-SCH23390 mirtazepine 4167 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
59647 D5 CLONED HUMAN 3H-SCH23390 SK&F 83959 2.1 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
256 5-HT1A CORTEX RAT 3H-8-OH-DPAT DHE 19 McCARTHY & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
69376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 1202 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
13312 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT CITALOPRAM >10000 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
80896 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
83200 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LSD 2.78 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85760 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide 230 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
27136 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CP-132,484 8410 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94208 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine 3300 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
37632 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(1-Naphthalenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.6 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
257 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DILTIAZEM >10000 PEROUTKA, 1988 Jan 15, 2025 Jan 15, 2025
67841 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
69377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPHENAZINE 145 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
13313 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT INDALPINE 9120.1 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
82689 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85761 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87041 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 2000 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 365 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24577 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.8 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
90881 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane 50.1187 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27137 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CP-132,484(4b) 287 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94209 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-benzyloxy-2,5-dimethoxyphenethylamine 2700 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
101377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 22 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37633 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(4-Chloro-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 433 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
258 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DMT 119.51 PIERCE & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
514 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 32.76 HALL ET AL., 1985 Jan 15, 2025 Jan 15, 2025
69378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CHLORPROMAZINE 3115 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
13314 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT PAROXETINE >10000 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
24578 5-HT1A FR. CORTEX RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 4.2 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
27138 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N,N-dimethyl derivative 562 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94210 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-allyloxy-2,5-dimethoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
37634 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(4-Methyl-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 58.6 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
515 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 45.12 COSSERY ET AL.,1986 Jan 15, 2025 Jan 15, 2025
69379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RACLOPRIDE >10000 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
13315 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT Femoxetine 3162.27 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
27139 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
37635 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[3-[4-(2,3-Dichlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 117 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
260 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT DMT 140.74 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
516 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 48.07 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
69380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 427 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
80644 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
86788 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide 590 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87044 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one 58.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
27140 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94212 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
37636 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 123 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
261 5-HT1A CORTEX RAT 3H-8-OH-DPAT DMT 245 TAYLOR ET AL,. 1987 Jan 15, 2025 Jan 15, 2025
517 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIPERONE 54 FOZARD ET AL., 1987 Jan 15, 2025 Jan 15, 2025
3333 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Amphetamine,(+) 6606 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 105 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
83205 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DMT 450 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
86789 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide 325 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90885 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 42.658 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27141 5-HT1A CLONED HUMAN 3H-8-OH-DPAT AL-37350A >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94213 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
37637 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide 78.7 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
262 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB 3770 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
67846 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3334 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SKF 82958 1781 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT OLANZAPINE 2063 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
83206 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOM >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85766 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide 495 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
27142 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOI,(-) 3843 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94214 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-isopropoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
101382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 48 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37638 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 19.8 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
3335 5-HT1A CLONED HUMAN 3H-8-OH-DPAT APOMORPHINE 4929 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Quetiapine 431 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
85767 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide 500 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87047 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one 196.2 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
94215 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,4,5-trimethoxyamphetamine >10000 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
31495 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) 1584.89 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
33287 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37639 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 7.5 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
264 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DOB 6326.73 PIERCE & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
520 5-HT1A CELLS C0S-7 3H-8-OH-DPAT SPIPERONE 63 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3336 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BROMOCRIPTINE,(+) 25 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
80392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 3215 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
89352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 3842 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89608 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 0.47863 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
94216 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-Bromo-2,5-dimethoxyphenethylamine 311 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
31496 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) 1000 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
37640 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide 4.5 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
265 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB 3770 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
521 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 66.1 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
3337 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CARBAMAZEPINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
81161 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
90889 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 20.4174 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
37641 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[3-[4-(4-Chlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 850 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
266 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB,R(-) 2332 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68106 5-HT1A UNDEFINED UNDEFINED 3H-8-OH-DPAT ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
3338 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CGS 12066B 44 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
14602 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SB-277011-A 5011.87 Reavill C., et al., 2000 Jan 15, 2025 Jan 15, 2025
83722 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 9987 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
86794 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide 219 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87050 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 193.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
26890 5-HT1A CLONED HUMAN 3H-8-OH-DPAT xanomeline 63.0957 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
37642 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 397 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
267 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB,S(+) 4041 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
523 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 66.1 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
67851 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3339 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CHLORPROMAZINE 3115 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78603 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
81675 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 15, 2025
83211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN 6510 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
86795 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide 331 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
89355 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 802 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
101387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 35 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37643 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[5-[4-(4-Chlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide 850 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
268 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOBU 4178 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
524 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 66.1 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3340 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOMIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
82188 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one 62 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
83212 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ro 60-0175 6680 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85772 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
31244 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PPP, S(-)-3 1730 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37644 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dimethylphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 268 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
269 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOET 3930 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3341 5-HT1A CLONED HUMAN 3H-8-OH-DPAT COCAINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
85773 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87053 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on 98 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89613 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 2.5704 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90893 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane 36.3078 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
25869 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27405 5-HT1A CLONED HUMAN 3H-8-OH-DPAT APOMORPHINE 117.49 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
37645 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(1-Naphthalenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 0.43 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
270 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOI 2355 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3342 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CYPROHEPTADINE 59 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
89614 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.86209 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27406 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BROMOCRIPTINE 12.8825 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
37646 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(1-Isoquinolyl)piperazin-1-yl]butyl]-3-methoxybenzamide 12.7 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
271 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT GEPIRONE 70 GLENNON ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3343 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DEPRENYL >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
27407 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Cabergoline 19.9526 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
37647 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(1,2-Benzisoxazol-3-yl)piperazin-1-yl]butyl]-3-methoxybenzamide 7730 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
67856 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3344 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DESIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80656 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82448 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine 0.6 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
86800 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide 99.1 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87056 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one 69.1 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
27408 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LISURIDE 0.147911 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95248 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 192.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 482 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37648 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-bromo-1-methoxy-2-naphthalenecarboxamide 1000 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
273 5-HT1A CORTEX PIG 3H-8-OH-DPAT GEPIRONE 89.1 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
3345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DHE 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
83217 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SB242087 9300 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
86801 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide 100 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
88593 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 140 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
90897 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one 64.5654 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27409 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PERGOLIDE 1.90546 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95249 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 182 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37649 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-methoxy-2-naphthalenecarboxamide 575 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
530 5-HT1A HIPPOCAMPUS HUMAN 3H-8-OH-DPAT SPIPERONE 100.92 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
83218 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide 1.21 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85778 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide 443 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
21778 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT CLOZAPINE 1700 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
89362 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 6631 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
27410 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piribedil 446.684 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
27666 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
95250 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 728.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37650 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-naphthalenecarboxamide 335 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
275 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT HALOPERIDOL 2761.11 GOZLAN ET AL., 1983 Jan 15, 2025 Jan 15, 2025
531 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 101 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
3347 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOPAMINE 8248 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
85779 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide 52.7 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87059 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 82.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
21779 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT HALOPERIDOL 2500 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
89619 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1.25893 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27411 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Pramipexole 691.831 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95251 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 82.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37651 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-quinolinecarboxamide 88.5 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
532 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIPERONE 120 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
3348 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 8-OH-DPAT 6.9 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78100 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80404 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
21780 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT Amisulpride >10000 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
89620 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.562341 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27412 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Quinelorane >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95252 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 212.6 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31252 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PPP, R(+)-3 868.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33556 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CELECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37652 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-(1,1'-biphenyl)-4-carboxamide 1000 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
277 5-HT1A CORTEX PIG 3H-8-OH-DPAT HALOPERIDOL 4790 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
533 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT SPIPERONE 130.76 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
67861 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 146 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3349 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ETICLOPRIDE,S(-) 1790 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
77845 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
13845 5-HT1A BRAIN RAT 3H-8-OH-DPAT CLOZAPINE 150 Tang AH, et al., 1996 Jan 15, 2025 Jan 15, 2025
82709 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
89365 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 6064 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
90901 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one 323.594 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27413 5-HT1A CLONED HUMAN 3H-8-OH-DPAT QUINPIROLE 1698.24 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95253 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 2600 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101397 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 20 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37653 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-benzofurancarboxamide36 126 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
534 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIPERONE 140 SCHLEGEL & PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
3350 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPENTHIXOL, Alpha 8028 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
86806 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide 9.19 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87062 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(3-(4-(6-fluoro benzo[d]isoxazol-3-yl)piperidin-1-yl)- 1-hydroxypropyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 19.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
27414 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ropinirole 288.403 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95254 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 158 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
33046 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT GBR-12909 3600 Andersen PH, et al., 1989 Jan 15, 2025 Jan 15, 2025
37654 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide 1660 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
535 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 148.4 HALL ET AL., 1986 Jan 15, 2025 Jan 15, 2025
3351 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPHENAZINE 2829 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
86807 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide 0.0113 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
27415 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Roxindole 0.114815 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95255 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 298 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37655 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indole-3-carboxamide 1110 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
50711 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 0.15 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
280 5-HT1A CELLS C0S-7 3H-8-OH-DPAT HISTAMINE 6011 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
536 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT SPIPERONE 155.56 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
68376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT GBR-12909 4677 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
85784 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl)picolinamide 44.1 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88600 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
89624 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 0.616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27416 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Talipexole 1698.24 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95256 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 2500 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37656 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indazole-3-carboxamide 621 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
39192 5-HT2B CLONED HUMAN 3H-8-OH-DPAT ATC0065 266 Chaki S, et al., 2005 Jan 15, 2025 Jan 15, 2025
50712 5-HT1B HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 643 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
68377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3353 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ondansetron HCl >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
85785 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-OH-DPAT 0.8 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87065 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 79.1 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89625 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90905 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 52.4807 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27417 5-HT1A CLONED HUMAN 3H-8-OH-DPAT TERGURIDE 3.46737 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95257 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 196.3 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31257 5-HT1A C.H.O. HUMAN 3H-8-OH-DPAT Ropinirole 288.403 Millan MJ, et. al., 2004 Jan 15, 2025 Jan 15, 2025
99865 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride 138 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
37657 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide 5500 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
38937 5-HT1A CORTEX RAT 3H-8-OH-DPAT QUIPAZINE,8-Me 1700 Glennon RA, et al., 1989 Jan 15, 2025 Jan 15, 2025
39193 5-HT2B CLONED HUMAN 3H-8-OH-DPAT ATC0175 9.66 Chaki S, et al., 2005 Jan 15, 2025 Jan 15, 2025
50713 5-HT1D HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 88.3 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
67866 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 66 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3354 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 5084 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
17178 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METHYLPHENIDATE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27418 5-HT1A CLONED HUMAN 3H-8-OH-DPAT TL99 3801.89 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95258 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 199.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101402 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 47 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37658 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-7-methoxy-2-benzofurancarboxamide 184 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
50714 5-HT1E HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
68379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.25893 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3355 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IBOGAINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
83739 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 8590 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
95259 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 229.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37659 5-HT1A Hippocampal RAT 3H-8-OH-DPAT 8-OH-DPAT 2.1 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
50715 5-HT2A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 4975 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
540 5-HT1A CELLS C0S-7 3H-8-OH-DPAT SPIROXATRINE 1.8 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 6.60693 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3356 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ICS 205-930 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
77596 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80668 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
86812 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(furoyl)piperazin-1-yl)propyl)isonicotinamide 779 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87068 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 84.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89372 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 2630 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
95260 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 365.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101148 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone 272 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50716 5-HT2B HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 73.6 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
68381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3357 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IDAZOXAN 662 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
86813 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
88605 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
90909 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 26.9153 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
95261 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 210.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
99869 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride 7 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
101149 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone 350 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50717 5-HT2C HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
542 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIROXATRINE 2.56 ALEXANDER & WOOD, 1988 Jan 15, 2025 Jan 15, 2025
68382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3358 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IMIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
13854 5-HT1A BRAIN RAT 3H-8-OH-DPAT PNU-96415E 134 Tang AH, et al., 1996 Jan 15, 2025 Jan 15, 2025
83486 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
89630 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0645654 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95262 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 218 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
99870 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride 22 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
50718 5-HT3 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
67871 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 91 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3359 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
87071 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 81.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89375 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 1836 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89631 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0147911 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95263 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide 476 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101407 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 28 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
50719 5-HT5A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
68384 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3360 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDL 72222 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
77344 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
80416 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
95264 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide 130 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31520 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(2-(1-(3,4-Dichloro-benzene sulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine 316.228 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
101152 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50720 5-HT6 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
545 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIROXATRINE 8.91 SCHOEFFTER AND HOYER,1988 Jan 15, 2025 Jan 15, 2025
68385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 1.25893 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3361 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDA,R(-) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
90913 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 37.1535 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
95265 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide 2000 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31521 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(2-(1-(3-bromo-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine 398.107 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
33057 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT BUPROPION >10000 Andersen PH, et al., 1989 Jan 15, 2025 Jan 15, 2025
101153 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone 33.5 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
38945 5-HT1A CORTEX RAT 3H-8-OH-DPAT QUIPAZINE 2000 Glennon RA, et al., 1989 Jan 15, 2025 Jan 15, 2025
50721 5-HT7 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 12.9 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
68386 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 6.60693 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3362 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDMA, R(-) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
82210 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one 20 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
18466 D3 BRAIN pigeon 3H-8-OH-DPAT WAY 100,635 370 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
86818 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide 0.13 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87074 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile 473.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
25378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ARIPIPRAZOLE 5.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25890 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Norephedrine, (+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
95266 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide 314.8 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
50722 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
547 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIROXATRINE,(+) 21 NIKAM ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3363 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METHAMPHETAMINE (+) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18467 D3 BRAIN pigeon 3H-8-OH-DPAT WAY 100,135 >10000 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
20259 5-HT1A CORTEX RAT 3H-8-OH-DPAT Benzamil 1900 Garritsen A et al., 1991 Jan 15, 2025 Jan 15, 2025
86819 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide 1060 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
89635 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0338844 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95267 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide 484.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
50723 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 6.75 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
67876 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 147 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68388 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piperazine 1.28825 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3364 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 5-HT,2-Me 3074 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
77092 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
82468 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(Indolin-1-yl)-2-(2-((pyridin-3-yloxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
18468 D3 BRAIN pigeon 3H-8-OH-DPAT DU125530 11 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
20260 5-HT1A CORTEX RAT 3H-8-OH-DPAT Amiloride >10000 Garritsen A et al., 1991 Jan 15, 2025 Jan 15, 2025
89636 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NLX-101 2.18776 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95268 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide 2300 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101156 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone 1684 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
101412 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 3569 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
50724 Beta2 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
293 5-HT1A CORTEX RAT 3H-8-OH-DPAT HISTAMINE >10000 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
549 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIROXATRINE,(-) 1.9 NIKAM ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68389 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 22.9087 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3365 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METHYLPHENIDATE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
12325 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 14489 0.61 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18469 D2 BRAIN pigeon 3H-8-OH-DPAT PINDOLOL,(+/-) >10000 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87077 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 54.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
90917 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane 69.1831 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
95269 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide 62.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101157 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone 81.8 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50725 Alpha2A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 96 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
550 5-HT1A CELLS C0S-7 3H-8-OH-DPAT SULPIRIDE 589 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68390 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 0.831764 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3366 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METOCLOPRAMIDE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
12326 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 15535 1.77 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18470 D2 BRAIN pigeon 3H-8-OH-DPAT NAN-190 14 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
89382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 160 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
95270 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide 30.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
50726 Alpha2B HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 238 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
68391 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 4-hydroxy piperid-1-yl] 5-fluoroindan-1-01 1000 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3367 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MIANSERIN 2592 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11303 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 420 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12327 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 15931 1.51 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18471 D2 BRAIN pigeon 3H-8-OH-DPAT S 15535 132 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
88615 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 658 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
89639 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 8-OH-DPAT 0.812831 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95271 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 9.4 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
40743 5-HT1A CLONED HUMAN 3H-8-OH-DPAT URB 597 >10000 Gobbi G, et al., 2005 Jan 15, 2025 Jan 15, 2025
50727 Alpha2C HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 15.4 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
296 5-HT1A CELLS C0S-7 3H-8-OH-DPAT ICS 205-930 1788 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperid-1-yl] indan-1-01 0.707946 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3368 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NAN-190 3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11304 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 9-OH-risperidone 590 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
76840 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
12328 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT Eltoprazine 9.33 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
80680 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5E)-5-((4-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one 6927 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
18472 D2 BRAIN pigeon 3H-8-OH-DPAT (S)-UH-301 7080 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85800 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-1 542 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
89640 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BUSPIRONE 5.01187 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95272 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT DPAT 2.3 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101160 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-(4-phenyl-1-piperazinyl)-1-propanone 1074 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50728 BZP HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
297 5-HT1A CORTEX PIG 3H-8-OH-DPAT ICS 205-930 >10000 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
553 5-HT1A CORTEX RAT 3H-8-OH-DPAT SUMATRIPTAN 100 McCARTHY & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
67881 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 147 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68393 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piperidine 0.288403 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3369 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NOMIFENSINE 1183 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11305 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 1500 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12329 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT MDL 73005 EF 1.25 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
82729 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
18473 D2 BRAIN pigeon 3H-8-OH-DPAT WAY 100,635 78 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85801 5-HT2A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-1 630 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
87081 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 53.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 152 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89641 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.51356 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90921 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 24.5471 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
101161 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 101 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
101417 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 172 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
50729 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
298 5-HT1A CORTEX PIG 3H-8-OH-DPAT ICS 205-930 >10000 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
554 5-HT1A CORTEX PIG 3H-8-OH-DPAT SUMATRIPTAN 741 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
68394 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) piperid-1-yl] 6-nitroindan-1-01 0.74131 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3370 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NOREPINEPHRINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11306 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PIPAMPERONE 2770 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12330 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT BMY 7378 1.99 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18474 D2 BRAIN pigeon 3H-8-OH-DPAT WAY 100,135 245 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
50730 AMPA HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
555 5-HT1A CORTEX RAT 3H-8-OH-DPAT SUMATRIPTAN 741 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
68395 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S 15535 0.794328 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3371 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PHENTOLAMINE 2151 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11307 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUSPIRILENE 56 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12331 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT NAN-190 0.7 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18475 D2 BRAIN pigeon 3H-8-OH-DPAT DU125530 5.2 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85803 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-2 2145 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
25643 5-HT1A CLONED HUMAN 3H-8-OH-DPAT COCAINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33323 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piroxicam >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
50731 NET HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
556 5-HT1A CELLS C0S-7 3H-8-OH-DPAT TFMPP 32.1 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3372 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PIMOZIDE 650 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11308 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 140 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12332 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT ALPRENOLOL,(-) 19.95 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
80428 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-4-((1H-indol-3-yl)methylene)-2-amino-1-methyl-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
83500 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
18476 BRAIN pigeon 3H-8-OH-DPAT NAN-190 0.7 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87084 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 31.8 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
31276 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDL 100907 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33068 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT NOMIFENSINE >10000 Andersen PH, et al., 1989 Jan 15, 2025 Jan 15, 2025
101164 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone 142 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50732 NK1 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
557 5-HT1A CORTEX RAT 3H-8-OH-DPAT TFMPP 75 SCHLEGEL & PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
3373 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PPP, S(-)-3 4174 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11309 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ZOTEPINE 330 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12333 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT TERTATOLOL(-) 8.31 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18477 BRAIN pigeon 3H-8-OH-DPAT PINDOLOL,(+/-) 7585 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
90925 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 43.6516 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
101165 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone 302 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50733 NK2 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
558 5-HT1A CORTEX RAT 3H-8-OH-DPAT TFMPP 130 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
67886 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 111 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3374 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PROPRANOLOL 272 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11310 5-HT1A CLONED HUMAN 3H-8-OH-DPAT OLANZAPINE 2720 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12334 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT WAY 100,135 32.35 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18478 BRAIN pigeon 3H-8-OH-DPAT S 15535 144 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85806 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-3 158 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
89646 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 389.045 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
101422 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 373 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
50734 NK3 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
559 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT TFMPP 148.15 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
3375 5-HT1A CLONED HUMAN 3H-8-OH-DPAT QUINPIROLE 1713 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11311 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Quetiapine 320 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12335 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 114.81 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18479 BRAIN pigeon 3H-8-OH-DPAT (S)-UH-301 3630 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87087 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 12 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89647 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 0.524807 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
28207 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Norfenfluramine (+) 1950 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
50735 Sigma 1 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 59.1 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
560 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT TFMPP 173 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
3376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT QUIPAZINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
72496 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(5-fluoro-4-(1-(3-fluorophenyl)ethoxy)pyrimidin-2-yl)-1,4-diazepane 578 Kim J et al 2019 Jan 15, 2025 Jan 15, 2025
11312 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ORG-5222 10 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12336 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SDZ 216,525 1.58 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
18480 BRAIN pigeon 3H-8-OH-DPAT WAY 100,635 120 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
89392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 163 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
101168 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone 15.2 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50736 V1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
561 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT TFMPP 175 GLENNON ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RESERPINE 1832 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
72497 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(5-fluoro-4-(1-(4-fluorophenyl)ethoxy)pyrimidin-2-yl)-1,4-diazepane 1066 Kim J et al 2019 Jan 15, 2025 Jan 15, 2025
11313 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SERTINDOLE 280 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
18481 BRAIN pigeon 3H-8-OH-DPAT WAY 100,135 790 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85809 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-4 204 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
90929 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 60.256 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
101169 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(4-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50737 V2 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
3378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RITANSERIN 2919 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
72498 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 5-fluoro-4-[(4-fluorophenyl)methoxy]-2-[(2R)-2methylpiperazin-1-yl]pyrimidine 271 Kim J et al 2019 Jan 15, 2025 Jan 15, 2025
11314 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ziprasidone 12 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
18482 BRAIN pigeon 3H-8-OH-DPAT DU125530 6.4 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87090 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 7-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 25.3 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89650 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 35.4813 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
50738 V1B HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
563 5-HT1A BRAIN RAT 3H-8-OH-DPAT TFMPP 230 ARNT & HYTTEL,1989 Jan 15, 2025 Jan 15, 2025
67891 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 120 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SCH 23390,R(+) 661 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
81203 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
18483 5-HT1A BRAIN pigeon 3H-8-OH-DPAT DU125530 0.7 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
89395 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 105 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89651 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 208.93 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
101427 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one 19 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
49715 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Pramipexole 6514 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
50739 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
3380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
80692 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5E)-5-((5-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one 2513 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82228 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one 1.5 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
18484 5-HT1B BRAIN pigeon 3H-8-OH-DPAT DU125530 890 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
20276 5-HT1A CORTEX RAT 3H-8-OH-DPAT HMA >10000 Garritsen A et al., 1991 Jan 15, 2025 Jan 15, 2025
85812 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-5 1246 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
101172 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(2-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50740 CB1 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
309 5-HT1A CORTEX RAT 3H-8-OH-DPAT ICYANOPINDOLOL 2.33 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
565 5-HT1A CORTEX PIG 3H-8-OH-DPAT TFMPP 288 SCHOEFFTER & HOYER, 1989 Jan 15, 2025 Jan 15, 2025
3381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SKF 38393 3096 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78645 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
18485 5-HT1D BRAIN pigeon 3H-8-OH-DPAT DU125530 1200 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87093 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 19.1 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
25141 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 427 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90933 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 144.544 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
26165 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Pseudonorephedrine, (-) [cathine, (-)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
101173 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(4-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50741 CB2 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
310 5-HT1A CORTEX PIG 3H-8-OH-DPAT ICYANOPINDOLOL 5.39 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
566 5-HT1A CORTEX PIG 3H-8-OH-DPAT TFMPP 288 SCHOEFFTER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SKF 77434 2107 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18486 5-HT2A BRAIN pigeon 3H-8-OH-DPAT DU125530 240 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
50742 D1 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
311 5-HT1A CORTEX RAT 3H-8-OH-DPAT IDAZOXAN 145.29 FOZARD ET AL., 1987 Jan 15, 2025 Jan 15, 2025
567 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT TFMPP 326.94 COSSERY ET AL.,1986 Jan 15, 2025 Jan 15, 2025
3383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SKF 81297 5516 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18487 5-HT2C BRAIN pigeon 3H-8-OH-DPAT DU125530 750 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85815 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-7 479 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
27703 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Fenfluramine 673 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33079 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT IMIPRAMINE >10000 Andersen PH, et al., 1989 Jan 15, 2025 Jan 15, 2025
50743 D2 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
312 5-HT1A CORTEX RAT 3H-8-OH-DPAT IDAZOXAN 162.89 KWONG ET AL., 1986 Jan 15, 2025 Jan 15, 2025
67896 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 25 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3384 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SPIPERONE 61 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
80440 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-2-amino-4-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one 3445 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82488 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-1-(Indolin-1-yl)-2-(2-((pyridin-3-yloxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
18488 5-HT3 BRAIN pigeon 3H-8-OH-DPAT DU125530 1100 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87096 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
88632 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 317 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
89656 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 199.526 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
101176 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(2-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50744 D3 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
3385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SULPIRIDE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
83513 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
18489 5-HT1A BRAIN pigeon 3H-8-OH-DPAT WAY 100,135 10 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
89657 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 3.80189 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90937 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-N-phenyl-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide 33.1131 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
101177 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(2-Pyridyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50745 KA HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
570 5-HT1A CELLS C0S-7 3H-8-OH-DPAT TFMPP 737 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3386 5-HT1A CLONED HUMAN 3H-8-OH-DPAT TRANYLCYPROMINE 5963 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78394 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
18490 5-HT1A BRAIN pigeon 3H-8-OH-DPAT WAY 100,635 0.5 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85818 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-8 1241 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
89402 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 126 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
50746 D4 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 21.8 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
315 5-HT1A CORTEX RAT 3H-8-OH-DPAT IMILOXAN 5538.14 KWONG ET AL., 1986 Jan 15, 2025 Jan 15, 2025
3387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT YM-09151-2 15 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18491 5-HT1A BRAIN pigeon 3H-8-OH-DPAT (S)-UH-301 81 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87099 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(6-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)hexanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 168.2 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
33595 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ETORICOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
101179 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(2-Pyrimidyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50747 D5 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
316 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT IMIPRAMINE >10000 GOZLAN ET AL., 1983 Jan 15, 2025 Jan 15, 2025
3388 5-HT1A CLONED HUMAN 3H-8-OH-DPAT YOHIMBINE 642 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18492 5-HT1A BRAIN pigeon 3H-8-OH-DPAT S 15535 1.9 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
26428 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Isoquercitrin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
101180 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(Phenylmethyl)-1-(4-phenyl-1-piperazinyl)propan-1-one 938 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
50748 SLC6A3 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
317 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT IMIPRAMINE >10000 SCHOEMAKER AND LANGER., 1986 Jan 15, 2025 Jan 15, 2025
67901 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 37 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3389 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ZIMELIDINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
82749 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
18493 5-HT1A BRAIN pigeon 3H-8-OH-DPAT NAN-190 1.3 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
85821 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-10 2326 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
89405 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 86 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
90941 5-HT1A HeLa HUMAN 3H-8-OH-DPAT N-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide 79.4328 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
50749 DOR HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
3390 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BUTACLAMOL,(+) 528 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78142 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
18494 5-HT1A BRAIN pigeon 3H-8-OH-DPAT PINDOLOL,(+/-) 47 Mos J et al., 1997 Jan 15, 2025 Jan 15, 2025
87102 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(6-Fuorobenzo[d]isoxazol-3-yl)- piperidin-1-yl) propyl)-5,6-dihydro-1H-pyrrolo [3,2,1-ij]quinolin4(2H)-one 38.7 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89662 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 13.8038 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
50750 HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP >10000 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
64574 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SSR181507 4.5 Claustre Y, et.al., 2003 Jan 15, 2025 Jan 15, 2025