The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 7,001-8,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
22739D1CLONEDHUMAN3H-SCH23390L-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
33491D5CLONEDHUMAN3H-SCH23390Meloxicam sodium>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41683D5CLONEDHUMAN3H-SCH23390ORG-522222.7PDSP Certified DataJan 15, 2025Jan 15, 2025
42451D1CLONEDHUMAN3H-SCH233903-methoxy-dibenz[d,g]azecine28.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46547D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
71892D1testtest3H-SCH2339010-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
78036D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79316D5CLONEDHUMAN3H-SCH233904-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
82644D1CLONEDHUMAN3H-SCH23390(S)-1-(Indolin-1-yl)-2-(2-((3-methoxyphenoxy)methyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
83668D1HEK293 cellsHUMAN3H-SCH23390Methamphetamine>10000Simmler LD et al 2013Jan 15, 2025Jan 28, 2025
84180D1CLONEDHUMAN3H-SCH23390(±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2465PDSP Certified DataJan 15, 2025Jan 28, 2025
22740D1CLONEDHUMAN3H-SCH23390D-methionine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
39636D1STRIATUMRAT3H-SCH23390SCH 391663.6Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
46548D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid1824Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70357D1CLONEDHUMAN3H-SCH23390N-Octyl-3-(3-hydroxyphenyl)pyrrolidine170Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
70613D1CLONEDHUMAN3H-SCH23390MRP3172>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
71381D5CLONEDHUMAN3H-SCH233905-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
78037D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79317D5CLONEDHUMAN3H-SCH23390DMT>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
81109D1CLONEDHUMAN3H-SCH23390N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
82645D5CLONEDHUMAN3H-SCH23390(S)-1-(Indolin-1-yl)-2-(2-((3-methoxyphenoxy)methyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
22741D1CLONEDHUMAN3H-SCH23390L-methionine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
25301D5CLONEDHUMAN3H-SCH23390Ziprasidone152PDSP Certified DataJan 15, 2025Jan 15, 2025
26837D1BRAINHUMAN3H-SCH23390mCPP7000Hamik A, et. al., 1989Jan 15, 2025Jan 15, 2025
28117D5CLONEDHUMAN3H-SCH23390Fenfluramine (-)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
39637D1STRIATUMRAT3H-SCH23390SCH 233900.4Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
46549D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70358D5CLONEDHUMAN3H-SCH23390N-Octyl-3-(3-hydroxyphenyl)pyrrolidine286Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
70614D5CLONEDHUMAN3H-SCH23390MRP3172>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
71894D5testtest3H-SCH2339010-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
79318D5CLONEDHUMAN3H-SCH233904-Hydroxy-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
81110D5CLONEDHUMAN3H-SCH23390N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
25558D1CLONEDHUMAN3H-SCH23390pdspTestCompound3628PDSP Certified DataJan 15, 2025Jan 15, 2025
25814D5CLONEDHUMAN3H-SCH23390Pseudoephedrine, (-)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
39638D1STRIATUMRAT3H-SCH23390HALOPERIDOL781Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
42454D1CLONEDHUMAN3H-SCH233904-chloro-3-hydroxy-dibenz[d,g]azecine0.83Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46550D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
74967D1CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
79319D5CLONEDHUMAN3H-SCH23390DMT,5-MeO>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
46551D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
74968D5CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77784D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79320D5CLONEDHUMAN3H-SCH23390N,N-Diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
24792D5CLONEDHUMAN3H-SCH23390CHLORPROMAZINE133PDSP Certified DataJan 15, 2025Jan 15, 2025
46552D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
58072D1CLONEDHUMAN3H-SCH23390Memantine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
71897D5testtest3H-SCH233906-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
77785D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79321D5CLONEDHUMAN3H-SCH233905-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
42457D5CLONEDHUMAN3H-SCH233904-chloro-3-hydroxy-dibenz[d,g]azecine0.057Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46553D5CLONEDHUMAN3H-SCH23390(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
71898D1testtest3H-SCH233906-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
75994D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
79322D5CLONEDHUMAN3H-SCH23390N,N-Dipropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
42458D1CLONEDHUMAN3H-SCH233902,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine3.2Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46554D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
59866D1CLONEDHUMAN3H-SCH233904-(2-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
71899D5testtest3H-SCH233906-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
75995D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
79323D5CLONEDHUMAN3H-SCH233904-Ethylthio-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
84187D1CLONEDHUMAN3H-SCH23390(±)-4-bromo-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide3135PDSP Certified DataJan 15, 2025Jan 28, 2025
38875D1CLONEDHUMAN3H-SCH23390MDL 11,939327.2Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
46555D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
71900D1testtest3H-SCH23390N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
77532D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79324D5CLONEDHUMAN3H-SCH233906-Fluoro-N,N-dimethyltryptamine6291Ray TS 2010 Jan 15, 2025Jan 28, 2025
84188D5CLONEDHUMAN3H-SCH23390(±)-4-bromo-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide8550PDSP Certified DataJan 15, 2025Jan 28, 2025
25820D1CLONEDHUMAN3H-SCH23390Pseudoephedrine, (-)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
28380D1CLONEDHUMAN3H-SCH23390ERGOTAMINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
33756D1CLONEDHUMAN3H-SCH23390N-(4-Acetamidophenyl)indomethacinamide>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
38876D1CLONEDHUMAN3H-SCH23390SR 46349B>10000Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
42460D1CLONEDHUMAN3H-SCH233902-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine9.3Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46556D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
58076D5CLONEDHUMAN3H-SCH23390Memantine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
70365D1CLONEDHUMAN3H-SCH23390N-Nonyl-3-(3-Hydroxyphenyl)Pyrrolidine174Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71901D2testtest3H-SCH23390N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
77533D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79325D5CLONEDHUMAN3H-SCH23390LISURIDE77Ray TS 2010 Jan 15, 2025Jan 28, 2025
38877D1CLONEDHUMAN3H-SCH23390MDL 1009072964Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
46557D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70366D5CLONEDHUMAN3H-SCH23390N-Nonyl-3-(3-Hydroxyphenyl)Pyrrolidine101Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71902D5testtest3H-SCH23390N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
79326D5CLONEDHUMAN3H-SCH23390(±)-2,5-Dimethoxy-4-iodoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
94942D1CLONEDHUMAN3H-SCH233904-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid520Jung et al 2021Jan 15, 2025Jan 28, 2025
42462D5CLONEDHUMAN3H-SCH233902-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine226.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46558D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
59870D5CLONEDHUMAN3H-SCH233904-(2-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
79327D5CLONEDHUMAN3H-SCH233901-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16095D5CLONEDHUMAN3H-SCH23390SKF-82526, (+)15Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82143D1CLONEDHUMAN3H-SCH233906-methoxy-2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)isoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
94943D1CLONEDHUMAN3H-SCH233904-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
33759D5CLONEDHUMAN3H-SCH23390N-(4-Acetamidophenyl)indomethacinamide>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
38367D1BRAINRAT3H-SCH23390MCL-2040.11Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42463D1CLONEDHUMAN3H-SCH233902-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine8.9Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46559D5CLONEDHUMAN3H-SCH23390(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
69344D1CLONEDHUMAN3H-SCH23390HALOPERIDOL83Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
71904D1testtest3H-SCH23390N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
77280D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79328D5CLONEDHUMAN3H-SCH23390(±)-2,5-Dimethoxy-4-methylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16096D5CLONEDHUMAN3H-SCH23390SKF 38393100Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82144D5CLONEDHUMAN3H-SCH233906-methoxy-2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)isoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
94944D1CLONEDHUMAN3H-SCH233904′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38368D1BRAINRAT3H-SCH23390SCH 233900.12Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46560D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
69345D1CLONEDHUMAN3H-SCH23390FLUPHENAZINE24Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
70369D1CLONEDHUMAN3H-SCH23390N-Decyl-3-(3-hydroxyphenyl)pyrrolidine128Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
72673D1CLONEDHUMAN3H-SCH233902,3-dihydrohinokiflavone>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
77281D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79329D5CLONEDHUMAN3H-SCH23390(±)-3,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16097D5CLONEDHUMAN3H-SCH23390Ergocryptine, beta113Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
87521D1CLONEDHUMAN3H-SCH233901,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
94945D1CLONEDHUMAN3H-SCH233905-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31713D1STRIATUMRAT3H-SCH23390OLANZAPINE31Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
38369D1BRAINRAT3H-SCH23390MCL-2030.19Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46561D5CLONEDHUMAN3H-SCH23390(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
69346D1CLONEDHUMAN3H-SCH23390CHLORPROMAZINE112Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
70370D5CLONEDHUMAN3H-SCH23390N-Decyl-3-(3-hydroxyphenyl)pyrrolidine143Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71906D5testtest3H-SCH23390N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
72674D5CLONEDHUMAN3H-SCH233902,3-dihydrohinokiflavone>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
79330D5CLONEDHUMAN3H-SCH23390(±)-2,5-Dimethoxy-4-ethylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16098D5CLONEDHUMAN3H-SCH23390APOMORPHINE363Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
83682D1HEK293 cellsHUMAN3H-SCH23390pyrovalerone>10000Simmler LD et al 2013Jan 15, 2025Jan 28, 2025
87522D5CLONEDHUMAN3H-SCH233901,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
94946D1CLONEDHUMAN3H-SCH233904′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31714D1STRIATUMRAT3H-SCH23390CLOZAPINE85Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
38370D1BRAINRAT3H-SCH23390MCL-2070.46Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42466D5CLONEDHUMAN3H-SCH233902-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine42.3Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46562D5CLONEDHUMAN3H-SCH23390N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
69347D1CLONEDHUMAN3H-SCH23390RACLOPRIDE>10000Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
71907D5testtest3H-SCH233902-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-1-ol>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
79331D5CLONEDHUMAN3H-SCH23390(±)-2,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16099D5CLONEDHUMAN3H-SCH23390BROMOCRIPTINE454Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82403D1CLONEDHUMAN3H-SCH23390(R)-1-(Indolin-1-yl)-2-(2-(((4-methylpyridin-2-yl)oxy)methyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
26083D1CLONEDHUMAN3H-SCH23390Methcathinone, (-)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
28387D5CLONEDHUMAN3H-SCH23390ERGOTAMINE170PDSP Certified DataJan 15, 2025Jan 15, 2025
94947D1CLONEDHUMAN3H-SCH233904′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31715D1STRIATUMRAT3H-SCH23390REMOXIPRIDE>10000Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
38371D1BRAINRAT3H-SCH23390MCL-2020.49Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
38883D5CLONEDHUMAN3H-SCH23390MDL 11,9392869Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
42467D1CLONEDHUMAN3H-SCH233902-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine82Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46563D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47331D1CLONEDHUMAN3H-SCH23390WAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
69348D1CLONEDHUMAN3H-SCH23390RISPERIDONE267Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
71908D5testtest3H-SCH233901,2-dimethoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
72420D1CLONEDHUMAN3H-SCH233905,6-methylenedioxy-2-aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 28, 2025
72932D1CLONEDHUMAN3H-SCH23390vicenin-2>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
75748D1CLONEDHUMAN3H-SCH233903-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77028D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79332D5CLONEDHUMAN3H-SCH23390LYSERGIC ACID344.4Ray TS 2010 Jan 15, 2025Jan 28, 2025
16100D5CLONEDHUMAN3H-SCH23390SKF-76783530Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82404D5CLONEDHUMAN3H-SCH23390(R)-1-(Indolin-1-yl)-2-(2-(((4-methylpyridin-2-yl)oxy)methyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
25060D5CLONEDHUMAN3H-SCH23390OLANZAPINE90PDSP Certified DataJan 15, 2025Jan 15, 2025
94948D1CLONEDHUMAN3H-SCH233904′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31716D1STRIATUMRAT3H-SCH23390Quetiapine455Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
38372D1BRAINRAT3H-SCH23390MCL-2100.52Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
38884D5CLONEDHUMAN3H-SCH23390MDL 100907>10000Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
46564D5CLONEDHUMAN3H-SCH23390PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
69349D1CLONEDHUMAN3H-SCH23390CLOZAPINE189Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
72933D5CLONEDHUMAN3H-SCH23390vicenin-2>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
75749D5CLONEDHUMAN3H-SCH233903-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77029D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79333D5CLONEDHUMAN3H-SCH23390cis-2a1013Ray TS 2010 Jan 15, 2025Jan 28, 2025
16101D5CLONEDHUMAN3H-SCH23390SKF-82526, (-)800Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
86245D1CLONEDHUMAN3H-SCH23390JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
94949D1CLONEDHUMAN3H-SCH233904′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31717D1STRIATUMRAT3H-SCH23390ORG-52225Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
38373D1BRAINRAT3H-SCH23390MCL-2090.6Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46565D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
69350D1CLONEDHUMAN3H-SCH23390OLANZAPINE58Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
71910D1testtest3H-SCH233901-(cyclopropylmethoxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
74726D1CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
79334D5CLONEDHUMAN3H-SCH23390R,R-2b591.9Ray TS 2010 Jan 15, 2025Jan 28, 2025
16102D5CLONEDHUMAN3H-SCH23390ADTN, (+)909Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
86246D5CLONEDHUMAN3H-SCH23390JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
24806D1CLONEDHUMAN3H-SCH23390CHLORPROMAZINE112PDSP Certified DataJan 15, 2025Jan 15, 2025
94950D1CLONEDHUMAN3H-SCH233904′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31718D1STRIATUMRAT3H-SCH23390HALOPERIDOL25Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
38374D1BRAINRAT3H-SCH23390MCL-2141.1Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42470D1CLONEDHUMAN3H-SCH233901,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine25.3Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46566D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
59110D1CLONEDHUMAN3H-SCH23390Beta-LT>10000Buhler A, et al., 2007Jan 15, 2025Jan 15, 2025
69351D1CLONEDHUMAN3H-SCH23390Quetiapine712Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
74727D5CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
79335D5CLONEDHUMAN3H-SCH23390S,S-2c402.2Ray TS 2010 Jan 15, 2025Jan 28, 2025
16103D5CLONEDHUMAN3H-SCH23390PERGOLIDE918Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
84199D5CLONEDHUMAN3H-SCH23390(±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide6789PDSP Certified DataJan 15, 2025Jan 28, 2025
94951D1CLONEDHUMAN3H-SCH233904′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38375D1BRAINRAT3H-SCH23390SKF-839591.18Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46567D5CLONEDHUMAN3H-SCH23390(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47335D5CLONEDHUMAN3H-SCH23390WAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
72424D5CLONEDHUMAN3H-SCH233905,6-methylenedioxy-2-aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 28, 2025
76776D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79336D5CLONEDHUMAN3H-SCH233905-MeO-TMT>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16104D5CLONEDHUMAN3H-SCH23390N-0437986Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82664D1CLONEDHUMAN3H-SCH23390(R)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
84200D1CLONEDHUMAN3H-SCH23390(±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2703PDSP Certified DataJan 15, 2025Jan 28, 2025
25320D1CLONEDHUMAN3H-SCH23390Ziprasidone30PDSP Certified DataJan 15, 2025Jan 15, 2025
94952D1CLONEDHUMAN3H-SCH233904-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38376D1BRAINRAT3H-SCH23390MCL-2161.81Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46568D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70377D1CLONEDHUMAN3H-SCH23390(-)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine181Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
73193D1testtest3H-SCH233903-(piperazin-1-yl)-N-(m-tolyl)propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
76777D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
79337D5CLONEDHUMAN3H-SCH23390EMDT>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16105D5CLONEDHUMAN3H-SCH23390NPA1136Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82665D5CLONEDHUMAN3H-SCH23390(R)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
25065D1CLONEDHUMAN3H-SCH23390OLANZAPINE58PDSP Certified DataJan 15, 2025Jan 15, 2025
94953D1CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38377D1BRAINRAT3H-SCH23390SKF 812971.9Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42473D1CLONEDHUMAN3H-SCH233901-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine0.46Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46569D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70378D5CLONEDHUMAN3H-SCH23390(-)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine227Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71914D1testtest3H-SCH233901-(allyloxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
73194D5testtest3H-SCH233903-(piperazin-1-yl)-N-(m-tolyl)propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
74474D1CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
79338D5CLONEDHUMAN3H-SCH23390Salvinorin A>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
16106D5CLONEDHUMAN3H-SCH233905-Hydroxy Tryptamine3000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
94954D1CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
33258D1CLONEDHUMAN3H-SCH23390nimesulide>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
38378D1BRAINRAT3H-SCH23390MCL-2061.93Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46570D5CLONEDHUMAN3H-SCH23390(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
73451D1testtest3H-SCH23390N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
74475D5CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75499D1CLONEDHUMAN3H-SCH23390propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
16107D5CLONEDHUMAN3H-SCH23390NOREPINEPHRINE>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
94955D5CLONEDHUMAN3H-SCH233904-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid1440Jung et al 2021Jan 15, 2025Jan 28, 2025
38379D1BRAINRAT3H-SCH23390(R)(+)-BrAPB2.29Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46571D5CLONEDHUMAN3H-SCH23390PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
59627D1CLONEDHUMAN3H-SCH23390RU 24213>10000O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
66028D1CLONEDHUMAN3H-SCH23390Ondansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
71916D5testtest3H-SCH233901-(allyloxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
75500D5CLONEDHUMAN3H-SCH23390propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
16108D5CLONEDHUMAN3H-SCH23390LY-171555>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
94956D5CLONEDHUMAN3H-SCH233904-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38380D1BRAINRAT3H-SCH23390MCL-2054.41Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42476D5CLONEDHUMAN3H-SCH233901-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine0.98Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46572D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70381D1CLONEDHUMAN3H-SCH23390(+)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine>10000Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
76525D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
11501D1STRIATUMRAT3H-SCH23390Pifluthixol0.63Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
16109D5CLONEDHUMAN3H-SCH23390SCH 233900.3Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
21741D1STRIATUMRAT3H-SCH23390Amisulpride>10000Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
94957D5CLONEDHUMAN3H-SCH233904′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38381D1BRAINRAT3H-SCH23390SKF 829584.56Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42477D1CLONEDHUMAN3H-SCH233903-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine3.1Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
46573D5CLONEDHUMAN3H-SCH23390PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
70382D5CLONEDHUMAN3H-SCH23390(+)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine639Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71918D5testtest3H-SCH233902-methoxy-6-methyl-10-nitro-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
76526D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
16110D5CLONEDHUMAN3H-SCH23390SKF 835660.4Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
21742D1STRIATUMRAT3H-SCH23390HALOPERIDOL250Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
94958D5CLONEDHUMAN3H-SCH233905-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
33262D5CLONEDHUMAN3H-SCH23390nimesulide>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
38382D1BRAINRAT3H-SCH23390MCL-2118.66Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
46574D5CLONEDHUMAN3H-SCH23390PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
73455D5testtest3H-SCH23390N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
16111D5CLONEDHUMAN3H-SCH23390FLUPENTHIXOL, Alpha8Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
21743D1STRIATUMRAT3H-SCH23390CLOZAPINE590Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
94959D5CLONEDHUMAN3H-SCH233904′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38383D1BRAINRAT3H-SCH23390SKF 7743410.5Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
59631D5CLONEDHUMAN3H-SCH23390RU 24213>10000O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
59887D1CLONEDHUMAN3H-SCH233904-(4-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
66032D5CLONEDHUMAN3H-SCH23390Ondansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
71920D5testtest3H-SCH233901,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
12528D1Choroid PlexusCANINE3H-SCH233905-Hydroxy Tryptamine>10000NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
16112D5CLONEDHUMAN3H-SCH23390BUTACLAMOL,(+)27Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
83696D1HEK293 cellsHUMAN3H-SCH23390MDPV>10000Simmler LD et al 2013Jan 15, 2025Jan 28, 2025
94960D5CLONEDHUMAN3H-SCH233904′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38384D1BRAINRAT3H-SCH23390MCL-21219.3Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42480D5CLONEDHUMAN3H-SCH233903-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine4.9Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
12529D1Choroid PlexusCANINE3H-SCH23390MIANSERIN161NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
78833D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
16113D5CLONEDHUMAN3H-SCH23390SCH 2338835Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
94961D5CLONEDHUMAN3H-SCH233904′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38385D1BRAINRAT3H-SCH23390MCL-20121.3Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42481D1CLONEDHUMAN3H-SCH233901-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine8.7Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
67314D1CLONEDHUMAN3H-SCH233901-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
71410D1CLONEDHUMAN3H-SCH233904-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71922D5testtest3H-SCH233901-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
12530D1Choroid PlexusCANINE3H-SCH23390KETANSERIN166NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
78834D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
16114D5CLONEDHUMAN3H-SCH23390HALOPERIDOL48Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
94962D5CLONEDHUMAN3H-SCH233904′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38386D1BRAINRAT3H-SCH23390SKF 3839326.6Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
73715D1testtest3H-SCH23390[2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
12531D1Choroid PlexusCANINE3H-SCH23390DOPAMINE>10000NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
16115D5CLONEDHUMAN3H-SCH23390CHLORPROMAZINE133Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82163D1CLONEDHUMAN3H-SCH233905-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one2734Besnard J et al 2012Jan 15, 2025Jan 28, 2025
84211D1CLONEDHUMAN3H-SCH23390(±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2100PDSP Certified DataJan 15, 2025Jan 28, 2025
90099D1CLONEDHUMAN3H-SCH233904-Bromo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
25331D5CLONEDHUMAN3H-SCH23390ZOTEPINE248PDSP Certified DataJan 15, 2025Jan 15, 2025
94963D5CLONEDHUMAN3H-SCH233904′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
31731D1STRIATUMRAT3H-SCH23390RISPERIDONE75Bymaster F.P., et. al., 1996Jan 15, 2025Jan 15, 2025
98803D1CLONEDHUMAN3H-SCH233901-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
38387D1BRAINRAT3H-SCH23390MCL-21537.1Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
59635D1CLONEDHUMAN3H-SCH23390SK&F 838223.2O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
59891D5CLONEDHUMAN3H-SCH233904-(4-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
71156D1CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE1960Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71924D5testtest3H-SCH233901-(allyloxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
73972D1testtest3H-SCH233901-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
12532D1Choroid PlexusCANINE3H-SCH23390FLUPENTHIXOL, Alpha30NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
16116D5CLONEDHUMAN3H-SCH23390CLOZAPINE250Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82164D5CLONEDHUMAN3H-SCH233905-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
84212D5CLONEDHUMAN3H-SCH23390(±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide7178PDSP Certified DataJan 15, 2025Jan 28, 2025
90100D1CLONEDHUMAN3H-SCH233902-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
25332D1CLONEDHUMAN3H-SCH23390ZOTEPINE71PDSP Certified DataJan 15, 2025Jan 15, 2025
94964D5CLONEDHUMAN3H-SCH233904′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
98804D5CLONEDHUMAN3H-SCH233901-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine3016Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
38388D1BRAINRAT3H-SCH23390MCL-213128Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42484D1CLONEDHUMAN3H-SCH233904-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine7.6Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
67317D5CLONEDHUMAN3H-SCH233901-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
70389D1CLONEDHUMAN3H-SCH23390(Rac)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide831Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71157D1CLONEDHUMAN3H-SCH23390HALOPERIDOL120Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71925D5testtest3H-SCH233902-methoxy-6-methyl-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
73973D5testtest3H-SCH233901-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
12533D1Choroid PlexusCANINE3H-SCH23390BUTACLAMOL,(+)3.7NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
78581D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
16117D5CLONEDHUMAN3H-SCH23390THIORIDAZINE300Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
85237D1recombinantHUMAN3H-SCH23390Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
90101D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
94965D5CLONEDHUMAN3H-SCH233904-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
38389D1BRAINRAT3H-SCH23390MCL-2181238Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
70390D5CLONEDHUMAN3H-SCH23390(Rac)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide312Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
70902D1testtest3H-SCH233906-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione5.7Martini ML et al 2019Jan 15, 2025Jan 28, 2025
71158D1CLONEDHUMAN3H-SCH23390CLOZAPINE290Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71414D5CLONEDHUMAN3H-SCH233904-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
75254D1CLONEDHUMAN3H-SCH23390ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
12534D1Choroid PlexusCANINE3H-SCH23390BUTACLAMOL, (-)>10000NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
78582D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
16118D5CLONEDHUMAN3H-SCH23390KETANSERIN2500Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
90102D1CLONEDHUMAN3H-SCH233901-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
94966D5CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate3010Jung et al 2021Jan 15, 2025Jan 28, 2025
34294D1STRIATUMRAT3H-SCH23390Dihydrexidine, DHX10Salmi P, et al., 2004Jan 15, 2025Jan 15, 2025
38390D1BRAINRAT3H-SCH23390MCL-230A>10000Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
70903D5testtest3H-SCH233906-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione6.7Martini ML et al 2019Jan 15, 2025Jan 28, 2025
71159D1CLONEDHUMAN3H-SCH23390SYA013163Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
73719D5testtest3H-SCH23390[2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
75255D5CLONEDHUMAN3H-SCH23390ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
16119D5CLONEDHUMAN3H-SCH23390SPIPERONE4500Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82423D1CLONEDHUMAN3H-SCH23390(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((4-methylpyridin-2-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
90103D1CLONEDHUMAN3H-SCH233902,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
94967D5CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
33527D1CLONEDHUMAN3H-SCH23390Naproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
34295D1STRIATUMRAT3H-SCH23390Dihydrexidine, DHX9.7Salmi P, et al., 2004Jan 15, 2025Jan 15, 2025
36599D1STRIATUMRAT3H-SCH23390RISPERIDONE>10000Leysen JE, et.al., 1994Jan 15, 2025Jan 15, 2025
38391D1BRAINRAT3H-SCH23390MCL-217>10000Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
42487D1CLONEDHUMAN3H-SCH233903,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine2Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
59639D5CLONEDHUMAN3H-SCH23390RU 242133.1O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
70904D1testtest3H-SCH233901-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione10Martini ML et al 2019Jan 15, 2025Jan 28, 2025
71160D1CLONEDHUMAN3H-SCH23390SYA16263238Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71928D5testtest3H-SCH23390N-(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
76280D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
16120D5CLONEDHUMAN3H-SCH23390ETICLOPRIDE>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82424D5CLONEDHUMAN3H-SCH23390(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((4-methylpyridin-2-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
90104D1CLONEDHUMAN3H-SCH233904-iodo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
34296D1STRIATUMHUMAN3H-SCH23390Dihydrexidine, DHX35.7Salmi P, et al., 2004Jan 15, 2025Jan 15, 2025
36600D1STRIATUMRAT3H-SCH233909-OH-risperidone510Leysen JE, et.al., 1994Jan 15, 2025Jan 15, 2025
3833D1CLONEDRAT3H-SCH23390LY 344864>10000PHEBUS LA, ET AL, 1997Jan 15, 2025Jan 15, 2025
70649D1CLONEDHUMAN3H-SCH23390MRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
70905D5testtest3H-SCH233901-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione15Martini ML et al 2019Jan 15, 2025Jan 28, 2025
76281D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
16121D5CLONEDHUMAN3H-SCH23390SULPIRIDE,(+)>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
90105D1CLONEDHUMAN3H-SCH233902-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
25849D1CLONEDHUMAN3H-SCH23390Pseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
26361D1CLONEDHUMAN3H-SCH23390Hyperforin595.8Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
34297D1STRIATUMRAT3H-SCH23390Dihydrexidine, DHX2.3Salmi P, et al., 2004Jan 15, 2025Jan 15, 2025
70650D5CLONEDHUMAN3H-SCH23390MRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
78330D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
81402D1CLONEDHUMAN3H-SCH23390[1-(1-phenoxypropan-2-yl)piperidin-3-yl]-pyridin-3-ylmethanone>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16122D5CLONEDHUMAN3H-SCH23390SULPIRIDE,(-)>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
85242D5recombinantHUMAN3H-SCH23390Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
90106D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-propylphenyl)ethanamine8400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
26106D5CLONEDHUMAN3H-SCH23390Methcathinone, (-)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
34298D1STRIATUMRAT3H-SCH23390Dihydrexidine, DHX4.59Salmi P, et al., 2004Jan 15, 2025Jan 15, 2025
42490D5CLONEDHUMAN3H-SCH233903,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine1.68Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
70907D1testtest3H-SCH233906-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione70Martini ML et al 2019Jan 15, 2025Jan 28, 2025
71931D5testtest3H-SCH23390N-(1-(allyloxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
78331D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
16123D1CLONEDHUMAN3H-SCH23390SKF-82526, (+)28Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
90107D1CLONEDHUMAN3H-SCH233902-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
93947D1STRIATUMPIG3H-SCH23390compound 422500Ortega R et al 2011Jan 15, 2025Jan 28, 2025
33531D5CLONEDHUMAN3H-SCH23390Naproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
34299D1STRIATUMRAT3H-SCH23390Dihydrexidine, DHX6.2Salmi P, et al., 2004Jan 15, 2025Jan 15, 2025
36603D1CLONEDHUMAN3H-SCH23390HALOPERIDOL359Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
42491D1CLONEDHUMAN3H-SCH233903,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine9.4Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
59643D1CLONEDHUMAN3H-SCH23390SK&F 839590.5O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
70396D1CLONEDHUMAN3H-SCH23390(-)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide4589Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
70908D5testtest3H-SCH233906-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione171Martini ML et al 2019Jan 15, 2025Jan 28, 2025
74236D1testtest3H-SCH23390N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
16124D1CLONEDHUMAN3H-SCH23390SKF 38393150Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
82684D1CLONEDHUMAN3H-SCH23390(S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine8366Besnard J et al 2012Jan 15, 2025Jan 28, 2025
90108D1CLONEDHUMAN3H-SCH233902,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
93948D1STRIATUMPIG3H-SCH23390compound 432900Ortega R et al 2011Jan 15, 2025Jan 28, 2025
36604D1CLONEDHUMAN3H-SCH23390CLOZAPINE539Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
70397D5CLONEDHUMAN3H-SCH23390(-)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide955Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
71933D5testtest3H-SCH23390N-(2-methoxy-6-methyl-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide>10000Karki A et al., 2020Jan 15, 2025Jan 28, 2025
74237D5testtest3H-SCH23390N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
82685D5CLONEDHUMAN3H-SCH23390(S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine8525Besnard J et al 2012Jan 15, 2025Jan 28, 2025
90109D1CLONEDHUMAN3H-SCH233902-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
93949D1STRIATUMPIG3H-SCH233903,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one2100Ortega R et al 2011Jan 15, 2025Jan 28, 2025
36605D1CLONEDHUMAN3H-SCH23390OLANZAPINE118Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
3838D1CLONEDRAT3H-SCH23390ILOPERIDONE546KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
70398D5CLONEDHUMAN3H-SCH23390(+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide>10000Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
78078D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
81150D1CLONEDHUMAN3H-SCH23390N-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
16126D1CLONEDHUMAN3H-SCH23390DOPAMINE2340Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81918D1CLONEDHUMAN3H-SCH23390(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
90110D1CLONEDHUMAN3H-SCH23390MESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
93950D1STRIATUMPIG3H-SCH233907-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one2300Ortega R et al 2011Jan 15, 2025Jan 28, 2025
36606D1CLONEDHUMAN3H-SCH23390RISPERIDONE147Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
42494D5CLONEDHUMAN3H-SCH233903,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine12.6Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
3839D1CLONEDRAT3H-SCH23390RISPERIDONE550KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
70399D1CLONEDHUMAN3H-SCH23390(+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide>10000Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
70911D1testtest3H-SCH233901,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione93Martini ML et al 2019Jan 15, 2025Jan 28, 2025
78079D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
81151D5CLONEDHUMAN3H-SCH23390N-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
16127D1CLONEDHUMAN3H-SCH23390APOMORPHINE680Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81919D5CLONEDHUMAN3H-SCH23390(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
90111D1CLONEDHUMAN3H-SCH233902-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine9300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
93951D1STRIATUMPIG3H-SCH233903,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one640Ortega R et al 2011Jan 15, 2025Jan 28, 2025
36607D1CLONEDHUMAN3H-SCH23390mirtazepine4167Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
59647D5CLONEDHUMAN3H-SCH23390SK&F 839592.1O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
2565-HT1ACORTEXRAT3H-8-OH-DPATDHE19McCARTHY & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
693765-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL1202Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
133125-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATCITALOPRAM>10000Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
808965-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
832005-HT1ACLONEDHUMAN3H-8-OH-DPATLSD2.78Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
857605-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide230Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
271365-HT1ACLONEDHUMAN3H-8-OH-DPATCP-132,4848410May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942085-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine3300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
376325-HT1AHippocampalRAT3H-8-OH-DPATN-[2-[4-(1-Naphthalenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide0.6Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2575-HT1ACORTEXHUMAN3H-8-OH-DPATDILTIAZEM>10000PEROUTKA, 1988Jan 15, 2025Jan 15, 2025
678415-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
693775-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPHENAZINE145Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
133135-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATINDALPINE9120.1Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
826895-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
857615-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
870415-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one2000Cao X et al 2018Jan 15, 2025Jan 15, 2025
893455-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide365Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
245775-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT5-Hydroxy Tryptamine1.8Borsini F, et al., 1995Jan 15, 2025Jan 15, 2025
908815-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane50.1187Franchini S et al 2014Jan 15, 2025Jan 15, 2025
271375-HT1ACLONEDHUMAN3H-8-OH-DPATCP-132,484(4b)287May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942095-HT1ACLONEDHUMAN3H-8-OH-DPAT4-benzyloxy-2,5-dimethoxyphenethylamine2700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
1013775-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one22Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
376335-HT1AHippocampalRAT3H-8-OH-DPATN-[2-[4-(4-Chloro-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide433Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2585-HT1ACORTEXHUMAN3H-8-OH-DPATDMT119.51PIERCE & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
5145-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSPIPERONE32.76HALL ET AL., 1985Jan 15, 2025Jan 15, 2025
693785-HT1ACLONEDHUMAN3H-8-OH-DPATCHLORPROMAZINE3115Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
133145-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATPAROXETINE>10000Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
245785-HT1AFR. CORTEXRAT3H-8-OH-DPAT5-Hydroxy Tryptamine4.2Borsini F, et al., 1995Jan 15, 2025Jan 15, 2025
271385-HT1ACLONEDHUMAN3H-8-OH-DPATN,N-dimethyl derivative562May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942105-HT1ACLONEDHUMAN3H-8-OH-DPAT4-allyloxy-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
376345-HT1AHippocampalRAT3H-8-OH-DPATN-[2-[4-(4-Methyl-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide58.6Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
5155-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSPIPERONE45.12COSSERY ET AL.,1986Jan 15, 2025Jan 15, 2025
693795-HT1ACLONEDHUMAN3H-8-OH-DPATRACLOPRIDE>10000Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
133155-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATFemoxetine3162.27Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
271395-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942115-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
376355-HT1AHippocampalRAT3H-8-OH-DPATN-[3-[4-(2,3-Dichlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide117Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2605-HT1AHIPPOCAMPUSBOVINE3H-8-OH-DPATDMT140.74PEROUTKA, 1985Jan 15, 2025Jan 15, 2025
5165-HT1ACORTEXPIG3H-8-OH-DPATSPIPERONE48.07HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
693805-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE427Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
806445-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
867885-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide590Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
870445-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one58.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
271405-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942125-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
376365-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide123Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2615-HT1ACORTEXRAT3H-8-OH-DPATDMT245TAYLOR ET AL,. 1987Jan 15, 2025Jan 15, 2025
5175-HT1ACORTEXRAT3H-8-OH-DPATSPIPERONE54FOZARD ET AL., 1987Jan 15, 2025Jan 15, 2025
33335-HT1ACLONEDHUMAN3H-8-OH-DPATAmphetamine,(+)6606TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
693815-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE105Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
832055-HT1ACLONEDHUMAN3H-8-OH-DPATDMT450Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
867895-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide325Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
908855-HT1AHeLaHUMAN3H-8-OH-DPAT8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane42.658Franchini S et al 2014Jan 15, 2025Jan 15, 2025
271415-HT1ACLONEDHUMAN3H-8-OH-DPATAL-37350A>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942135-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
376375-HT1AHippocampalRAT3H-8-OH-DPATN-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide78.7Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2625-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOB3770TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
678465-HT1ACLONEDHUMAN3H-8-OH-DPATS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33345-HT1ACLONEDHUMAN3H-8-OH-DPATSKF 829581781TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
693825-HT1ACLONEDHUMAN3H-8-OH-DPATOLANZAPINE2063Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
832065-HT1ACLONEDHUMAN3H-8-OH-DPATDOM>10000Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
857665-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide495Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
271425-HT1ACLONEDHUMAN3H-8-OH-DPATDOI,(-)3843May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942145-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-isopropoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
1013825-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione48Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
376385-HT1AHippocampalRAT3H-8-OH-DPATN-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-3-methoxybenzamide19.8Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
33355-HT1ACLONEDHUMAN3H-8-OH-DPATAPOMORPHINE4929TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
693835-HT1ACLONEDHUMAN3H-8-OH-DPATQuetiapine431Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
857675-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide500Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
870475-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one196.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
942155-HT1ACLONEDHUMAN3H-8-OH-DPAT2,4,5-trimethoxyamphetamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
314955-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)1584.89Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
332875-HT1ACLONEDHUMAN3H-8-OH-DPATAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
376395-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide7.5Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2645-HT1ACORTEXHUMAN3H-8-OH-DPATDOB6326.73PIERCE & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
5205-HT1ACELLSC0S-73H-8-OH-DPATSPIPERONE63RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
33365-HT1ACLONEDHUMAN3H-8-OH-DPATBROMOCRIPTINE,(+)25TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
803925-HT1ACLONEDHUMAN3H-8-OH-DPAT(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one3215Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
893525-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide3842Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
896085-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone0.47863Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
942165-HT1ACLONEDHUMAN3H-8-OH-DPAT4-Bromo-2,5-dimethoxyphenethylamine311Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
314965-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)1000Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
376405-HT1AHippocampalRAT3H-8-OH-DPATN-[5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide4.5Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
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5215-HT1ACORTEXPIG3H-8-OH-DPATSPIPERONE66.1MARKSTEIN ET AL, 1986Jan 15, 2025Jan 15, 2025
33375-HT1ACLONEDHUMAN3H-8-OH-DPATCARBAMAZEPINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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908895-HT1AHeLaHUMAN3H-8-OH-DPAT8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane20.4174Franchini S et al 2014Jan 15, 2025Jan 15, 2025
376415-HT1AHippocampalRAT3H-8-OH-DPATN-[3-[4-(4-Chlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide850Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2665-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOB,R(-)2332TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
681065-HT1AUNDEFINEDUNDEFINED3H-8-OH-DPATABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
33385-HT1ACLONEDHUMAN3H-8-OH-DPATCGS 12066B44TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
146025-HT1ACLONEDHUMAN3H-8-OH-DPATSB-277011-A5011.87Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
837225-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide9987PDSP Certified DataJan 15, 2025Jan 15, 2025
867945-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide219Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
870505-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one193.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
268905-HT1ACLONEDHUMAN3H-8-OH-DPATxanomeline63.0957Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
376425-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide397Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2675-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOB,S(+)4041TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
5235-HT1ACORTEXPIG3H-8-OH-DPATSPIPERONE66.1ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
678515-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33395-HT1ACLONEDHUMAN3H-8-OH-DPATCHLORPROMAZINE3115TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
786035-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
816755-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
832115-HT1ACLONEDHUMAN3H-8-OH-DPATKETANSERIN6510Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
867955-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide331Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
893555-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide802Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
1013875-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione35Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
376435-HT1AHippocampalRAT3H-8-OH-DPATN-[5-[4-(4-Chlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide850Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2685-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOBU4178TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
5245-HT1ACORTEXPIG3H-8-OH-DPATSPIPERONE66.1SCHLICKER ET AL., 1989Jan 15, 2025Jan 15, 2025
33405-HT1ACLONEDHUMAN3H-8-OH-DPATCLOMIPRAMINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
821885-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one62Besnard J et al 2012Jan 15, 2025Jan 15, 2025
832125-HT1ACLONEDHUMAN3H-8-OH-DPATRo 60-01756680Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
857725-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
312445-HT1ACLONEDHUMAN3H-8-OH-DPATPPP, S(-)-31730PDSP Certified DataJan 15, 2025Jan 15, 2025
376445-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dimethylphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide268Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2695-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOET3930TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
33415-HT1ACLONEDHUMAN3H-8-OH-DPATCOCAINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
857735-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
870535-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on98Cao X et al 2018Jan 15, 2025Jan 15, 2025
896135-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone2.5704Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
908935-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane36.3078Franchini S et al 2014Jan 15, 2025Jan 15, 2025
258695-HT1ACLONEDHUMAN3H-8-OH-DPATPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
274055-HT1ACLONEDHUMAN3H-8-OH-DPATAPOMORPHINE117.49Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
376455-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(1-Naphthalenyl)piperazin-1-yl]butyl]-3-methoxybenzamide0.43Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2705-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOI2355TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
33425-HT1ACLONEDHUMAN3H-8-OH-DPATCYPROHEPTADINE59TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
896145-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1.86209Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274065-HT1ACLONEDHUMAN3H-8-OH-DPATBROMOCRIPTINE12.8825Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
376465-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(1-Isoquinolyl)piperazin-1-yl]butyl]-3-methoxybenzamide12.7Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2715-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATGEPIRONE70GLENNON ET AL., 1988Jan 15, 2025Jan 15, 2025
33435-HT1ACLONEDHUMAN3H-8-OH-DPATDEPRENYL>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
274075-HT1ACLONEDHUMAN3H-8-OH-DPATCabergoline19.9526Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
376475-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(1,2-Benzisoxazol-3-yl)piperazin-1-yl]butyl]-3-methoxybenzamide7730Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
678565-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33445-HT1ACLONEDHUMAN3H-8-OH-DPATDESIPRAMINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
783525-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
806565-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
824485-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine0.6Besnard J et al 2012Jan 15, 2025Jan 15, 2025
868005-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide99.1Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
870565-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one69.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
274085-HT1ACLONEDHUMAN3H-8-OH-DPATLISURIDE0.147911Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952485-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide192.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1013925-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione482Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
376485-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-bromo-1-methoxy-2-naphthalenecarboxamide1000Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2735-HT1ACORTEXPIG3H-8-OH-DPATGEPIRONE89.1HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
33455-HT1ACLONEDHUMAN3H-8-OH-DPATDHE1.5TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
832175-HT1ACLONEDHUMAN3H-8-OH-DPATSB2420879300Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
868015-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide100Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
885935-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE140Peprah K et al 2012Jan 15, 2025Jan 15, 2025
908975-HT1AHeLaHUMAN3H-8-OH-DPAT1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one64.5654Franchini S et al 2014Jan 15, 2025Jan 15, 2025
274095-HT1ACLONEDHUMAN3H-8-OH-DPATPERGOLIDE1.90546Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952495-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide182Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
376495-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-methoxy-2-naphthalenecarboxamide575Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
5305-HT1AHIPPOCAMPUSHUMAN3H-8-OH-DPATSPIPERONE100.92HOYER ET AL., 1986Jan 15, 2025Jan 15, 2025
832185-HT1ACLONEDHUMAN3H-8-OH-DPATCyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide1.21Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
857785-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide443Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
217785-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATCLOZAPINE1700Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
893625-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide6631Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
274105-HT1ACLONEDHUMAN3H-8-OH-DPATPiribedil446.684Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
276665-HT1ACLONEDHUMAN3H-8-OH-DPATMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
952505-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide728.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
376505-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-naphthalenecarboxamide335Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2755-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATHALOPERIDOL2761.11GOZLAN ET AL., 1983Jan 15, 2025Jan 15, 2025
5315-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSPIPERONE101TITELER ET AL., 1987Jan 15, 2025Jan 15, 2025
33475-HT1ACLONEDHUMAN3H-8-OH-DPATDOPAMINE8248TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
857795-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide52.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
870595-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one82.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
217795-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATHALOPERIDOL2500Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
896195-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1.25893Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274115-HT1ACLONEDHUMAN3H-8-OH-DPATPramipexole691.831Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952515-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide82.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
376515-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-quinolinecarboxamide88.5Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
5325-HT1ACORTEXRAT3H-8-OH-DPATSPIPERONE120PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
33485-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT6.9TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
781005-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
804045-HT1ACLONEDHUMAN3H-8-OH-DPAT(E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
217805-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATAmisulpride>10000Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
896205-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone0.562341Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274125-HT1ACLONEDHUMAN3H-8-OH-DPATQuinelorane>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952525-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide212.6Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
312525-HT1ACLONEDHUMAN3H-8-OH-DPATPPP, R(+)-3868.9PDSP Certified DataJan 15, 2025Jan 15, 2025
335565-HT1ACLONEDHUMAN3H-8-OH-DPATCELECOXIB>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
376525-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-(1,1'-biphenyl)-4-carboxamide1000Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
2775-HT1ACORTEXPIG3H-8-OH-DPATHALOPERIDOL4790HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
5335-HT1ACORTEXHUMAN3H-8-OH-DPATSPIPERONE130.76HOYER ET AL., 1986Jan 15, 2025Jan 15, 2025
678615-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)146Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33495-HT1ACLONEDHUMAN3H-8-OH-DPATETICLOPRIDE,S(-)1790TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
778455-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
138455-HT1ABRAINRAT3H-8-OH-DPATCLOZAPINE150Tang AH, et al., 1996Jan 15, 2025Jan 15, 2025
827095-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
893655-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide6064Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
909015-HT1AHeLaHUMAN3H-8-OH-DPAT2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one323.594Franchini S et al 2014Jan 15, 2025Jan 15, 2025
274135-HT1ACLONEDHUMAN3H-8-OH-DPATQUINPIROLE1698.24Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952535-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide2600Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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5345-HT1ACORTEXRAT3H-8-OH-DPATSPIPERONE140SCHLEGEL & PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
33505-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPENTHIXOL, Alpha8028TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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33515-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPHENAZINE2829TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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274155-HT1ACLONEDHUMAN3H-8-OH-DPATRoxindole0.114815Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952555-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide298Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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507115-HT1AHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP0.15Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
2805-HT1ACELLSC0S-73H-8-OH-DPATHISTAMINE6011RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
5365-HT1AHIPPOCAMPUSBOVINE3H-8-OH-DPATSPIPERONE155.56PEROUTKA, 1985Jan 15, 2025Jan 15, 2025
683765-HT1ACLONEDHUMAN3H-8-OH-DPATcis 1-hydroxyindane67.6083Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33525-HT1ACLONEDHUMAN3H-8-OH-DPATGBR-129094677TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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274165-HT1ACLONEDHUMAN3H-8-OH-DPATTalipexole1698.24Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
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391925-HT2BCLONEDHUMAN3H-8-OH-DPATATC0065266Chaki S, et al., 2005Jan 15, 2025Jan 15, 2025
507125-HT1BHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP643Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
683775-HT1ACLONEDHUMAN3H-8-OH-DPATtrans 1-hydroxyindane1.62181Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
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857855-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-OH-DPAT0.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
870655-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one79.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
896255-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0616595Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
909055-HT1AHeLaHUMAN3H-8-OH-DPAT8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane52.4807Franchini S et al 2014Jan 15, 2025Jan 15, 2025
274175-HT1ACLONEDHUMAN3H-8-OH-DPATTERGURIDE3.46737Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952575-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide196.3Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
312575-HT1AC.H.O.HUMAN3H-8-OH-DPATRopinirole288.403Millan MJ, et. al., 2004Jan 15, 2025Jan 15, 2025
998655-HT1AHIPPOCAMPUSMOUSE3H-8-OH-DPAT1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride138Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
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507135-HT1DHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP88.3Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
678665-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline66Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
683785-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol23.4423Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33545-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL5084TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
171785-HT1ACLONEDHUMAN3H-8-OH-DPATMETHYLPHENIDATE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
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952585-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide199.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1014025-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione47Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
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837395-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one8590PDSP Certified DataJan 15, 2025Jan 15, 2025
952595-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide229.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
376595-HT1AHippocampalRAT3H-8-OH-DPAT8-OH-DPAT2.1Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
507155-HT2AHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP4975Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
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683805-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol6.60693Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
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775965-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
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870685-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one84.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
893725-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide2630Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
952605-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide365.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1011485-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone272Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
507165-HT2BHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP73.6Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
683815-HT1ACLONEDHUMAN3H-8-OH-DPAT(-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol1.02329Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33575-HT1ACLONEDHUMAN3H-8-OH-DPATIDAZOXAN662TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
868135-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
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909095-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane26.9153Franchini S et al 2014Jan 15, 2025Jan 15, 2025
952615-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide210.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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896305-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone0.0645654Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952625-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide218Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
998705-HT1AHIPPOCAMPUSMOUSE3H-8-OH-DPAT7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride22Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
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678715-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline91Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
683835-HT1ACLONEDHUMAN3H-8-OH-DPAT1-hydroxyindane1.62181Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33595-HT1ACLONEDHUMAN3H-8-OH-DPATKETANSERIN>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
870715-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one81.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
893755-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1836Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
896315-HT1ACLONEDHUMAN3H-8-OH-DPAT(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0147911Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952635-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide476Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1014075-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione28Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
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315205-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-1-(2-(1-(3,4-Dichloro-benzene sulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine316.228Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
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5455-HT1ACORTEXPIG3H-8-OH-DPATSPIROXATRINE8.91SCHOEFFTER AND HOYER,1988Jan 15, 2025Jan 15, 2025
683855-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-011.25893Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33615-HT1ACLONEDHUMAN3H-8-OH-DPATMDA,R(-)>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
909135-HT1AHeLaHUMAN3H-8-OH-DPAT8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane37.1535Franchini S et al 2014Jan 15, 2025Jan 15, 2025
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315215-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-1-(2-(1-(3-bromo-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine398.107Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
330575-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATBUPROPION>10000Andersen PH, et al., 1989Jan 15, 2025Jan 15, 2025
1011535-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone33.5Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
389455-HT1ACORTEXRAT3H-8-OH-DPATQUIPAZINE2000Glennon RA, et al., 1989Jan 15, 2025Jan 15, 2025
507215-HT7HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP12.9Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
683865-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-016.60693Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33625-HT1ACLONEDHUMAN3H-8-OH-DPATMDMA, R(-)>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
822105-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one20Besnard J et al 2012Jan 15, 2025Jan 15, 2025
18466D3BRAINpigeon3H-8-OH-DPATWAY 100,635370Mos J et al., 1997Jan 15, 2025Jan 15, 2025
868185-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide0.13Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
870745-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile473.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
253785-HT1ACLONEDHUMAN3H-8-OH-DPATARIPIPRAZOLE5.6PDSP Certified DataJan 15, 2025Jan 15, 2025
258905-HT1ACLONEDHUMAN3H-8-OH-DPATNorephedrine, (+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
952665-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide314.8Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
50722HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
5475-HT1ACORTEXRAT3H-8-OH-DPATSPIROXATRINE,(+)21NIKAM ET AL., 1988Jan 15, 2025Jan 15, 2025
683875-HT1ACLONEDHUMAN3H-8-OH-DPAT(-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-011.02329Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33635-HT1ACLONEDHUMAN3H-8-OH-DPATMETHAMPHETAMINE (+)>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
18467D3BRAINpigeon3H-8-OH-DPATWAY 100,135>10000Mos J et al., 1997Jan 15, 2025Jan 15, 2025
202595-HT1ACORTEXRAT3H-8-OH-DPATBenzamil1900Garritsen A et al., 1991Jan 15, 2025Jan 15, 2025
868195-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide1060Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
896355-HT1ACLONEDHUMAN3H-8-OH-DPAT(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone0.0338844Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952675-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide484.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
50723HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP6.75Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
678765-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline147Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
683885-HT1ACLONEDHUMAN3H-8-OH-DPATPiperazine1.28825Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33645-HT1ACLONEDHUMAN3H-8-OH-DPAT5-HT,2-Me3074TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
770925-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
824685-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-1-(Indolin-1-yl)-2-(2-((pyridin-3-yloxy)methyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
18468D3BRAINpigeon3H-8-OH-DPATDU12553011Mos J et al., 1997Jan 15, 2025Jan 15, 2025
202605-HT1ACORTEXRAT3H-8-OH-DPATAmiloride>10000Garritsen A et al., 1991Jan 15, 2025Jan 15, 2025
896365-HT1ACLONEDHUMAN3H-8-OH-DPATNLX-1012.18776Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952685-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide2300Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1011565-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone1684Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1014125-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione3569Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
50724Beta2HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
2935-HT1ACORTEXRAT3H-8-OH-DPATHISTAMINE>10000PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
5495-HT1ACORTEXRAT3H-8-OH-DPATSPIROXATRINE,(-)1.9NIKAM ET AL., 1988Jan 15, 2025Jan 15, 2025
683895-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-0122.9087Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33655-HT1ACLONEDHUMAN3H-8-OH-DPATMETHYLPHENIDATE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
123255-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATS 144890.61Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
18469D2BRAINpigeon3H-8-OH-DPATPINDOLOL,(+/-)>10000Mos J et al., 1997Jan 15, 2025Jan 15, 2025
870775-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one54.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
909175-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane69.1831Franchini S et al 2014Jan 15, 2025Jan 15, 2025
952695-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide62.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1011575-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone81.8Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
50725Alpha2AHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP96Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
5505-HT1ACELLSC0S-73H-8-OH-DPATSULPIRIDE589RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
683905-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-010.831764Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33665-HT1ACLONEDHUMAN3H-8-OH-DPATMETOCLOPRAMIDE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
123265-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATS 155351.77Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
18470D2BRAINpigeon3H-8-OH-DPATNAN-19014Mos J et al., 1997Jan 15, 2025Jan 15, 2025
893825-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide160Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
952705-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide30.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
50726Alpha2BHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP238Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
683915-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 4-hydroxy piperid-1-yl] 5-fluoroindan-1-011000Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33675-HT1ACLONEDHUMAN3H-8-OH-DPATMIANSERIN2592TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113035-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE420Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123275-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATS 159311.51Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
18471D2BRAINpigeon3H-8-OH-DPATS 15535132Mos J et al., 1997Jan 15, 2025Jan 15, 2025
886155-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol658Sampson D et al 2014Jan 15, 2025Jan 15, 2025
896395-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT0.812831Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952715-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT5-Hydroxy Tryptamine9.4Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
407435-HT1ACLONEDHUMAN3H-8-OH-DPATURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
50727Alpha2CHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP15.4Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
2965-HT1ACELLSC0S-73H-8-OH-DPATICS 205-9301788RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
683925-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperid-1-yl] indan-1-010.707946Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33685-HT1ACLONEDHUMAN3H-8-OH-DPATNAN-1903TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113045-HT1ACLONEDHUMAN3H-8-OH-DPAT9-OH-risperidone590Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
768405-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
123285-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATEltoprazine9.33Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
806805-HT1ACLONEDHUMAN3H-8-OH-DPAT(5E)-5-((4-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one6927Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
18472D2BRAINpigeon3H-8-OH-DPAT(S)-UH-3017080Mos J et al., 1997Jan 15, 2025Jan 15, 2025
858005-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-1542Luethi D et al 2019Jan 15, 2025Jan 15, 2025
896405-HT1ACLONEDHUMAN3H-8-OH-DPATBUSPIRONE5.01187Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952725-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATDPAT2.3Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1011605-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-(4-phenyl-1-piperazinyl)-1-propanone1074Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
50728BZPHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
2975-HT1ACORTEXPIG3H-8-OH-DPATICS 205-930>10000MARKSTEIN ET AL, 1986Jan 15, 2025Jan 15, 2025
5535-HT1ACORTEXRAT3H-8-OH-DPATSUMATRIPTAN100McCARTHY & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
678815-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole147Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
683935-HT1ACLONEDHUMAN3H-8-OH-DPATPiperidine0.288403Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33695-HT1ACLONEDHUMAN3H-8-OH-DPATNOMIFENSINE1183TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113055-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL1500Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123295-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATMDL 73005 EF1.25Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
827295-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
18473D2BRAINpigeon3H-8-OH-DPATWAY 100,63578Mos J et al., 1997Jan 15, 2025Jan 15, 2025
858015-HT2AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-1630Luethi D et al 2019Jan 15, 2025Jan 15, 2025
870815-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one53.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
893855-HT1ACLONEDHUMAN3H-8-OH-DPATN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide152Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
896415-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1.51356Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
909215-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane24.5471Franchini S et al 2014Jan 15, 2025Jan 15, 2025
1011615-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone101Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1014175-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione172Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
50729HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
2985-HT1ACORTEXPIG3H-8-OH-DPATICS 205-930>10000HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
5545-HT1ACORTEXPIG3H-8-OH-DPATSUMATRIPTAN741SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
683945-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) piperid-1-yl] 6-nitroindan-1-010.74131Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33705-HT1ACLONEDHUMAN3H-8-OH-DPATNOREPINEPHRINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113065-HT1ACLONEDHUMAN3H-8-OH-DPATPIPAMPERONE2770Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123305-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATBMY 73781.99Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
18474D2BRAINpigeon3H-8-OH-DPATWAY 100,135245Mos J et al., 1997Jan 15, 2025Jan 15, 2025
50730AMPAHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
5555-HT1ACORTEXRAT3H-8-OH-DPATSUMATRIPTAN741SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
683955-HT1ACLONEDHUMAN3H-8-OH-DPATS 155350.794328Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33715-HT1ACLONEDHUMAN3H-8-OH-DPATPHENTOLAMINE2151TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113075-HT1ACLONEDHUMAN3H-8-OH-DPATFLUSPIRILENE56Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123315-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATNAN-1900.7Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
18475D2BRAINpigeon3H-8-OH-DPATDU1255305.2Mos J et al., 1997Jan 15, 2025Jan 15, 2025
858035-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-22145Luethi D et al 2019Jan 15, 2025Jan 15, 2025
256435-HT1ACLONEDHUMAN3H-8-OH-DPATCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
333235-HT1ACLONEDHUMAN3H-8-OH-DPATPiroxicam>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
50731NETHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
5565-HT1ACELLSC0S-73H-8-OH-DPATTFMPP32.1RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
33725-HT1ACLONEDHUMAN3H-8-OH-DPATPIMOZIDE650TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113085-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE140Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123325-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATALPRENOLOL,(-)19.95Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
804285-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((1H-indol-3-yl)methylene)-2-amino-1-methyl-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
835005-HT1AHEK293 cellsHUMAN3H-8-OH-DPATMBDB>10000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
18476BRAINpigeon3H-8-OH-DPATNAN-1900.7Mos J et al., 1997Jan 15, 2025Jan 15, 2025
870845-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one31.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
312765-HT1ACLONEDHUMAN3H-8-OH-DPATMDL 100907>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
330685-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATNOMIFENSINE>10000Andersen PH, et al., 1989Jan 15, 2025Jan 15, 2025
1011645-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone142Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
50732NK1HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
5575-HT1ACORTEXRAT3H-8-OH-DPATTFMPP75SCHLEGEL & PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
33735-HT1ACLONEDHUMAN3H-8-OH-DPATPPP, S(-)-34174TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113095-HT1ACLONEDHUMAN3H-8-OH-DPATZOTEPINE330Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123335-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATTERTATOLOL(-)8.31Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
18477BRAINpigeon3H-8-OH-DPATPINDOLOL,(+/-)7585Mos J et al., 1997Jan 15, 2025Jan 15, 2025
909255-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane43.6516Franchini S et al 2014Jan 15, 2025Jan 15, 2025
1011655-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone302Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
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282075-HT1ACLONEDHUMAN3H-8-OH-DPATNorfenfluramine (+)1950PDSP Certified DataJan 15, 2025Jan 15, 2025
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870935-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one19.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
251415-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE427PDSP Certified DataJan 15, 2025Jan 15, 2025
909335-HT1AHeLaHUMAN3H-8-OH-DPAT8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane144.544Franchini S et al 2014Jan 15, 2025Jan 15, 2025
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277035-HT1ACLONEDHUMAN3H-8-OH-DPATFenfluramine673PDSP Certified DataJan 15, 2025Jan 15, 2025
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678965-HT1ACLONEDHUMAN3H-8-OH-DPATS)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole25Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33845-HT1ACLONEDHUMAN3H-8-OH-DPATSPIPERONE61TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
804405-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-2-amino-4-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one3445Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
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184935-HT1ABRAINpigeon3H-8-OH-DPATNAN-1901.3Mos J et al., 1997Jan 15, 2025Jan 15, 2025
858215-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-102326Luethi D et al 2019Jan 15, 2025Jan 15, 2025
894055-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide86Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
909415-HT1AHeLaHUMAN3H-8-OH-DPATN-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide79.4328Franchini S et al 2014Jan 15, 2025Jan 15, 2025
50749DORHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
33905-HT1ACLONEDHUMAN3H-8-OH-DPATBUTACLAMOL,(+)528TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
781425-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
184945-HT1ABRAINpigeon3H-8-OH-DPATPINDOLOL,(+/-)47Mos J et al., 1997Jan 15, 2025Jan 15, 2025
871025-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(6-Fuorobenzo[d]isoxazol-3-yl)- piperidin-1-yl) propyl)-5,6-dihydro-1H-pyrrolo [3,2,1-ij]quinolin4(2H)-one38.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
896625-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone13.8038Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
50750HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
645745-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSSR1815074.5Claustre Y, et.al., 2003Jan 15, 2025Jan 15, 2025