The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 7,001-8,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
101895NETCLONEDHUMAN[3H]NisoxetineZiprasidone69PDSP Certified DataMar 24, 2025Jul 28, 2026
36615D2CLONEDHUMAN3H-SPIPERONEMIANSERIN2197Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102151DORCLONEDHUMAN[3H]DADLENEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
37895MPP-9CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione19Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38151CLONEDRAT3H-dexamethasoneC30H36NO31000von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
39175D4CLONEDHUMANR-SATN-DESMETHYLCLOZAPINE70Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39431V2CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396875-HT2BCLONEDHUMAN3H-5HTORG-1296291.2011Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40711mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one84Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41223CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41991M1CLONEDHUMAN3H-QNBDothiepin18Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42247CLONEDHUMAN125I-[Ile]Motilin[L-Bpa5,Ile13]Motilin50Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42759CLONEDUNDEFINEDFunctionalCyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-beta-Ala-Cys (O))-amide (S)>10000Song YL, et al., 2006Jan 15, 2025Jan 15, 2025
43015FYNCLONEDHUMAN3H-StaurosporineGleevec5500Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43271CLK1CLONEDHUMAN3H-StaurosporineSU11248100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43527FLT3CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43783CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44039STK36CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44295CaMKCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44551FLT4CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44807MAPK12CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45063PTK2CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45319CDK2CLONEDHUMANFunctionalkenpaullone670Bain J, et al., 2003Jan 15, 2025Jan 28, 2025
45575NETCLONEDHUMAN3H-NisoxetineDothiepin46Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458315-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46087Alpha2ACLONEDHUMAN3H-CLONIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46599SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46855M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47367Kainate receptorCLONEDHUMAN3H-Kainic acidLY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
48135Y2CLONEDHUMAN3H-Propionyl-NPYPP, human1000Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48647GNRHRCLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49159MORCLONEDRAT3H-DAMGOLYS32820Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49671SST5CLONEDHUMAN125I-LTT-SST-28L-796,778>10000Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
49927mGluR6CLONEDRATFunctionalD-Glutamate>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 15, 2025
50183mGluR3CLONEDHUMANFunctionalL-CCG-I2100Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50439SLC6A4CLONEDHUMAN3H-CITALOPRAM5-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine8Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581195-HT2ACLONEDHUMAN3H-KETANSERINN-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate427Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58375H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5755>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58631hERGCLONEDHUMAN3H-N-Me-DofetilideMRS5474>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
591435-HT2ACLONEDHUMAN3H-KETANSERINHALOPERIDOL30Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59399D2CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4-(2-thienyl)benzamide840Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59911D4CLONEDHUMAN3H-NMSP4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60167A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-4-(2-(Cyclohexylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60423GABAACLONEDHUMANFNZWY-S-2100Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60679GABAACLONEDHUMANFNZXHE-I-0938.9Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60935GABAACLONEDHUMANFNZ3 EBC1000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61191GABAACLONEDHUMANFNZQH-II-067a31Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61447GABAACLONEDHUMANFNZRY-05444Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617035-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine1507Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62215SLC6A3CLONEDHUMAN[3H] WIN35428Benzedrone1089Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62471M4CLONEDHUMAN3H-QNB2-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
62983GABAACLONEDRAT3H-RO-15-1788Zolpidem383Costanzo A et al., 2002Jan 15, 2025Jan 27, 2025
634955-HT2BCLONEDHUMAN3H-LSDRISPERIDONE35Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640075-HT6CLONEDHUMAN3H-LSD1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one125.8Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642635-HT2ACLONEDHUMAN3H-KETANSERINSERTINDOLE0.323594Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64519D2CLONEDHUMAN3H-N-MethylspiperonePROCHLORPERAZINE2.23872Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65287GABAACLONEDHUMAN[3H] FlunitrazepamSH-I-03011.04Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65544GABAACLONEDHUMAN[3H] FlunitrazepamMLT-I-701.1Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65800GABAACLONEDHUMAN[3H] FlunitrazepamYT-687.8Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
660565-HT1ACLONEDHUMAN3H-WAY100635Mellpaladine A7500Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66312Beta3CLONEDHUMANI-125-PindololFinazine>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66568Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride52Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
668245-HT7CLONEDHUMAN3H-LSDN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
670805-HT2ACLONEDHUMAN3H-KETANSERIN1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
678485-HT2ACLONEDHUMAN3H-KETANSERINS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline91Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33365-HT1ACLONEDHUMAN3H-8-OH-DPATBROMOCRIPTINE,(+)25TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68872SST5CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH279.4328Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
35925-HT2CCLONEDRAT3H-MESULERGINESKF 38393>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69128H3CLONEDHUMAN3H-HistamineHISTAMINE10Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
3848D2CLONEDRAT3H-SPIPERONEQuetiapine329KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69384H1CLONEDHUMAN3H-PYRILAMINEHALOPERIDOL4160Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4104KORCLONEDHUMAN3H-U69,593Leu-ENKEPHALIN>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69640Alpha2BCLONEDHUMAN3H-RAUWOLSCINEDPH4376Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43605-HT6CLONEDHUMAN3H-LSD8-OH-DPAT>10000KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69896D2CLONEDHUMAN3H-N-Methylspiperone4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4616SLC6A3CLONEDHUMAN3H-DA UPTAKEBUPROPION784PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48725-HT2BCLONEDHUMAN3H-5HTYOHIMBINE43.2WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70408Sigma 1CLONEDHUMAN3H-Pentazocine(+)MRP42685.5Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51285-HT2BCLONEDHUMAN3H-5HTTMA307NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70664NETCLONEDHUMAN3H-NisoxetineMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
53845-HT2BCLONEDHUMAN3H-5HTSB200646a630.95BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
709205-HT2BCLONEDHUMAN3H-LSD(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione840Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
56405-HT4CLONEDRAT3H-GR-1138085-CT9120.1CLAEYSEN S, ET AL., 1997Jan 15, 2025Jan 27, 2025
71176D5CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE2590Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5896Alpha2BCLONEDHUMAN3H-RAUWOLSCINEMIANSERIN27WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714325-HT5ACLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine5844Klein LM et al 2018Jan 15, 2025Jan 15, 2025
6152Alpha1BCLONEDRAT125I-HEATINDORAMINE226LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64085-HT3CLONEDGUINEA PIG3H-BIMU-1ZACOPRIDE,R>10000BONHAUS DW, ET AL., 1993Jan 15, 2025Jan 15, 2025
72200DATCLONEDHUMAN3H-WIN354282-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
69205-HT2ACLONEDHUMAN3H-KETANSERINMOLINDONE5800SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72712Alpha2CCLONEDHUMAN3H-RAUWOLSCINEnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7432MORCLONEDHUMAN3H-DAMGODIPRENORPHINE-HCl0.07Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
72968Alpha1DCLONEDHUMAN3H-PRAZOSINcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7688GABAACLONEDHUMAN3H-MUSCIMOLGamma-Aminobutyric acid8.7Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7944GABAACLONEDHUMAN3H-RO-15-178861000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8200SST5CLONEDHUMAN125I-LTT-SST-28Somatostatin-142.24Panetta R, et al., 1993Jan 15, 2025Jan 15, 2025
8456SST5CLONEDHUMAN125I-Tyr3-octreotideCGP 239962.08Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8712SST2CLONEDHUMAN125I-Tyr3-octreotideRC 1600.31Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8968SST1CLONEDHUMAN125I-SRIF-28L-363,301630.95Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
745045-HT6CLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9224SST2CLONEDMOUSE125I-MK-678MK 6780.18Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
9736MT2CLONEDHUMAN125I-Iodomelatonin8-M-PDOT3Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75272NOPCLONEDHUMAN3H-Nociceptinethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate9400Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
9992CB2CLONEDMOUSE3H-CP-55940SR 1445280.05Griffin G, Tao Q, Abood ME, 2000Jan 15, 2025Jan 15, 2025
755285-HT6CLONEDHUMAN3H-LSDpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10248CLONEDHAMSTER125I-HEATNiguldipine(+)501.18Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75784Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76040DORCLONEDHUMAN3H-DADLEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate627Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10760D2CLONEDRAT3H-LSDRACLOPRIDE1.99ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
76296SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
765525-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768085-HT7CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77064Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77320Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77576D2CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77832H1CLONEDHUMAN3H-PYRILAMINE(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78088M1CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78344M5CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78600DORCLONEDHUMAN3H-DADLE(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78856DORCLONEDHUMAN3H-DADLE(±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791125-HT5ACLONEDHUMAN3H-LSDLYSERGIC ACID9Ray TS 2010 Jan 15, 2025Jan 15, 2025
79368Alpha1ACLONEDHUMAN3H-PRAZOSINSalvinorin A>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14088Alpha2ACLONEDPIG3H-YohimbineIsoproterenol-l>10000Brink CB, et al., 2000Jan 15, 2025Jan 15, 2025
79624CLONEDHUMAN3H-CLONIDINE3,4,5-Trimethoxyphenethylamine2677.6Ray TS 2010 Jan 15, 2025Jan 15, 2025
79880M5CLONEDHUMAN3H-QNBDMT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14600D3CLONEDHUMAN125I-IODOSULPRIDESB-277011-A11.22Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80136CLONEDHUMAN3H-VASOPRESSINEMDT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14856D1CLONEDRATUNDEFINEDOLANZAPINE10Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
803925-HT1ACLONEDHUMAN3H-8-OH-DPAT(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one3215Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15112PTGFRCLONEDHUMAN3H-PGF2AlphaAGN 191365>10000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806485-HT2ACLONEDHUMAN3H-KETANSERIN(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153685-HT1BCLONEDHUMAN3H-5HTCGS 12066B2.08BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809045-HT4CLONEDHUMAN3H-GR113808(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one603Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
156245-HT2BCLONEDRAT3H-5HTAMESERGIDE10.71BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81160H4CLONEDHUMAN3H-HistamineN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
158805-HT7CLONEDRATUNDEFINED5-Methoxytryptamine0.93BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
814165-HT2ACLONEDHUMAN3H-KETANSERIN1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine>10000Weiss DR et al 2018Jan 15, 2025Jan 15, 2025
16136D1CLONEDHUMAN3H-SCH23390NOREPINEPHRINE>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81672D2CLONEDHUMAN3H-N-Methylspiperone(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
819285-HT1DCLONEDHUMAN3H-Cimetidine(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16648M1CLONEDHUMAN3H-QNBATR0.5Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82184D5CLONEDHUMAN3H-SCH233902-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82440Alpha1ACLONEDHUMAN3H-PRAZOSIN(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
826965-HT3CLONEDHUMAN3H-GR65630(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17672CLONEDHUMAN125I-VIPVIP [D-Thr7]162Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832085-HT2CCLONEDHUMAN125I-DOIDOM25.7Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83464M4CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+)35.4813Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83720DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
83976KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(3-bromobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide438PDSP Certified DataJan 15, 2025Jan 28, 2025
84232DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide2471PDSP Certified DataJan 15, 2025Jan 28, 2025
18952H1CLONEDGUINEA PIG3H-MEPYRAMINECLOZAPINE1.23Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84488KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84744DORCLONEDHUMAN3H-DADLEbenzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19464GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHhAc-MCH(6-16)-NH22.7Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
85000DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
86024D3CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
21000CLONEDRAT3H-NECA18250Shamim MT et al., 1989Jan 15, 2025Jan 15, 2025
86536A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
21512nAChRCLONEDXenopus3H-EpibatidineNNEP7.2Avalos M et al., 2002Jan 15, 2025Jan 27, 2025
87560Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
22280A1CLONEDHUMAN125I-Aba4a175Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
87816D2CLONEDHUMAN3H-RACLOPRIDE4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline505Staron J et al 2016Jan 15, 2025Jan 28, 2025
225365-HT1DCLONEDHUMAN3H-5CTSL6501557990Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
88072A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22792H2CLONEDHUMAN3H-TIOTIDINEL-cysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23048nAChRCLONEDHUMAN3H-EpibatidineL-homocysteine thiolactone>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
88584H1CLONEDHUMAN3H-PYRILAMINE1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine212Peprah K et al 2012Jan 15, 2025Jan 28, 2025
893525-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide3842Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240725-HT2ACLONEDHUMANUNDEFINEDRISPERIDONE0.21Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
896085-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone0.47863Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
90120D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
25096D1CLONEDHUMAN3H-SCH23390Quetiapine712Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90632A2BCLONEDHUMAN3H-PSB-6033-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
253525-HT1DCLONEDHUMAN3H-GR-125743ZOTEPINE175PDSP Certified DataJan 15, 2025Jan 15, 2025
25864mGluR6CLONEDRATFunctionalPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91400CB2CLONEDHUMAN3H-CP55940O-6617>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26120M3CLONEDHUMAN3H-QNBPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91656A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26376M5CLONEDHUMAN3H-QNBRutin35.13Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91912A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3-chlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26632MORCLONEDHUMAN3H-DiprenorphineHyperoside>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921685-HT6CLONEDHUMAN3H-LSDN-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)-8-quinolinesulfonamide504Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
26888M5CLONEDHUMAN3H-QNBxanomeline39.8107Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92424KORCLONEDHUMAN3H-U695939,13:15,16-diepoxylabdane-6β,15α-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92680M2CLONEDHUMAN3H-QNB9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27400Beta2CLONEDHUMAN3H-CGP-12177Talipexole>10000Millan MJ, et al., 2002Jan 15, 2025Jan 28, 2025
929365-HT6CLONEDHUMAN3H-LSDWA-1323Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276565-HT7CLONEDHUMAN3H-LSDMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279125-HT2ACLONEDHUMAN3H-KETANSERINDMT,5-Me1325Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
93704A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester26.4Federico S et al 2018Jan 15, 2025Jan 15, 2025
28424mGluR5CLONEDHUMAN3H-QuisqualateQuisqualate29Mutel V, et.al., 2000Jan 15, 2025Jan 28, 2025
93960D2CLONEDHUMAN3H-SPIPERONEcompound 433.9Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28680D1CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE1960Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942165-HT1ACLONEDHUMAN3H-8-OH-DPAT4-Bromo-2,5-dimethoxyphenethylamine311Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29192SST2CLONEDHUMANUNDEFINEDNC8-120.024Patel YC, 1999Jan 15, 2025Jan 15, 2025
947285-HT2ACLONEDHUMAN3H-KETANSERIN4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94984D3CLONEDHUMAN3H-N-Methylspiperone5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29960H4CLONEDHUMAN3H-Histamine(1H-Indol-2-yl)-(piperazin-1-yl)-methanone38Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30216D1CLONEDRATUNDEFINEDDuloxetine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 15, 2025
957525-HT5ACLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96008NETCLONEDHUMAN3H-Nisoxetine6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30728CLONEDRATUNDEFINEDAtomoxetine1000Bymaster F.P., et. al., 2002Jan 15, 2025Jan 15, 2025
96264Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96520Alpha1ACLONEDHUMAN[3H]-prazosin6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
31240Alpha1ACLONEDHUMAN3H-PRAZOSINMDL 1009071199PDSP Certified DataJan 15, 2025Jan 15, 2025
96776D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314965-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)1000Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97032D2CLONEDHUMAN[3H]N-methylspiperoneFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97288MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o24.4Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97544A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32776NK1CLONEDHUMAN3H-Sar9,Met(O2)11-Substance PSR 48968273Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98312D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride1087Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985685-HT2BCLONEDHUMAN[3H]-LSD4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide587Ofon E et al 2016aJan 15, 2025Jan 15, 2025
332885-HT1BCLONEDHUMAN3H-GR-125743Acetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98824DORCLONEDHUMAN3H-DADLE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33544Alpha2ACLONEDHUMAN3H-CLONIDINENaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99080Beta1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99336D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol963Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34056P2X3CLONEDHUMAN3H-A-317491Cibacron blue2530Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99592A1CLONEDHUMAN3H-CCPA8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine1.22Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34312nAChRCLONEDRAT3H-EpibatidineABT-418803Grinevich VP, et al., 2004Jan 15, 2025Jan 28, 2025
99848Alpha2CCLONEDHUMAN[125I] iodoclonidine(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide280Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
1001045-HT2CCLONEDHUMAN3H-MESULERGINEQuetiapine3624PDSP Certified DataJan 15, 2025Jan 15, 2025
34824CLONEDRAT3H-CP-55940Rinvanil, Phenyl-propionyl>10000Jan 15, 2025Jan 15, 2025
100360NETCLONEDHUMAN3H-NisoxeneCariprazine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100616CGRPCLONEDHUMANFunctionalN2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100872Beta2CLONEDHUMAN3H-CGP-121771-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1)2Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
35592CLONEDHUMAN3H-SQ 29548CARBACYCLIN>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35848Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester33Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013845-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione476Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101640D4CLONEDHUMAN[3H]-N-methylspiperonePerospirone3.2PDSP Certified DataMar 21, 2025Jul 28, 2026
101896DATCLONEDHUMAN[3H]WIN35428Ziprasidone424PDSP Certified DataMar 24, 2025Jul 28, 2026
36616D3CLONEDHUMAN125I-IODOSULPRIDE(2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin293Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102152KORCLONEDHUMAN[3H]U69593NEMONAPRIDE2713PDSP Certified DataMar 25, 2025Jul 28, 2026
37896MPP-2CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-nitro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione16Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38152CLONEDRAT3H-dexamethasoneC57H79N2O9590von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
39432Calcium channelCLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396885-HT2BCLONEDHUMAN3H-5HTORG-3768442.658Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40712mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one4530Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41224CLONEDHUMAN125I-Chemokine5-(4-Butyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41992M1CLONEDHUMAN3H-QNBDOXEPIN38Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42248CLONEDHUMAN125I-[Ile]Motilincyanogen bromide, CNBr0.85Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42760CLONEDUNDEFINEDFunctionalCyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Cys (O))-amide (S)>10000Song YL, et al., 2006Jan 15, 2025Jan 15, 2025
43016FYNCLONEDHUMAN3H-StaurosporineZD-64745700Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43272CLK1CLONEDHUMAN3H-StaurosporineMLN-5181400Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43528FLT4CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43784KDRCLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44040STK38LCLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44296CaMKCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44552FRKCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44808AAK1CLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45064PTK6CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45320CLONEDHUMANFunctionalkenpaullone230Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45576SLC6A3CLONEDHUMAN3H-WIN 35,428Dothiepin5310Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458325-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46088Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46600SLC6A3CLONEDHUMAN3H-WIN 35,428PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46856M5CLONEDHUMAN3H-QNB(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47368Kainate receptorCLONEDHUMAN3H-Kainic acidLY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
48136Y2CLONEDHUMAN3H-Propionyl-NPYPP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human500Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48648CLONEDHUMANFunctional1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride400Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49160MORCLONEDRAT3H-DAMGOLYS2275.3Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49672Y2CLONEDChicken[125I] - Peptide YYPYY, chicken0.630957Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49928CLONEDRATFunctional(S)-2-Aminoadipic acid>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 15, 2025
50184mGluR3CLONEDHUMANFunctional1S, 3R-ACPD>10000Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50440SLC6A4CLONEDHUMAN3H-CITALOPRAMN,N-Dimethyl-4-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine519Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581205-HT2ACLONEDHUMAN125I-DOIN-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate11.2Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58376H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5202>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
591445-HT2ACLONEDHUMAN3H-KETANSERINKETANSERIN2Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59400D4CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4-(3-thienyl)benzamide2Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59912D5CLONEDHUMAN3H-SCH233904-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60168A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-4-(6-(3-Chlorobenzylamino)-2-((3,4- difluorophenyl)ethynyl)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide3.49Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60424GABAACLONEDHUMANFNZWY-S-2124Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60680GABAACLONEDHUMANFNZXHE-I-0931107Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60936GABAACLONEDHUMANFNZDM-146247Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61192GABAACLONEDHUMANFNZQH-II-067a16Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61448GABAACLONEDHUMANFNZRY-05459Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617045-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine2234Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62216NETCLONEDHUMAN[3H] NisoxetineNaphyrone96Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62472M4CLONEDHUMAN3H-QNB3-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
62984GABAACLONEDRAT3H-RO-15-17883-(2-Thienylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 5-oxide8.6Costanzo A et al., 2002Jan 15, 2025Jan 27, 2025
63496Alpha1BCLONEDHUMAN3H-PRAZOSINRISPERIDONE9Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640085-HT6CLONEDHUMAN3H-LSD1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one124.5Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642645-HT2ACLONEDHUMAN3H-KETANSERINSULPIRIDE4786.3Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64520CLONEDHUMAN3H-Estradiol17beta-Estradiol380Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65288GABAACLONEDHUMAN[3H] FlunitrazepamSH-I-03019.09Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65545GABAACLONEDHUMAN[3H] FlunitrazepamMLT-I-7040.3Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65801GABAACLONEDHUMAN[3H] FlunitrazepamYT-660.49Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
660575-HT1ACLONEDHUMAN3H-WAY100635Mellpaladine B652Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66313Beta2CLONEDHUMAN3H-CGP12177Finazine>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66569Beta1CLONEDHUMANI-125-Pindolol3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66825Alpha1ACLONEDHUMAN3H-PRAZOSINN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
670815-HT2BCLONEDHUMAN3H-LSD1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate969Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
673375-HT1ACLONEDHUMAN3H-WAY1006351-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride58Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
678495-HT6CLONEDHUMAN3H-LSDS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline1483Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33375-HT1ACLONEDHUMAN3H-8-OH-DPATCARBAMAZEPINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68873SST1CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH21000Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
35935-HT2CCLONEDRAT3H-MESULERGINESKF 774343037TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69129H3CLONEDHUMAN3H-HistamineN-alpha-methylhistamine3.98107Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
3849D2CLONEDRAT3H-SPIPERONEHALOPERIDOL13KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69385H1CLONEDHUMAN3H-PYRILAMINEFLUPHENAZINE67Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4105KORCLONEDHUMAN3H-U69,593Beta-Endorphin11.4TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69641Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43615-HT6CLONEDHUMAN3H-LSDOCTOCLOTHEPIN,(-)1.8KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69897D2CLONEDHUMAN3H-N-Methylspiperone4-[1-(4-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4617SLC6A3CLONEDHUMAN3H-DA UPTAKEDOPAMINE1770PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48735-HT2BCLONEDHUMAN3H-5HTLY 538571.53WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704095-HT7CLONEDHUMAN3H-LSDMRP4268600Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51295-HT2BCLONEDHUMAN3H-5HTMEM763NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70665DORCLONEDHUMAN3H-DADLEMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
53855-HT2BCLONEDHUMAN3H-5HT5-Hydroxy Tryptamine0.79BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
709215-HT2BCLONEDHUMAN3H-LSD(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione2051Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
56415-HT4CLONEDHUMAN3H-GR-113808RS 1002350.00057544CLAEYSEN S, ET AL., 1997Jan 15, 2025Jan 27, 2025
71177D5CLONEDHUMAN3H-SCH23390HALOPERIDOL147Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5897Alpha2BCLONEDHUMAN3H-RAUWOLSCINECORYNANTHINE77WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714335-HT6CLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine1791Klein LM et al 2018Jan 15, 2025Jan 15, 2025
6153Alpha1BCLONEDRAT125I-HEATCORYNANTHINE517LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64095-HT3CLONEDGUINEA PIG3H-BIMU-1BIMU 127.5BONHAUS DW, ET AL., 1993Jan 15, 2025Jan 15, 2025
6665D2CLONEDHUMAN3H-NEMONAPRIDECHLORPROMAZINE14SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
72201DORCLONEDHUMAN3H-DADLE2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69215-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE5.8SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
7433MORCLONEDHUMAN3H-DAMGONaloxone(-)0.93Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
72969Alpha2ACLONEDHUMAN3H-RAUWOLSCINEcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7689GABAACLONEDHUMAN3H-MUSCIMOLMuscimol2.88Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7945GABAACLONEDHUMAN3H-RO-15-178881000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8201SST5CLONEDHUMAN125I-LTT-SST-28SRIF-D-Trp80.28Panetta R, et al., 1993Jan 15, 2025Jan 15, 2025
8457SST5CLONEDHUMAN125I-Tyr3-octreotideoctreotide0.33Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8713SST2CLONEDHUMAN125I-Tyr3-octreotideoctreotide0.79Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8969SST2CLONEDHUMAN125I-SRIF-28Somatostatin-140.19Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
745055-HT7CLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9225SST2CLONEDMOUSE125I-MK-678L-363,3018.6Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74761D1CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75017M1CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9737MT2CLONEDHUMAN125I-IodomelatoninN-Acetyltryptamine12.7Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
9993CB2CLONEDMOUSE3H-CP-55940JWH-015431Griffin G, Tao Q, Abood ME, 2000Jan 15, 2025Jan 15, 2025
755295-HT7CLONEDHUMAN3H-LSDpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10249CLONEDHAMSTER125I-HEATPHENTOLAMINE79.43Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75785Beta 1CLONEDHUMAN125I-Pindolol1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76041KORCLONEDHUMAN3H-U69593Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate207Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
107615-HT2CCLONEDRAT3H-LSDCLOZAPINE6.3ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
76297NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765535-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76809Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one6390Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77065Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77321Beta 2CLONEDHUMAN3H-CGP12177(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77577D3CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
778335-HT1DCLONEDHUMAN3H-Cimetidine(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78089M2CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78345NETCLONEDHUMAN3H-Nisoxetine(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78601KORCLONEDHUMAN3H-U69593(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide490Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78857KORCLONEDHUMAN3H-U69593(±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide30Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791135-HT5ACLONEDHUMAN3H-LSDcis-2a16.4Ray TS 2010 Jan 15, 2025Jan 15, 2025
79369Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14089Alpha2ACLONEDPIG3H-YohimbineUK-14,304478.63Brink CB, et al., 2000Jan 15, 2025Jan 15, 2025
79625CLONEDHUMAN3H-CLONIDINE4-Bromo-2,5-dimethoxyphenethylamine2155.3Ray TS 2010 Jan 15, 2025Jan 15, 2025
79881M5CLONEDHUMAN3H-QNBDMT,5-MeO>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14601D2CLONEDHUMAN125I-IODOSULPRIDESB-277011-A1047.12Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80137CLONEDHUMAN3H-VASOPRESSIN5-MeO-TMT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14857D1CLONEDRATUNDEFINEDRISPERIDONE21Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
803935-HT1ECLONEDHUMAN3H-5-CT(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15113PTGFRCLONEDHUMAN3H-PGF2AlphaAGN 1913668128Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806495-HT2BCLONEDHUMAN3H-LSD(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one1274Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153695-HT1BCLONEDHUMAN3H-5HTSUMATRIPTAN7.76BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809055-HT5ACLONEDHUMAN3H-LSD(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one3324Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
156255-HT2BCLONEDRAT3H-5HTKETANSERIN3548.13BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
811615-HT1ACLONEDHUMAN3H-8-OH-DPATN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158815-HT7CLONEDRATUNDEFINED5-Hydroxy Tryptamine0.6BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81417D2CLONEDHUMAN3H-N-Methylspiperone1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine6787Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16137D1CLONEDHUMAN3H-SCH23390LY-171555>10000Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81673D3CLONEDHUMAN3H-N-Methylspiperone(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
81929H3CLONEDHUMAN3H-Alpha-methylhistamine(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16649M1CLONEDHUMAN3H-QNBSCOPOLAMINE1.1Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82185D2CLONEDHUMAN3H-N-Methylspiperone2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one1112Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82441Alpha1BCLONEDHUMAN3H-PRAZOSIN(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
826975-HT4CLONEDHUMAN3H-GR113808(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17673CLONEDHUMAN125I-VIPVIP [D-Phe6]288Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832095-HT2CCLONEDHUMAN125I-DOIKETANSERIN117Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83465M3CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+)30.903Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83721DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
83977KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide2362PDSP Certified DataJan 15, 2025Jan 28, 2025
84233KORCLONEDHUMAN3H-U69593(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide205PDSP Certified DataJan 15, 2025Jan 28, 2025
18953H1CLONEDGUINEA PIG3H-MEPYRAMINEtrans-H2-PAT(-)1.15Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84489KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19209CLONEDRAT125I-VIP[Phe1]PACAP-27300Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84745KORCLONEDHUMAN3H-U69593benzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19465GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Nle818Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
85001MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
86025D4CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86281A1CLONEDHUMAN3H-CCPA8-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione41.7Koch P et al 2018Jan 15, 2025Jan 15, 2025
21001CLONEDRAT3H-NECA19210Shamim MT et al., 1989Jan 15, 2025Jan 15, 2025
86537A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
21513nAChRCLONEDXenopus3H-EpibatidineNFEP2.1Avalos M et al., 2002Jan 15, 2025Jan 27, 2025
87561Beta 1CLONEDHUMAN125I-Pindolol2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
22281A1CLONEDHUMAN125I-Aba4c3030Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878175-HT6CLONEDHUMAN3H-LSD4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline90Staron J et al 2016Jan 15, 2025Jan 15, 2025
22537hERGCLONEDHUMAN3H-MethylspiperoneQuetiapine5765Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88073A1CLONEDHUMAN3H-CCPA9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22793H2CLONEDHUMAN3H-TIOTIDINEL-homocysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23049nAChRCLONEDHUMAN3H-EpibatidineD-homocysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
88585M1CLONEDHUMAN3H-QNB1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
23561H3CLONEDRAT3H-NAMHA-3041212.51189Esbenshade TA, et al., 2003Jan 15, 2025Jan 15, 2025
893535-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide87Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240735-HT2ACLONEDHUMANUNDEFINEDSERTINDOLE0.3Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89865nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride378Liu J et al 2010Jan 15, 2025Jan 29, 2025
90121D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine4100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24841D5CLONEDHUMAN3H-SCH23390CLOZAPINE235PDSP Certified DataJan 15, 2025Jan 15, 2025
90633A2BCLONEDHUMAN3H-PSB-6033-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide801 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
253535-HT1ECLONEDHUMAN3H-5HTZOTEPINE1080PDSP Certified DataJan 15, 2025Jan 15, 2025
25609M2CLONEDHUMAN3H-QNBCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91145A1CLONEDHUMAN3H-DPCPXN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25865M2CLONEDHUMAN3H-QNBPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91401CB2CLONEDHUMAN3H-CP55940O-6618>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26121nAChR7CLONEDHUMAN3H-EpibatidinePseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91657A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26377GABAACLONEDRAT3H-RO-15-1788Amentoflavone6.17Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91913A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (2-chlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26633MORCLONEDHUMAN3H-DiprenorphineRutin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921695-HT6CLONEDHUMAN3H-LSD4-Fluoro-N-(1-{2-[2-(methylsulfanyl)phenoxy]ethyl} pyrrolidin-3-yl)benzenesulfonamide357Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268895-HT4CLONEDPIGLET125I-SB-207710xanomeline251.189Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92425KORCLONEDHUMAN3H-U695939,13:15,16-diepoxylabdane-6β,16β-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92681M1CLONEDHUMAN3H-QNB9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27401Beta2CLONEDHUMAN3H-CGP-12177TERGURIDE19.9526Millan MJ, et al., 2002Jan 15, 2025Jan 28, 2025
929375-HT6CLONEDHUMAN3H-LSD(RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine21Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276575-HT6CLONEDHUMAN3H-LSDMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279135-HT2ACLONEDHUMAN3H-DOBDMT,5-Me90Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28169H1CLONEDHUMAN3H-PYRILAMINEMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93705A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester15.7Federico S et al 2018Jan 15, 2025Jan 15, 2025
28425CLONEDHUMAN3H-QuisqualateL-Glutamate340Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93961D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one3.2Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28681D2CLONEDHUMAN3H-NMSPARIPIPRAZOLE0.74Shapiro DA, et.al., 2003Jan 15, 2025Jan 27, 2025
942175-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-ethoxyphenethylamine670Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29193SST2CLONEDHUMANUNDEFINEDBIM 2326815.1Patel YC, 1999Jan 15, 2025Jan 15, 2025
947295-HT2ACLONEDHUMAN3H-KETANSERIN4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94985D3CLONEDHUMAN3H-N-Methylspiperone4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29961H4CLONEDHUMAN3H-Histamine(4-Ethyl-piperazin-1-yl)-(1H-indol-2-yl)-methanone260Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30217KORCLONEDBOVINEUNDEFINEDDuloxetine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 27, 2025
957535-HT6CLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30473CLONEDXenopusUNDEFINED(S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-4-yl)methyl)amino]benzenepropaneamide bis(trifluoroacetate)330Kromann H, et. al., 2002aJan 15, 2025Jan 15, 2025
96009NETCLONEDHUMAN3H-NisoxetineTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30729CCK1CLONEDMOUSEUNDEFINEDAtomoxetine1000Bymaster F.P., et. al., 2002Jan 15, 2025Jan 15, 2025
96265Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30985Beta1CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
96521Alpha1BCLONEDHUMAN[3H]-prazosin6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
31241Alpha1BCLONEDHUMAN3H-PRAZOSINMDL 100907424.7PDSP Certified DataJan 15, 2025Jan 15, 2025
96777D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine7700Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314975-HT1BCLONEDHUMAN3H-5HT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)3162.28Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97033D3CLONEDHUMAN[3H]N-methylspiperoneFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97289MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o191Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97545A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32777NK2CLONEDHUMAN3H-NEUROKININ ASCH 2062720.4Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98313D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride418Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985695-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,723Ofon E et al 2016aJan 15, 2025Jan 15, 2025
332895-HT1DCLONEDHUMAN3H-GR-125743Acetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98825KORCLONEDHUMAN3H-U695931-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33545Alpha2BCLONEDHUMAN3H-CLONIDINENaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99081Beta1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99337D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(quinolin-3-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol244Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34057P2X3CLONEDHUMAN3H-A-317491Suramin1090Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99593A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine3.29Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34313nAChRCLONEDRAT3H-EpibatidineMCC969Grinevich VP, et al., 2004Jan 15, 2025Jan 28, 2025
99849D2CLONEDHUMAN[3H]N-methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide2200Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
1001055-HT3CLONEDHUMAN3H-GR65630Quetiapine4330PDSP Certified DataJan 15, 2025Jan 15, 2025
34825CLONEDRAT3H-CP-55940PhAR, epoxy>10000Jan 15, 2025Jan 15, 2025
100361Alpha2CCLONEDHUMAN3H-RAUWOLSCINEILOPERIDONE5.6PDSP Certified DataJan 15, 2025Jan 28, 2025
100617CGRPCLONEDHUMANFunctionalN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100873Beta1CLONEDHUMAN125I-Pindolol1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1)6Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
35593CLONEDHUMAN3H-SQ 29548SQ 295484.1Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35849Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester9.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013855-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione34Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101641D5CLONEDHUMAN[3H]-SCH23390Perospirone1742PDSP Certified DataMar 21, 2025Jul 28, 2026
101897MORCLONEDHUMAN[3H]-DAMGOZiprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
36617D3CLONEDHUMAN125I-IODOSULPRIDEHALOPERIDOL4.4Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102153GABAACLONEDHUMAN[3H]-MuscimolNEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
37897MPP-9CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-nitro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione57Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38153CLONEDRAT3H-dexamethasoneC57H79N2O9Na310von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
39433Calcium channelCLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 28, 2025
396895-HT2BCLONEDHUMAN3H-5HTPINDOLOL,(+/-)2187.76Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40713mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one101Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41225CLONEDHUMAN125I-Chemokine5-(4-Hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41993M1CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42249CLONEDHUMANFunctionalcyanogen bromide, CNBr8.4Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42505CLONEDRABBITUNDEFINEDMotilin0.977237Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43017GAKCLONEDHUMAN3H-StaurosporineStaurosporine68Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43273CLK1CLONEDHUMAN3H-StaurosporineRoscovitine2100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43529FYNCLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43785JAK1CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44041STK4CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44297CaMKCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44553FYNCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44809ACK1CLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45065RIPK2CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45321LCKCLONEDHUMANFunctionalkenpaullone470Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45577SLC6A4CLONEDHUMAN3H-IMIPRAMINEDOXEPIN68Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458335-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46089Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46601SLC6A3CLONEDHUMAN3H-WIN 35,428(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46857M5CLONEDHUMAN3H-QNB(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47369Kainate receptorCLONEDHUMAN3H-Kainic acidLY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
47881SST1CLONEDHUMAN3H-thymidineBIM-239263.6Zatelli MC, et.al., 2002Jan 15, 2025Jan 15, 2025
48137Y2CLONEDHUMAN3H-Propionyl-NPYNPY [hPP(1-17), Ala31,Aib32], human500Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48649CLONEDHUMANFunctional1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.2Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49161MORCLONEDRAT3H-DAMGOLYS3220.92Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49673Y2CLONEDChicken[125I] - Peptide YYNPY, porcine0.346737Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49929mGluR2CLONEDRATFunctional(S)-2-Aminoadipic acid>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 28, 2025
50185Kainate receptorCLONEDUNDEFINED3H-AMPALY 3828844000Bortolotto, Z., et al., 1999Jan 15, 2025Jan 15, 2025
50441SLC6A4CLONEDHUMAN3H-CITALOPRAMN,N-Dimethyl-5-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine401Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581215-HT2ACLONEDHUMAN125I-DOIN-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate2.63Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58377H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5923>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58889nAChR7CLONEDHUMAN3H-EpibatidineNicotine323.5Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
591455-HT1ACLONEDHUMAN3H-WAY100635KETANSERIN1044Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59401D2CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4-(3-thienyl)benzamide1200Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59913H1CLONEDHUMAN3H-PYRILAMINE4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60169A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (phenylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide0.85Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60425GABAACLONEDHUMANFNZWY-S-230Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60681GABAACLONEDHUMANFNZXHE-I-09320Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60937GABAACLONEDHUMANFNZDM-1464.23Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61193GABAACLONEDHUMANFNZCD-21416.4Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61449GABAACLONEDHUMANFNZRY-03120.4Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617055-HT2ACLONEDHUMAN3H-KETANSERIN(Z)-N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-4-phenylbut-3-en-1-amine226Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62217SerotoninCLONEDHUMAN[3H] CitalopramNaphyrone41Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62473M4CLONEDHUMAN3H-QNB4-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
62985GABAACLONEDRAT3H-RO-15-1788DIAZEPAM9.8Costanzo A et al., 2002Jan 15, 2025Jan 27, 2025
63497Alpha2CCLONEDHUMAN3H-RAUWOLSCINERISPERIDONE9.1Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640095-HT6CLONEDHUMAN3H-LSD1-[1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one107.4Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642655-HT2ACLONEDHUMAN3H-KETANSERINTHIORIDAZINE19.0546Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64521CLONEDHUMAN3H-Estradiol4-hydroxytamoxifen100Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65289GABAACLONEDHUMAN[3H] FlunitrazepamSH-I-0301.89Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65546GABAACLONEDHUMAN[3H] FlunitrazepamMLT-I-701000Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65802GABAACLONEDHUMAN[3H] FlunitrazepamYT-61.039Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
660585-HT1BCLONEDHUMAN3H-5-CTMellpaladine B590Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66314D1CLONEDHUMAN3H-SCH233930Finazine1431Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66570Beta3CLONEDHUMANI-125-Pindolol3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66826Alpha1BCLONEDHUMAN3H-PRAZOSINN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
670825-HT3CLONEDHUMAN3H-GR1138081-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate671Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
673385-HT1BCLONEDHUMAN3H-5-CT1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67850D2CLONEDHUMAN3H-RACLOPRIDES)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
33385-HT1ACLONEDHUMAN3H-8-OH-DPATCGS 12066B44TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68874SST2CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH21000Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
35945-HT2CCLONEDRAT3H-MESULERGINESKF 812971510TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69130H3CLONEDHUMAN3H-HistamineAlpha-Methylhistamine-R6.30957Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
38505-HT2ACLONEDRAT3H-SPIPERONEILOPERIDONE3.1KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69386H1CLONEDHUMAN3H-PYRILAMINECHLORPROMAZINE0.18Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4106KORCLONEDHUMAN3H-U69,593NALTRINDOLE10.1TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69642Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43625-HT6CLONEDHUMAN3H-LSDCLOZAPINE9.5KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69898D2CLONEDHUMAN3H-N-Methylspiperone4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4618SLC6A3CLONEDHUMAN3H-DA UPTAKENOREPINEPHRINE8500PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48745-HT2BCLONEDHUMAN3H-5HT1-NP3.25WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704105-HT2BCLONEDHUMAN3H-LSDMRP42688.6Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51305-HT2BCLONEDHUMAN3H-5HTDOAc313NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70666KORCLONEDHUMAN3H-U69,593MRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
53865-HT2BCLONEDRAT3H-5HTYOHIMBINE50.11BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
709225-HT2BCLONEDHUMAN3H-LSD(4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione231Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
71178D5CLONEDHUMAN3H-SCH23390CLOZAPINE454Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5898Alpha2BCLONEDHUMAN3H-RAUWOLSCINEKETANSERIN199WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714345-HT7CLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine724Klein LM et al 2018Jan 15, 2025Jan 15, 2025
6154Alpha1BCLONEDRAT125I-HEATWB 410128.6LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64105-HT3CLONEDGUINEA PIG3H-BIMU-1BIMU 820BONHAUS DW, ET AL., 1993Jan 15, 2025Jan 15, 2025
6666D4CLONEDHUMAN3H-NEMONAPRIDECHLORPROMAZINE22SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
69225-HT2ACLONEDHUMAN3H-KETANSERINPERLAPINE30SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72714D1CLONEDHUMAN3H-SCH23390naringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7434MORCLONEDHUMAN3H-DAMGONALTREXONE-HCl1Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
72970Alpha2BCLONEDHUMAN3H-RAUWOLSCINEcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7690GABAACLONEDHUMAN3H-MUSCIMOLThiomuscimol13.18Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7946GABAACLONEDHUMAN3H-RO-15-178891162He X, et al., 1999Jan 15, 2025Jan 27, 2025
8202SST5CLONEDHUMAN125I-LTT-SST-28SMS 201-99514.16Panetta R, et al., 1993Jan 15, 2025Jan 15, 2025
8458SST5CLONEDHUMAN125I-Tyr3-octreotideoctreotide-Tyr33.89Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8714SST2CLONEDHUMAN125I-Tyr3-octreotideCGP 239961.12Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8970SST2CLONEDHUMAN125I-SRIF-28SS-250.31Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74506Alpha1ACLONEDHUMAN3H-PRAZOSIN(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9226SST2CLONEDMOUSE125I-MK-678L-363,57226Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74762D5CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9482MT1CLONEDHUMAN125I-IodomelatoninMELATONIN0.56Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
75018M2CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9738MT2CLONEDHUMAN125I-IodomelatoninMelatonin,6-Methoxy3.5Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
752745-HT1ACLONEDHUMAN3H-WAY100635Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9994CB2CLONEDMOUSE3H-CP-55940JWH-0510.72Griffin G, Tao Q, Abood ME, 2000Jan 15, 2025Jan 15, 2025
75530Alpha1ACLONEDHUMAN3H-PRAZOSINpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10250CLONEDHAMSTER125I-HEATPRAZOSIN0.12Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75786Beta3CLONEDHUMAN125I-Pindolol1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76042MORCLONEDHUMAN3H-DAMGOEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate1770Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
107625-HT2CCLONEDRAT3H-LSDRILAPINE25.11ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
76298NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
765545-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76810Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77066Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77322D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77578D4CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77834H3CLONEDHUMAN3H-Alpha-methylhistamine(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78090M3CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78346SERTCLONEDHUMAN3H-CITALOPRAM(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78602MORCLONEDHUMAN3H-DAMGO(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78858KORCLONEDHUMAN3H-U69593(±)-(4aR,8S,8aR)-N-(2,6-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791145-HT5ACLONEDHUMAN3H-LSDR,R-2b12.7Ray TS 2010 Jan 15, 2025Jan 15, 2025
79370Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-3,4-Methylenedioxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14090Alpha2ACLONEDPIG3H-Yohimbinep-AMINOCLONIDINE288.4Brink CB, et al., 2000Jan 15, 2025Jan 15, 2025
79626CLONEDHUMAN3H-CLONIDINEDMT650.3Ray TS 2010 Jan 15, 2025Jan 15, 2025
79882M5CLONEDHUMAN3H-QNB4-Ethyl-2,5-dimethoxyphenethylamine1725Ray TS 2010 Jan 15, 2025Jan 15, 2025
146025-HT1ACLONEDHUMAN3H-8-OH-DPATSB-277011-A5011.87Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80138V2CLONEDHUMAN3H-VASOPRESSIN(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14858D1CLONEDRATUNDEFINEDQuetiapine390Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
803945-HT1BCLONEDHUMAN3H-5-CT(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15114PTGFRCLONEDHUMAN3H-PGF2AlphaAGN 190910>10000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806505-HT2CCLONEDHUMAN3H-MESULERGINE(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153705-HT1BCLONEDHUMAN3H-5HT5-Hydroxy Tryptamine4.26BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809065-HT6CLONEDHUMAN3H-LSD(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
156265-HT2BCLONEDRAT3H-5HTRITANSERIN5.12BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
811625-HT1BCLONEDHUMAN3H-5-CTN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158825-HT7CLONEDRATUNDEFINEDMETERGOLINE63.09BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81418H1CLONEDHUMAN3H-PYRILAMINE1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16138D1CLONEDHUMAN3H-SCH23390SCH 233900.35Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81674D4CLONEDHUMAN3H-N-Methylspiperone(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
81930H4CLONEDHUMAN3H-Histamine(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16650M1CLONEDHUMAN3H-QNBTrihexyphenidyl1.6Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82186D3CLONEDHUMAN3H-N-Methylspiperone2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one56Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82442Alpha1DCLONEDHUMAN3H-PRAZOSIN(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
826985-HT5ACLONEDHUMAN3H-LSD(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17674CLONEDHUMAN125I-VIPVIP [D-Asp8]110Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832105-HT2ACLONEDHUMAN125I-DOIKETANSERIN7.6Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83466M2CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+)13.8038Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
837225-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide9987PDSP Certified DataJan 15, 2025Jan 15, 2025
83978KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide3216PDSP Certified DataJan 15, 2025Jan 28, 2025
18954H1CLONEDGUINEA PIG3H-MEPYRAMINEtrans-H2-PAT(+/-)1.53Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84490DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19210CLONEDRAT125I-VIPVIP [D-His1]200Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84746DORCLONEDHUMAN3H-DADLEphenyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19466GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Leu945Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
85002MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19722D2CLONEDHUMANUNDEFINEDBENPERIDOL0.027Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
86026M1CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
21002CLONEDRAT3H-NECA205300Shamim MT et al., 1989Jan 15, 2025Jan 15, 2025
86538A1CLONEDHUMAN3H-CCPA1-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione2440Koch P et al 2018Jan 15, 2025Jan 15, 2025
21514nAChRCLONEDXenopus3H-EpibatidineNEP11Avalos M et al., 2002Jan 15, 2025Jan 27, 2025
87562Beta3CLONEDHUMAN125I-Pindolol2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
22282A1CLONEDHUMAN125I-Aba4d6.82Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878185-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline79Staron J et al 2016Jan 15, 2025Jan 15, 2025
22538hERGCLONEDHUMAN3H-MethylspiperoneOLANZAPINE6013Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88074A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22794H2CLONEDHUMAN3H-TIOTIDINED-homocysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23050nAChRCLONEDHUMAN3H-EpibatidineL-homocysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
88586Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine45.1Peprah K et al 2012Jan 15, 2025Jan 28, 2025
23562H3CLONEDHUMAN3H-NAMHA-304121758.578Esbenshade TA, et al., 2003Jan 15, 2025Jan 15, 2025
893545-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide44Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240745-HT2ACLONEDHUMANUNDEFINEDTHIORIDAZINE1.1Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89610D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89866nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride133Liu J et al 2010Jan 15, 2025Jan 29, 2025
90122D1CLONEDHUMAN3H-SCH23390Mescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
248425-HT6CLONEDHUMAN3H-LSDCLOZAPINE17PDSP Certified DataJan 15, 2025Jan 15, 2025
90378A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide193Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90634A2BCLONEDHUMAN3H-PSB-6033-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25354H2CLONEDHUMAN3H-TIOTIDINEZOTEPINE500PDSP Certified DataJan 15, 2025Jan 15, 2025
91146A2ACLONEDHUMAN3H-CGS-21680N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide3310Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25866D2CLONEDHUMAN3H-NMSPPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91402CB1CLONEDHUMAN3H-CP55940O-661889Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91658A3CLONEDHUMAN3H-PSB-11N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26378NETCLONEDHUMAN3H-NisoxetineHyperforin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91914A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3,4-dichlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26634MORCLONEDHUMAN3H-DiprenorphineQuercetin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921705-HT6CLONEDHUMAN3H-LSD4-Fluoro-N-{1-[2-(phenoxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide248Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268905-HT1ACLONEDHUMAN3H-8-OH-DPATxanomeline63.0957Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92426KORCLONEDHUMAN3H-U695939,13:15,16-diepoxylabdane-6β,16α-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92682H1CLONEDHUMAN3H-PYRILAMINE(5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
27402Beta1CLONEDHUMAN3H-CGP-12177TERGURIDE660.693Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929385-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine16Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276585-HT5ACLONEDHUMAN3H-LSDMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279145-HT2ACLONEDHUMAN3H-KETANSERINDOI52Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28170D4CLONEDHUMAN3H-NMSPMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93706A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester6.73Federico S et al 2018Jan 15, 2025Jan 15, 2025
28426mGluR5CLONEDHUMAN3H-QuisqualateL-Glutamate700Mutel V, et.al., 2000Jan 15, 2025Jan 28, 2025
93962D2CLONEDHUMAN3H-SPIPERONE7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one26Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28682D2CLONEDHUMAN3H-NMSPARIPIPRAZOLE3.3Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942185-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-methallyloxyphenethylamine40Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29194SST2CLONEDHUMANUNDEFINEDseglitide0.1Patel YC, 1999Jan 15, 2025Jan 15, 2025
947305-HT2ACLONEDHUMAN3H-KETANSERIN4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94986D3CLONEDHUMAN3H-N-Methylspiperone4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29962H4CLONEDHUMAN3H-Histamine+-(1H-Indol-2-yl)-(3-methyl-piperazin-1-yl)-methanone202Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30218GABAACLONEDBOVINEUNDEFINEDDuloxetine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 15, 2025
957545-HT7CLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96010NETCLONEDHUMAN3H-NisoxetineTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30730CCK2CLONEDMOUSEUNDEFINEDAtomoxetine1000Bymaster F.P., et. al., 2002Jan 15, 2025Jan 15, 2025
96266Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30986Beta2CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 28, 2025
96522Alpha2ACLONEDHUMAN3H-RAUWOLSCINE6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jul 30, 2025
31242H1CLONEDHUMAN3H-PYRILAMINEMDL 10090766.7PDSP Certified DataJan 15, 2025Jan 15, 2025
96778D1CLONEDHUMAN[3H]SCH233901-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314985-HT1BCLONEDHUMAN3H-5HT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)3981.07Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97034D4CLONEDHUMAN[3H]N-methylspiperoneFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97290MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol29.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97546A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (789Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32778NK2CLONEDHUMAN3H-NEUROKININ ACP 99994>10000Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98314D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985705-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride358Ofon E et al 2016aJan 15, 2025Jan 15, 2025
332905-HT2ACLONEDHUMAN3H-KETANSERINAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98826M1CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
33546Alpha2CCLONEDHUMAN3H-CLONIDINENaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99082Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99338D2CLONEDHUMAN[3H]N-methylspiperonePG648746Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34058P2X3CLONEDHUMAN3H-A-317491PPADS3470Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99594A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine1.52Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34314nAChRCLONEDRAT3H-EpibatidineSIB-1508Y991Grinevich VP, et al., 2004Jan 15, 2025Jan 28, 2025
99850D2CLONEDHUMAN[3H]N-methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
1001065-HT5ACLONEDHUMAN3H-LSDQuetiapine2300PDSP Certified DataJan 15, 2025Jan 15, 2025
34826CLONEDRAT3H-CP-55940PhAR, Cycloproyl>10000Jan 15, 2025Jan 15, 2025
100362DATCLONEDHUMAN3H-WIN35428ILOPERIDONE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100618CGRPCLONEDHUMANFunctionalN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamine>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100874Beta1CLONEDHUMAN125I-Pindolol1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)7Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
35594CLONEDHUMAN3H-SQ 29548U4661935Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35850SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester2.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
101386D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione118Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
101642SERTCLONEDHUMAN[3H]CitalopramPerospirone984PDSP Certified DataMar 21, 2025Jul 28, 2026
101898DORCLONEDHUMAN[3H]DADLEZiprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
36618D3CLONEDHUMAN125I-IODOSULPRIDECLOZAPINE242Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102154H1CLONEDHUMAN[3H]PyrilamineNEMONAPRIDE741PDSP Certified DataMar 25, 2025Jul 28, 2026
37898MPP-2CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-iodo-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione86Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38154CLONEDRAT3H-dexamethasoneC55H77N2O81000von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
39434Calcium channelCLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 28, 2025
396905-HT2BCLONEDHUMAN3H-5HTQUINPIROLE301.995Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40714mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one901Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41226CLONEDHUMAN125I-Chemokine1-(4-Cyano-4,4-diphenylbutyl)-4-phenylpiperidine-4-carbonitrile >10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41994M1CLONEDHUMAN3H-QNBFemoxetine92Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42250CLONEDHUMAN125I-[Ile]MotilinK368,374C0.6Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42506CLONEDRABBITUNDEFINED[Nle13]-Motilin0.851138Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43018GAKCLONEDHUMAN3H-StaurosporineSB202190650Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43274CLK1CLONEDHUMAN3H-StaurosporineFlavopiridol2200Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43530HCKCLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43786PKMYT1CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44042SykCLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44298CaMKCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44554GAKCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44810STK6CLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45066RPS6KA3CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45322CDK2CLONEDHUMANFunctionalalsterpaullone80Bain J, et al., 2003Jan 15, 2025Jan 28, 2025
45578NETCLONEDHUMAN3H-NisoxetineDOXEPIN29.5Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458345-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46090Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46602SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46858M5CLONEDHUMAN3H-QNBPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47114M3CLONEDHUMAN3H-NMSIodophenpropit3700Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47370Grik5CLONEDHUMAN3H-Kainic acidLY 46619550Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47882SST2CLONEDHUMAN3H-thymidineBIM-239261000Zatelli MC, et.al., 2002Jan 15, 2025Jan 15, 2025
48138Y2CLONEDHUMAN3H-Propionyl-NPYNPY [Ala31, Aib32], porcine500Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48650CLONEDHUMANFunctional1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.3Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
48906Y1CLONEDChicken[125I] - Peptide YYPYY, chicken5.12861Holmberg, SK et al., 2002Jan 15, 2025Jan 15, 2025
49162CCK1CLONEDHUMAN125I-CCK-8LYS201>10000Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49674Y2CLONEDChicken[125I] - Peptide YYNPY2-36, porcine0.549541Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49930mGluR4CLONEDRATFunctional(S)-2-Aminoadipic acid>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 28, 2025
50186Kainate receptorCLONEDUNDEFINED3H-AMPALY 382884>10000Bortolotto, Z., et al., 1999Jan 15, 2025Jan 28, 2025
50442SLC6A4CLONEDHUMAN3H-CITALOPRAMN,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine445Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581225-HT2ACLONEDHUMAN3H-KETANSERINN-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate21.4Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58378H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5930>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58890nAChR7CLONEDHUMAN3H-EpibatidineKodiak extract202.1Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
591465-HT2ACLONEDHUMAN3H-KETANSERINMETHYSERGIDE3.25Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59402D4CLONEDHUMAN3H-N-MethylspiporoneN-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(2-thienyl)benzamide24Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59914H2CLONEDHUMAN3H-Cimetidine4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60170A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-4-(2-(Biphenyl-4-ylethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide3.1Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60426GABAACLONEDHUMANFNZWY-S-6120Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60682GABAACLONEDHUMANFNZXHE-I-0931162Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60938GABAACLONEDHUMANFNZDM-146148Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61194GABAACLONEDHUMANFNZCD-21448.2Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61450GABAACLONEDHUMANFNZRY-03127Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617065-HT2ACLONEDHUMAN3H-KETANSERINCLOZAPINE15Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
61962CLONEDHUMANUNDEFINEDazimilide1400Busch ,AE et al., 1998Jan 15, 2025Jan 15, 2025
62218SerotoninCLONEDHUMAN[3H] CitalopramI-Naphyrone34Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62474M5CLONEDHUMAN3H-QNBDiphenidine1653Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
62986GABAACLONEDRAT3H-RO-15-1788Zolpidem>10000Costanzo A et al., 2002Jan 15, 2025Jan 27, 2025
63498H1CLONEDHUMAN3H-PYRILAMINERISPERIDONE27Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640105-HT6CLONEDHUMAN3H-LSD1-[1-(Naphthalene-1-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one51.7Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642665-HT2ACLONEDHUMAN3H-KETANSERINtiotixene89.1251Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64522CLONEDHUMAN3H-Estradiolraloxifene18Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65290GABAACLONEDHUMAN[3H] FlunitrazepamXLI-34813.56Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65547GABAACLONEDHUMAN[3H] FlunitrazepamXHE-III-041.2Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65803GABAACLONEDHUMAN[3H] FlunitrazepamPWZ-09611.1Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
660595-HT1DCLONEDHUMAN3H-5-CTMellpaladine B489Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66315D2CLONEDHUMAN3H-N-MethylspiperoneFinazine1412Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66571Beta2CLONEDHUMAN3H-CGP121773-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66827Alpha1DCLONEDHUMAN3H-PRAZOSINN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
670835-HT2CCLONEDHUMAN3H-MESULERGINE1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
673395-HT1DCLONEDHUMAN3H-5-CT1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride4549Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
678515-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33395-HT1ACLONEDHUMAN3H-8-OH-DPATCHLORPROMAZINE3115TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68875SST3CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH21000Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
35955-HT2CCLONEDRAT3H-MESULERGINESPIPERONE4094TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69131H3CLONEDHUMAN3H-HistamineAlpha-Methylhistamine-S63.0957Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
38515-HT2ACLONEDRAT3H-SPIPERONERISPERIDONE1.4KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69387H1CLONEDHUMAN3H-PYRILAMINERACLOPRIDE8430Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4107KORCLONEDHUMAN3H-U69,593BNTX3.7TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69643Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43635-HT6CLONEDHUMAN3H-LSDOLANZAPINE10KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69899D2CLONEDHUMAN3H-N-Methylspiperone4-[1-(3-methylphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4619SLC6A3CLONEDHUMAN3H-DA UPTAKE5-Hydroxy Tryptamine>10000PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48755-HT2BCLONEDHUMAN3H-RAUWOLSCINELSD,2-Bromo7.47WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704115-HT1ACLONEDHUMAN3H-WAY100635MRP42685.6Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51315-HT2BCLONEDHUMAN3H-5HTDON166NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70667MORCLONEDHUMAN3H-DAMGOMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
53875-HT2BCLONEDRAT3H-5HTmCPP25.11BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
709235-HT7CLONEDHUMAN3H-LSD(4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione2765Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
71179D5CLONEDHUMAN3H-SCH23390SYA162631451Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5899Alpha2BCLONEDHUMAN3H-RAUWOLSCINEOXYMETAZOLINE213WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
71435SERTCLONEDHUMAN3H-CITALOPRAM4-acetoxy-N,N-diallyltryptamine1089Klein LM et al 2018Jan 15, 2025Jan 28, 2025
6155Alpha1CCLONEDBOVINE125I-HEATEPINEPHRINE6250LOMASNEY JW, ET AL., 1991Jan 15, 2025Jan 15, 2025
64115-HT3CLONEDRAT3H-BIMU-15-Hydroxy Tryptamine501BONHAUS DW, ET AL., 1993Jan 15, 2025Jan 15, 2025
72203H1CLONEDHUMAN3H-PYRILAMINE2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69235-HT2ACLONEDHUMAN3H-KETANSERINRACLOPRIDE5400SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72715D5CLONEDHUMAN3H-SCH23390naringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7435MORCLONEDHUMAN3H-DAMGOBeta C N A0.9Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
72971Alpha2CCLONEDHUMAN3H-RAUWOLSCINEcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7691GABAACLONEDHUMAN3H-MUSCIMOLTHIP46.77Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7947GABAACLONEDHUMAN3H-RO-15-1788101000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8203SST5CLONEDHUMAN125I-LTT-SST-28MK 6785.02Panetta R, et al., 1993Jan 15, 2025Jan 15, 2025
8459SST5CLONEDHUMAN125I-Tyr3-octreotideL-362,8550.67Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8715SST2CLONEDHUMAN125I-Tyr3-octreotideL-362,8551.62Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8971SST2CLONEDHUMAN125I-SRIF-28somatostatin-280.19Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74507Alpha1BCLONEDHUMAN3H-PRAZOSIN(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9227SST2CLONEDMOUSE125I-MK-678L-363,376356Raynor K, et al., 1993aJan 15, 2025Jan 15, 2025
74763D2CLONEDHUMAN3H-N-Methylspiperone(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9483MT1CLONEDHUMAN125I-IodomelatoninN-Acetyltryptamine870Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
75019M3CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9739MT2CLONEDHUMAN125I-IodomelatoninSerotonin,N-acetyl189Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
752755-HT1BCLONEDHUMAN3H-5-CTEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9995CB2CLONEDHUMAN3H-CP-55940WIN 35,4281.19Griffin G, Tao Q, Abood ME, 2000Jan 15, 2025Jan 15, 2025
75531Alpha1BCLONEDHUMAN3H-PRAZOSINpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10251CLONEDHAMSTER125I-HEATSPIPERONE31.62Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
75787Beta 2CLONEDHUMAN3H-CGP121771S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
107635-HT2CCLONEDRAT3H-LSDFLUPERLAPINE19.95ROTH ET AL., 1993Jan 15, 2025Jan 15, 2025
765555-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76811Alpha1DCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77067Beta 1CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77323D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77579DATCLONEDHUMAN3H-WIN 35,428(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77835H4CLONEDHUMAN3H-Histamine(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78091M4CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78347Sigma 1CLONEDHUMAN3H-Pentazocine(+)(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
786035-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78859DORCLONEDHUMAN3H-DADLE(±)-(4aR,8S,8aR)-N-(2,6-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791155-HT5ACLONEDHUMAN3H-LSDS,S-2c27.3Ray TS 2010 Jan 15, 2025Jan 15, 2025
79371Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14091Alpha2ACLONEDPIG3H-YohimbineB-HT 9201000Brink CB, et al., 2000Jan 15, 2025Jan 15, 2025
79627CLONEDHUMAN3H-CLONIDINE4-Hydroxy-N,N-dimethyltryptamine792.2Ray TS 2010 Jan 15, 2025Jan 15, 2025
79883M5CLONEDHUMAN3H-QNB4-Ethylthio-2,5-dimethoxyphenethylamine1502Ray TS 2010 Jan 15, 2025Jan 15, 2025
146035-HT1BCLONEDHUMAN3H-5HTSB-277011-A6309.57Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
80139V2CLONEDHUMAN3H-VASOPRESSIN3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14859D1CLONEDRATUNDEFINEDZiprasidone9.5Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
803955-HT1DCLONEDHUMAN3H-5-CT(E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15115PTGFRCLONEDHUMAN3H-PGF2AlphaAGN 190911>10000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806515-HT3CLONEDHUMAN3H-GR-65630(Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153715-HT1BCLONEDHUMAN3H-5HTMETHYSERGIDE25.11BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809075-HT7CLONEDHUMAN3H-LSD(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
156275-HT2BCLONEDRAT3H-5HTMIANSERIN52.48BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
811635-HT1DCLONEDHUMAN3H-5-CTN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158835-HT7CLONEDRATUNDEFINEDLSD9.54BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81419H1CLONEDHUMAN3H-PYRILAMINEN-[[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-methylmethanamine>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16139D1CLONEDHUMAN3H-SCH23390SKF 835660.3Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
816755-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
81931KORCLONEDHUMAN3H-U69593(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16651M1CLONEDHUMAN3H-QNBProcyclidine4.6Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82187D4CLONEDHUMAN3H-N-Methylspiperone2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one264Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82443D1CLONEDHUMAN3H-SCH23390(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
826995-HT6CLONEDHUMAN3H-LSD(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17675CLONEDHUMAN125I-VIPVIP [D-Asn9]1.1Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832115-HT1ACLONEDHUMAN3H-8-OH-DPATKETANSERIN6510Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83467M1CLONEDHUMAN3H-NMS1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+)5.01187Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83723NETCLONEDHUMAN3H-Nisoxetine(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5904PDSP Certified DataJan 15, 2025Jan 15, 2025
184435-HT1ACLONEDHUMAN3H-5HT1-NP9.2Jorand-Lebrun C et al., 1997aJan 15, 2025Jan 15, 2025
83979KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-cyclohexyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one6292PDSP Certified DataJan 15, 2025Jan 28, 2025
84235M2CLONEDHUMAN3H-QNB(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide8259PDSP Certified DataJan 15, 2025Jan 15, 2025
18955H1CLONEDGUINEA PIG3H-MEPYRAMINEtrans-H2-PAT(+)23Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84491MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19211CLONEDRAT125I-VIPVIP(2-28)200Ciccarelli E et al., 1994Jan 15, 2025Jan 15, 2025
84747DORCLONEDHUMAN3H-DADLES-phenyl (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbothioate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19467GPR145CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Gly1037Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
85003DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19723D2CLONEDHUMANUNDEFINEDBROMOCRIPTINE2Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
86027M2CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86283A2BCLONEDHUMAN3H-PSB-6038-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
21003CLONEDRAT3H-NECA245600Shamim MT et al., 1989Jan 15, 2025Jan 15, 2025
86539A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione149Koch P et al 2018Jan 15, 2025Jan 15, 2025
87563Beta 2CLONEDHUMAN3H-CGP121772-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
22283A1CLONEDHUMAN125I-Aba51660Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
87819D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline691Staron J et al 2016Jan 15, 2025Jan 28, 2025
22539D2CLONEDHUMAN3H-MethylspiperoneSERTINDOLE6.55Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88075A1CLONEDHUMAN3H-CCPA9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3800Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
22795H2CLONEDHUMAN3H-TIOTIDINED-homocysteine thiolactone>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
23051nAChRCLONEDHUMAN3H-EpibatidineL-cysteine sulfinic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 27, 2025
88587Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine194.5Peprah K et al 2012Jan 15, 2025Jan 28, 2025
23563GPR10CLONEDHUMAN125I-PrRP20NPY18-367400Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
893555-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide802Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240755-HT2ACLONEDHUMANUNDEFINEDTrifluperazine7.4Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89611D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89867nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride3400Liu J et al 2010Jan 15, 2025Jan 29, 2025
90123D1CLONEDHUMAN3H-SCH23390LSD310Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24843M5CLONEDHUMAN3H-QNBCLOZAPINE94PDSP Certified DataJan 15, 2025Jan 15, 2025
90379A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide452Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25099H1CLONEDHUMAN3H-PYRILAMINEQuetiapine7.5PDSP Certified DataJan 15, 2025Jan 15, 2025
90635A2BCLONEDHUMAN3H-PSB-6032-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
253555-HT2ACLONEDRAT3H-KETANSERINZOTEPINE6PDSP Certified DataJan 15, 2025Jan 15, 2025
256115-HT3CLONEDHUMAN3H-ZACOPRIDECOCAINE1950PDSP Certified DataJan 15, 2025Jan 15, 2025
91147A3CLONEDHUMAN125I-AB-MECAN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25867mGluR8CLONEDRATFunctionalPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91403CB1CLONEDHUMAN3H-SR144528O-661844Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
261235-HT1BCLONEDHUMAN3H-GR-125743Pseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91659A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide174Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26379SLC6A3CLONEDBOVINE3H-WIN 35,428Amentoflavone877.4Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91915A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (2,4-dichlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
26635MORCLONEDHUMAN3H-DiprenorphineQuercitrin>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
921715-HT6CLONEDHUMAN3H-LSD4-Fluoro-N-{1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide96Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
268915-HT1BCLONEDHUMAN3H-5HTxanomeline50.1187Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
92427KORCLONEDHUMAN3H-U695939,13-epoxylabd-5-en-7-on-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92683H1CLONEDHUMAN3H-PYRILAMINE9,13:15,16-diepoxylabdane-6b,15a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
27403Beta1CLONEDHUMAN3H-CGP-12177TL99>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929395-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine6Sudol S et al 2020Jan 15, 2025Jan 15, 2025
276595-HT3CLONEDHUMAN3H-ZACOPRIDEMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279155-HT2ACLONEDHUMAN3H-DOBDOI3.1Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
28171D5CLONEDHUMAN3H-SCH23390METHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93707A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester4.88Federico S et al 2018Jan 15, 2025Jan 15, 2025
28427CLONEDHUMAN3H-QuisqualateDHPG900Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93963D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one38Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28683D3CLONEDHUMAN3H-NMSPARIPIPRAZOLE9.7Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942195-HT2ACLONEDHUMAN3H-KETANSERIN4-allyloxy-2,5-dimethoxyphenethylamine140Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29195SST2CLONEDHUMANUNDEFINEDVapreotide5.4Patel YC, 1999Jan 15, 2025Jan 15, 2025
947315-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94987D3CLONEDHUMAN3H-N-Methylspiperone4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29963H4CLONEDHUMAN3H-Histamine(1H-Indol-2-yl)-(4-phenethyl-piperazin-1-yl)-methanone7000Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30219GABAACLONEDBOVINEUNDEFINEDVenlafaxine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 15, 2025
957555-HT5ACLONEDHUMAN3H-LSDN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30475CLONEDXenopusUNDEFINED(S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-cyclohexylmethyl)amino]benzenepropaneamide bis(trifluoroacetate)240Kromann H, et. al., 2002aJan 15, 2025Jan 15, 2025
96011NETCLONEDHUMAN3H-Nisoxetine6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
30731NK1CLONEDRATUNDEFINEDAtomoxetine1000Bymaster F.P., et. al., 2002Jan 15, 2025Jan 15, 2025
96267Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30987A1CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
96523Beta1CLONEDHUMAN[125I]-Pindolol6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
31243H4CLONEDHUMAN3H-HistamineMDL 100907>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
96779D1CLONEDHUMAN[3H]SCH233901-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA8800Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314995-HT1DCLONEDHUMAN3H-5HT(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)501.187Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97035D5CLONEDHUMAN[3H]SCH23390Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97291MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o135Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97547A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate721Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
32779NK2CLONEDHUMAN3H-NEUROKININ ASR 489680.4Anthes, JC et al., 2002Jan 15, 2025Jan 15, 2025
98315D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline5647Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985715-HT2BCLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride232Ofon E et al 2016aJan 15, 2025Jan 15, 2025
332915-HT2BCLONEDHUMAN3H-LSDAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98827M2CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
33547M2CLONEDHUMAN3H-QNBNaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99083Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99339D2CLONEDHUMAN[3H]N-methylspiperoneOMO5-057321Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34059P2X3CLONEDHUMAN3H-A-317491KN-62>10000Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99595A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine2.43Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
34315nAChRCLONEDRAT3H-EpibatidineGTS-211290Grinevich VP, et al., 2004Jan 15, 2025Jan 28, 2025
99851D3CLONEDHUMAN[3H]N-methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
1001075-HT6CLONEDHUMAN3H-LSDQuetiapine1777PDSP Certified DataJan 15, 2025Jan 15, 2025
34827CLONEDRAT3H-CP-55940PhAR, Di-hydro>10000Jan 15, 2025Jan 15, 2025
100363NETCLONEDHUMAN3H-NisoxetineILOPERIDONE535PDSP Certified DataJan 15, 2025Jan 15, 2025
100619CGRPCLONEDHUMANFunctionalN2-[3,5-Dibromo-N-(4-phenyl-1-oxybutyl)-L-tyrosyl]-L-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
1008755-HT1ACLONEDHUMAN3H-WAY1006351-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)24.6Stephenson, K. et. al., 2008Jan 15, 2025Jan 15, 2025
35595CLONEDHUMAN3H-SQ 29548AH-23848592Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35851Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole47Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013875-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione35Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101643NETCLONEDHUMAN[3H] NisoxetinePerospirone303PDSP Certified DataMar 21, 2025Jul 28, 2026
101899KORCLONEDHUMAN[3H]U69593Ziprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
36619D3CLONEDHUMAN125I-IODOSULPRIDEOLANZAPINE43Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102155H2CLONEDHUMAN[3H]TiotidineNEMONAPRIDE2108PDSP Certified DataMar 25, 2025Jul 28, 2026
37899MPP-9CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-iodo-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione10Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38155CLONEDRAT3H-dexamethasoneC54H76NO71000von Geldern TW, et al, 2004Jan 15, 2025Jan 15, 2025
39435CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396915-HT2BCLONEDHUMAN3H-5HTQUIPAZINE85.1138Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40459mGluR5CLONEDRATFunctional(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40715mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4'-ethylphenyl)-3H-1,3,6-triazafluoren-4-one1460Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41227CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)piperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41995M1CLONEDHUMAN3H-QNBFLUOXETINE1030Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42251CLONEDHUMANFunctionalK368,374C0.3Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42507CLONEDRABBITUNDEFINEDerythromycin-A190.546Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
43019GAKCLONEDHUMAN3H-StaurosporineSB20358039Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43275CLK2CLONEDHUMAN3H-StaurosporineEKB-569700Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43531INSRCLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43787MAPK12CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44043TEKCLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44299CaMKCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44555HCKCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44811AURKCCLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45067SLKCLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45323CLONEDHUMANFunctionalalsterpaullone110Bain J, et al., 2003Jan 15, 2025Jan 15, 2025
45579SLC6A3CLONEDHUMAN3H-WIN 35,428DOXEPIN>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458355-HT2BCLONEDHUMAN3H-LSD(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46091Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46603SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46859M5CLONEDHUMAN3H-QNB(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47115M3CLONEDHUMAN3H-NMSThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47371Grik5CLONEDHUMAN3H-Kainic acidLY 4576911550Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47883SST3CLONEDHUMAN3H-thymidineBIM-239261000Zatelli MC, et.al., 2002Jan 15, 2025Jan 15, 2025
48139Y2CLONEDHUMAN3H-Propionyl-NPYNPY, human0.04Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48651CLONEDHUMANFunctional1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride12.1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
48907Y1CLONEDChicken[125I] - Peptide YYNPY, porcine0.213796Holmberg, SK et al., 2002Jan 15, 2025Jan 15, 2025
49163CCK1CLONEDHUMAN125I-CCK-8TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-1-Adoc840Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49675Y2CLONEDChicken[125I] - Peptide YYNPY 3-36, porcine0.74131Salaneck E, et al., 2000Jan 15, 2025Jan 15, 2025
49931mGluR6CLONEDRATFunctional(S)-2-Aminoadipic acid>10000Brauner-Osborne H, et.al., 1996Jan 15, 2025Jan 15, 2025
50187Kainate receptorCLONEDUNDEFINED3H-Kainic acidLY 382884>10000Bortolotto, Z., et al., 1999Jan 15, 2025Jan 28, 2025
50443SLC6A4CLONEDHUMAN3H-CITALOPRAMN,N-Dimethyl-5-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine7Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
581235-HT2ACLONEDHUMAN3H-KETANSERINN-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate5.25Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58379H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5474>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58891nAChR7CLONEDHUMAN3H-EpibatidineCamel Snus extract195.3Harris A, et al., 2015Jan 15, 2025Jan 15, 2025
591475-HT1ACLONEDHUMAN3H-WAY100635METHYSERGIDE25Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025