30087 SST3 CLONED RAT 125I-SOMATOSTATIN Somatostatin-14 1.33 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
7312 V2 CLONED RAT 3H-AVP OPC-41061 1.33 Yamamura Y, et al., 1998 Jan 15, 2025 Jan 15, 2025
65558 GABAA CLONED HUMAN [3H] Flunitrazepam PWZ-009A1 1.34 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
5966 Alpha2A CELLS HT29 3H-RAUWOLSCINE BAM 1303 1.34 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
12886 CLONED HUMAN 3H-RAUWOLSCINE BAM 1303 1.34 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
8305 SST4 CLONED HUMAN 125I-CGP23996 Somatostatin-14 1.34 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
7816 GABAA CLONED HUMAN 3H-RO-15-1788 15 1.34 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
6538 5-HT7B CLONED HUMAN 3H-5CT METHIOTHEPIN 1.34 JASPER JR,ET AL., Jan 15, 2025 Jan 15, 2025
5021 5-HT2A CLONED HUMAN 3H-KETANSERIN KETANSERIN 1.34 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
6309 5-HT7 CORTEX GUINEA PIG 3H-5CT 5-Hydroxy Tryptamine 1.34 TO ZP, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
60630 GABAA CLONED HUMAN FNZ PWZ-009A1 1.34 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
9710 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl-2-Me 1.34 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
42508 CLONED RABBIT 35S-GTPGammaS Motilin 1.34896 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
26405 GAL2 CLONED RAT 125I-GALANIN Galanin rat 1.34896 Smith KE, et. al., 1998 Jan 15, 2025 Jan 15, 2025
97849 5-HT2C Membranes HUMAN 3H-MESULERGINE Eplivanserin 1.34896 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
63339 CRF1 CLONED HUMAN 125I-Astressin + GTP GammaS NBI 35965 1.34896 Hoare SR, et al., 2003 Jan 15, 2025 Jan 15, 2025
27320 Alpha1D CLONED HUMAN 3H-PRAZOSIN Roxindole 1.34896 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
27856 D3 CLONED HUMAN 3H-SPIPERONE GR218231 1.34896 Millan MJ, et al., 2000b Jan 15, 2025 Jan 15, 2025
63716 D2 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 1.34896 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
2316 5-HT3 ENTO CORTEX RAT 3H-ZACOPRIDE GR 65630 1.35 BARNES ET AL., 1988 Jan 15, 2025 Jan 15, 2025
99358 D3 CLONED HUMAN [3H]N-methylspiperone 6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline 1.35 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
2897 5-HT2A CORTEX RAT 125I-LSD LSD 1.35 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
35947 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN 8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 1.35 Campiani G, et al., 2005 Jan 15, 2025 Jan 15, 2025
886 5-HT2C Choroid Plexus HUMAN 3H-MESULERGINE METITEPIN 1.35 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
12665 MOR BE(2)-C HUMAN 3H-DAMGO Naloxone(-) 1.35 Standifer KM, et al., 1994 Jan 15, 2025 Jan 15, 2025
41871 H3 CLONED RAT 3H-Alpha-Me-histamine 4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 1.35 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
24476 CLONED RAT 3H-R214127 R214127 1.35 Lavreysen, H, et al., 2003 Jan 15, 2025 Jan 15, 2025
67490 Beta 1 CLONED HUMAN I125- Iodopindolol PROPRANOLOL 1.35 Song, Gang et., al. 2017 Jan 15, 2025 Jan 15, 2025
40938 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-88 1.35 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
8208 SST4 CLONED HUMAN 125I-LTT-SST-28 SMS 201-995 1.36 Demchyshyn L, et al., 1993 Jan 15, 2025 Jan 15, 2025
41365 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione 1.36 Kumar JS, et al., 2006 Jan 15, 2025 Jan 15, 2025
24477 CLONED RAT 3H-R214127 NPS 2390 1.36 Lavreysen, H, et al., 2003 Jan 15, 2025 Jan 15, 2025
70065 D3 CLONED HUMAN 3H-SPIPERONE (-)-5-OH-DPAT 1.36 Ghosh, B. et, al 2010 Jan 15, 2025 Jan 28, 2025
25582 Alpha2A CLONED HUMAN 3H-CLONIDINE OXYMETAZOLINE 1.36 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
65839 GABAA CLONED HUMAN [3H] Flunitrazepam DM-II-72 (C15H10N20BrCl) 1.37 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
13365 D4 CLONED HUMAN 35S-GTPGammaS HALOPERIDOL 1.37 Newman-Tancredi A, et al., 1997 Jan 15, 2025 Jan 27, 2025
61265 GABAA CLONED HUMAN FNZ DM-II-72 1.37 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
10075 MOR BRAIN MOUSE 125I-Endomorphin-2 Endomorphin 2 1.37 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
136 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.37 COSSERY ET AL.,1986 Jan 15, 2025 Jan 15, 2025
9352 GABAA CEREBRAL CORTEX RAT FNZ Flunitrazepam 1.37 Giorgi,Lecca,Cancedda,Giuliana,Corda,1995 Jan 15, 2025 Jan 15, 2025
9387 GABAA Parotid gland RAT 3H-PK11195 PK11195 1.37 Yamagishi H, et al., 1998 Jan 15, 2025 Jan 15, 2025
13488 LUNG RAT 3H-QNB 4-DAMP 1.37 Gies JP, et al., 1989 Jan 15, 2025 Jan 15, 2025
18916 H1 CLONED GUINEA PIG 3H-trans-H2-PAT,(-) trans-H2-PAT(+/-) 1.37 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
2856 5-HT2A CORTEX RAT 3H-KETANSERIN KETANSERIN 1.38 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
2857 5-HT2A CORTEX RAT 3H-KETANSERIN KETANSERIN 1.38 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
2858 5-HT2A CORTEX RAT 3H-KETANSERIN KETANSERIN 1.38 HOYER, 1988 (TIPS) Jan 15, 2025 Jan 15, 2025
2859 5-HT2A CORTEX RAT 3H-KETANSERIN KETANSERIN 1.38 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
8753 SST2 CORTEX HUMAN 125I-Tyr3-octreotide BIM 23014 1.38 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
16970 D3 CLONED HUMAN 3H-SPIPERONE GR218231 1.38 Cussac D, et al., 2000 Jan 15, 2025 Jan 15, 2025
57439 CB1 UNDEFINED UNDEFINED UNDEFINED Rimonabant 1.38 Donohue SR et al., 2009 Jan 15, 2025 Jan 15, 2025
41065 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-129 1.38 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
41068 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-147 1.38 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
3970 5-HT4 Colliculus Neurons MOUSE 3H-GR-113808 RN 76186 1.38 CLAEYSEN S, ET AL., 1996 Jan 15, 2025 Jan 27, 2025
2979 5-HT2A CORTEX HUMAN 3H-KETANSERIN METITEPIN 1.38 HOYER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
4805 5-HT4 Colliculus Neurons MOUSE 3H-GR-113808 RN 76186 1.38 ANSANAY H, ET AL.,1996 Jan 15, 2025 Jan 15, 2025
10963 SLC6A3 BRAIN RAT 3H-WIN 35,428 BINDING RTI-147 1.38 DAMAJ MI, et al., 1999 Jan 15, 2025 Jan 15, 2025
5090 5-HT2C CLONED HUMAN 3H-MESULERGINE MIANSERIN 1.38 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
32258 M2 HEART RAT 3H-NMS Secoverine 1.38038 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
83468 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 1.38038 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
39819 5-HT2B CLONED HUMAN 3H-MESULERGINE LISURIDE 1.38038 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
64652 H1 CLONED HUMAN 3H-PYRILAMINE MAPROTILINE 1.38038 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
27297 Alpha1B CLONED HUMAN 3H-PRAZOSIN BROMOCRIPTINE 1.38038 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
67753 5-HT2C Choroid Plexus PIG 3H-5-HT MESULERGINE 1.38038 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
63672 Alpha1 CLONED HUMAN 3H-PRAZOSIN RISPERIDONE 1.38038 Schmidt, AW. et, al. 2001 Jan 15, 2025 Jan 15, 2025
34339 nAChR7 CLONED RAT 3H-MLA Methyllycaconitine 1.39 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 15, 2025
7724 GABAA CLONED RAT 3H-FMZ flumazenil 1.39 Renard S, et al., 1999 Jan 15, 2025 Jan 27, 2025
99639 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[3-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine 1.39 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
3171 5-HT7 CLONED RAT 3H-LSD RISPERIDONE 1.39 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
22420 A2B CLONED HUMAN 3H-ZM241385 20 1.39 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
92827 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1.39 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
23714 MC1 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH Gamma3-MSH 1.39 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
22493 MC1 CLONED HUMAN 125I-NDP-MSH Gamma3-MSH 1.39 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
73472 Sigma 1 test RODENT 3H-Pentazocine(+) 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 1.4 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
4097 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl NALBzoH 1.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
102145 D3 CLONED HUMAN [3H]N-methylspiperone NEMONAPRIDE 1.4 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
13571 M4 CORTICAL RAT 3H-cAMP 4-DAMP 1.4 McKinney M, et al., 1991 Jan 15, 2025 Jan 15, 2025
51722 NR3C1 UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline 1.4 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
3851 5-HT2A CLONED RAT 3H-SPIPERONE RISPERIDONE 1.4 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
100365 Alpha1A CLONED HUMAN 3H-PRAZOSIN ILOPERIDONE 1.4 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
63502 D2 CLONED RAT 3H-N-Methylspiperone ARIPIPRAZOLE 1.4 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
16655 M2 CLONED HUMAN 3H-QNB BENZTROPINE 1.4 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
35603 D2 CLONED HUMAN 3H-SPIPERONE RISPERIDONE 1.4 Phillips ST, et. al., 1995 Jan 15, 2025 Jan 27, 2025
48149 Y5 CLONED HUMAN 3H-Propionyl-NPY PP, human 1.4 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
62742 SST5 Ovary HAMSTER UNKNOWN Somatostatin-14 1.4 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
12567 Mesenteric artery RAT 125I-Angiotensin II L-158,809 1.4 Kushida H, et al., 1995 Jan 15, 2025 Jan 15, 2025
42263 CLONED HUMAN 125I-Motilin Delta 17-20 1.4 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
45592 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE IMIPRAMINE 1.4 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
29980 BRAIN RAT 3H-CLONIDINE OXYMETAZOLINE 1.4 Greenberg, DA et al., 1976 Jan 15, 2025 Jan 15, 2025
36381 Platelets HUMAN 3H-SQ 29548 BM 613 1.4 Hanson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
12318 AORTA RAT 3H-PRAZOSIN PHENTOLAMINE 1.4 Jones SB, et al., 1987 Jan 15, 2025 Jan 15, 2025
20773 D2 BRAIN CALF 3H-Haloperidol Ergocristine 1.4 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
13862 MOR Striatal Membranes BOVINE 3H-DAMGO MC-CAM 1.4 McLaughlin, et al., 1998 Jan 15, 2025 Jan 15, 2025
31783 M1 CLONED HUMAN 3H-NMS CLOZAPINE 1.4 Bymaster F.P., et. al., 1996 Jan 15, 2025 Jan 15, 2025
40999 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-114 1.4 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
55591 KOR UNDEFINED HUMAN UNDEFINED clocinnamox 1.4 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
11048 H3 CLONED RAT 3H-methylhistamine Immepip 1.4 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
23848 CRF1 CLONED HUMAN 125I-oCRF hrCRF 1.4 Zhang, GE. et al., 2003 Jan 15, 2025 Jan 15, 2025
66090 CB1 CEREBELLUM RAT 3H-CP55940 Arachidonyl-2-chloro-ethylamide 1.4 Hillard CJ, et al., 1999 Jan 15, 2025 Jan 28, 2025
54058 Kcnn3 UNDEFINED RAT UNDEFINED UCL-1848 1.4 Sørensen US et al., 2008 Jan 15, 2025 Jan 15, 2025
10286 TP Placenta Membranes HUMAN 125I-BOP 227I-BOP 1.4 D'AngeloDavis MG, Ali S, Dorn GW, 1994 Jan 15, 2025 Jan 15, 2025
4144 KOR BRAIN GUINEA PIG 3H-U69,593 DYNORPHIN(1-8)-OH 1.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
35889 SLC6A4 CLONED HUMAN 3H-PAROXETINE 7-Methoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole 1.4 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
14899 CLONED RAT UNDEFINED SERTINDOLE 1.4 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
10294 MOR CLONED HUMAN 3H-DAMGO Naloxone(-) 1.4 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
4663 SLC6A3 CLONED HUMAN 3H-GBR 12,935 BINDING GBR-12909 1.4 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
64568 D2 STRIATUM RAT 3H-SPIPERONE HALOPERIDOL 1.4 Claustre Y, et.al., 2003 Jan 15, 2025 Jan 15, 2025
13881 A1 HEART Chick 125I-Aba CHA 1.4 Leung E, et al., 1987 Jan 15, 2025 Jan 15, 2025
47931 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 1.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
10300 MOR CLONED HUMAN 3H-DAMGO DAMGO 1.4 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
14908 CLONED RAT UNDEFINED SERTINDOLE 1.4 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
37438 D3 CLONED primate 3H-YM 09151-2 NGB 2904 1.4 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
98112 CB1 CLONED HUMAN [3H]CP55940 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(1-methylethyl)sulfonyl]piperazin-1-yl}-9H-purine 1.4 Amato GS et al 2018 Jan 15, 2025 Jan 28, 2025
22337 A1 BRAIN BOVINE 3H-DPCPX CPT 1.4 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
53058 DOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan 1.4 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
10311 MOR CLONED HUMAN 3H-DAMGO Bremazocine 1.4 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
37447 D3 CLONED primate 3H-YM 09151-2 N-{4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl}(9-oxofluoren-4-yl)carboxamide 1.4 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
81225 Alpha1B test test 3H-PRAZOSIN 5’-Iodo-HEAT HCl 1.4 Petrie EC et al 2012 Jan 15, 2025 Jan 28, 2025
81226 Alpha1D test test 3H-PRAZOSIN 5’-Iodo-HEAT HCl 1.4 Petrie EC et al 2012 Jan 15, 2025 Jan 28, 2025
13387 D3 CLONED HUMAN 3H-thymidine CF 25-397 1.4 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
90955 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (S)-5-((3-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride 1.4 Sun H et al 2016 Jan 15, 2025 Jan 28, 2025
51275 SLC6A4 UNDEFINED RAT UNDEFINED 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol 1.4 Keith JM et al., 2007 Jan 15, 2025 Jan 15, 2025
81228 Alpha2B test test 3H-CLONIDINE 5’-Iodo-HEAT HCl 1.4 Petrie EC et al 2012 Jan 15, 2025 Jan 28, 2025
38735 CLONED RAT 3H-dexamethasone RU 38486 1.4 Link JT, et al., 2005 Jan 15, 2025 Jan 15, 2025
52047 SLC6A4 UNDEFINED HUMAN UNDEFINED N-(4-(4-(3,4-dichlorophenoxy)-3-((methylamino)methyl)phenyl)but-3-ynyl)cyclopropanamine 1.4 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
66130 CLONED HUMAN 3H-PRAZOSIN RISPERIDONE 1.4 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
100690 5-HT1D CLONED HUMAN 125I-aminopotentidine Pizotyline 1.4 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
13395 D3 CLONED HUMAN 3H-thymidine DOPAMINE 1.4 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
22099 PMNL RAT 3H-Leukotriene B4 BIIL-315 1.4 Birke FW, et al., 2001 Jan 15, 2025 Jan 15, 2025
28501 D2 CLONED HUMAN 3H-NMSP PERPHENAZINE 1.4 Kroeze WK, et.al., 2003 Jan 15, 2025 Jan 15, 2025
68950 GABAA CLONED RAT 3H-Ro15-1788 3-(2,4-Difluorophenyl)-5-[3-(3,5-difluoropyridin-2-yl)-4-fluorophenyl]pyridazine 1.4 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
13399 D2 CLONED HUMAN 125I-IODOSULPRIDE LISURIDE 1.4 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
98136 CB1 CLONED HUMAN [3H]CP55940 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclohexylpiperazine-1-carboxamide 1.4 Amato GS et al 2018 Jan 15, 2025 Jan 28, 2025
20825 D2 BRAIN CALF 3H-Haloperidol METHIOTHEPIN 1.4 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
30553 A1 BRAIN RAT 3H-R-PIA C19H21ClN5O4 1.4 Thompson RD et al., 1991 Jan 15, 2025 Jan 15, 2025
20826 D2 BRAIN CALF 3H-Haloperidol HALOPERIDOL 1.4 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
20827 D2 BRAIN CALF 3H-Haloperidol Bromoperidol 1.4 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
3677 MOR BRAIN GUINEA PIG 3H-DAMGO Methadone-HCL,(-) 1.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
31839 D1 retina RAT 3H-SCH23390 SCH 23390 1.4 Bymaster F.P., et. al., 1999 Jan 15, 2025 Jan 15, 2025
70240 MOR CLONED MOUSE 3H-DAMGO DAMGO 1.4 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
39520 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
59744 PBR KIDNEY RAT 3H-PK11195 2-[5,7-Dimethyl-2-(4’-propoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-N,N-diethylacetamide 1.4 Reynolds, A. et. al., 2010 Jan 15, 2025 Jan 15, 2025
29025 SST5 CLONED HUMAN 125I-LTT-SST-28 BIM 23050 1.4 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
38242 CLONED RAT 3H-dexamethasone C30H36NO3 1.4 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
78948 5-HT1D CLONED HUMAN 3H-5-CT 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane 1.4 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
97637 SST1 CLONED HUMAN 125I-LTT-SST-28 L-797,591 1.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
38245 CLONED RAT 3H-dexamethasone C55H77N2O8 1.4 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
52069 SLC6A4 UNDEFINED HUMAN UNDEFINED (5-(4-(4-isopropylpiperazin-1-yl)butyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine 1.4 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
53861 PGR UNDEFINED HUMAN UNDEFINED Mpa 1.4 Pedram B et al., 2008 Jan 15, 2025 Jan 15, 2025
12135 D2 BRAIN HUMAN UNDEFINED PERPHENAZINE 1.4 Richelson E., 1988 Jan 15, 2025 Jan 15, 2025
2664 5-HT2A CAUDATE BOVINE 125I-LSD SPIPERONE 1.4 HARTIG ET AL., 1985 Jan 15, 2025 Jan 15, 2025
85608 nAChR FOREBRAIN RAT 3H-Epibatidine Isopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate 1.4 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
11369 5-HT2A CLONED HUMAN 125I-R091150 Ziprasidone 1.4 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
13417 D3 CLONED HUMAN 125I-IODOSULPRIDE CF 25-397 1.4 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
50795 SLC6A3 UNDEFINED HUMAN UNDEFINED methyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate 1.4 Froimowitz M et al., 2007 Jan 15, 2025 Jan 15, 2025
56941 DOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-iodo)benzamido]morphinan-oxalate 1.4 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
59245 CLONED RAT 3H-5HT 4-Chloro-3-{3-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 1.4 Smid P, et al., 2005 Jan 15, 2025 Jan 15, 2025
56942 DOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-t-butyl)benzamido]morphinan-oxalate 1.4 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
68976 GABAA CLONED RAT 3H-Ro15-1788 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3-fluoropyridin-2-yl)pyridazine 1.4 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
90992 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (S)-5-((3-Chlorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride 1.4 Sun H et al 2016 Jan 15, 2025 Jan 28, 2025
20852 D2 STRIATUM CALF 3H-Haloperidol HALOPERIDOL 1.4 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
59254 CLONED RAT 3H-5HT 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2,2-dimethyl-2H-1,4-benzoxazin-3(4H)-one 1.4 Smid P, et al., 2005 Jan 15, 2025 Jan 15, 2025
70267 MOR CLONED MOUSE 3H-DAMGO NALOXONE 1.4 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
13436 CEREBELLUM RAT FNZ Beta CCM 1.4 Massotti M, et al., 1991 Jan 15, 2025 Jan 15, 2025
31868 M1 CLONED HUMAN 3H-QNB CLOZAPINE 1.4 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
49020 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (+)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-butyl]piperidine hydrochloride 1.4 Berardi, F et al., 2003 Jan 15, 2025 Jan 15, 2025
31613 D1 Striatal Membranes RAT 3H-SCH23390 C19H23ClN2S dimaleate (54) 1.4 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
66174 D2 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 1.4 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 28, 2025
21376 A2A CLONED HUMAN 125I-APE ZM 241385 1.4 Linden J et al., 1999 Jan 15, 2025 Jan 15, 2025
70274 MOR CLONED MOUSE 3H-DAMGO Morphine 1.4 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
29315 Y5 CLONED Rat 6B 125I-PYY PYY 3-36, rat 1.4 Hu Y, et al., 1996 Jan 15, 2025 Jan 15, 2025
3720 MOR CLONED HUMAN 3H-DAMGO Naloxone(-) 1.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
47752 Y1 CLONED RAT [125I] - Peptide YY NPY 28-36, [P30, Y32, L34] 1.4 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
137 5-HT1A CORTEX RAT 3H-5-MeO-DPAC 5-Hydroxy Tryptamine 1.4 COSSERY ET AL., 1987 Jan 15, 2025 Jan 15, 2025
85897 TAAR1 HEK293 cells RAT 3H-RO5166017 2C-BI-11 1.4 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
23690 SLC6A4 CLONED HUMAN 3H-CITALOPRAM Fluoxetine-R-(-) 1.4 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
25226 D2 CLONED HUMAN 3H-NMSP THIOTHIXENE 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
51597 Alpha1D UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide 1.4 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
62093 CLONED HUMAN 3H- LSD 5-HT7 1.4 Herth, Matthis et. al. 2015 Jan 15, 2025 Jan 15, 2025
48015 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 1.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
51090 Alpha1A UNDEFINED HUMAN UNDEFINED 3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 1.4 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
45204 M1 CORTEX RAT 3H-PIRENZEPINE (1RS,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate 1.4 Naito R, et al., 2005 Jan 15, 2025 Jan 15, 2025
97685 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 1.4 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
14742 PAF Washed Platelets HUMAN 3H-PAF CV-6209 1.4 Tahraoui L, et al., 1990 Jan 15, 2025 Jan 15, 2025
36759 H1 CLONED HUMAN 3H-PYRILAMINE (+)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 1.4 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
34968 nAChR CLONED UNDEFINED 3H-Epibatidine 5-(1-Hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 1.4 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
10907 D4 CLONED HUMAN 3H-SPIPERONE SPIPERONE 1.4 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
70302 MOR CLONED MOUSE 3H-Diprenorphine Naltrexone 1.4 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
18595 PANCREAS RAT 125I-CCK-33 22 1.4 Evans BE et al., 1986 Jan 15, 2025 Jan 15, 2025
29091 SST3 CLONED HUMAN 125I-LTT-SST-28 BIM 23058 1.4 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
48803 D3 CLONED HUMAN 3H-SPIPERONE BP-897 1.4 Bettinetti L, et al., 2002 Jan 15, 2025 Jan 15, 2025
18597 PANCREAS RAT 125I-CCK-33 20 1.4 Evans BE et al., 1986 Jan 15, 2025 Jan 15, 2025
99751 DOR CLONED HUMAN 3H-DPDPE (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
15016 5-HT7 CLONED RAT 3H-LSD RISPERIDONE 1.4 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
26280 5-HT1B CLONED HUMAN 3H-5HT 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-mesitylenepiperazin-1-yl)ethanone 1.4 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
100264 5-HT2B CLONED HUMAN 3H-LSD SERTINDOLE 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
5801 Alpha2A CELLS HT29 3H-RAUWOLSCINE WY26703 1.4 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
45486 NMDA CLONED HUMAN 3H-Glycine L-701,324 1.4 Buchstaller HP, et al., 2006 Jan 15, 2025 Jan 28, 2025
2992 5-HT2A CORTEX RAT 3H-KETANSERIN MIANSERIN 1.4 LEYSON ET AL., 1982 Jan 15, 2025 Jan 15, 2025
32945 SST4 CLONED HUMAN 125I-Tyr11-SRIF Somatostatin-14 1.4 Ankersen M, et. al.,1998 Jan 15, 2025 Jan 15, 2025
100785 PDE4d CLONED HUMAN Functional 2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide 1.4 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
10679 M3 CLONED HUMAN 3H-NMS HX 1.4 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
42938 EGFR CLONED HUMAN 3H-Staurosporine Tarceva 1.4 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
7355 DOR CLONED HUMAN 3H-Naltrindole ETORPHINE - HCI 1.4 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
14779 D2 Striatal Membranes CALF 3H-Haloperidol BROMPERIDOL 1.4 Creese I, et al., 1976 Jan 15, 2025 Jan 15, 2025
65724 GABAA CLONED HUMAN [3H] Flunitrazepam TG-4-39 1.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
14780 D2 Striatal Membranes CALF 3H-Haloperidol THIOTHIXENE,cis- 1.4 Creese I, et al., 1976 Jan 15, 2025 Jan 15, 2025
18876 A2A CLONED HUMAN 3H-MRE 3008F20 ZM 241385 1.4 Gessi S et al., 2002 Jan 15, 2025 Jan 15, 2025
42940 EGFR CLONED HUMAN 3H-Staurosporine CI-1033 1.4 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
12222 BRAIN HUMAN UNDEFINED CHLORPROMAZINE 1.4 Richelson E., 1988 Jan 15, 2025 Jan 15, 2025
17598 T47D HUMAN 125I-VIP VIP Ala9 1.4 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
36798 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 1.4 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 27, 2025
53951 D3 UNDEFINED HUMAN UNDEFINED Naphthalene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide 1.4 Leopoldo M et al., 2009 Jan 15, 2025 Jan 15, 2025
2496 5-HT3 ENTO CORTEX RAT 3H-GR-65630 QUIPAZINE 1.4 Kilpatrick et al., 1987 Jan 15, 2025 Jan 15, 2025
11200 D2 STRIATUM RAT 3H-Haloperidol HALOPERIDOL 1.4 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
24258 V2 CLONED RAT 125I-VIP VIP Ala27 1.4 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
53700 D2 UNDEFINED HUMAN UNDEFINED HALOPERIDOL 1.4 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
55750 5-HT1D UNDEFINED HUMAN UNDEFINED N1,N13-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tridecanediamide 1.4 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
55239 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 1.4 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
70089 5-HT3 CORTICAL MEMBRANES RAT 3H-GR-65630 1.4 Van Wijingaarden, I. et, al. 1993 Jan 15, 2025 Jan 15, 2025
1738 5-HT2A CORTEX HUMAN 3H-KETANSERIN CHLORPROMAZINE 1.4 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
39115 D3 CLONED HUMAN R-SAT FLUPHENAZINE 1.4 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
41675 5-HT6 CLONED HUMAN 3H-LSD ORG-5222 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
10960 SLC6A3 BRAIN RAT 3H-WIN 35,428 BINDING RTI-114 1.4 DAMAJ MI, et al., 1999 Jan 15, 2025 Jan 15, 2025
41680 D2 CLONED HUMAN 3H-NMSP ORG-5222 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
55248 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 1.4 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
64978 H1 BRAIN GUINEA PIG 3H-MEPYRAMINE CHLORPHENIRAMINE-d 1.4 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
11738 D2 CAUDATE NUCLEUS HUMAN 3H-SPIPERONE PERPHENAZINE 1.4 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
18906 A3 CLONED HUMAN 3H-MRE 3008F20 MRE 3062F20 1.4 Gessi S et al., 2002 Jan 15, 2025 Jan 15, 2025
37853 BRAIN GUINEA PIG 3H-Cyprodime NALOXONE 1.4 Marki A, et al., 1999 Jan 15, 2025 Jan 15, 2025
59614 5-HT7 CLONED HUMAN 3H-LSD RA-7 1.4 Hedlund, P. et. al., 2010 Jan 15, 2025 Jan 15, 2025
66274 Sigma 1 BRAIN RAT 3H-Haloperidol 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 1.4 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
54242 CB1 UNDEFINED UNDEFINED UNDEFINED 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2-difluorobutyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 1.4 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
60642 GABAA CLONED HUMAN FNZ TG-4-39 1.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
14820 D2 Corpus Striatum CALF 3H-Haloperidol HALOPERIDOL 1.4 Creese I, et al., 1976 Jan 15, 2025 Jan 15, 2025
12005 H1 CORTICAL MEMBRANES HUMAN 3H-doxepin Trimipramine 1.4 Kanba S, et al., 1984 Jan 15, 2025 Jan 15, 2025
3304 D3 CLONED HUMAN 3H-YM 09151-2 BUTACLAMOL,(+) 1.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
4073 DOR CLONED HUMAN 3H-DPDPE-Cl WIN 44,441(-) 1.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
100073 5-HT1A CLONED HUMAN 3H-WAY100635 Cariprazine 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
32747 5-HT2C CLONED RAT 3H-MESULERGINE MIANSERIN 1.4 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
16623 Y2 CLONED HUMAN [125I] - Peptide YY Des-AA11-18[Cys7,21,D-Lys9 (Ac)]-NPY 1.4 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
99824 DOR CLONED HUMAN [3H]DPDPE (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
16625 Y2 CLONED HUMAN [125I] - Peptide YY Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26]-NPY 1.4 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
6130 Alpha1C CLONED HUMAN 125I-HEAT PHENTOLAMINE 1.4 HIRASAWA A, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
89843 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 1.4 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
5108 5-HT2A CLONED HUMAN 125I-DOI DOC 1.4 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
35830 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 1.4 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
62712 SST2 COLON RAT UNKNOWN (4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 1.4 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
27899 5-HT2A CLONED HUMAN 3H-DOB LISURIDE 1.4 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
49147 DOR CLONED HUMAN 3H-DPDPE LYS401 1.4 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
29180 SST1 CLONED HUMAN UNDEFINED L-797,591 1.4 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
63740 nAChR BRAIN MICE 3H-NICOTINE Nicotine 1.4 Damaj, MI et al., 1998 Jan 15, 2025 Jan 15, 2025
2322 5-HT3 HIPPOCAMPUS HUMAN 3H-ZACOPRIDE GRANISETRON 1.41 BARNES ET AL., 1988 Jan 15, 2025 Jan 15, 2025
2323 5-HT3 CELLS N1E-115 3H-ICS 205-930 GRANISETRON 1.41 HOYER & NEIJT, 1988 Jan 15, 2025 Jan 15, 2025
8754 SST2 CORTEX HUMAN 125I-Tyr3-octreotide RC 160 1.41 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
54074 MOR UNDEFINED UNDEFINED UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan 1.41 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
45641 NET CLONED HUMAN 3H-Nisoxetine Protriptyline 1.41 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
4961 5-HT2A CLONED RAT 3H-KETANSERIN ERGOTAMINE 1.41 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
2956 5-HT2A CORTEX PIG 3H-KETANSERIN METHERGINE 1.41 HOYER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
90512 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1.41 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
8854 GABAA Submandibular gland RAT 3H-PK11195 PK11195 1.41 Yamagishi H, et al., 1998 Jan 15, 2025 Jan 15, 2025
30113 SST5 CLONED HUMAN 125I-SOMATOSTATIN Somatostatin-14 1.41 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
5039 5-HT2A CLONED HUMAN 3H-KETANSERIN SPIPERONE 1.41 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
13493 HEART RAT 3H-QNB ATR 1.41 Gies JP, et al., 1989 Jan 15, 2025 Jan 15, 2025
8632 SST4 CLONED MOUSE 125I-Tyr11-SRIF CGP 23996 1.41 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
8380 SST2 CLONED HUMAN 125I-Tyr3-octreotide CST17 1.41 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
10941 DOR BRAIN MOUSE 3H-DPDPE BU 95 1.41 TRAYNOR, JR., et al., 1999 Jan 15, 2025 Jan 15, 2025
30163 A3 CLONED RAT 3H-AB-MECA 2-Chloro-N6-(3-iodobenzyl)-adenosine 1.41 Kim HO et al., 1994 Jan 15, 2025 Jan 15, 2025
50148 KA BRAIN RABBIT 3H-Methylglutamate-4-(2S,4R) Kainate 1.41 Toms, NJ et al., 1997 Jan 15, 2025 Jan 15, 2025
51965 KOR UNDEFINED HUMAN UNDEFINED 1'-(p-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1.41 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
22017 LHRH Pituitary RAT UNDEFINED 25 1.41254 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
32280 M2 HEART RAT 3H-NMS SCOPOLAMINE 1.41254 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
26939 5-HT6 CLONED HUMAN 3H-LSD METHIOTHEPIN 1.41254 Hirst WD, et.al.,2003 Jan 15, 2025 Jan 15, 2025
26958 5-HT6 CLONED RAT 3H-LSD SB-357134 1.41254 Hirst WD, et.al.,2003 Jan 15, 2025 Jan 15, 2025
32347 M4 LUNG RABBIT 3H-NMS 4-DAMP 1.41254 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
64376 H1 CLONED HUMAN 3H-PYRILAMINE OLANZAPINE 1.41254 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
64135 D3 CLONED RAT 3H-N-Methylspiperone FLUPHENAZINE 1.41254 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
39610 5-HT2B CLONED HUMAN Functional DOI 1.41254 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
32230 M1 CORTEX RAT 3H-PIRENZEPINE Secoverine 1.41254 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
21999 LHRH Pituitary RAT UNDEFINED 7 1.41254 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
22006 LHRH Pituitary RAT UNDEFINED 14 1.41254 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
41857 H3 CLONED RAT 3H-Alpha-Me-histamine 6-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 1.42 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
99720 D3 CLONED HUMAN [3H]spiperone (S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol 1.42 Luo D et al 2016 Jan 15, 2025 Jan 28, 2025
24492 CLONED RAT 3H-Quisqualate (S)-3,5-DHPG 1.42 Lavreysen, H, et al., 2003 Jan 15, 2025 Jan 15, 2025
64941 CLONED HUMAN 3H-PRAZOSIN RISPERIDONE 1.42 Ishibashi, Tadashi. et. al, 2010 Jan 15, 2025 Jan 15, 2025
65565 GABAA CLONED HUMAN [3H] Flunitrazepam Alprazolam 1.43 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
30062 SST2 CLONED RAT 125I-SOMATOSTATIN Somatostatin-14 1.43 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
30075 SST2 CLONED MOUSE 125I-SOMATOSTATIN Somatostatin-14 1.43 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
60558 GABAA CLONED HUMAN FNZ Alprazolam 1.43 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
49574 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 1.43 Shimon I, et.al., 1997 Jan 15, 2025 Jan 15, 2025
14294 SLC6A3 STRIATUM RAT 3H-DA UPTAKE GBR-12909 1.43 Letchworth SR, et al., 2000 Jan 15, 2025 Jan 15, 2025
12889 CLONED HUMAN 3H-RAUWOLSCINE OXYMETAZOLINE 1.44 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
55150 D2 UNDEFINED HUMAN UNDEFINED FLUPHENAZINE 1.44 von Coburg Y et al., 2009 Jan 15, 2025 Jan 15, 2025
5055 5-HT2B CLONED HUMAN 3H-5HT MESULERGINE 1.44 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
56046 MOR UNDEFINED UNDEFINED UNDEFINED (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-2-carboxylate 1.44 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
34103 H3 BRAIN CORTEX RAT 3H-Alpha-Me-histamine A-349821 1.44544 Esbenshade TA, et al., 2004 Jan 15, 2025 Jan 15, 2025
64084 H3 CORTEX RAT 3H-Alpha-Me-histamine A-349821 1.44544 Esbenshade TA, et al., 2004 Jan 15, 2025 Jan 15, 2025
63330 CRF1 CLONED HUMAN 125I-Sauvagine NBI 35965 1.44544 Hoare SR, et al., 2003 Jan 15, 2025 Jan 15, 2025
64181 CLONED HUMAN 3H-PRAZOSIN CHLORPROMAZINE 1.44544 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
26818 GAL2 CLONED HUMAN 125I-GALANIN M32 1.44544 Borowsky Beth, et. al., 1998 Jan 15, 2025 Jan 15, 2025
6917 5-HT2A CLONED HUMAN 3H-KETANSERIN ISOCLOZAPINE 1.45 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
60191 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-((4,5-Dimethylfuran-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide 1.45 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
5967 Alpha2A CELLS HT29 3H-RAUWOLSCINE OXYMETAZOLINE 1.45 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
12664 MOR BE(2)-C HUMAN 3H-DAMGO Methadone-HCL,(-) 1.45 Standifer KM, et al., 1994 Jan 15, 2025 Jan 15, 2025
1929 5-HT2A CORTEX RAT 125I-LSD ERGOTAMINE 1.45 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
7314 V1A CLONED RAT 3H-AVP AVP 1.45 Yamamura Y, et al., 1998 Jan 15, 2025 Jan 15, 2025
90522 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) HALOPERIDOL 1.45 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
10939 DOR BRAIN MOUSE 3H-DPDPE BU 47 1.45 TRAYNOR, JR., et al., 1999 Jan 15, 2025 Jan 15, 2025
47585 PKCα CLONED HUMAN 3H-PDBU CH2OCOC(CH3)3 1.45 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
63903 CLONED HUMAN 123I-ADAM 2-[(2-Amino-4-fluorophenyl)thio]-N,N-dimethylbenzenemethanamine 1.46 Huang Y et al., 2005 Jan 15, 2025 Jan 15, 2025
185 5-HT1A CORTEX PIG 3H-8-OH-DPAT 8-OH-DPAT 1.46 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
45527 NMDA CLONED HUMAN 3H-Glycine 2-Chloro-4-hydroxy-3-isopropyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 1.46 Buchstaller HP, et al., 2006 Jan 15, 2025 Jan 28, 2025
7184 NOP CLONED MOUSE 35S-GTPGammaS Ac-RYYKWR-NH2 1.47 Dooley CT, et al., 1997 Jan 15, 2025 Jan 15, 2025
99357 D3 CLONED HUMAN [3H]N-methylspiperone 5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole 1.47 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
45625 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NORFLUOXETINE 1.47 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
6985 GAL3 CLONED RAT 125I-p Galanin Galanin (1-29), rat 1.47 WANG S, ET AL., 12/1997 Jan 15, 2025 Jan 15, 2025
41071 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-208 1.47 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
30067 SST2 CLONED RAT 125I-SOMATOSTATIN BIM 23014 1.47 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
41872 H3 CLONED RAT 3H-Alpha-Me-histamine 3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 1.47 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
91557 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide 1.47 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
11519 DOR NG108-15 MOUSE 3H-DPDPE NALTRINDOLE 1.47 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
83482 M5 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 1.47911 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
39821 5-HT2C CLONED HUMAN 3H-MESULERGINE RS-102221 1.47911 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
64666 H1 CLONED HUMAN 3H-PYRILAMINE Trimipramine 1.47911 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
39841 5-HT2B CLONED HUMAN 3H-MESULERGINE SB-215505 1.47911 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
24768 Y2 CLONED HUMAN 125I-PYY PYY13-36, porcine 1.47911 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
27335 CORTEX RAT 3H-RX821002 TERGURIDE 1.47911 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
18669 H3 CLONED RAT 3H-Alpha-Me-histamine Iodophenpropit 1.47911 Wieland K et al., 2001 Jan 15, 2025 Jan 15, 2025
17153 5-HT2A BRAIN HUMAN 3H-KETANSERIN OLANZAPINE 1.48 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
58117 5-HT2A CLONED HUMAN 125I-DOI N-(3-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 1.48 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
22334 A1 BRAIN PIG 3H-DPCPX XAC 1.48 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
35134 5-HT2A CORTEX RAT 3H-KETANSERIN ST1460 1.48 Campiani G, et al., 2002 Jan 15, 2025 Jan 15, 2025
7000 GAL2 CLONED RAT 125I-p Galanin Galanin (1-29), rat 1.48 WANG S, ET AL., 12/1997 Jan 15, 2025 Jan 15, 2025
34648 5-HT2A CORTEX RAT 3H-KETANSERIN ST1469 1.48 Campiani G, et al., 2004 Jan 15, 2025 Jan 15, 2025
66188 CORTEX RAT 3H-KETANSERIN (+)-7-Chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3] benzothiazepine 1.48 Campiani G, et al., 1998 Jan 15, 2025 Jan 15, 2025
22412 A2B CLONED HUMAN 3H-ZM241385 12 1.48 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
9418 MT1 CLONED HUMAN 125I-Mel MELATONIN 1.48 Reppert, Godson, Mahle, Weaver, Slaugenhaupt, 1995 Jan 15, 2025 Jan 15, 2025
53033 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(2',3',4',6'-tetra-O-benzyl-D-glucopyranosyl)acetamido]morphinan 1.49 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
10049 MOR CLONED RAT 125I-Endomorphin-2 DAMGO 1.49 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
30058 SST2 CLONED MOUSE 125I-SOMATOSTATIN BIM 23268 1.49 Meyerhof W, 1998 Jan 15, 2025 Jan 15, 2025
45456 NET CLONED HUMAN 3H-Nisoxetine NORTRYPTYLINE 1.49 Vaishnavi SN, et al., 2004 Jan 15, 2025 Jan 15, 2025
92829 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide 1.49 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
13799 NK1 CLONED HUMAN 125I-Bolton Hunter FK 888 1.49 Kudlacz EM, et al., 1996 Jan 15, 2025 Jan 15, 2025
47616 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
51458 Alpha1A UNDEFINED HUMAN UNDEFINED 3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 1.5 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
12293 Spinal cord RAT 3H-NICOTINE Nicotine-L (base) 1.5 Khan IM, et al., 1994 Jan 15, 2025 Jan 15, 2025
61958 HEART GUINEA PIG UNDEFINED ASTEMIZOLE 1.5 Salata, JJ et al., 1995 Jan 15, 2025 Jan 15, 2025
56071 CB1 UNDEFINED HUMAN UNDEFINED HU-210 1.5 Fan H et al., 2009 Jan 15, 2025 Jan 15, 2025
61452 GABAA CLONED HUMAN FNZ RY-031 1.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
47630 ADK recombinant HUMAN Functional 4-N-(4-Methylphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
7183 NOP CLONED MOUSE 35S-GTPGammaS Ac-RYYRIK-NH2 1.5 Dooley CT, et al., 1997 Jan 15, 2025 Jan 15, 2025
3345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DHE 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
19473 GPR145 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH MCH 1.5 Sailer AW et al., 2001 Jan 15, 2025 Jan 15, 2025
47633 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(5-azido-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
57363 CHRNA4 UNDEFINED RAT UNDEFINED Nicotine 1.5 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
93972 D2 CLONED HUMAN 3H-SPIPERONE compound 43 1.5 Ortega R et al 2011 Jan 15, 2025 Jan 29, 2025
30487 M3 CLONED HUMAN 3H-QNB 3-Ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 1.5 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
38935 5-HT3 CORTEX RAT 3H-QUIPAZINE QUIPAZINE 1.5 Glennon RA, et al., 1989 Jan 15, 2025 Jan 15, 2025
32792 D2 CLONED HUMAN 3H-SPIPERONE CHLORPROMAZINE 1.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
47644 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 1.5 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
59420 D4 CLONED HUMAN 3H-N-Methylspiporone N-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide 1.5 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
19231 NB-OK-1 HUMAN 125-[AcHis1]Pacap PACAP(6-38) 1.5 Vandermeers A et al., 1992 Jan 15, 2025 Jan 15, 2025
35871 SLC6A4 CLONED HUMAN 3H-PAROXETINE 7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 1.5 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
60192 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-((5-Ethylfuran-2-yl)ethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1.5 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
32801 D2 STRIATUM CANINE 3H-SPIPERONE OCTOCLOTHEPIN-S 1.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
93219 D4 CHO cells HUMAN 3H-SPIPERONE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1.5 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
11050 H3 CLONED RAT 3H-methylhistamine N-methylhistamine 1.5 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
12074 5-HT1D CLONED HUMAN 3H-GR-125743 Naratriptan 1.5 Domenech T, et al., 1997 Jan 15, 2025 Jan 15, 2025
53292 CHRNA4 UNDEFINED RAT UNDEFINED Nicotine 1.5 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
88622 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1.5 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
2609 5-HT2A CORTEX RAT 3H-KETANSERIN XYLAMIDINE 1.5 LEYSON ET AL., 1982 Jan 15, 2025 Jan 15, 2025
9777 MT2 CLONED HUMAN 125I-Iodomelatonin 4-P-PDOT 1.5 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
41010 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-122 1.5 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
10803 D2 CLONED HUMAN 125I-IODOSULPRIDE FLUPENTHIXOL, Alpha 1.5 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
23859 D2 CLONED HUMAN UNDEFINED Dopamine, D2 high 1.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
56627 NR3C1 UNDEFINED HUMAN UNDEFINED (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(5-methylthiophen-2-yl)-ethanol 1.5 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
82228 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one 1.5 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
42804 CLONED HUMAN 125I-ghrelin 6-[(Benzyloxy)methyl]-5-(4-{[(2-chloropyridin-4-yl)methyl]amino}phenyl)pyrimidine-2,4-diamine 1.5 Serby MD, et al., 2006 Jan 15, 2025 Jan 15, 2025
10807 D3 CLONED HUMAN 125I-IODOSULPRIDE HALOPERIDOL 1.5 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
100919 AChE BRAIN HUMAN Functional [5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]carbamic acid 2-(1H-indol-3-yl)ethyl Ester 1.5 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
11066 H3 CORTEX RAT 3H-methylhistamine R-alpha-methylhistamine 1.5 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
48698 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 1.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
9531 SLC6A4 CLONED HUMAN 3H-CITALOPRAM CITALOPRAM 1.5 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
101947 H1 CLONED HUMAN [3H] Pyrilamine ZOTEPINE 1.5 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
54846 SLC6A4 UNDEFINED RAT UNDEFINED (3R)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 1.5 Hatzenbuhler NT et al., 2008 Jan 15, 2025 Jan 15, 2025
70975 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 1.5 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
51263 SLC6A4 UNDEFINED RAT UNDEFINED 7-(3-(4-ethylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 1.5 Keith JM et al., 2007 Jan 15, 2025 Jan 15, 2025
21057 A1 BRAIN RAT 3H-R-PIA 19 1.5 Shamim MT et al., 1989 Jan 15, 2025 Jan 15, 2025
10312 MOR CLONED HUMAN 3H-DAMGO NALTREXONE-HCl 1.5 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
7242 ETA CLONED HUMAN 125I-ENDOTHELIN SB 217242 1.5 Ohlstein EH, et al., 1998 Jan 15, 2025 Jan 15, 2025
23628 5-HT2A CLONED HUMAN 3H-KETANSERIN Cyamemazine 1.5 Hameg A. et al., 2003 Jan 15, 2025 Jan 15, 2025
100172 5-HT1A CLONED HUMAN 3H-WAY100635 Ziprasidone 1.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
101196 MOR CLONED HUMAN 3H-Diprenorphine (S)-1-((5-(3,4-Dihydroisoquinolin-2(1H)-yl)pentyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate 1.5 Henry S,et al., 2021 Jan 15, 2025 Jan 28, 2025
3405 MOR CLONED HUMAN 3H-DAMGO BUPRENORPHINE 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
43342 GAK CLONED HUMAN 3H-Staurosporine EKB-569 1.5 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
47702 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Indatraline 1.5 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
19032 NB-OK-1 HUMAN 125-AcHis1-PACAP(1-27) PACAP(6-38) 1.5 Robberecht P et al., 1992 Jan 15, 2025 Jan 15, 2025
20824 D2 BRAIN CALF 3H-Haloperidol cis-Thiothixene 1.5 Burt DR et al., 1976 Jan 15, 2025 Jan 15, 2025
9049 SST4 CLONED RAT 125I-CGP23996 DC23-60 1.5 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
29017 SST2 CLONED HUMAN 125I-LTT-SST-28 MK 678 1.5 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
37465 D3 CLONED HUMAN 3H-SPIPERONE benzofuranyl 1.5 Newman AH, et al., 2005 Jan 15, 2025 Jan 15, 2025
18269 D2 BRAIN RAT 3H-NPA CHLORPROMAZINE 1.5 Hall H et al., 1986 Jan 15, 2025 Jan 27, 2025
19806 D4 CLONED HUMAN UNDEFINED THIORIDAZINE 1.5 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
10847 D3 CLONED HUMAN 125I-IODOSULPRIDE ADTN DIMETHYL 6,7 1.5 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
12383 KOR CEREBELLUM RAT 3H-flumazenil Bretazenil 1.5 Giusti P, et al., 1993 Jan 15, 2025 Jan 27, 2025
99170 A1 CLONED RAT [3H]CCPA 1,3-Dimethyl-8-phenyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1.5 Brunschweiger A et al 2016 Jan 15, 2025 Jan 15, 2025
61026 GABAA CLONED HUMAN FNZ XHE-II-002 1.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
62562 Sigma 1 BRAIN RAT 3H-Pentazocine (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-methyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one 1.5 Mcleod, Michael C. et. al., 2016 Jan 15, 2025 Jan 28, 2025
63075 MC4 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-c[Cys-Glu-His-D(2')Nal-Arg-Trp-Gly-Cys]-Pro-Pro-Lys-Asp-NH2 1.5 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
33124 SLC6A4 BRAIN RAT UNDEFINED DESIPRAMINE 1.5 Muth, EA et al., 1986 Jan 15, 2025 Jan 15, 2025
17765 CLONED RAT 125I-VIP VIP [D-Lys15] 1.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
68969 GABAA CLONED RAT 3H-Ro15-1788 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3,5-difluoropyridin-2-yl)pyridazine5-[4-Fluoro-3-(3,5-difluoropyridin-2-yl)-phenyl]-3-(3,5-difluoropyridin-2-yl)pyridazine 1.5 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
17770 CLONED RAT 125I-VIP VIP [D-Lys20] 1.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
94058 5-HT1A CLONED HUMAN [3H]-8-OH-DPAT LSD 1.5 Luethi D et al 2018 Jan 15, 2025 Jan 15, 2025
91755 A2B CLONED HUMAN 3H-MRS-1754 8-(1-{2-Oxo-2-[4-(3-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 1.5 Basu S et al 2017 Jan 15, 2025 Jan 15, 2025
6253 EP3 CLONED MOUSE 3H-PGE2 PGE1,11-DEOXY 1.5 Kiriyama M, et al., 1997 Jan 15, 2025 Jan 15, 2025
51567 Alpha1D UNDEFINED HUMAN UNDEFINED 4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 1.5 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
17778 CLONED RAT 125I-VIP VIP [D-Asn28] 1.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
22131 MOR BRAIN RAT 3H-Naloxone/+NaCl Cyclazocine 1.5 Pert CB, et al., 1974 Jan 15, 2025 Jan 15, 2025
31603 D1 Striatal Membranes RAT 3H-SCH23390 C23H26F4N2 (44) 1.5 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
54899 5-HT1A UNDEFINED HUMAN UNDEFINED (R)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide 1.5 Hatzenbuhler NT et al., 2008 Jan 15, 2025 Jan 15, 2025
41332 D5 CLONED HUMAN 3H-SCH23390 LE400 1.5 Hoefgen B, et al., 2006 Jan 15, 2025 Jan 15, 2025
70262 MOR CLONED MOUSE 3H-DAMGO Morphine 1.5 Pan YX, et al., 2005 Jan 15, 2025 Jan 29, 2025
3703 KOR CLONED HUMAN 3H-U69,593 LEVORPHANOL-tartarate 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
59255 CLONED RAT 3H-5HT 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2,4-dimethyl-2H-1,4-benzoxazin-3(4H)-one 1.5 Smid P, et al., 2005 Jan 15, 2025 Jan 15, 2025
16248 M1 CLONED HUMAN 3H-NMS a 1.5 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
31864 M2 CLONED HUMAN 3H-QNB ATR 1.5 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
40571 MOB BRAIN BOVINE UNDEFINED 1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1.5 Chimenti F, et al., 2005 Jan 15, 2025 Jan 15, 2025
22140 MOR BRAIN RAT 3H-Naloxone/-NaCl Nalorphine 1.5 Pert CB, et al., 1974 Jan 15, 2025 Jan 15, 2025
382 5-HT1A HIPPOCAMPUS HUMAN 3H-8-OH-DPAT METHERGINE 1.5 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
16255 M2 CLONED HUMAN 3H-NMS Ipratropium 1.5 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
16256 M2 CLONED HUMAN 3H-NMS ATR 1.5 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
19840 D3 CLONED HUMAN UNDEFINED THIORIDAZINE 1.5 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
16769 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE CITALOPRAM 1.5 Millan MJ, et al., 2001 Jan 15, 2025 Jan 15, 2025
3714 KOR BRAIN GUINEA PIG 3H-U69,593 BUPRENORPHINE 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
13447 CEREBELLUM RAT 3H-Clonazepam Beta CCM 1.5 Massotti M, et al., 1991 Jan 15, 2025 Jan 15, 2025
41351 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-phenyl-7-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine 1.5 Ugarkar BG, et al., 2003 Jan 15, 2025 Jan 15, 2025
18312 D2 BRAIN RAT 3H-domperidone A 38120 1.5 Hall H et al., 1986 Jan 15, 2025 Jan 27, 2025
65416 nAChR CLONED HUMAN [3H] Flunitrazepam XHE-II-002 1.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
3721 MOR BRAIN GUINEA PIG 3H-DAMGO Naloxone(-) 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
54154 NR3C1 UNDEFINED HUMAN UNDEFINED prednisolone 1.5 Yang BV et al., 2009 Jan 15, 2025 Jan 15, 2025
40587 MOB BRAIN BOVINE UNDEFINED (+/-)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1.5 Chimenti F, et al., 2005 Jan 15, 2025 Jan 15, 2025
22156 MOR BRAIN RAT 3H-Naloxone/+NaCl NALOXONE 1.5 Pert CB, et al., 1974 Jan 15, 2025 Jan 15, 2025
6797 Y2 CLONED HUMAN 125I-PYY PYY13-36, porcine 1.5 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
88463 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
36753 5-HT2C CLONED HUMAN 3H-MESULERGINE (+)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 1.5 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
22163 MOR BRAIN RAT 3H-Naloxone/-NaCl NALOXONE 1.5 Pert CB, et al., 1974 Jan 15, 2025 Jan 15, 2025
23958 D3 CLONED HUMAN UNDEFINED THIORIDAZINE 1.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
100502 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 1.5 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
45208 M1 CORTEX RAT 3H-PIRENZEPINE quinuclidin-3-yl benzhydrylcarbamate 1.5 Naito R, et al., 2005 Jan 15, 2025 Jan 15, 2025
52377 CHRNA4 UNDEFINED HUMAN UNDEFINED Nicotine 1.5 Carroll FI et al., 2007 Jan 15, 2025 Jan 15, 2025
56221 5-HT1A UNDEFINED HUMAN UNDEFINED (2S)-2-{[4-(6-Fluoroquinolin-2-yl)-1,4-diazepan-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline 1.5 Zhou D et al., 2009 Jan 15, 2025 Jan 15, 2025
48798 D3 CLONED HUMAN 3H-SPIPERONE N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide 1.5 Bettinetti L, et al., 2002 Jan 15, 2025 Jan 15, 2025
4513 D2 BRAIN RAT 3H-SPIPERONE RISPERIDONE 1.5 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
57762 SLC6A4 UNDEFINED HUMAN UNDEFINED (R)-7-[8-(2-Oxo-1,2,3,4-tetrahydro-quinolin-7-ylmethyl)-3-aza-bicyclo[3.2.1]oct-3-ylmethyl]-7,8-dihydro-3H-1,6,9-trioxa-3-aza-cyclopenta[a]naphthalen-2-one 1.5 Yan Y et al., 2010 Jan 15, 2025 Jan 15, 2025
16035 AMPA CEREBRAL CORTEX RAT 3H-Kainic acid domoic acid 1.5 Sakai R, et al., 2001 Jan 15, 2025 Jan 15, 2025
18854 V1B CLONED HUMAN 3H-AVP SSR149415 1.5 Serradeil-Le Gal C et al., 2002 Jan 15, 2025 Jan 15, 2025
9642 SLC6A4 CORTEX RAT 3H-CITALOPRAM Fluvoxamine 1.5 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
3758 MOR CLONED HUMAN 3H-DAMGO DYNORPHIN(1-11)-OH 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
10672 M2 CLONED HUMAN 3H-NMS ATR 1.5 Buckley NJ,Bonner, Buckley, Brann, 1989 Jan 15, 2025 Jan 15, 2025
31666 5-HT2A CORTICAL MEMBRANES RAT 3H-KETANSERIN C22H27FN2 (45) 1.5 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
55730 5-HT1D UNDEFINED HUMAN UNDEFINED 4-fluoro-N-{3-[1-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethyl)piperidin-4-yl]-1H-indol-5-yl}benzamide 1.5 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
10936 MOR BRAIN MOUSE 3H-DAMGO BU 96 1.5 TRAYNOR, JR., et al., 1999 Jan 15, 2025 Jan 15, 2025
3259 D2 CLONED HUMAN 3H-YM 09151-2 FLUPENTHIXOL, Alpha 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
24251 V2 CLONED RAT 125I-VIP VIP Ala20 1.5 Igarashi H, et al., 2002 Jan 15, 2025 Jan 27, 2025
14781 D2 Striatal Membranes CALF 3H-Haloperidol HALOPERIDOL 1.5 Creese I, et al., 1976 Jan 15, 2025 Jan 15, 2025
70846 5-HT2A test test 3H- Ketanserin N-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride (3) 1.5 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
51390 M3 UNDEFINED HUMAN UNDEFINED {3-[(2-adamantan-1-yl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-dimethyl-amine 1.5 Sonda S et al., 2007 Jan 15, 2025 Jan 15, 2025
72127 nAChR CLONED HUMAN 3H-Epibatidine 2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 1.5 Magnus CJ et al 2019 Jan 15, 2025 Jan 29, 2025
19391 A3 CLONED HUMAN 3H-NECA 5 1.5 Klotz KN et al., 1999 Jan 15, 2025 Jan 15, 2025
66241 Ghrelin CLONED HUMAN 125I-ghrelin 6-[(Benzyloxy)methyl]-5-(4-{[(2-chloropyridin-4-yl)methyl]amino}phenyl)pyrimidine-2,4-diamine 1.5 Serby MD, et al., 2006 Jan 15, 2025 Jan 15, 2025
72130 nAChR CLONED HUMAN 3H-Epibatidine 2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 1.5 Magnus CJ et al 2019 Jan 15, 2025 Jan 29, 2025
11202 D2 STRIATUM RAT 3H-Haloperidol FLUSPIRILENE 1.5 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
56002 CB1 UNDEFINED HUMAN UNDEFINED 9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophenyl)-9H-purin-6-amine 1.5 Griffith DA et al., 2009 Jan 15, 2025 Jan 15, 2025
3780 MOR BRAIN GUINEA PIG 3H-DAMGO ETORPHINE - HCI 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
56005 CB1 UNDEFINED HUMAN UNDEFINED 9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine 1.5 Griffith DA et al., 2009 Jan 15, 2025 Jan 15, 2025
32714 5-HT2A CORTEX RAT 3H-KETANSERIN MIANSERIN 1.5 Wikstrom HV, et al., 2002 Jan 15, 2025 Jan 15, 2025
55244 OPRL1 UNDEFINED HUMAN UNDEFINED 3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 1.5 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
63437 Alpha1A CEREBRAL CORTEX RAT 3H-PRAZOSIN Y-931 1.5 Morimoto, T et al., 2002 Jan 15, 2025 Jan 28, 2025
9935 M2 CLONED RAT 3H-MQNB(-) Dexetimide 1.5 Kovacs, Yamamura, Waite, Varga, Roeske, 1998 Jan 15, 2025 Jan 15, 2025
18897 A3 CLONED HUMAN 3H-MRE 3008F20 MRE 3046F20 1.5 Gessi S et al., 2002 Jan 15, 2025 Jan 15, 2025
42450 D5 CLONED HUMAN 3H-SCH23390 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
63187 Beta2 CEREBELLUM RAT 125I-Pindolol ICI 118,551 1.5 Rainbow, TC et al., 1984 Jan 15, 2025 Jan 28, 2025
4052 DOR CLONED HUMAN 3H-DPDPE-Cl DELTORPHIN-II 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
24023 D4 CLONED HUMAN UNDEFINED THIORIDAZINE 1.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
60631 GABAA CLONED HUMAN FNZ DM-239 1.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
5848 Alpha2B LUNG NEONATAL RAT 3H-RAUWOLSCINE Tetrahydroalstonine 1.5 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
19160 HIPPOCAMPUS RAT 125I-PACAP(1-27) PACAP(1-27) 1.5 Gourlet P et al., 1991 Jan 15, 2025 Jan 15, 2025
32984 D2 CLONED HUMAN 3H-RACLOPRIDE CHLORPROMAZINE 1.5 Stormann TM, et al., 1990 Jan 15, 2025 Jan 15, 2025
4062 DOR CLONED HUMAN 3H-DPDPE-Cl ETORPHINE - HCI 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
10207 M2 CLONED RAT 3H-MQNB(-) ATR 1.5 Wei,Roeske,Lai,Wanibuchi,Hidaka,Usuda,Yamamura1992 Jan 15, 2025 Jan 15, 2025
65503 GABAA CLONED HUMAN [3H] Flunitrazepam DM-239 1.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
11490 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SPIROXATRINE 1.5 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
51938 MOR UNDEFINED HUMAN UNDEFINED BUPRENORPHINE 1.5 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
68582 D3 CLONED HUMAN 125I-IABN 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 1.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
13030 H1 BRAIN RAT 3H-MEPYRAMINE Pyrathiazine 1.5 Tran VT, et al., 1978 Jan 15, 2025 Jan 15, 2025
57834 KOR UNDEFINED HUMAN UNDEFINED 2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl-cyclohexyl)-acetamide 1.5 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
98031 SST3 CLONED HUMAN 125I-LTT-SRIF28 KE108 1.5 Reubi JC, et.al.,2002 Jan 15, 2025 Jan 15, 2025
56559 MOR UNDEFINED UNDEFINED UNDEFINED Naloxone(-) 1.5 Mathew SC et al., 2009 Jan 15, 2025 Jan 15, 2025
34544 nAChR CLONED RAT 3H-Epibatidine Cytisine 1.5 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
58096 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(3-Methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 1.5 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
40177 TNFα whole blood assay (WBA) HUMAN Functional 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 1.5 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40178 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 1.5 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
16627 Y5 CLONED HUMAN [125I] - Peptide YY NPY 1.5 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
53241 Alpha1D UNDEFINED HUMAN UNDEFINED 1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1.5 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
4090 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl DYNORPHIN(1-8)-OH 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
54266 CB1 UNDEFINED HUMAN UNDEFINED 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2,2-trifluoroethyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 1.5 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
101885 5-HT1A CLONED HUMAN [3H]-8-OH-DPAT Ziprasidone 1.5 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
6911 D4 CLONED HUMAN 3H-SPIPERONE THIORIDAZINE 1.5 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
51199 CHRNA4 UNDEFINED RAT UNDEFINED 2-(6-chloro-3-pyridinyl)-2,6-diazabicyclo[3.2.1]octane 1.5 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
65835 GABAA CLONED HUMAN [3H] Flunitrazepam XLi351 C21H21ClN2OSi 1.507 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
60637 GABAA CLONED HUMAN FNZ XLi351 1.507 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
58112 5-HT2A CLONED HUMAN 125I-DOI N-(2-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine hydrochloride 1.51 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
4865 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 1.51 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
8474 SST3 CLONED HUMAN 125I-LTT-SRIF28 CGP 23996 1.51 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
539 5-HT1A HIPPOCAMPUS RAT 125I-BH-8-MeO-N-PA SPIROXATRINE 1.51 GOZLAN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12327 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 15931 1.51 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
3923 5-HT6 CLONED RAT 3H-LSD METHIOTHEPIN 1.51 BOESS FG, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
2904 5-HT2A CORTEX RAT 125I-LSD LSD, IODO 1.51 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
17006 NOP CLONED HUMAN Leucyl-3H-NC J-113397 1.51 Hashiba E, et al., 2001 Jan 15, 2025 Jan 15, 2025
2703 5-HT2A CORTEX RAT 3H-SPIPERONE PROPERICIAZINE 1.51 LEYSEN ET AL., 1978 Jan 15, 2025 Jan 15, 2025
15827 5-HT7 CLONED RAT 3H-5HT 5-Hydroxy Tryptamine 1.51 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
89641 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.51356 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
63580 Alpha2A Ovary HAMSTER 3H-RX821002 RX811059 1.51356 Pauwels, Petrus J. et. al, 2003 Jan 15, 2025 Jan 28, 2025
32349 M4 LUNG RABBIT 3H-NMS Dicyclomine 1.51356 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
28775 SST3 CLONED HUMAN 125I-LTT-SRIF28 CGP 23996 1.51356 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
27511 5-HT1B STRIATUM GUINEA PIG 3H-GR-125743 DHE 1.51356 Millan MJ, et al., 2002a Jan 15, 2025 Jan 15, 2025
39827 5-HT2C CLONED HUMAN 3H-MESULERGINE MIANSERIN 1.51356 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39589 5-HT2A CLONED HUMAN Functional DOB 1.51356 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
99594 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine 1.52 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
7451 BB2 CELLS MOUSE 125I-[DTyr6,BetaAla11,Phe13,Nle14]Bn(6-14) GRP 1.52 Katsuno T, et al., 1999 Jan 15, 2025 Jan 15, 2025
7730 GABAA CLONED RAT 3H-FMZ flumazenil 1.52 Renard S, et al., 1999 Jan 15, 2025 Jan 27, 2025
12413 D3 CLONED RAT 125I-NCQ 298 PIMOZIDE 1.52 Boundy VA, et al., 1993 Jan 15, 2025 Jan 15, 2025
9349 GABAA CEREBRAL CORTEX Newborn rats FNZ Flunitrazepam 1.52 Giorgi,Lecca,Cancedda,Giuliana,Corda,1995 Jan 15, 2025 Jan 15, 2025
22428 A2B CLONED HUMAN 3H-ZM241385 28 1.52 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
47056 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-03I 1.52 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
7633 GABAA CLONED RAT 3H-FMZ flumazenil 1.52 Renard S, et al., 1999 Jan 15, 2025 Jan 27, 2025
4320 5-HT7 CLONED RAT 3H-5HT 5-Hydroxy Tryptamine 1.52 SHEN Y, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
11520 KOR CEREBELLUM GUINEA PIG 3H-U69,593 Spiradoline 1.53 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
4873 5-HT2B CLONED HUMAN 3H-5HT LY 53857 1.53 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
18954 H1 CLONED GUINEA PIG 3H-MEPYRAMINE trans-H2-PAT(+/-) 1.53 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
18970 H1 CLONED HUMAN 3H-MEPYRAMINE Triprolidine 1.53 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
38442 D5 CLONED HUMAN 3H-SCH23390 MCL-202 1.53 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
70191 BRAIN Zebrafish 3H-Diprenorphine Dynorphin A 1.53 Gonzalez-Nunez V, et al., 2006 Jan 15, 2025 Jan 15, 2025
14713 LUNG GUINEA PIG 3H-LTD4 LTE4 1.53 Shirley JT and Cheng JB, 1991 Jan 15, 2025 Jan 15, 2025
25472 SLC6A3 CLONED HUMAN 3H-WIN 35,428 pdspTestCompound1 1.53 MM Goodman, et. al., 2000 Jan 15, 2025 Jan 15, 2025
2459 5-HT3 AREA POSTREMA RAT 3H-GR-65630 ONDANSETRON 1.53 Kilpatrick et al., 1989 Jan 15, 2025 Jan 15, 2025
60081 A3 CLONED HUMAN 125I-AB-MECA (1S,2R,3S,4R,5S)-4-(6-(cyclobutylamino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide 1.53 Tosh, Dipip et. al., 2015 Jan 15, 2025 Jan 15, 2025
27078 MOR BRAIN MOUSE 3H-DAMGO Tyr-d-Ala-Phe-Phe-NH2 1.53 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
2299 5-HT3 CORTEX RAT 3H-ICS 205-930 DAU 6287 1.53 GIRALDO ET AL., 1989 Jan 15, 2025 Jan 15, 2025
65556 GABAA CLONED HUMAN [3H] Flunitrazepam FG8205 1.54 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65566 GABAA CLONED HUMAN [3H] Flunitrazepam Alprazolam 1.54 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
55091 H3 UNDEFINED HUMAN UNDEFINED {3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine 1.54 von Coburg Y et al., 2009 Jan 15, 2025 Jan 15, 2025
60525 GABAA CLONED HUMAN FNZ FG 8205 1.54 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
138 5-HT1A HIPPO:LESIONED RAT 3H-WB4101 5-Hydroxy Tryptamine 1.54 MORROW ET AL., 1985 Jan 15, 2025 Jan 15, 2025
60559 GABAA CLONED HUMAN FNZ Alprazolam 1.54 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
5046 5-HT2B CLONED HUMAN 3H-5HT CYPROHEPTADINE 1.54 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
5057 5-HT2B CLONED HUMAN 3H-5HT METHIOTHEPIN 1.54 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
59330 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Fluoro-5-(4-fluoro-3-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 1.54 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
29127 SST3 CLONED HUMAN 125I-LTT-SST-28 BIM 23068 1.54 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
18929 H1 CLONED HUMAN 3H-trans-H2-PAT,(-) CLOZAPINE 1.54 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
2346 5-HT3 NG108-15 NG 3H-ICS 205-930 ICS 205-930 1.55 NEIJT ET AL, 1988 Jan 15, 2025 Jan 15, 2025
15933 CB2 CLONED MOUSE 3H-CP-55940 JTE-907 1.55 Iwamura H, et al., 2000 Jan 15, 2025 Jan 15, 2025
41341 CLONED HUMAN UNDEFINED SKF 64139 1.55 Wu Q, et al., 2005 Jan 15, 2025 Jan 15, 2025
29126 SST2 CLONED HUMAN 125I-LTT-SST-28 BIM 23068 1.55 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
14582 CB1 BRAIN RAT 3H-CP-55940 XVI 1.55 Compton DR, et al., 1993 Jan 15, 2025 Jan 15, 2025
14623 CB1 BRAIN RAT 3H-CP-55940 DMHP, 1', 2' 1.56 Compton DR, et al., 1993 Jan 15, 2025 Jan 15, 2025
65832 GABAA CLONED HUMAN [3H] Flunitrazepam XLi352 C18H13ClN2O 1.56 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
94534 A1 C.H.O. test 3H-CCPA 2-chloro-5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine 1.56 Petrelli R et al 2018 Jan 15, 2025 Jan 15, 2025
60638 GABAA CLONED HUMAN FNZ XLi352 1.56 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
10052 MOR BRAIN MOUSE 125I-Endomorphin-1 Endomorphin 2 1.57 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
59269 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-methyl-7-azabicyclo[2.2.1]heptane 1.57 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
99718 D3 CLONED RAT [3H]spiperone (S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol 1.57 Luo D et al 2016 Jan 15, 2025 Jan 28, 2025
61320 GABAA CLONED HUMAN FNZ JYI-04 1.57 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
59281 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methoxyphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 1.57 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
2993 5-HT2A FR. CORTEX RAT 3H-KETANSERIN MIANSERIN 1.57 LEYSEN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
7603 Alpha2B CLONED HUMAN 3H-MK912 SPIROXATRINE 1.57 Uhlen S, et al., 1994 Jan 15, 2025 Jan 15, 2025
65762 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-04 (C12H23N3O3) 1.57 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65292 GABAA CLONED HUMAN [3H] Flunitrazepam XLI-348 1.578 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
61134 GABAA CLONED HUMAN FNZ XLI-348 1.578 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
15366 5-HT1B CLONED HUMAN 3H-5HT 5-CT 1.58 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
5397 5-HT2C CLONED HUMAN 3H-MESULERGINE METHYSERGIDE 1.58 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
8981 SST2 CLONED HUMAN 125I-SRIF-28 RC 160II 1.58 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
10779 D2 CLONED RAT 3H-LSD CLOROTEPINE (+) 1.58 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
5410 5-HT2C CLONED RAT 3H-MESULERGINE RITANSERIN 1.58 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
10788 D2 CLONED RAT 3H-LSD RISPERIDONE 1.58 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
2860 5-HT2A CORTEX RAT 125I-LSD KETANSERIN 1.58 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
12336 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SDZ 216,525 1.58 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
11834 Alpha2A CLONED HUMAN 3H-RX821002 PHENTOLAMINE 1.58 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
9019 SST5 CLONED HUMAN 125I-SRIF-28 BIM 23052 1.58 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
829 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.58 HOYER, 1988 or 9 (book) Jan 15, 2025 Jan 15, 2025
11842 Alpha2C CLONED HUMAN 3H-RX821002 Fluparoxan 1.58 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
54596 A2B UNDEFINED HUMAN UNDEFINED 1-Ethyl-8-(4-(4-(4-methylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1.58 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
15433 5-HT1B CLONED RAT 125I-ICYP RU 24969 1.58 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
54109 KOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-isoquinolyl)acetamido]morphinan 1.58 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
11879 5-HT2A CLONED HUMAN 3H-KETANSERIN MIANSERIN 1.58 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
12906 LUNG RAT 3H-RAUWOLSCINE ARC-239 1.58 O'Rourke MF, et al., 1993 Jan 15, 2025 Jan 15, 2025
18548 M1 CLONED HUMAN 3H-NMS TRIPITRAMINE 1.58 Maggio R et al., 1994 Jan 15, 2025 Jan 15, 2025
11893 D3 CLONED HUMAN 3H-SPIPERONE 7-OH-DPAT 1.58 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
41845 H3 CLONED RAT 3H-Alpha-Me-histamine (6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 1.58 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
6774 Y2 CLONED HUMAN 125I-PYY NPY2-36, human 1.58 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
12678 KOR BE(2)-C HUMAN 3H-NalBzoH Mr2266 1.58 Standifer KM, et al., 1994 Jan 15, 2025 Jan 27, 2025
8590 SST2 CLONED MOUSE 125I-Tyr11-SRIF BIM 23014 1.58 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
2981 5-HT2A CORTEX PIG 3H-KETANSERIN METITEPIN 1.58 HOYER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
2982 5-HT2A CORTEX RAT 125I-LSD METITEPIN 1.58 ENGEL ET AL, 1984 Jan 15, 2025 Jan 15, 2025
6310 5-HT7 CORTEX GUINEA PIG 3H-5CT 5-Methoxytryptamine 1.58 TO ZP, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
12223 BRAIN HUMAN UNDEFINED CLOZAPINE 1.58 Richelson E., 1988 Jan 15, 2025 Jan 15, 2025
8664 SST5 CLONED RAT 125I-Tyr11-SRIF RC 160 1.58 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
5337 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 RS 67506 1.58 EGLEN RM, ET AL, 1995 Jan 15, 2025 Jan 15, 2025
15579 5-HT2A CLONED HUMAN 3H-DOI DOI 1.58 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
5373 5-HT2A CLONED RAT 3H-KETANSERIN METHYSERGIDE 1.58 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
69138 H3 CLONED HUMAN 3H-Histamine Imetit 1.58489 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
68885 SST3 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Ala-Phe-Thr-Ser-Cys}-NH2 1.58489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
32033 5-HT2B CLONED HUMAN 3H-5HT MIANSERIN 1.58489 Bonhaus, DW et. al., 1999 Jan 15, 2025 Jan 15, 2025
68905 SST3 CLONED HUMAN 125I-SRIF Cyclo[HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe] 1.58489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
97848 5-HT2C Membranes HUMAN 3H-MESULERGINE ACP-103 1.58489 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
68923 SST1 CLONED HUMAN 125I-SRIF Cyclo[(diaminoethylcarbamoyl)HyPro-Tyr-D-Trp-Lys-Tyr(Bzl)-Phe] 1.58489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
39996 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C14H15FN2·C4H4O4 1.58489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
68938 SST1 CLONED HUMAN 125I-SRIF Cyclo[(N,N-dimethyldiaminoethylcarbamoyl)HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe 1.58489 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
40279 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.58489 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
86624 5-HT2A CLONED HUMAN 3H-KETANSERIN METHYSERGIDE 1.58489 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
63351 Y5 CLONED HUMAN 125I-PYY CGP 71683A 1.58489 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
31370 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE METERGOLINE 1.58489 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
24753 Y2 CLONED HUMAN 125I-PYY NPY2-36, human 1.58489 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
31423 5-HT7 CLONED RAT 125I-LSD 5-Methoxytryptamine 1.58489 Eglen RM et al., 1997 Jan 15, 2025 Jan 27, 2025
69313 D3 CLONED HUMAN 125I-IODOSULPRIDE trans-3-(2-(4-((3-(3-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine 1.58489 Macdonald G, et al., 2003 Jan 15, 2025 Jan 15, 2025
34762 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methylthio-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 1.58489 Bromidge SM, et al., 2000 Jan 15, 2025 Jan 15, 2025
69326 D3 CLONED HUMAN 125I-IODOSULPRIDE trans-3-(2-(4-((3-(2-Cyanophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine 1.58489 Macdonald G, et al., 2003 Jan 15, 2025 Jan 15, 2025
99342 D3 CLONED HUMAN [3H]N-methylspiperone 1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2-methoxyphenyl)piperazine 1.59 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
14624 CB1 BRAIN RAT 3H-CP-55940 THC-DMH 1.59 Compton DR, et al., 1993 Jan 15, 2025 Jan 15, 2025
5486 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 1.59 WAINSCOTT DB, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
12663 MOR BE(2)-C HUMAN 3H-DAMGO TAPS 1.59 Standifer KM, et al., 1994 Jan 15, 2025 Jan 15, 2025
38281 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N-Dimethyl-2-(2'-aminophenylthio)benzylamine 1.59 Jarkas N, et al., 2005 Jan 15, 2025 Jan 15, 2025
56042 MOR UNDEFINED UNDEFINED UNDEFINED (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-3-carboxylate 1.59 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
51456 Alpha1A UNDEFINED HUMAN UNDEFINED 2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 1.6 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
35842 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 1.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
24839 Alpha1A CLONED HUMAN 125I-HEAT CLOZAPINE 1.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
51465 Alpha1A UNDEFINED HUMAN UNDEFINED 5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 1.6 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
16650 M1 CLONED HUMAN 3H-QNB Trihexyphenidyl 1.6 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
2317 5-HT3 ENTO CORTEX RAT 3H-GR-65630 GR 65630 1.6 Kilpatrick et al., 1987 Jan 15, 2025 Jan 15, 2025
6413 5-HT3 CLONED RAT 3H-BIMU-1 ICS 205-930 1.6 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
51213 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-chloro-5-hydroxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane 1.6 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
27150 5-HT2A BRAIN RAT 125I-DOI 5-HT, alpha,Omega-dimethyl 1.6 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
6416 5-HT3 CLONED RAT 3H-BIMU-1 BIMU 1 1.6 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
65040 H1 BRAIN GUINEA PIG 3H-MEPYRAMINE AMITRIPTYLINE 1.6 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
71954 D4 test test 3H-N-Methylspiperone 8-(4-(1H-Indol-3-yl)butyl)-1-phenyl-1,3,8-triazaspiro[4.5] decan-4-one 1.6 Etukala JR et al 2016 Jan 15, 2025 Jan 28, 2025
96786 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.6 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
9235 SST2 CLONED MOUSE 125I-MK-678 BIM 23014 1.6 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
51475 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 1.6 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
12564 LIVER RAT 125I-Angiotensin II Saralasin 1.6 Keiser JA, et al., 1995 Jan 15, 2025 Jan 15, 2025
56852 CB1 UNDEFINED HUMAN UNDEFINED Rimonabant 1.6 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
30486 M2 CLONED HUMAN 3H-QNB 3-Ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 1.6 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
51222 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-methyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 1.6 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
65815 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-13 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
42266 CLONED HUMAN 125I-Motilin Delta 26-28 1.6 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
47903 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
38688 UNDEFINED HUMAN 3H-hypoxanthine Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(3-thiophen-3-yl-benzyloxymethyl)-propylcarbamoyl]-2-methyl-propyl}-amide 1.6 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
65570 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-082 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
93986 D3 CLONED HUMAN 3H-SPIPERONE 7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one 1.6 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
35876 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(2-phenoxyethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 1.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
56100 MOR UNDEFINED HUMAN UNDEFINED Nalbuphine 1.6 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
57385 CB1 UNDEFINED HUMAN UNDEFINED N-Cyclohexyl-4-[(2,4-dichlorophenyl)(phenyl)methyl]-piperazine-1-carboxamide 1.6 Meng T et al., 2010 Jan 15, 2025 Jan 15, 2025
33835 STRIATUM RAT 3H-RX821002 Brimonidine GTP 1.6 Bylund DB, et al., 2001 Jan 15, 2025 Jan 15, 2025
11820 FR. CORTEX HUMAN 3H-RAUWOLSCINE YOHIMBINE 1.6 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
56364 CHRNA4 UNDEFINED RAT UNDEFINED 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine 1.6 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
2861 5-HT2A CORTEX RAT 3H-MESULERGINE KETANSERIN 1.6 CLOSSE, 1983 Jan 15, 2025 Jan 15, 2025
98094 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide 1.6 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
11056 H3 CLONED HUMAN 3H-methylhistamine Immepip 1.6 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
36656 H1 CLONED HUMAN 3H-PYRILAMINE mirtazepine 1.6 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
50485 5-HT2A CORTEX RAT 125I-DOI SPIPERONE 1.6 MCKENNA & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
24119 VPAC1 T47D HUMAN 125I-VIP Vasoactive intestinal polypeptide 1.6 Igarashi H, et al., 2002 Jan 15, 2025 Jan 15, 2025
16442 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE YOHIMBINE 1.6 Naselsky DP, et al., 2001 Jan 15, 2025 Jan 15, 2025
37179 Y5 BRAIN RAT 125I-hPP CP732925 1.6 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
5948 Alpha2B LUNG RAT 3H-RAUWOLSCINE ARC-239 1.6 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
9533 SLC6A4 CLONED HUMAN 3H-CITALOPRAM Fluvoxamine 1.6 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
23357 A1 BRAIN BOVINE 3H-DPCPX R-PIA 1.6 Klotz KN et al., 1991 Jan 15, 2025 Jan 27, 2025
8000 GABAA CLONED HUMAN 3H-RO-15-1788 24 1.6 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
58944 D2 CLONED HUMAN 3H-N-Methylspiporone 4-[5-trans-hydroxy-5-cis-(4′-chlorophenyl)-2-azabicyclo[3.2.1]octanyl]-4″-fluorobutyrophenone 1.6 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
23873 D2 CLONED HUMAN UNDEFINED SERTINDOLE 1.6 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
60996 GABAA CLONED HUMAN FNZ XHE-III-13 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
85573 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate 1.6 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
28998 SST3 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 1.6 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
9799 retina RABBIT 3H-Dopamine release 4-P-ADOT 1.6 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
32844 D4 STRIATUM CANINE 3H-SPIPERONE OCTOCLOTHEPIN-R 1.6 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
53836 5-HT1A UNDEFINED RAT UNDEFINED 2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole 1.6 Siracusa MA et al., 2008 Jan 15, 2025 Jan 15, 2025
17486 PANCREAS GUINEA PIG 125I-VIP VIP Ala9 1.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
51278 SLC6A4 UNDEFINED RAT UNDEFINED 7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 1.6 Keith JM et al., 2007 Jan 15, 2025 Jan 15, 2025
54350 CB2 UNDEFINED HUMAN UNDEFINED N-(Adamant-1-yl)-4-oxo-1-pentyl-7-(phenylthio)-1,4-dihydroquinoline-3-carboxamide 1.6 Pasquini S et al., 2008 Jan 15, 2025 Jan 15, 2025
10832 D3 CLONED HUMAN 125I-IODOSULPRIDE 7-OH-DPAT 1.6 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
35921 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 2,2-Dimethyl-propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 1.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
53585 SLC6A4 UNDEFINED RAT UNDEFINED 3-{4-[(1,4-cis)-4-(1H-Indol-4-yl)-pipera-zinyl-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 1.6 Zhou D et al., 2008 Jan 15, 2025 Jan 15, 2025
58962 Alpha1A CLONED HUMAN 3H-PRAZOSIN CLOZAPINE 1.6 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
3667 MOR BRAIN GUINEA PIG 3H-DAMGO ETONITAZENE 1.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
72531 DAT CLONED HUMAN 3H-WIN 35,428 sakurantin 1.6 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
23891 D2 CLONED HUMAN 3H-RACLOPRIDE RACLOPRIDE 1.6 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
5717 Alpha2C KIDNEY OPOSSUM 3H-RAUWOLSCINE WB 4101 1.6 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
6741 D2 CLONED HUMAN 3H-RACLOPRIDE RISPERIDONE 1.6 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
94037 Alpha1A CORTEX PIG 3H-PRAZOSIN 3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 1.6 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
68438 H1 CLONED HUMAN [11C]R107474 mirtazapine 1.6 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
65111 GABAA CLONED HUMAN [3H] Flunitrazepam TG-II-82 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
4696 5-HT1D CLONED HUMAN 3H-5HT 5-CT 1.6 WEINSHANK RL, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
6746 D2 CLONED HUMAN 3H-RACLOPRIDE THIORIDAZINE 1.6 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
15194 LUNG RAT 3H-RAUWOLSCINE PIPEROXAN 1.6 Boyajian CL, et al., 1987 Jan 15, 2025 Jan 15, 2025
23898 D2 CLONED HUMAN 3H-RACLOPRIDE Trifluperazine 1.6 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
55899 MOR UNDEFINED HUMAN UNDEFINED 3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 1.6 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
67682 A2A STRIATUM RAT 3H-CGS21680 N-Ethyl-l-deoxy-1-[6-amino-2-(3-phenyl-l-propyn-lyl)-9H-purin-9-yI]-beta-D-ribofuranuronamide 1.6 Cristalli G, et al., 1994 Jan 15, 2025 Jan 15, 2025
31589 D1 Striatal Membranes RAT 3H-SCH23390 C22H27ClN2 1.5maleate (38) 1.6 Bogeso, K.P., et al., 1995 Jan 15, 2025 Jan 15, 2025
2665 5-HT2A CORTEX RAT 3H-KETANSERIN SPIPERONE 1.6 GLASER & TRABER, 1985 Jan 15, 2025 Jan 15, 2025
2666 5-HT2A CORTEX RAT 3H-KETANSERIN SPIPERONE 1.6 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
19818 D4 CLONED HUMAN 3H-Olanzapine OLANZAPINE 1.6 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
100970 D2 CLONED HUMAN 3H-Methylspiperone ARIPIPRAZOLE 1.6 Snyder et al., 2015 Jan 15, 2025 Jan 28, 2025
59242 CLONED RAT 3H-5HT 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-6-fluoro-1H-indole 1.6 Smid P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59755 D2 CLONED HUMAN 3H-N-Methylspiporone 4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)-1-butanone 1.6 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
65645 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-III-13 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
17773 CLONED RAT 125I-VIP VIP [D-Leu23] 1.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
33901 D1 STRIATUM RAT 125I-SCH 23982 (1R,3S)-1-(Aminomethyl)-3,4-dihydro-5,6-dihydroxy-3-phenyl-1H-2-benzopyran Hydrochloride 1.6 DeNinno MP, et al., 1991 Jan 15, 2025 Jan 27, 2025
20078 A1 BRAIN RAT 3H-PIA 1-deaza-2-Cl-CPA (2b) 1.6 Cristalli G et al., 1988 Jan 15, 2025 Jan 15, 2025
58224 Alpha1A CLONED HUMAN 3H-PRAZOSIN CLOZAPINE 1.6 Chen X, et al., 2015 Jan 15, 2025 Jan 15, 2025
71794 Sigma 2 test test 3H-DTG Cimbiâ€701 1.6 LEstrade Elina T et al 2019 Jan 15, 2025 Jan 28, 2025
94068 5-HT2A CLONED HUMAN [3H]-ketanserin 2,5-dimethoxy-4-benzylthiophenethylamine 1.6 Luethi D et al 2018 Jan 15, 2025 Jan 15, 2025
19831 D4 CLONED HUMAN UNDEFINED FLUPENTHIXOL, Alpha 1.6 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
20344 CEREBRAL CORTEX RAT 3H-CCK8 Caerulein 1.6 Van Dijk A et al., 1984 Jan 15, 2025 Jan 15, 2025
19833 D4 CLONED HUMAN 3H-Clozapine CLOZAPINE 1.6 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
100217 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Blonanserin 1.6 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
101498 H2 CLONED HUMAN [3H]Tiotidine Asenapine 1.6 PDSP Certified Data Mar 20, 2025 Mar 20, 2025
3712 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl BUPRENORPHINE 1.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18306 D2 BRAIN RAT 3H-domperidone ETICLOPRIDE 1.6 Hall H et al., 1986 Jan 15, 2025 Jan 27, 2025
62854 Brain Frontal Cortex HUMAN 3H-RAUWOLSCINE YOHIMBINE 1.6 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 15, 2025
14983 D3 CLONED HUMAN 3H-RACLOPRIDE SERTINDOLE 1.6 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
39559 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1.6 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
48007 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
23689 SLC6A4 CLONED HUMAN 3H-CITALOPRAM CITALOPRAM 1.6 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
36747 5-HT2A CLONED HUMAN 125I-R091150 (+)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 1.6 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
98445 5-HT7 CLONED HUMAN [3H]-LSD 2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one, 1.6 Ofon E et al 2016 Jan 15, 2025 Jan 15, 2025
34191 D2 STRIATUM RAT 3H-domperidone BUTACLAMOL,(+) 1.6 Grandy DK, et al., 1989 Jan 15, 2025 Jan 15, 2025
19346 NK3 CLONED GUINEA PIG 125I-[MePhe7]-NKB SB 235375 1.6 Hay DW et al., 2002 Jan 15, 2025 Jan 15, 2025
36754 NET CLONED RAT 3H-Nisoxetine (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 1.6 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39062 D2 CLONED HUMAN R-SAT Sultopride 1.6 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
34967 nAChR CLONED UNDEFINED 3H-Epibatidine 5-(1-Ethynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 1.6 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
15002 5-HT7 CLONED MOUSE 3H-5HT RISPERIDONE 1.6 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
3746 MOR CLONED HUMAN 3H-DAMGO Beta-Endorphin 1.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
47522 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY CP732925 1.6 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
17573 PANC1 HUMAN 125I-VIP VIP Ala8 1.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
90021 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
11174 5-HT7 CLONED MOUSE 3H-5HT RISPERIDONE 1.6 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
2983 5-HT2A CORTEX RAT 3H-KETANSERIN METITEPIN 1.6 PAZOS ET AL, 1984 Jan 15, 2025 Jan 15, 2025
99752 DOR CLONED HUMAN 3H-DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl] propyl}-Nmethylpropanamide 1.6 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
39084 D3 CLONED HUMAN R-SAT BUTACLAMOL 1.6 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
55471 D2 UNDEFINED HUMAN UNDEFINED 4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 1.6 Sikazwe DM et al., 2009 Jan 15, 2025 Jan 15, 2025
29365 CCR5 CLONED RAT 3H-Epibatidine Lobeline 1.6 Jensen AA, et al., 2003 Jan 15, 2025 Jan 15, 2025
17590 T47D HUMAN 125I-VIP Vasoactive intestinal polypeptide 1.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
3511 5-HT2A CLONED RAT 3H-KETANSERIN KETANSERIN 1.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
65720 GABAA CLONED HUMAN [3H] Flunitrazepam TG-4-39 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
100281 5-HT2C CLONED HUMAN 3H-MESULERGINE SERTINDOLE 1.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
51129 Alpha1D UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide 1.6 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
186 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 8-OH-DPAT 1.6 COSSERY ET AL.,1986 Jan 15, 2025 Jan 15, 2025
79036 5-HT2B CLONED HUMAN 3H-LSD (±)-4-Ethylthio-2,5-dimethoxyamphetamine 1.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
7872 GABAA CLONED HUMAN 3H-RO-15-1788 3 1.6 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
52420 SLC6A4 UNDEFINED RAT UNDEFINED 7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 1.6 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
63428 5-HT2A CEREBRAL CORTEX RAT 125I-DOI OLANZAPINE 1.6 Morimoto, T et al., 2002 Jan 15, 2025 Jan 15, 2025
51909 D3 UNDEFINED HUMAN UNDEFINED (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-imidazo[1,2-a]pyridine 1.6 Leopoldo M et al., 2007 Jan 15, 2025 Jan 15, 2025
13766 SLC6A3 STRIATUM RAT 3H-GBR 12,935 BINDING GBR-12935 1.6 Garreau L, et al., 1997 Jan 15, 2025 Jan 15, 2025
55238 OPRL1 UNDEFINED HUMAN UNDEFINED 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 1.6 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
56006 CB1 UNDEFINED HUMAN UNDEFINED 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine 1.6 Griffith DA et al., 2009 Jan 15, 2025 Jan 15, 2025
51143 Alpha1D UNDEFINED HUMAN UNDEFINED 5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 1.6 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
24008 D4 CLONED HUMAN UNDEFINED CLOZAPINE 1.6 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
56522 CB2 UNDEFINED HUMAN UNDEFINED (R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide 1.6 Silvestri R et al., 2009 Jan 15, 2025 Jan 15, 2025
70092 5-HT3 CORTICAL MEMBRANES RAT 3H-GR-65630 ONDANSETRON 1.6 Van Wijingaarden, I. et, al. 1993 Jan 15, 2025 Jan 15, 2025
24014 D4 CLONED HUMAN UNDEFINED OLANZAPINE 1.6 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
39118 D3 CLONED HUMAN R-SAT RISPERIDONE 1.6 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
55760 5-HT1A UNDEFINED UNDEFINED UNDEFINED 2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine 1.6 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
55761 5-HT1F UNDEFINED HUMAN UNDEFINED 4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-benzamide 1.6 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
53714 D2 UNDEFINED HUMAN UNDEFINED 4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 1.6 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
18643 D3 CLONED RAT 3H-RACLOPRIDE SERTINDOLE 1.6 Strange PG 2001 Jan 15, 2025 Jan 15, 2025
28883 SST2 CLONED RAT 125I-Tyr11-somatostatin DC-25-100 1.6 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
14293 SLC6A3 STRIATUM RAT 3H-DA UPTAKE PTT(-) 1.6 Letchworth SR, et al., 2000 Jan 15, 2025 Jan 15, 2025
18647 Platelet membrane HUMAN 3H-PGD2 S-5751 1.6 Arimura A et al., 2001 Jan 15, 2025 Jan 15, 2025
17627 CLONED RAT 125I-VIP VIP Ala17 1.6 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
37083 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Lecozotan 1.6 Schechter LE, et al., 2005 Jan 15, 2025 Jan 15, 2025
45531 NMDA CLONED HUMAN 3H-Glycine 2-Chloro-4-hydroxy-3-methoxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 1.6 Buchstaller HP, et al., 2006 Jan 15, 2025 Jan 28, 2025
67553 nAChR FOREBRAIN RAT 3H-Epibatidine (1R)-2-(3-Pyridinyl)-8-azabicyclo[3/2/1]oct-2-ene 1.6 Gohlke, H et al., 2003 Jan 15, 2025 Jan 15, 2025
37092 AChE serum BOVINE Functional N,N-Bis[3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl]-N-allylamine 1.6 Campiani G, et al., 2005a Jan 15, 2025 Jan 15, 2025
62692 SST2 COLON RAT UNKNOWN (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 1.6 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
60646 GABAA CLONED HUMAN FNZ TG-4-39 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60647 GABAA CLONED HUMAN FNZ TG-II-82 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
5865 Alpha2B LUNG NEONATAL RAT 3H-RAUWOLSCINE ARC-239 1.6 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
40172 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 1.6 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
53229 Alpha1D UNDEFINED HUMAN UNDEFINED 1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1.6 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
4078 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl Leu-ENKEPHALIN 1.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
98030 SST4 CLONED HUMAN 125I-LTT-SRIF28 KE108 1.6 Reubi JC, et.al.,2002 Jan 15, 2025 Jan 15, 2025
41966 GABAA CLONED HUMAN 3H-RO-15-1788 3-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine 1.6 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
4079 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl Beta-Endorphin 1.6 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
99823 DOR CLONED HUMAN [3H]DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 1.6 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
54256 CB1 UNDEFINED HUMAN UNDEFINED Rimonabant 1.6 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
6897 D4 CLONED HUMAN 3H-SPIPERONE CLOZAPINE 1.6 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
49137 DOR CLONED HUMAN 35S-GTPGammaS DPDPE 1.6 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
60660 GABAA CLONED HUMAN FNZ QH-II-082 1.6 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
1781 5-HT2A CORTEX HUMAN 3H-KETANSERIN CLOZAPINE 1.6 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
63480 D3 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 1.6 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
17407 NOP BRAIN MOUSE 125I-Tyr14-OFQ OFQ/N (1-11),[Tyr10] 1.6 Mogil JS, Pasternak GW., 2001 Jan 15, 2025 Jan 15, 2025
94536 A1 C.H.O. test 3H-CCPA 2-chloro-5′-chloro-5′-deoxyN6 -(±)-endo-norbornyl-adenosine 1.61 Petrelli R et al 2018 Jan 15, 2025 Jan 15, 2025
8715 SST2 CLONED HUMAN 125I-Tyr3-octreotide L-362,855 1.62 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
99612 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1.62 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
60193 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-(Benzofuran-2-ylethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1.62 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
58160 5-HT2C CLONED HUMAN 125I-DOI N-(3-Bromobenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 1.62 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
830 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
831 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
832 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
833 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 HOYER & KARPF, 1988 Jan 15, 2025 Jan 15, 2025
834 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 HOYER, 1988 Jan 15, 2025 Jan 15, 2025
835 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 HOYER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
836 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.62 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
5452 5-HT4B CLONED HUMAN 3H-GR-113808 ML10375 1.62 BLONDEL O, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
65144 GABAA CLONED HUMAN [3H] Flunitrazepam CM-A87 1.62 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
8351 SST2 CLONED HUMAN 125I-Tyr10-CST14 L-362,855 1.62 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
68799 5-HT3 NG108-15 PIG 3H-DAU 6215 ZACOPRIDE,R 1.62 Schiavi, GB et al., 1994 Jan 15, 2025 Jan 15, 2025
8387 SST2 CLONED HUMAN 125I-Tyr3-octreotide L-362,855 1.62 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
15339 5-HT1D CLONED Dog 3H-5HT SUMATRIPTAN 1.62 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
8687 SST2 CLONED HUMAN 125I-Tyr3-octreotide L-362,855 1.62 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
60657 GABAA CLONED HUMAN FNZ CM-A87 1.62 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60414 GABAA CLONED HUMAN FNZ CM-A-87 1.62 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
68377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
28788 SST2 CLONED HUMAN 125I-Tyr10-CST14 L-362,855 1.62181 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
42109 Alpha2B CLONED HUMAN 35S-GTPGammaS RX821002 1.62181 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
64127 D2 CLONED HUMAN 3H-N-Methylspiperone Trifluperazine 1.62181 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
39828 5-HT2C CLONED HUMAN 3H-MESULERGINE RITANSERIN 1.62181 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
26791 GAL2 CLONED HUMAN 125I-GALANIN Galanin rat 1.62181 Borowsky Beth, et. al., 1998 Jan 15, 2025 Jan 15, 2025
18656 H3 CLONED HUMAN 3H-Alpha-Me-histamine Imetit 1.62181 Wieland K et al., 2001 Jan 15, 2025 Jan 15, 2025
32240 M1 CORTEX RAT 3H-PIRENZEPINE Cyclopentolate 1.62181 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
60434 GABAA CLONED HUMAN FNZ WY-TSC-4 1.63 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65575 GABAA CLONED HUMAN [3H] Flunitrazepam WY-TSC-4 (WYS8) 1.63 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
37185 BRAIN RAT 3H-14-methoxymetopon NALOXONE 1.63 Spetea M.,et.al.,2003 Jan 15, 2025 Jan 15, 2025
5489 5-HT2B CLONED HUMAN 3H-5HT LY 53857 1.63 WAINSCOTT DB, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
55665 AChE UNDEFINED HUMAN UNDEFINED 1,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene 1.63 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
13225 BRAIN RAT 3H-CLONIDINE IDAZOXAN 1.63 Boyajian CL, et al., 1987 Jan 15, 2025 Jan 15, 2025
14256 D3 CLONED RAT 3H-SPIPERONE DM 1451 1.63 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 15, 2025
18931 H1 CLONED HUMAN 3H-MEPYRAMINE CLOZAPINE 1.63 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
65618 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-60 (C17H11N2OF) 1.635 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
60819 GABAA CLONED HUMAN FNZ JYI-60 1.635 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
4869 5-HT2B CLONED HUMAN 3H-5HT RITANSERIN 1.64 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
51974 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 1.64 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
101205 MOR CLONED HUMAN 3H-Diprenorphine (S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperidin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate 1.64 Henry S,et al., 2021 Jan 15, 2025 Jan 28, 2025
10856 M2 BRAINSTEM RAT 3H-QNB ATR 1.64 McKinney M, ET AL., 1989 Jan 15, 2025 Jan 15, 2025
2667 5-HT2A CORTEX RAT 125I-LSD SPIPERONE 1.64 HARTIG ET AL., 1983 Jan 15, 2025 Jan 15, 2025
2668 5-HT2A CORTEX RAT 125I-LSD SPIPERONE 1.64 KADAN ET AL., 1984 Jan 15, 2025 Jan 15, 2025
28546 Alpha1A CLONED HUMAN 3H-PRAZOSIN CLOZAPINE 1.64 Kroeze WK, et.al., 2003 Jan 15, 2025 Jan 15, 2025
50437 SLC6A4 CLONED HUMAN 3H-CITALOPRAM MADAM 1.65 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
60176 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-((3,4-Difluorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane- 1-carboxamide 1.65 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
65821 GABAA CLONED HUMAN [3H] Flunitrazepam CM-D45 C19H21N3O4 1.65 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
52776 5-HT2A UNDEFINED HUMAN UNDEFINED N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide 1.65 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
8756 SST2 CORTEX HUMAN 125I-Tyr3-octreotide CGP 23996 1.65 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
21561 A1 BRAIN RAT 3H-cyclohexyladenosine 5 1.65 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
18780 CCK1 PANCREAS RAT 125I-CCK CCK 1.65 Gully D et al., 1993 Jan 15, 2025 Jan 15, 2025
10084 MOR BRAIN MOUSE 125I-Endomorphin-2 DADLE-OH 1.65 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
139 5-HT1A CORTEX RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.65 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
24493 CLONED RAT 3H-Quisqualate (S)-4C3HPG 1.65 Lavreysen, H, et al., 2003 Jan 15, 2025 Jan 15, 2025
5058 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 1.65 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
61397 GABAA CLONED HUMAN FNZ CM-D45 1.65 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
69356 D2 CLONED HUMAN 3H-NMSP RISPERIDONE 1.65 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
18930 H1 CLONED HUMAN 3H-trans-H2-PAT,(-) trans-H2-PAT(-) 1.65 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
48924 Y5 CLONED Chicken [125I] - Peptide YY NPY18-36, porcine 1.65959 Holmberg, SK et al., 2002 Jan 15, 2025 Jan 15, 2025
34101 H3 CLONED RAT 3H-Alpha-Me-histamine A-349821 1.65959 Esbenshade TA, et al., 2004 Jan 15, 2025 Jan 15, 2025
64649 H1 CLONED HUMAN 3H-PYRILAMINE Levomepromazine 1.65959 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
87124 D3 olfactory tubercle RAT 3H-7-OH-DPAT 8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 1.66 Cao X et al 2018 Jan 15, 2025 Jan 28, 2025
12721 Adrenal Membranes RAT 125I-Angiotensin II L-159,530 1.66 Beauchamp HT, et al., 1995 Jan 15, 2025 Jan 15, 2025
98260 DOR BRAIN MOUSE 3H-DPDPE N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide 1.66 Nakajima R et al 2015 Jan 15, 2025 Jan 28, 2025
16881 A1 CLONED Chick 125I-Aba CHA 1.66 Durand IH, Green RD. 2001 Jan 15, 2025 Jan 15, 2025
16378 Y2 CLONED RAT [125I] - Peptide YY PYY, N-alpha-Ac, 22-36 1.66 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
59140 5-HT2A CLONED HUMAN 3H-KETANSERIN CYPROHEPTADINE 1.67 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
2610 5-HT2A FR. CORTEX RAT 3H-KETANSERIN XYLAMIDINE 1.67 LEYSEN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
55100 H1 UNDEFINED HUMAN UNDEFINED MAPROTILINE 1.67 von Coburg Y et al., 2009 Jan 15, 2025 Jan 15, 2025
65809 GABAA CLONED HUMAN [3H] Flunitrazepam XLI-2TC 1.673 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
60805 GABAA CLONED HUMAN FNZ XLI-2TC 1.673 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
99590 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine 1.68 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
11527 CCK1 PANCREAS RAT 3H-CCK8 CCK8 1.68 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
85774 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide 1.68 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
40992 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-193 1.68 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
60201 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-(Cyclohexylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1.68 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
10063 MOR BRAIN MOUSE 125I-Endomorphin-1 MORPHINE-SULFATE 1.68 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
61067 GABAA CLONED HUMAN FNZ RY-098 1.68 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
140 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.68 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
64930 D2 CLONED HUMAN 3H-N-Methylspiperone Lurasidone 1.68 Ishibashi, Tadashi. et. al, 2010 Jan 15, 2025 Jan 28, 2025
65703 GABAA CLONED HUMAN [3H] Flunitrazepam RY-098 1.68 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
55988 SLC6A4 UNDEFINED RAT UNDEFINED (R)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride 1.68 Manning JR et al., 2009 Jan 15, 2025 Jan 15, 2025
42490 D5 CLONED HUMAN 3H-SCH23390 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1.68 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
12864 Beta2 CLONED HUMAN 125I-ICYP TMQ, 3'-Iodo 1.69 Fraundorfer PF, et al., 1994 Jan 15, 2025 Jan 28, 2025
41296 D5 CLONED HUMAN Functional LE400 1.69 Hoefgen B, et al., 2006 Jan 15, 2025 Jan 15, 2025
8276 SST4 CLONED HUMAN 125I-LTT-SRIF28 CGP 23996 1.69 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
15467 5-HT1B CLONED RAT 3H-5HT 5-Methoxytryptamine 1.69 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
8813 SST5 CLONED HUMAN 125I-CGP23996 L-361,301 1.69 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
6013 M4 CLONED HUMAN M4 3H-QNB 4-DAMP 1.69 CHELALA JL, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
8328 SST2 CLONED HUMAN 125I-LTT-SRIF28 CST14-Tyr10 1.69 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
27040 MOR ILEUM GUINEA PIG 3H-DAMGO DALDA 1.69 Schiller P,et,al.,2000 Jan 15, 2025 Jan 15, 2025
12226 BRAIN HUMAN UNDEFINED LOXAPINE 1.69 Richelson E., 1988 Jan 15, 2025 Jan 15, 2025
10954 SLC6A3 BRAIN RAT 3H-WIN 35,428 BINDING RTI-51 1.69 DAMAJ MI, et al., 1999 Jan 15, 2025 Jan 15, 2025
27091 MOR BRAIN MOUSE 3H-DAMGO DALDA 1.69 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
5086 5-HT2C CLONED HUMAN 3H-MESULERGINE MESULERGINE 1.69 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
51935 MOR UNDEFINED HUMAN UNDEFINED 7alpha-[(cinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 1.69 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
40937 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 RTI-51 1.69 Carroll FI, et al., 1995 Jan 15, 2025 Jan 15, 2025
9455 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-OH 1.69 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
8442 SST5 CLONED HUMAN 125I-CGP23996 L-363,301 1.69 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
65826 GABAA CLONED HUMAN [3H] Flunitrazepam YT-5 1.695 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
60532 GABAA CLONED HUMAN FNZ YT-5 1.695 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
42509 CLONED RABBIT 35S-GTPGammaS [Nle13]-Motilin 1.69824 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
17936 CRF1 BRAIN RAT 125-Tyr0 ovine SSR125543A 1.69824 Gully D et al., 2001 Jan 15, 2025 Jan 15, 2025
32336 M4 HEART Chick 3H-NMS Biperiden 1.69824 Lazareno, S et al., 1990 Jan 15, 2025 Jan 15, 2025
28833 SST2 CLONED HUMAN 125I-LTT-SRIF28 Tyr10-cortistatin 1.69824 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
28861 SST4 CLONED HUMAN 125I-LTT-SRIF28 CGP 23996 1.69824 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
101888 5-HT1E CLONED HUMAN 3H-5HT Ziprasidone 1.7 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
38144 CLONED RAT 3H-dexamethasone C56H80NO8 1.7 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
17666 PANC1 HUMAN 125I-VIP Vasoactive intestinal polypeptide 1.7 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
64771 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 3beta-(p-methylphenyl)tropane-2beta-carboxylic acid methyl ester 1.7 Carroll FI, et al., 2004 Jan 15, 2025 Jan 15, 2025
64773 SLC6A3 Striatal Membranes RAT 3H-WIN 35,428 (1R)-3alpha-(4-Bromophenyl)tropane-2beta-carboxylic Acid Methyl Ester Tosylate 1.7 Carroll FI, et al., 2004 Jan 15, 2025 Jan 15, 2025
8204 SST5 CLONED HUMAN 125I-LTT-SST-28 RC 160 1.7 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
62733 SST2 COLON RAT UNKNOWN RC-121 1.7 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
12559 AT1 LIVER RAT 125I-Angiotensin II Saralasin 1.7 Keiser JA, et al., 1995 Jan 15, 2025 Jan 15, 2025
32784 NK3 CLONED HUMAN 125I-MePhe7-NKB SR 142801 1.7 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
51218 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(5-cyano-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 1.7 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
62738 SST4 Ovary HAMSTER UNKNOWN Somatostatin-14 1.7 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
96790 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
4119 KOR CLONED HUMAN 3H-U69,593 DYNORPHIN(1-17)-OH 1.7 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
93983 D3 CLONED HUMAN 3H-SPIPERONE compound 42 1.7 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
65568 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-082 1.7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
37155 STRIATUM RAT 3H-CGS-21680 N-Ethyl-l-deoxy-1-[6-amino-2-(3-hydroxy-3-phenyl-1-butyn-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide 1.7 Cristalli G, et al., 1994 Jan 15, 2025 Jan 15, 2025
100902 BchE serum HUMAN Functional 1H-indole-3-carboxylic acid [6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]amide 1.7 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 15, 2025
12073 5-HT1D CLONED HUMAN 3H-GR-125743 5-Methoxytryptamine 1.7 Domenech T, et al., 1997 Jan 15, 2025 Jan 15, 2025
16172 D2 CLONED RAT 125I-IODOSULPRIDE Amisulpride 1.7 Sokoloff P, et al., 1990 Jan 15, 2025 Jan 15, 2025
67885 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 1.7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
4141 KOR BRAIN GUINEA PIG 3H-U69,593 NALORPHINE - HCI 1.7 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
49453 SLC6A4 BRAIN RAT 3H-CN-IMI SERTRALINE 1.7 Kovachich GB, et al., 1988 Jan 15, 2025 Jan 15, 2025
13614 WHOLE BRAIN GUINEA PIG 125I-Neurotensin SR 48527 1.7 Betancur C, et al., 1995 Jan 15, 2025 Jan 15, 2025
100910 BchE serum HUMAN Functional 2-(5-Bromo-1H-indol-3-yl)-N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]acetamide 1.7 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 15, 2025
64815 CCR5 CLONED UNDEFINED 125I-RANTES (S)-(-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 1.7 Seto M, et al., 2006 Jan 15, 2025 Jan 28, 2025
20528 A1 myocardial membranes BOVINE 3H-DPCPX DPX 1.7 Lohse MJ et al., 1987 Jan 15, 2025 Jan 15, 2025
35633 STRIATUM RAT 3H-SPIPERONE KETANSERIN 1.7 Bogeso KP, et al., 1988 Jan 15, 2025 Jan 15, 2025
36657 H1 CLONED HUMAN 3H-PYRILAMINE MIANSERIN 1.7 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
32818 D2 STRIATUM CANINE 3H-SPIPERONE ADTN 1.7 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
4147 KOR BRAIN GUINEA PIG 3H-U69,593 DYNORPHIN(1-17)-OH 1.7 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
63283 A3 Ovary HAMSTER [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamide (1S,2R,3S,4R,5S)-4-(5-((5-chlorothiophen-2-yl)ethynyl)-7-(ethylamino)-3H-imidazo[4,5- b]pyridin-3-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1.7 Tosh, Dilip et. al., 2015 Jan 15, 2025 Jan 15, 2025
64819 CCR5 CLONED UNDEFINED 125I-RANTES (S)-(-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-1-benzazocine-5-carboxamide 1.7 Seto M, et al., 2006 Jan 15, 2025 Jan 28, 2025
66100 5-HT1A CLONED HUMAN 3H-WAY100635 ARIPIPRAZOLE 1.7 Hirose, Tsuyoshi. et. al, 2005 Jan 15, 2025 Jan 15, 2025
98100 CB1 CHO cells HUMAN 3H-CP-55940 N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide 1.7 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
94008 5-HT1A CORTEX PIG [3H]WAY 600135 compound 43 1.7 Ortega R et al 2011 Jan 15, 2025 Jan 15, 2025
13882 A1 HEART Chick 125I-Aba R-PIA 1.7 Leung E, et al., 1987 Jan 15, 2025 Jan 15, 2025
24122 VPAC1 PANC1 HUMAN 125I-VIP Vasoactive intestinal polypeptide 1.7 Igarashi H, et al., 2002 Jan 15, 2025 Jan 15, 2025
94010 5-HT1A CORTEX PIG [3H]WAY 600135 7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one 1.7 Ortega R et al 2011 Jan 15, 2025 Jan 15, 2025
53306 MOR UNDEFINED HUMAN UNDEFINED (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-phenylpropanoic acid 1.7 Le Bourdonnec B et al., 2008 Jan 15, 2025 Jan 15, 2025
2877 5-HT2A CORTEX HUMAN 3H-KETANSERIN LOXAPINE 1.7 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
16190 D3 CLONED RAT 125I-IODOSULPRIDE Thioproperazine 1.7 Sokoloff P, et al., 1990 Jan 15, 2025 Jan 15, 2025
24126 VPAC1 CLONED HUMAN 125I-VIP [Lys15, Arg16, Leu27]VIP(1-7)GRF(8-27) 1.7 Igarashi H, et al., 2002 Jan 15, 2025 Jan 15, 2025
3395 MOR CLONED HUMAN 3H-DAMGO NORMORPHINE-HClO4 1.7 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
3399 MOR CLONED HUMAN 3H-DAMGO DIHYDROMORPHINE 1.7 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
41800 CLONED HUMAN 3H-Estradiol 1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1.7 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
34378 MOR FOREBRAIN RAT 3H-DAMGO Methadone 1.7 Codd EE et al, 1995 Jan 15, 2025 Jan 15, 2025
16715 M5 CLONED HUMAN 3H-QNB ATR 1.7 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
10319 MOR CLONED RAT 3H-DAMGO Beta-Endorphin 1.7 Raynor,Kong,Mestek,Bye,Tian,Liu,Yu,Reisine 1995 Jan 15, 2025 Jan 15, 2025
22096 PMNL Monkey 3H-Leukotriene B4 CGS 25019 C 1.7 Birke FW, et al., 2001 Jan 15, 2025 Jan 15, 2025
53072 KOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-[(3'-dimethylamino)benzamido]morphinan 1.7 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
23890 D2 CLONED HUMAN 3H-RACLOPRIDE PROCHLORPERAZINE 1.7 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
68947 GABAA CLONED RAT 3H-Ro15-1788 5-[3-(3,5-Difluoropyridin2-yl)-4-fluorophenyl]-3-(2-fluorophenyl)pyridazine 1.7 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
65620 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-60 (C17H11N2OF) 1.7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
73558 Sigma 1 test RODENT 3H-Pentazocine(+) 3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride 1.7 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
91482 5-HT2A CLONED HUMAN 125I-DOI (6bS,11aS)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophenyl)-1-butanone 1.7 Li P et al 2014 Jan 15, 2025 Jan 15, 2025
34138 Beta1 CLONED HUMAN 125I-CYP Carvedilol 1.7 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
85595 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate 1.7 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
101211 MOR CLONED HUMAN 3H-Diprenorphine (S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopro-pan-2-aminium Trifluoroacetate 1.7 Henry S,et al., 2021 Jan 15, 2025 Jan 28, 2025
10845 D3 CLONED HUMAN 125I-IODOSULPRIDE ADTN 6,7 1.7 Freedman SB, et al., 1994 Jan 15, 2025 Jan 15, 2025
97630 SST4 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 1.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
47967 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
22113 PMNL HUMAN 3H-Leukotriene B4 BIIL-260 1.7 Birke FW, et al., 2001 Jan 15, 2025 Jan 15, 2025
39521 S1P1 CLONED HUMAN 35S-GTPGammaS 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid 1.7 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
60002 mGluR5 Ovary HAMSTER 3H-Inostitol 2-Methyl-6-[(5-phenyl-3-pyridinyl)ethynyl]pyridine 1.7 Alagille, D. et. al, 2005 Jan 15, 2025 Jan 28, 2025
53859 5-HT1A UNDEFINED RAT UNDEFINED 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzothiazole 1.7 Siracusa MA et al., 2008 Jan 15, 2025 Jan 15, 2025
13414 D3 CLONED HUMAN 125I-IODOSULPRIDE LISURIDE 1.7 Sautel F, et al., 1995 Jan 15, 2025 Jan 15, 2025
18279 D2 BRAIN RAT 3H-NPA A 37843 1.7 Hall H et al., 1986 Jan 15, 2025 Jan 27, 2025
52072 SLC6A4 UNDEFINED HUMAN UNDEFINED (5-bromo-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine 1.7 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
30825 KOR CORTEX RAT 3H-Indiplon Indiplon 1.7 Sullivan SK et al., 2004 Jan 15, 2025 Jan 27, 2025
52073 H3 UNDEFINED HUMAN UNDEFINED N-methyl(2-(4-(methylthio)phenoxy)-5-(4-(piperidin-1-yl)but-1-ynyl)phenyl)methanamine 1.7 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
100202 5-HT1D CLONED HUMAN 3H-5CT Ziprasidone 1.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
53611 5-HT1A UNDEFINED HUMAN UNDEFINED 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole 1.7 Zhou D et al., 2008 Jan 15, 2025 Jan 15, 2025
68979 GABAA CLONED RAT 3H-Ro15-1788 5-[3-(3,5-Difluoropyridin-2-yl)-4-fluorophenyl]-3-(3-fluoropyridin-2-yl)pyridazine 1.7 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
39027 D2 CLONED HUMAN R-SAT CHLORPROMAZINE 1.7 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
61814 5-HT2C CLONED HUMAN 3H-MESULERGINE FECIMBI-36 1.7 Prabhakaran, Jaya et. al. 2015 Jan 15, 2025 Jan 15, 2025
16506 CLONED HUMAN 3H-RACLOPRIDE RISPERIDONE 1.7 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
7804 GABAA CLONED HUMAN 3H-RO-15-1788 3 1.7 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
51326 H3 UNDEFINED HUMAN UNDEFINED N,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine 1.7 Keith JM et al., 2007 Jan 15, 2025 Jan 15, 2025
30848 BB2 CLONED HUMAN 125I-[Tyr4]Bn [D-Tyr6,NAlpha-acetyl-Dap11,Phe13,Nle14]Bn(6-14) 1.7 Mantey, SA et. al., 2004 Jan 15, 2025 Jan 15, 2025
49024 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (-)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-2-methyl-propyl]piperidine hydrochloride 1.7 Berardi, F et al., 2003 Jan 15, 2025 Jan 15, 2025
14980 D2 CLONED HUMAN 3H-RACLOPRIDE RISPERIDONE 1.7 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 27, 2025
36740 D2 CLONED HUMAN 3H-SPIPERONE (-)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin 1.7 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
10374 nAChR M10 Cells Mammalian 3H-Epibatidine ABT-418 1.7 Whiteaker P, Sharples CG, Wonnacott S, 1998 Jan 15, 2025 Jan 15, 2025
16267 M5 CLONED HUMAN 3H-NMS Ipratropium 1.7 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
141 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.7 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
16269 M1 CLONED RAT 3H-PIRENZEPINE a 1.7 Hirose H, et al., 2001 Jan 15, 2025 Jan 15, 2025
101012 5-HT2B CLONED HUMAN 3H- LSD N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine 1.7 Kapadia N et al 2016 Jan 15, 2025 Jan 15, 2025
37524 D3 CLONED RAT 3H-SPIROPERIDOL N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 1.7 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
60821 GABAA CLONED HUMAN FNZ JYI-60 1.7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
8088 GABAA CLONED HUMAN 3H-RO-15-1788 26 1.7 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
52891 CB2 UNDEFINED HUMAN UNDEFINED N-cyclohexyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide 1.7 Silvestri R et al., 2008 Jan 15, 2025 Jan 15, 2025
9372 GABAA CLONED HUMAN FNZ Clonazepam 1.7 Pritchett DB, Luddens H, Seeburg PH, 1989 Jan 15, 2025 Jan 27, 2025