101895 NET CLONED HUMAN [3H]Nisoxetine Ziprasidone 69 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36615 D2 CLONED HUMAN 3H-SPIPERONE MIANSERIN 2197 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102151 DOR CLONED HUMAN [3H]DADLE NEMONAPRIDE >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37895 MPP-9 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 19 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38151 CLONED RAT 3H-dexamethasone C30H36NO3 1000 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
39175 D4 CLONED HUMAN R-SAT N-DESMETHYLCLOZAPINE 70 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39431 V2 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39687 5-HT2B CLONED HUMAN 3H-5HT ORG-12962 91.2011 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40711 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one 84 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41223 CLONED HUMAN 125I-Chemokine 5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41991 M1 CLONED HUMAN 3H-QNB Dothiepin 18 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42247 CLONED HUMAN 125I-[Ile]Motilin [L-Bpa5,Ile13]Motilin 50 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42759 CLONED UNDEFINED Functional Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-beta-Ala-Cys (O))-amide (S) >10000 Song YL, et al., 2006 Jan 15, 2025 Jan 15, 2025
43015 FYN CLONED HUMAN 3H-Staurosporine Gleevec 5500 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43271 CLK1 CLONED HUMAN 3H-Staurosporine SU11248 100 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43527 FLT3 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43783 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44039 STK36 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44295 CaMK CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44551 FLT4 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44807 MAPK12 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45063 PTK2 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45319 CDK2 CLONED HUMAN Functional kenpaullone 670 Bain J, et al., 2003 Jan 15, 2025 Jan 28, 2025
45575 NET CLONED HUMAN 3H-Nisoxetine Dothiepin 46 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45831 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46087 Alpha2A CLONED HUMAN 3H-CLONIDINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46599 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46855 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47367 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
48135 Y2 CLONED HUMAN 3H-Propionyl-NPY PP, human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48647 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49159 MOR CLONED RAT 3H-DAMGO LYS328 20 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
49671 SST5 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
49927 mGluR6 CLONED RAT Functional D-Glutamate >10000 Brauner-Osborne H, et.al., 1996 Jan 15, 2025 Jan 15, 2025
50183 mGluR3 CLONED HUMAN Functional L-CCG-I 2100 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50439 SLC6A4 CLONED HUMAN 3H-CITALOPRAM 5-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 8 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
58119 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 427 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58375 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5755 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58631 hERG CLONED HUMAN 3H-N-Me-Dofetilide MRS5474 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
59143 5-HT2A CLONED HUMAN 3H-KETANSERIN HALOPERIDOL 30 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59399 D2 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4-(2-thienyl)benzamide 840 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59911 D4 CLONED HUMAN 3H-NMSP 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60167 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-4-(2-(Cyclohexylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60423 GABAA CLONED HUMAN FNZ WY-S-2 100 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60679 GABAA CLONED HUMAN FNZ XHE-I-093 8.9 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60935 GABAA CLONED HUMAN FNZ 3 EBC 1000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61191 GABAA CLONED HUMAN FNZ QH-II-067a 31 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61447 GABAA CLONED HUMAN FNZ RY-054 44 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61703 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine 1507 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62215 SLC6A3 CLONED HUMAN [3H] WIN35428 Benzedrone 1089 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62471 M4 CLONED HUMAN 3H-QNB 2-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
62983 GABAA CLONED RAT 3H-RO-15-1788 Zolpidem 383 Costanzo A et al., 2002 Jan 15, 2025 Jan 27, 2025
63495 5-HT2B CLONED HUMAN 3H-LSD RISPERIDONE 35 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64007 5-HT6 CLONED HUMAN 3H-LSD 1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 125.8 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64263 5-HT2A CLONED HUMAN 3H-KETANSERIN SERTINDOLE 0.323594 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64519 D2 CLONED HUMAN 3H-N-Methylspiperone PROCHLORPERAZINE 2.23872 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65287 GABAA CLONED HUMAN [3H] Flunitrazepam SH-I-030 11.04 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65544 GABAA CLONED HUMAN [3H] Flunitrazepam MLT-I-70 1.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65800 GABAA CLONED HUMAN [3H] Flunitrazepam YT-6 87.8 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66056 5-HT1A CLONED HUMAN 3H-WAY100635 Mellpaladine A 7500 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66312 Beta3 CLONED HUMAN I-125-Pindolol Finazine >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66568 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 52 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66824 5-HT7 CLONED HUMAN 3H-LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67080 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67848 5-HT2A CLONED HUMAN 3H-KETANSERIN S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 91 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3336 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BROMOCRIPTINE,(+) 25 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68872 SST5 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 79.4328 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
3592 5-HT2C CLONED RAT 3H-MESULERGINE SKF 38393 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69128 H3 CLONED HUMAN 3H-Histamine HISTAMINE 10 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3848 D2 CLONED RAT 3H-SPIPERONE Quetiapine 329 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69384 H1 CLONED HUMAN 3H-PYRILAMINE HALOPERIDOL 4160 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4104 KOR CLONED HUMAN 3H-U69,593 Leu-ENKEPHALIN >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69640 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE DPH 4376 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4360 5-HT6 CLONED HUMAN 3H-LSD 8-OH-DPAT >10000 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69896 D2 CLONED HUMAN 3H-N-Methylspiperone 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4616 SLC6A3 CLONED HUMAN 3H-DA UPTAKE BUPROPION 784 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4872 5-HT2B CLONED HUMAN 3H-5HT YOHIMBINE 43.2 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70408 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) MRP4268 5.5 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5128 5-HT2B CLONED HUMAN 3H-5HT TMA 307 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70664 NET CLONED HUMAN 3H-Nisoxetine MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5384 5-HT2B CLONED HUMAN 3H-5HT SB200646a 630.95 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
70920 5-HT2B CLONED HUMAN 3H-LSD (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 840 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
5640 5-HT4 CLONED RAT 3H-GR-113808 5-CT 9120.1 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
71176 D5 CLONED HUMAN 3H-SCH23390 ARIPIPRAZOLE 2590 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5896 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE MIANSERIN 27 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71432 5-HT5A CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 5844 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6152 Alpha1B CLONED RAT 125I-HEAT INDORAMINE 226 LOMASNEY JW, ET AL., 1991 Jan 15, 2025 Jan 15, 2025
6408 5-HT3 CLONED GUINEA PIG 3H-BIMU-1 ZACOPRIDE,R >10000 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
72200 DAT CLONED HUMAN 3H-WIN35428 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 15, 2025
6920 5-HT2A CLONED HUMAN 3H-KETANSERIN MOLINDONE 5800 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72712 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7432 MOR CLONED HUMAN 3H-DAMGO DIPRENORPHINE-HCl 0.07 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72968 Alpha1D CLONED HUMAN 3H-PRAZOSIN catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7688 GABAA CLONED HUMAN 3H-MUSCIMOL Gamma-Aminobutyric acid 8.7 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7944 GABAA CLONED HUMAN 3H-RO-15-1788 6 1000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8200 SST5 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.24 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
8456 SST5 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 2.08 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8712 SST2 CLONED HUMAN 125I-Tyr3-octreotide RC 160 0.31 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8968 SST1 CLONED HUMAN 125I-SRIF-28 L-363,301 630.95 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74504 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9224 SST2 CLONED MOUSE 125I-MK-678 MK 678 0.18 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9736 MT2 CLONED HUMAN 125I-Iodomelatonin 8-M-PDOT 3 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75272 NOP CLONED HUMAN 3H-Nociceptin ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate 9400 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
9992 CB2 CLONED MOUSE 3H-CP-55940 SR 144528 0.05 Griffin G, Tao Q, Abood ME, 2000 Jan 15, 2025 Jan 15, 2025
75528 5-HT6 CLONED HUMAN 3H-LSD propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10248 CLONED HAMSTER 125I-HEAT Niguldipine(+) 501.18 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75784 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76040 DOR CLONED HUMAN 3H-DADLE Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate 627 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10760 D2 CLONED RAT 3H-LSD RACLOPRIDE 1.99 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
76296 SERT CLONED HUMAN 3H-CITALOPRAM (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76552 5-HT3 CLONED HUMAN 3H-GR-65630 (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76808 5-HT7 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77064 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77320 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77576 D2 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77832 H1 CLONED HUMAN 3H-PYRILAMINE (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78088 M1 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78344 M5 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78600 DOR CLONED HUMAN 3H-DADLE (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78856 DOR CLONED HUMAN 3H-DADLE (±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79112 5-HT5A CLONED HUMAN 3H-LSD LYSERGIC ACID 9 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79368 Alpha1A CLONED HUMAN 3H-PRAZOSIN Salvinorin A >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14088 Alpha2A CLONED PIG 3H-Yohimbine Isoproterenol-l >10000 Brink CB, et al., 2000 Jan 15, 2025 Jan 15, 2025
79624 CLONED HUMAN 3H-CLONIDINE 3,4,5-Trimethoxyphenethylamine 2677.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79880 M5 CLONED HUMAN 3H-QNB DMT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14600 D3 CLONED HUMAN 125I-IODOSULPRIDE SB-277011-A 11.22 Reavill C., et al., 2000 Jan 15, 2025 Jan 15, 2025
80136 CLONED HUMAN 3H-VASOPRESSIN EMDT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14856 D1 CLONED RAT UNDEFINED OLANZAPINE 10 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
80392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 3215 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15112 PTGFR CLONED HUMAN 3H-PGF2Alpha AGN 191365 >10000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80648 5-HT2A CLONED HUMAN 3H-KETANSERIN (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15368 5-HT1B CLONED HUMAN 3H-5HT CGS 12066B 2.08 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80904 5-HT4 CLONED HUMAN 3H-GR113808 (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 603 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15624 5-HT2B CLONED RAT 3H-5HT AMESERGIDE 10.71 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81160 H4 CLONED HUMAN 3H-Histamine N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
15880 5-HT7 CLONED RAT UNDEFINED 5-Methoxytryptamine 0.93 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81416 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 15, 2025
16136 D1 CLONED HUMAN 3H-SCH23390 NOREPINEPHRINE >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81672 D2 CLONED HUMAN 3H-N-Methylspiperone (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81928 5-HT1D CLONED HUMAN 3H-Cimetidine (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16648 M1 CLONED HUMAN 3H-QNB ATR 0.5 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82184 D5 CLONED HUMAN 3H-SCH23390 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82440 Alpha1A CLONED HUMAN 3H-PRAZOSIN (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82696 5-HT3 CLONED HUMAN 3H-GR65630 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17672 CLONED HUMAN 125I-VIP VIP [D-Thr7] 162 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83208 5-HT2C CLONED HUMAN 125I-DOI DOM 25.7 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83464 M4 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 35.4813 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83720 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83976 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N-(3-bromobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 438 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84232 DOR CLONED HUMAN 3H-DADLE (±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide 2471 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18952 H1 CLONED GUINEA PIG 3H-MEPYRAMINE CLOZAPINE 1.23 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84488 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84744 DOR CLONED HUMAN 3H-DADLE benzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19464 GPR145 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH hAc-MCH(6-16)-NH2 2.7 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
85000 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86024 D3 CLONED HUMAN 3H-Alpha-methylhistamine (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
21000 CLONED RAT 3H-NECA 18 250 Shamim MT et al., 1989 Jan 15, 2025 Jan 15, 2025
86536 A2B CLONED HUMAN 3H-PSB-603 1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1000 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
21512 nAChR CLONED Xenopus 3H-Epibatidine NNEP 7.2 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
87560 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
22280 A1 CLONED HUMAN 125I-Aba 4a 175 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87816 D2 CLONED HUMAN 3H-RACLOPRIDE 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 505 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
22536 5-HT1D CLONED HUMAN 3H-5CT SL650155 7990 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
88072 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22792 H2 CLONED HUMAN 3H-TIOTIDINE L-cysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23048 nAChR CLONED HUMAN 3H-Epibatidine L-homocysteine thiolactone >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88584 H1 CLONED HUMAN 3H-PYRILAMINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 212 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
89352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 3842 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24072 5-HT2A CLONED HUMAN UNDEFINED RISPERIDONE 0.21 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89608 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 0.47863 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90120 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
25096 D1 CLONED HUMAN 3H-SCH23390 Quetiapine 712 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90632 A2B CLONED HUMAN 3H-PSB-603 3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25352 5-HT1D CLONED HUMAN 3H-GR-125743 ZOTEPINE 175 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25864 mGluR6 CLONED RAT Functional Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91400 CB2 CLONED HUMAN 3H-CP55940 O-6617 >10000 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26120 M3 CLONED HUMAN 3H-QNB Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91656 A3 CLONED HUMAN 3H-PSB-11 4-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide 1000 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26376 M5 CLONED HUMAN 3H-QNB Rutin 35.13 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91912 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3-chlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26632 MOR CLONED HUMAN 3H-Diprenorphine Hyperoside >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92168 5-HT6 CLONED HUMAN 3H-LSD N-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)-8-quinolinesulfonamide 504 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26888 M5 CLONED HUMAN 3H-QNB xanomeline 39.8107 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92424 KOR CLONED HUMAN 3H-U69593 9,13:15,16-diepoxylabdane-6β,15α-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92680 M2 CLONED HUMAN 3H-QNB 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27400 Beta2 CLONED HUMAN 3H-CGP-12177 Talipexole >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 28, 2025
92936 5-HT6 CLONED HUMAN 3H-LSD WA-13 23 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
27656 5-HT7 CLONED HUMAN 3H-LSD MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27912 5-HT2A CLONED HUMAN 3H-KETANSERIN DMT,5-Me 1325 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93704 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 26.4 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28424 mGluR5 CLONED HUMAN 3H-Quisqualate Quisqualate 29 Mutel V, et.al., 2000 Jan 15, 2025 Jan 28, 2025
93960 D2 CLONED HUMAN 3H-SPIPERONE compound 43 3.9 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
28680 D1 CLONED HUMAN 3H-SCH23390 ARIPIPRAZOLE 1960 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94216 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-Bromo-2,5-dimethoxyphenethylamine 311 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29192 SST2 CLONED HUMAN UNDEFINED NC8-12 0.024 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94728 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94984 D3 CLONED HUMAN 3H-N-Methylspiperone 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29960 H4 CLONED HUMAN 3H-Histamine (1H-Indol-2-yl)-(piperazin-1-yl)-methanone 38 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
30216 D1 CLONED RAT UNDEFINED Duloxetine 1000 Bymaster F.P., et. al., 2001 Jan 15, 2025 Jan 15, 2025
95752 5-HT5A CLONED HUMAN 3H-LSD 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96008 NET CLONED HUMAN 3H-Nisoxetine 6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
30728 CLONED RAT UNDEFINED Atomoxetine 1000 Bymaster F.P., et. al., 2002 Jan 15, 2025 Jan 15, 2025
96264 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96520 Alpha1A CLONED HUMAN [3H]-prazosin 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 29, 2025
31240 Alpha1A CLONED HUMAN 3H-PRAZOSIN MDL 100907 1199 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96776 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31496 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) 1000 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97032 D2 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97288 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 24.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97544 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
32776 NK1 CLONED HUMAN 3H-Sar9,Met(O2)11-Substance P SR 48968 273 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98312 D2 CLONED HUMAN [3H]-N-methylspiperone 5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 1087 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98568 5-HT2B CLONED HUMAN [3H]-LSD 4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide 587 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33288 5-HT1B CLONED HUMAN 3H-GR-125743 Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98824 DOR CLONED HUMAN 3H-DADLE 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33544 Alpha2A CLONED HUMAN 3H-CLONIDINE Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99080 Beta1 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99336 D2 CLONED HUMAN [3H]N-methylspiperone 4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol 963 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34056 P2X3 CLONED HUMAN 3H-A-317491 Cibacron blue 2530 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99592 A1 CLONED HUMAN 3H-CCPA 8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine 1.22 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
34312 nAChR CLONED RAT 3H-Epibatidine ABT-418 803 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 28, 2025
99848 Alpha2C CLONED HUMAN [125I] iodoclonidine (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 280 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100104 5-HT2C CLONED HUMAN 3H-MESULERGINE Quetiapine 3624 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34824 CLONED RAT 3H-CP-55940 Rinvanil, Phenyl-propionyl >10000 Jan 15, 2025 Jan 15, 2025
100360 NET CLONED HUMAN 3H-Nisoxene Cariprazine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100616 CGRP CLONED HUMAN Functional N2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100872 Beta2 CLONED HUMAN 3H-CGP-12177 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1) 2 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 28, 2025
35592 CLONED HUMAN 3H-SQ 29548 CARBACYCLIN >10000 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35848 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester 33 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101384 5-HT6 CLONED HUMAN 3H-LSD 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 476 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
101640 D4 CLONED HUMAN [3H]-N-methylspiperone Perospirone 3.2 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101896 DAT CLONED HUMAN [3H]WIN35428 Ziprasidone 424 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36616 D3 CLONED HUMAN 125I-IODOSULPRIDE (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 293 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102152 KOR CLONED HUMAN [3H]U69593 NEMONAPRIDE 2713 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37896 MPP-2 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-nitro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 16 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38152 CLONED RAT 3H-dexamethasone C57H79N2O9 590 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
39432 Calcium channel CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39688 5-HT2B CLONED HUMAN 3H-5HT ORG-37684 42.658 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40712 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one 4530 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41224 CLONED HUMAN 125I-Chemokine 5-(4-Butyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41992 M1 CLONED HUMAN 3H-QNB DOXEPIN 38 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42248 CLONED HUMAN 125I-[Ile]Motilin cyanogen bromide, CNBr 0.85 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42760 CLONED UNDEFINED Functional Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Cys (O))-amide (S) >10000 Song YL, et al., 2006 Jan 15, 2025 Jan 15, 2025
43016 FYN CLONED HUMAN 3H-Staurosporine ZD-6474 5700 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43272 CLK1 CLONED HUMAN 3H-Staurosporine MLN-518 1400 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43528 FLT4 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43784 KDR CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44040 STK38L CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44296 CaMK CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44552 FRK CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44808 AAK1 CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45064 PTK6 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45320 CLONED HUMAN Functional kenpaullone 230 Bain J, et al., 2003 Jan 15, 2025 Jan 15, 2025
45576 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Dothiepin 5310 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45832 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46088 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46600 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46856 M5 CLONED HUMAN 3H-QNB (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47368 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
48136 Y2 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48648 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 400 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49160 MOR CLONED RAT 3H-DAMGO LYS227 5.3 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
49672 Y2 CLONED Chicken [125I] - Peptide YY PYY, chicken 0.630957 Salaneck E, et al., 2000 Jan 15, 2025 Jan 15, 2025
49928 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1996 Jan 15, 2025 Jan 15, 2025
50184 mGluR3 CLONED HUMAN Functional 1S, 3R-ACPD >10000 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50440 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N-Dimethyl-4-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine 519 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
58120 5-HT2A CLONED HUMAN 125I-DOI N-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 11.2 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58376 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5202 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
59144 5-HT2A CLONED HUMAN 3H-KETANSERIN KETANSERIN 2 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59400 D4 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4-(3-thienyl)benzamide 2 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59912 D5 CLONED HUMAN 3H-SCH23390 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60168 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(6-(3-Chlorobenzylamino)-2-((3,4- difluorophenyl)ethynyl)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide 3.49 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60424 GABAA CLONED HUMAN FNZ WY-S-2 124 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60680 GABAA CLONED HUMAN FNZ XHE-I-093 1107 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60936 GABAA CLONED HUMAN FNZ DM-146 247 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61192 GABAA CLONED HUMAN FNZ QH-II-067a 16 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61448 GABAA CLONED HUMAN FNZ RY-054 59 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61704 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine 2234 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62216 NET CLONED HUMAN [3H] Nisoxetine Naphyrone 96 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62472 M4 CLONED HUMAN 3H-QNB 3-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
62984 GABAA CLONED RAT 3H-RO-15-1788 3-(2-Thienylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 5-oxide 8.6 Costanzo A et al., 2002 Jan 15, 2025 Jan 27, 2025
63496 Alpha1B CLONED HUMAN 3H-PRAZOSIN RISPERIDONE 9 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64008 5-HT6 CLONED HUMAN 3H-LSD 1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one 124.5 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64264 5-HT2A CLONED HUMAN 3H-KETANSERIN SULPIRIDE 4786.3 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64520 CLONED HUMAN 3H-Estradiol 17beta-Estradiol 380 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
65288 GABAA CLONED HUMAN [3H] Flunitrazepam SH-I-030 19.09 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65545 GABAA CLONED HUMAN [3H] Flunitrazepam MLT-I-70 40.3 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65801 GABAA CLONED HUMAN [3H] Flunitrazepam YT-6 60.49 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66057 5-HT1A CLONED HUMAN 3H-WAY100635 Mellpaladine B 652 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66313 Beta2 CLONED HUMAN 3H-CGP12177 Finazine >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66569 Beta1 CLONED HUMAN I-125-Pindolol 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66825 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67081 5-HT2B CLONED HUMAN 3H-LSD 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 969 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67337 5-HT1A CLONED HUMAN 3H-WAY100635 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 58 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67849 5-HT6 CLONED HUMAN 3H-LSD S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 1483 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3337 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CARBAMAZEPINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68873 SST1 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 1000 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
3593 5-HT2C CLONED RAT 3H-MESULERGINE SKF 77434 3037 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69129 H3 CLONED HUMAN 3H-Histamine N-alpha-methylhistamine 3.98107 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3849 D2 CLONED RAT 3H-SPIPERONE HALOPERIDOL 13 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69385 H1 CLONED HUMAN 3H-PYRILAMINE FLUPHENAZINE 67 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4105 KOR CLONED HUMAN 3H-U69,593 Beta-Endorphin 11.4 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69641 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 2-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4361 5-HT6 CLONED HUMAN 3H-LSD OCTOCLOTHEPIN,(-) 1.8 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69897 D2 CLONED HUMAN 3H-N-Methylspiperone 4-[1-(4-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4617 SLC6A3 CLONED HUMAN 3H-DA UPTAKE DOPAMINE 1770 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4873 5-HT2B CLONED HUMAN 3H-5HT LY 53857 1.53 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70409 5-HT7 CLONED HUMAN 3H-LSD MRP4268 600 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5129 5-HT2B CLONED HUMAN 3H-5HT MEM 763 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70665 DOR CLONED HUMAN 3H-DADLE MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5385 5-HT2B CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 0.79 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
70921 5-HT2B CLONED HUMAN 3H-LSD (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 2051 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
5641 5-HT4 CLONED HUMAN 3H-GR-113808 RS 100235 0.00057544 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
71177 D5 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 147 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5897 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE CORYNANTHINE 77 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71433 5-HT6 CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 1791 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6153 Alpha1B CLONED RAT 125I-HEAT CORYNANTHINE 517 LOMASNEY JW, ET AL., 1991 Jan 15, 2025 Jan 15, 2025
6409 5-HT3 CLONED GUINEA PIG 3H-BIMU-1 BIMU 1 27.5 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
6665 D2 CLONED HUMAN 3H-NEMONAPRIDE CHLORPROMAZINE 14 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
72201 DOR CLONED HUMAN 3H-DADLE 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6921 5-HT2A CLONED HUMAN 3H-KETANSERIN OLANZAPINE 5.8 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
7433 MOR CLONED HUMAN 3H-DAMGO Naloxone(-) 0.93 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72969 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7689 GABAA CLONED HUMAN 3H-MUSCIMOL Muscimol 2.88 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7945 GABAA CLONED HUMAN 3H-RO-15-1788 8 1000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8201 SST5 CLONED HUMAN 125I-LTT-SST-28 SRIF-D-Trp8 0.28 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
8457 SST5 CLONED HUMAN 125I-Tyr3-octreotide octreotide 0.33 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8713 SST2 CLONED HUMAN 125I-Tyr3-octreotide octreotide 0.79 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8969 SST2 CLONED HUMAN 125I-SRIF-28 Somatostatin-14 0.19 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74505 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9225 SST2 CLONED MOUSE 125I-MK-678 L-363,301 8.6 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
74761 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75017 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9737 MT2 CLONED HUMAN 125I-Iodomelatonin N-Acetyltryptamine 12.7 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
9993 CB2 CLONED MOUSE 3H-CP-55940 JWH-015 431 Griffin G, Tao Q, Abood ME, 2000 Jan 15, 2025 Jan 15, 2025
75529 5-HT7 CLONED HUMAN 3H-LSD propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10249 CLONED HAMSTER 125I-HEAT PHENTOLAMINE 79.43 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75785 Beta 1 CLONED HUMAN 125I-Pindolol 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76041 KOR CLONED HUMAN 3H-U69593 Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate 207 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10761 5-HT2C CLONED RAT 3H-LSD CLOZAPINE 6.3 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
76297 NET CLONED HUMAN [3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76553 5-HT5A CLONED HUMAN 3H-LSD (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76809 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 6390 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77065 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77321 Beta 2 CLONED HUMAN 3H-CGP12177 (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77577 D3 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77833 5-HT1D CLONED HUMAN 3H-Cimetidine (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78089 M2 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78345 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78601 KOR CLONED HUMAN 3H-U69593 (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 490 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78857 KOR CLONED HUMAN 3H-U69593 (±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 30 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79113 5-HT5A CLONED HUMAN 3H-LSD cis-2a 16.4 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79369 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-2,5-Dimethoxy-4-bromoamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14089 Alpha2A CLONED PIG 3H-Yohimbine UK-14,304 478.63 Brink CB, et al., 2000 Jan 15, 2025 Jan 15, 2025
79625 CLONED HUMAN 3H-CLONIDINE 4-Bromo-2,5-dimethoxyphenethylamine 2155.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79881 M5 CLONED HUMAN 3H-QNB DMT,5-MeO >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14601 D2 CLONED HUMAN 125I-IODOSULPRIDE SB-277011-A 1047.12 Reavill C., et al., 2000 Jan 15, 2025 Jan 15, 2025
80137 CLONED HUMAN 3H-VASOPRESSIN 5-MeO-TMT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14857 D1 CLONED RAT UNDEFINED RISPERIDONE 21 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
80393 5-HT1E CLONED HUMAN 3H-5-CT (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15113 PTGFR CLONED HUMAN 3H-PGF2Alpha AGN 191366 8128 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80649 5-HT2B CLONED HUMAN 3H-LSD (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one 1274 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15369 5-HT1B CLONED HUMAN 3H-5HT SUMATRIPTAN 7.76 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80905 5-HT5A CLONED HUMAN 3H-LSD (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one 3324 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15625 5-HT2B CLONED RAT 3H-5HT KETANSERIN 3548.13 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81161 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
15881 5-HT7 CLONED RAT UNDEFINED 5-Hydroxy Tryptamine 0.6 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81417 D2 CLONED HUMAN 3H-N-Methylspiperone 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine 6787 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16137 D1 CLONED HUMAN 3H-SCH23390 LY-171555 >10000 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81673 D3 CLONED HUMAN 3H-N-Methylspiperone (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81929 H3 CLONED HUMAN 3H-Alpha-methylhistamine (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16649 M1 CLONED HUMAN 3H-QNB SCOPOLAMINE 1.1 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82185 D2 CLONED HUMAN 3H-N-Methylspiperone 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 1112 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82441 Alpha1B CLONED HUMAN 3H-PRAZOSIN (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82697 5-HT4 CLONED HUMAN 3H-GR113808 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17673 CLONED HUMAN 125I-VIP VIP [D-Phe6] 288 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83209 5-HT2C CLONED HUMAN 125I-DOI KETANSERIN 117 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83465 M3 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 30.903 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83721 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83977 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2362 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84233 KOR CLONED HUMAN 3H-U69593 (±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide 205 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18953 H1 CLONED GUINEA PIG 3H-MEPYRAMINE trans-H2-PAT(-) 1.15 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84489 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19209 CLONED RAT 125I-VIP [Phe1]PACAP-27 300 Ciccarelli E et al., 1994 Jan 15, 2025 Jan 15, 2025
84745 KOR CLONED HUMAN 3H-U69593 benzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19465 GPR145 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Nle8 18 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
85001 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86025 D4 CLONED HUMAN 3H-Alpha-methylhistamine (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86281 A1 CLONED HUMAN 3H-CCPA 8-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 41.7 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
21001 CLONED RAT 3H-NECA 19 210 Shamim MT et al., 1989 Jan 15, 2025 Jan 15, 2025
86537 A3 CLONED HUMAN 3H-PSB-11 1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione >10000 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
21513 nAChR CLONED Xenopus 3H-Epibatidine NFEP 2.1 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
87561 Beta 1 CLONED HUMAN 125I-Pindolol 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
22281 A1 CLONED HUMAN 125I-Aba 4c 3030 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87817 5-HT6 CLONED HUMAN 3H-LSD 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 90 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22537 hERG CLONED HUMAN 3H-Methylspiperone Quetiapine 5765 Kongsamut, S, et. al., 2002 Jan 15, 2025 Jan 15, 2025
88073 A1 CLONED HUMAN 3H-CCPA 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22793 H2 CLONED HUMAN 3H-TIOTIDINE L-homocysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23049 nAChR CLONED HUMAN 3H-Epibatidine D-homocysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88585 M1 CLONED HUMAN 3H-QNB 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
23561 H3 CLONED RAT 3H-NAMH A-304121 2.51189 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
89353 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 87 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24073 5-HT2A CLONED HUMAN UNDEFINED SERTINDOLE 0.3 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89865 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 378 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90121 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 4100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24841 D5 CLONED HUMAN 3H-SCH23390 CLOZAPINE 235 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90633 A2B CLONED HUMAN 3H-PSB-603 3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 801 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25353 5-HT1E CLONED HUMAN 3H-5HT ZOTEPINE 1080 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25609 M2 CLONED HUMAN 3H-QNB COCAINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91145 A1 CLONED HUMAN 3H-DPCPX N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide >10000 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
25865 M2 CLONED HUMAN 3H-QNB Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91401 CB2 CLONED HUMAN 3H-CP55940 O-6618 >10000 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26121 nAChR7 CLONED HUMAN 3H-Epibatidine Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91657 A3 CLONED HUMAN 3H-PSB-11 4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide 1000 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26377 GABAA CLONED RAT 3H-RO-15-1788 Amentoflavone 6.17 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91913 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (2-chlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26633 MOR CLONED HUMAN 3H-Diprenorphine Rutin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92169 5-HT6 CLONED HUMAN 3H-LSD 4-Fluoro-N-(1-{2-[2-(methylsulfanyl)phenoxy]ethyl} pyrrolidin-3-yl)benzenesulfonamide 357 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26889 5-HT4 CLONED PIGLET 125I-SB-207710 xanomeline 251.189 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92425 KOR CLONED HUMAN 3H-U69593 9,13:15,16-diepoxylabdane-6β,16β-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92681 M1 CLONED HUMAN 3H-QNB 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27401 Beta2 CLONED HUMAN 3H-CGP-12177 TERGURIDE 19.9526 Millan MJ, et al., 2002 Jan 15, 2025 Jan 28, 2025
92937 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine 21 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
27657 5-HT6 CLONED HUMAN 3H-LSD MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27913 5-HT2A CLONED HUMAN 3H-DOB DMT,5-Me 90 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28169 H1 CLONED HUMAN 3H-PYRILAMINE METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93705 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 15.7 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28425 CLONED HUMAN 3H-Quisqualate L-Glutamate 340 Mutel V, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93961 D2 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 3.2 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
28681 D2 CLONED HUMAN 3H-NMSP ARIPIPRAZOLE 0.74 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 27, 2025
94217 5-HT2A CLONED HUMAN 3H-KETANSERIN 2,5-dimethoxy-4-ethoxyphenethylamine 670 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29193 SST2 CLONED HUMAN UNDEFINED BIM 23268 15.1 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94729 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94985 D3 CLONED HUMAN 3H-N-Methylspiperone 4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29961 H4 CLONED HUMAN 3H-Histamine (4-Ethyl-piperazin-1-yl)-(1H-indol-2-yl)-methanone 260 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
30217 KOR CLONED BOVINE UNDEFINED Duloxetine 1000 Bymaster F.P., et. al., 2001 Jan 15, 2025 Jan 27, 2025
95753 5-HT6 CLONED HUMAN 3H-LSD 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
30473 CLONED Xenopus UNDEFINED (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-4-yl)methyl)amino]benzenepropaneamide bis(trifluoroacetate) 330 Kromann H, et. al., 2002a Jan 15, 2025 Jan 15, 2025
96009 NET CLONED HUMAN 3H-Nisoxetine Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
30729 CCK1 CLONED MOUSE UNDEFINED Atomoxetine 1000 Bymaster F.P., et. al., 2002 Jan 15, 2025 Jan 15, 2025
96265 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30985 Beta1 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96521 Alpha1B CLONED HUMAN [3H]-prazosin 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 29, 2025
31241 Alpha1B CLONED HUMAN 3H-PRAZOSIN MDL 100907 424.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96777 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 7700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31497 5-HT1B CLONED HUMAN 3H-5HT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) 3162.28 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97033 D3 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97289 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 191 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97545 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
32777 NK2 CLONED HUMAN 3H-NEUROKININ A SCH 206272 0.4 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98313 D2 CLONED HUMAN [3H]-N-methylspiperone 5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 418 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98569 5-HT2B CLONED HUMAN [3H]-LSD 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride, 723 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33289 5-HT1D CLONED HUMAN 3H-GR-125743 Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98825 KOR CLONED HUMAN 3H-U69593 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33545 Alpha2B CLONED HUMAN 3H-CLONIDINE Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99081 Beta1 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99337 D2 CLONED HUMAN [3H]N-methylspiperone 1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(quinolin-3-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol 244 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34057 P2X3 CLONED HUMAN 3H-A-317491 Suramin 1090 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99593 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine 3.29 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
34313 nAChR CLONED RAT 3H-Epibatidine MCC 969 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 28, 2025
99849 D2 CLONED HUMAN [3H]N-methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 2200 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
100105 5-HT3 CLONED HUMAN 3H-GR65630 Quetiapine 4330 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34825 CLONED RAT 3H-CP-55940 PhAR, epoxy >10000 Jan 15, 2025 Jan 15, 2025
100361 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE ILOPERIDONE 5.6 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100617 CGRP CLONED HUMAN Functional N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100873 Beta1 CLONED HUMAN 125I-Pindolol 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1) 6 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 28, 2025
35593 CLONED HUMAN 3H-SQ 29548 SQ 29548 4.1 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35849 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester 9.8 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101385 5-HT7 CLONED HUMAN 3H-5-CT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 34 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
101641 D5 CLONED HUMAN [3H]-SCH23390 Perospirone 1742 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101897 MOR CLONED HUMAN [3H]-DAMGO Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36617 D3 CLONED HUMAN 125I-IODOSULPRIDE HALOPERIDOL 4.4 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102153 GABAA CLONED HUMAN [3H]-Muscimol NEMONAPRIDE >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37897 MPP-9 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-nitro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 57 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38153 CLONED RAT 3H-dexamethasone C57H79N2O9Na 310 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
39433 Calcium channel CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 28, 2025
39689 5-HT2B CLONED HUMAN 3H-5HT PINDOLOL,(+/-) 2187.76 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40713 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one 101 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41225 CLONED HUMAN 125I-Chemokine 5-(4-Hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41993 M1 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42249 CLONED HUMAN Functional cyanogen bromide, CNBr 8.4 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42505 CLONED RABBIT UNDEFINED Motilin 0.977237 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
43017 GAK CLONED HUMAN 3H-Staurosporine Staurosporine 68 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43273 CLK1 CLONED HUMAN 3H-Staurosporine Roscovitine 2100 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43529 FYN CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43785 JAK1 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44041 STK4 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44297 CaMK CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44553 FYN CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44809 ACK1 CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45065 RIPK2 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45321 LCK CLONED HUMAN Functional kenpaullone 470 Bain J, et al., 2003 Jan 15, 2025 Jan 15, 2025
45577 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE DOXEPIN 68 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45833 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46089 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46601 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46857 M5 CLONED HUMAN 3H-QNB (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47369 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
47881 SST1 CLONED HUMAN 3H-thymidine BIM-23926 3.6 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
48137 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48649 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49161 MOR CLONED RAT 3H-DAMGO LYS322 0.92 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
49673 Y2 CLONED Chicken [125I] - Peptide YY NPY, porcine 0.346737 Salaneck E, et al., 2000 Jan 15, 2025 Jan 15, 2025
49929 mGluR2 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50185 Kainate receptor CLONED UNDEFINED 3H-AMPA LY 382884 4000 Bortolotto, Z., et al., 1999 Jan 15, 2025 Jan 15, 2025
50441 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N-Dimethyl-5-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine 401 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
58121 5-HT2A CLONED HUMAN 125I-DOI N-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 2.63 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58377 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5923 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58889 nAChR7 CLONED HUMAN 3H-Epibatidine Nicotine 323.5 Harris A, et al., 2015 Jan 15, 2025 Jan 15, 2025
59145 5-HT1A CLONED HUMAN 3H-WAY100635 KETANSERIN 1044 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59401 D2 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4-(3-thienyl)benzamide 1200 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59913 H1 CLONED HUMAN 3H-PYRILAMINE 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60169 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (phenylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide 0.85 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60425 GABAA CLONED HUMAN FNZ WY-S-2 30 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60681 GABAA CLONED HUMAN FNZ XHE-I-093 20 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60937 GABAA CLONED HUMAN FNZ DM-146 4.23 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61193 GABAA CLONED HUMAN FNZ CD-214 16.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61449 GABAA CLONED HUMAN FNZ RY-031 20.4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61705 5-HT2A CLONED HUMAN 3H-KETANSERIN (Z)-N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-4-phenylbut-3-en-1-amine 226 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62217 Serotonin CLONED HUMAN [3H] Citalopram Naphyrone 41 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62473 M4 CLONED HUMAN 3H-QNB 4-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
62985 GABAA CLONED RAT 3H-RO-15-1788 DIAZEPAM 9.8 Costanzo A et al., 2002 Jan 15, 2025 Jan 27, 2025
63497 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE RISPERIDONE 9.1 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64009 5-HT6 CLONED HUMAN 3H-LSD 1-[1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 107.4 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64265 5-HT2A CLONED HUMAN 3H-KETANSERIN THIORIDAZINE 19.0546 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64521 CLONED HUMAN 3H-Estradiol 4-hydroxytamoxifen 100 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
65289 GABAA CLONED HUMAN [3H] Flunitrazepam SH-I-030 1.89 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65546 GABAA CLONED HUMAN [3H] Flunitrazepam MLT-I-70 1000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65802 GABAA CLONED HUMAN [3H] Flunitrazepam YT-6 1.039 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66058 5-HT1B CLONED HUMAN 3H-5-CT Mellpaladine B 590 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66314 D1 CLONED HUMAN 3H-SCH233930 Finazine 1431 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66570 Beta3 CLONED HUMAN I-125-Pindolol 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66826 Alpha1B CLONED HUMAN 3H-PRAZOSIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67082 5-HT3 CLONED HUMAN 3H-GR113808 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 671 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67338 5-HT1B CLONED HUMAN 3H-5-CT 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67850 D2 CLONED HUMAN 3H-RACLOPRIDE S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
3338 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CGS 12066B 44 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68874 SST2 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 1000 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
3594 5-HT2C CLONED RAT 3H-MESULERGINE SKF 81297 1510 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69130 H3 CLONED HUMAN 3H-Histamine Alpha-Methylhistamine-R 6.30957 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3850 5-HT2A CLONED RAT 3H-SPIPERONE ILOPERIDONE 3.1 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69386 H1 CLONED HUMAN 3H-PYRILAMINE CHLORPROMAZINE 0.18 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4106 KOR CLONED HUMAN 3H-U69,593 NALTRINDOLE 10.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69642 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 3-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4362 5-HT6 CLONED HUMAN 3H-LSD CLOZAPINE 9.5 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69898 D2 CLONED HUMAN 3H-N-Methylspiperone 4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4618 SLC6A3 CLONED HUMAN 3H-DA UPTAKE NOREPINEPHRINE 8500 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4874 5-HT2B CLONED HUMAN 3H-5HT 1-NP 3.25 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70410 5-HT2B CLONED HUMAN 3H-LSD MRP4268 8.6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5130 5-HT2B CLONED HUMAN 3H-5HT DOAc 313 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70666 KOR CLONED HUMAN 3H-U69,593 MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5386 5-HT2B CLONED RAT 3H-5HT YOHIMBINE 50.11 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
70922 5-HT2B CLONED HUMAN 3H-LSD (4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 231 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
71178 D5 CLONED HUMAN 3H-SCH23390 CLOZAPINE 454 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5898 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE KETANSERIN 199 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71434 5-HT7 CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 724 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6154 Alpha1B CLONED RAT 125I-HEAT WB 4101 28.6 LOMASNEY JW, ET AL., 1991 Jan 15, 2025 Jan 15, 2025
6410 5-HT3 CLONED GUINEA PIG 3H-BIMU-1 BIMU 8 20 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
6666 D4 CLONED HUMAN 3H-NEMONAPRIDE CHLORPROMAZINE 22 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
6922 5-HT2A CLONED HUMAN 3H-KETANSERIN PERLAPINE 30 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72714 D1 CLONED HUMAN 3H-SCH23390 naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7434 MOR CLONED HUMAN 3H-DAMGO NALTREXONE-HCl 1 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72970 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7690 GABAA CLONED HUMAN 3H-MUSCIMOL Thiomuscimol 13.18 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7946 GABAA CLONED HUMAN 3H-RO-15-1788 9 1162 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8202 SST5 CLONED HUMAN 125I-LTT-SST-28 SMS 201-995 14.16 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
8458 SST5 CLONED HUMAN 125I-Tyr3-octreotide octreotide-Tyr3 3.89 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8714 SST2 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 1.12 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8970 SST2 CLONED HUMAN 125I-SRIF-28 SS-25 0.31 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74506 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9226 SST2 CLONED MOUSE 125I-MK-678 L-363,572 26 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
74762 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9482 MT1 CLONED HUMAN 125I-Iodomelatonin MELATONIN 0.56 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
75018 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9738 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Methoxy 3.5 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75274 5-HT1A CLONED HUMAN 3H-WAY100635 Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9994 CB2 CLONED MOUSE 3H-CP-55940 JWH-051 0.72 Griffin G, Tao Q, Abood ME, 2000 Jan 15, 2025 Jan 15, 2025
75530 Alpha1A CLONED HUMAN 3H-PRAZOSIN propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10250 CLONED HAMSTER 125I-HEAT PRAZOSIN 0.12 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75786 Beta3 CLONED HUMAN 125I-Pindolol 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76042 MOR CLONED HUMAN 3H-DAMGO Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate 1770 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10762 5-HT2C CLONED RAT 3H-LSD RILAPINE 25.11 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
76298 NOP CLONED HUMAN 3H-Nociceptin (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
76554 5-HT6 CLONED HUMAN 3H-LSD (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76810 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77066 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77322 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77578 D4 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77834 H3 CLONED HUMAN 3H-Alpha-methylhistamine (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78090 M3 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78346 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78602 MOR CLONED HUMAN 3H-DAMGO (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78858 KOR CLONED HUMAN 3H-U69593 (±)-(4aR,8S,8aR)-N-(2,6-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79114 5-HT5A CLONED HUMAN 3H-LSD R,R-2b 12.7 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79370 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-3,4-Methylenedioxyamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14090 Alpha2A CLONED PIG 3H-Yohimbine p-AMINOCLONIDINE 288.4 Brink CB, et al., 2000 Jan 15, 2025 Jan 15, 2025
79626 CLONED HUMAN 3H-CLONIDINE DMT 650.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79882 M5 CLONED HUMAN 3H-QNB 4-Ethyl-2,5-dimethoxyphenethylamine 1725 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14602 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SB-277011-A 5011.87 Reavill C., et al., 2000 Jan 15, 2025 Jan 15, 2025
80138 V2 CLONED HUMAN 3H-VASOPRESSIN (±)-2,5-Dimethoxy-4-bromoamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14858 D1 CLONED RAT UNDEFINED Quetiapine 390 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
80394 5-HT1B CLONED HUMAN 3H-5-CT (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15114 PTGFR CLONED HUMAN 3H-PGF2Alpha AGN 190910 >10000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80650 5-HT2C CLONED HUMAN 3H-MESULERGINE (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15370 5-HT1B CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 4.26 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80906 5-HT6 CLONED HUMAN 3H-LSD (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15626 5-HT2B CLONED RAT 3H-5HT RITANSERIN 5.12 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81162 5-HT1B CLONED HUMAN 3H-5-CT N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
15882 5-HT7 CLONED RAT UNDEFINED METERGOLINE 63.09 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81418 H1 CLONED HUMAN 3H-PYRILAMINE 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16138 D1 CLONED HUMAN 3H-SCH23390 SCH 23390 0.35 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81674 D4 CLONED HUMAN 3H-N-Methylspiperone (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81930 H4 CLONED HUMAN 3H-Histamine (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16650 M1 CLONED HUMAN 3H-QNB Trihexyphenidyl 1.6 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82186 D3 CLONED HUMAN 3H-N-Methylspiperone 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 56 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82442 Alpha1D CLONED HUMAN 3H-PRAZOSIN (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82698 5-HT5A CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17674 CLONED HUMAN 125I-VIP VIP [D-Asp8] 110 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83210 5-HT2A CLONED HUMAN 125I-DOI KETANSERIN 7.6 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83466 M2 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 13.8038 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83722 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 9987 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83978 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3216 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18954 H1 CLONED GUINEA PIG 3H-MEPYRAMINE trans-H2-PAT(+/-) 1.53 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84490 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19210 CLONED RAT 125I-VIP VIP [D-His1] 200 Ciccarelli E et al., 1994 Jan 15, 2025 Jan 15, 2025
84746 DOR CLONED HUMAN 3H-DADLE phenyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19466 GPR145 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Leu9 45 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
85002 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19722 D2 CLONED HUMAN UNDEFINED BENPERIDOL 0.027 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
86026 M1 CLONED HUMAN 3H-QNB (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
21002 CLONED RAT 3H-NECA 20 5300 Shamim MT et al., 1989 Jan 15, 2025 Jan 15, 2025
86538 A1 CLONED HUMAN 3H-CCPA 1-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione 2440 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
21514 nAChR CLONED Xenopus 3H-Epibatidine NEP 11 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
87562 Beta3 CLONED HUMAN 125I-Pindolol 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
22282 A1 CLONED HUMAN 125I-Aba 4d 6.82 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87818 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€4â€iodoâ€Nâ€(2â€phenylethyl)aniline 79 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22538 hERG CLONED HUMAN 3H-Methylspiperone OLANZAPINE 6013 Kongsamut, S, et. al., 2002 Jan 15, 2025 Jan 15, 2025
88074 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22794 H2 CLONED HUMAN 3H-TIOTIDINE D-homocysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23050 nAChR CLONED HUMAN 3H-Epibatidine L-homocysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88586 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 45.1 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
23562 H3 CLONED HUMAN 3H-NAMH A-304121 758.578 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
89354 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 44 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24074 5-HT2A CLONED HUMAN UNDEFINED THIORIDAZINE 1.1 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89610 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89866 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 133 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90122 D1 CLONED HUMAN 3H-SCH23390 Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24842 5-HT6 CLONED HUMAN 3H-LSD CLOZAPINE 17 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90378 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide 193 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90634 A2B CLONED HUMAN 3H-PSB-603 3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25354 H2 CLONED HUMAN 3H-TIOTIDINE ZOTEPINE 500 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91146 A2A CLONED HUMAN 3H-CGS-21680 N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide 3310 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
25866 D2 CLONED HUMAN 3H-NMSP Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91402 CB1 CLONED HUMAN 3H-CP55940 O-6618 89 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
91658 A3 CLONED HUMAN 3H-PSB-11 N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide 1000 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26378 NET CLONED HUMAN 3H-Nisoxetine Hyperforin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91914 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3,4-dichlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26634 MOR CLONED HUMAN 3H-Diprenorphine Quercetin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92170 5-HT6 CLONED HUMAN 3H-LSD 4-Fluoro-N-{1-[2-(phenoxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 248 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26890 5-HT1A CLONED HUMAN 3H-8-OH-DPAT xanomeline 63.0957 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92426 KOR CLONED HUMAN 3H-U69593 9,13:15,16-diepoxylabdane-6β,16α-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92682 H1 CLONED HUMAN 3H-PYRILAMINE (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27402 Beta1 CLONED HUMAN 3H-CGP-12177 TERGURIDE 660.693 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92938 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 16 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
27658 5-HT5A CLONED HUMAN 3H-LSD MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27914 5-HT2A CLONED HUMAN 3H-KETANSERIN DOI 52 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28170 D4 CLONED HUMAN 3H-NMSP METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93706 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 6.73 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28426 mGluR5 CLONED HUMAN 3H-Quisqualate L-Glutamate 700 Mutel V, et.al., 2000 Jan 15, 2025 Jan 28, 2025
93962 D2 CLONED HUMAN 3H-SPIPERONE 7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one 26 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
28682 D2 CLONED HUMAN 3H-NMSP ARIPIPRAZOLE 3.3 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94218 5-HT2A CLONED HUMAN 3H-KETANSERIN 2,5-dimethoxy-4-methallyloxyphenethylamine 40 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29194 SST2 CLONED HUMAN UNDEFINED seglitide 0.1 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94730 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94986 D3 CLONED HUMAN 3H-N-Methylspiperone 4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29962 H4 CLONED HUMAN 3H-Histamine +-(1H-Indol-2-yl)-(3-methyl-piperazin-1-yl)-methanone 202 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
30218 GABAA CLONED BOVINE UNDEFINED Duloxetine 1000 Bymaster F.P., et. al., 2001 Jan 15, 2025 Jan 15, 2025
95754 5-HT7 CLONED HUMAN 3H-LSD 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96010 NET CLONED HUMAN 3H-Nisoxetine Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
30730 CCK2 CLONED MOUSE UNDEFINED Atomoxetine 1000 Bymaster F.P., et. al., 2002 Jan 15, 2025 Jan 15, 2025
96266 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30986 Beta2 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 28, 2025
96522 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jul 30, 2025
31242 H1 CLONED HUMAN 3H-PYRILAMINE MDL 100907 66.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96778 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31498 5-HT1B CLONED HUMAN 3H-5HT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) 3981.07 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97034 D4 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97290 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97546 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 789 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
32778 NK2 CLONED HUMAN 3H-NEUROKININ A CP 99994 >10000 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98314 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline >10000 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98570 5-HT2B CLONED HUMAN [3H]-LSD 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride 358 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33290 5-HT2A CLONED HUMAN 3H-KETANSERIN Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98826 M1 CLONED HUMAN 3H-QNB 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
33546 Alpha2C CLONED HUMAN 3H-CLONIDINE Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99082 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99338 D2 CLONED HUMAN [3H]N-methylspiperone PG648 746 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34058 P2X3 CLONED HUMAN 3H-A-317491 PPADS 3470 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99594 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine 1.52 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
34314 nAChR CLONED RAT 3H-Epibatidine SIB-1508Y 991 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 28, 2025
99850 D2 CLONED HUMAN [3H]N-methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
100106 5-HT5A CLONED HUMAN 3H-LSD Quetiapine 2300 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34826 CLONED RAT 3H-CP-55940 PhAR, Cycloproyl >10000 Jan 15, 2025 Jan 15, 2025
100362 DAT CLONED HUMAN 3H-WIN35428 ILOPERIDONE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100618 CGRP CLONED HUMAN Functional N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamine >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100874 Beta1 CLONED HUMAN 125I-Pindolol 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1) 7 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 28, 2025
35594 CLONED HUMAN 3H-SQ 29548 U46619 35 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35850 SLC6A4 CLONED HUMAN 3H-PAROXETINE 3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester 2.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101386 D2 CLONED HUMAN 3H-RACLOPRIDE 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 118 Zareba P, et al., 2019 Jan 15, 2025 Jan 28, 2025
101642 SERT CLONED HUMAN [3H]Citalopram Perospirone 984 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101898 DOR CLONED HUMAN [3H]DADLE Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36618 D3 CLONED HUMAN 125I-IODOSULPRIDE CLOZAPINE 242 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102154 H1 CLONED HUMAN [3H]Pyrilamine NEMONAPRIDE 741 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37898 MPP-2 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-iodo-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 86 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38154 CLONED RAT 3H-dexamethasone C55H77N2O8 1000 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
39434 Calcium channel CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 28, 2025
39690 5-HT2B CLONED HUMAN 3H-5HT QUINPIROLE 301.995 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40714 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one 901 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41226 CLONED HUMAN 125I-Chemokine 1-(4-Cyano-4,4-diphenylbutyl)-4-phenylpiperidine-4-carbonitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41994 M1 CLONED HUMAN 3H-QNB Femoxetine 92 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42250 CLONED HUMAN 125I-[Ile]Motilin K368,374C 0.6 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42506 CLONED RABBIT UNDEFINED [Nle13]-Motilin 0.851138 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
43018 GAK CLONED HUMAN 3H-Staurosporine SB202190 650 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43274 CLK1 CLONED HUMAN 3H-Staurosporine Flavopiridol 2200 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43530 HCK CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43786 PKMYT1 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44042 Syk CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44298 CaMK CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44554 GAK CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44810 STK6 CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45066 RPS6KA3 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45322 CDK2 CLONED HUMAN Functional alsterpaullone 80 Bain J, et al., 2003 Jan 15, 2025 Jan 28, 2025
45578 NET CLONED HUMAN 3H-Nisoxetine DOXEPIN 29.5 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45834 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46090 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46602 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46858 M5 CLONED HUMAN 3H-QNB PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47114 M3 CLONED HUMAN 3H-NMS Iodophenpropit 3700 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47370 Grik5 CLONED HUMAN 3H-Kainic acid LY 466195 50 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47882 SST2 CLONED HUMAN 3H-thymidine BIM-23926 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
48138 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48650 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48906 Y1 CLONED Chicken [125I] - Peptide YY PYY, chicken 5.12861 Holmberg, SK et al., 2002 Jan 15, 2025 Jan 15, 2025
49162 CCK1 CLONED HUMAN 125I-CCK-8 LYS201 >10000 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
49674 Y2 CLONED Chicken [125I] - Peptide YY NPY2-36, porcine 0.549541 Salaneck E, et al., 2000 Jan 15, 2025 Jan 15, 2025
49930 mGluR4 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50186 Kainate receptor CLONED UNDEFINED 3H-AMPA LY 382884 >10000 Bortolotto, Z., et al., 1999 Jan 15, 2025 Jan 28, 2025
50442 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine 445 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
58122 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 21.4 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58378 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5930 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58890 nAChR7 CLONED HUMAN 3H-Epibatidine Kodiak extract 202.1 Harris A, et al., 2015 Jan 15, 2025 Jan 15, 2025
59146 5-HT2A CLONED HUMAN 3H-KETANSERIN METHYSERGIDE 3.25 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59402 D4 CLONED HUMAN 3H-N-Methylspiporone N-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(2-thienyl)benzamide 24 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59914 H2 CLONED HUMAN 3H-Cimetidine 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60170 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-(Biphenyl-4-ylethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 3.1 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60426 GABAA CLONED HUMAN FNZ WY-S-6 120 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60682 GABAA CLONED HUMAN FNZ XHE-I-093 1162 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60938 GABAA CLONED HUMAN FNZ DM-146 148 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61194 GABAA CLONED HUMAN FNZ CD-214 48.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61450 GABAA CLONED HUMAN FNZ RY-031 27 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61706 5-HT2A CLONED HUMAN 3H-KETANSERIN CLOZAPINE 15 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
61962 CLONED HUMAN UNDEFINED azimilide 1400 Busch ,AE et al., 1998 Jan 15, 2025 Jan 15, 2025
62218 Serotonin CLONED HUMAN [3H] Citalopram I-Naphyrone 34 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62474 M5 CLONED HUMAN 3H-QNB Diphenidine 1653 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
62986 GABAA CLONED RAT 3H-RO-15-1788 Zolpidem >10000 Costanzo A et al., 2002 Jan 15, 2025 Jan 27, 2025
63498 H1 CLONED HUMAN 3H-PYRILAMINE RISPERIDONE 27 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64010 5-HT6 CLONED HUMAN 3H-LSD 1-[1-(Naphthalene-1-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 51.7 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64266 5-HT2A CLONED HUMAN 3H-KETANSERIN tiotixene 89.1251 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64522 CLONED HUMAN 3H-Estradiol raloxifene 18 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
65290 GABAA CLONED HUMAN [3H] Flunitrazepam XLI-348 13.56 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65547 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-III-04 1.2 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65803 GABAA CLONED HUMAN [3H] Flunitrazepam PWZ-096 11.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66059 5-HT1D CLONED HUMAN 3H-5-CT Mellpaladine B 489 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66315 D2 CLONED HUMAN 3H-N-Methylspiperone Finazine 1412 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66571 Beta2 CLONED HUMAN 3H-CGP12177 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66827 Alpha1D CLONED HUMAN 3H-PRAZOSIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67083 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67339 5-HT1D CLONED HUMAN 3H-5-CT 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 4549 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67851 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3339 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CHLORPROMAZINE 3115 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68875 SST3 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 1000 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
3595 5-HT2C CLONED RAT 3H-MESULERGINE SPIPERONE 4094 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69131 H3 CLONED HUMAN 3H-Histamine Alpha-Methylhistamine-S 63.0957 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3851 5-HT2A CLONED RAT 3H-SPIPERONE RISPERIDONE 1.4 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69387 H1 CLONED HUMAN 3H-PYRILAMINE RACLOPRIDE 8430 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4107 KOR CLONED HUMAN 3H-U69,593 BNTX 3.7 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69643 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 4-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4363 5-HT6 CLONED HUMAN 3H-LSD OLANZAPINE 10 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69899 D2 CLONED HUMAN 3H-N-Methylspiperone 4-[1-(3-methylphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4619 SLC6A3 CLONED HUMAN 3H-DA UPTAKE 5-Hydroxy Tryptamine >10000 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4875 5-HT2B CLONED HUMAN 3H-RAUWOLSCINE LSD,2-Bromo 7.47 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70411 5-HT1A CLONED HUMAN 3H-WAY100635 MRP4268 5.6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5131 5-HT2B CLONED HUMAN 3H-5HT DON 166 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70667 MOR CLONED HUMAN 3H-DAMGO MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5387 5-HT2B CLONED RAT 3H-5HT mCPP 25.11 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
70923 5-HT7 CLONED HUMAN 3H-LSD (4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 2765 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
71179 D5 CLONED HUMAN 3H-SCH23390 SYA16263 1451 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5899 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE OXYMETAZOLINE 213 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71435 SERT CLONED HUMAN 3H-CITALOPRAM 4-acetoxy-N,N-diallyltryptamine 1089 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
6155 Alpha1C CLONED BOVINE 125I-HEAT EPINEPHRINE 6250 LOMASNEY JW, ET AL., 1991 Jan 15, 2025 Jan 15, 2025
6411 5-HT3 CLONED RAT 3H-BIMU-1 5-Hydroxy Tryptamine 501 BONHAUS DW, ET AL., 1993 Jan 15, 2025 Jan 15, 2025
72203 H1 CLONED HUMAN 3H-PYRILAMINE 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6923 5-HT2A CLONED HUMAN 3H-KETANSERIN RACLOPRIDE 5400 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72715 D5 CLONED HUMAN 3H-SCH23390 naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7435 MOR CLONED HUMAN 3H-DAMGO Beta C N A 0.9 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72971 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7691 GABAA CLONED HUMAN 3H-MUSCIMOL THIP 46.77 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7947 GABAA CLONED HUMAN 3H-RO-15-1788 10 1000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8203 SST5 CLONED HUMAN 125I-LTT-SST-28 MK 678 5.02 Panetta R, et al., 1993 Jan 15, 2025 Jan 15, 2025
8459 SST5 CLONED HUMAN 125I-Tyr3-octreotide L-362,855 0.67 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8715 SST2 CLONED HUMAN 125I-Tyr3-octreotide L-362,855 1.62 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8971 SST2 CLONED HUMAN 125I-SRIF-28 somatostatin-28 0.19 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74507 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9227 SST2 CLONED MOUSE 125I-MK-678 L-363,376 356 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
74763 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9483 MT1 CLONED HUMAN 125I-Iodomelatonin N-Acetyltryptamine 870 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
75019 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9739 MT2 CLONED HUMAN 125I-Iodomelatonin Serotonin,N-acetyl 189 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75275 5-HT1B CLONED HUMAN 3H-5-CT Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9995 CB2 CLONED HUMAN 3H-CP-55940 WIN 35,428 1.19 Griffin G, Tao Q, Abood ME, 2000 Jan 15, 2025 Jan 15, 2025
75531 Alpha1B CLONED HUMAN 3H-PRAZOSIN propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10251 CLONED HAMSTER 125I-HEAT SPIPERONE 31.62 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75787 Beta 2 CLONED HUMAN 3H-CGP12177 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10763 5-HT2C CLONED RAT 3H-LSD FLUPERLAPINE 19.95 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
76555 5-HT7 CLONED HUMAN 3H-LSD (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76811 Alpha1D CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77067 Beta 1 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77323 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77579 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77835 H4 CLONED HUMAN 3H-Histamine (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78091 M4 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78347 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78603 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78859 DOR CLONED HUMAN 3H-DADLE (±)-(4aR,8S,8aR)-N-(2,6-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79115 5-HT5A CLONED HUMAN 3H-LSD S,S-2c 27.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79371 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-3,4-Methylenedioxymethamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14091 Alpha2A CLONED PIG 3H-Yohimbine B-HT 920 1000 Brink CB, et al., 2000 Jan 15, 2025 Jan 15, 2025
79627 CLONED HUMAN 3H-CLONIDINE 4-Hydroxy-N,N-dimethyltryptamine 792.2 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79883 M5 CLONED HUMAN 3H-QNB 4-Ethylthio-2,5-dimethoxyphenethylamine 1502 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14603 5-HT1B CLONED HUMAN 3H-5HT SB-277011-A 6309.57 Reavill C., et al., 2000 Jan 15, 2025 Jan 15, 2025
80139 V2 CLONED HUMAN 3H-VASOPRESSIN 3,4,5-Trimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14859 D1 CLONED RAT UNDEFINED Ziprasidone 9.5 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
80395 5-HT1D CLONED HUMAN 3H-5-CT (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15115 PTGFR CLONED HUMAN 3H-PGF2Alpha AGN 190911 >10000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80651 5-HT3 CLONED HUMAN 3H-GR-65630 (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15371 5-HT1B CLONED HUMAN 3H-5HT METHYSERGIDE 25.11 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80907 5-HT7 CLONED HUMAN 3H-LSD (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15627 5-HT2B CLONED RAT 3H-5HT MIANSERIN 52.48 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81163 5-HT1D CLONED HUMAN 3H-5-CT N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
15883 5-HT7 CLONED RAT UNDEFINED LSD 9.54 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81419 H1 CLONED HUMAN 3H-PYRILAMINE N-[[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-methylmethanamine >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16139 D1 CLONED HUMAN 3H-SCH23390 SKF 83566 0.3 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81675 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 15, 2025
81931 KOR CLONED HUMAN 3H-U69593 (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16651 M1 CLONED HUMAN 3H-QNB Procyclidine 4.6 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82187 D4 CLONED HUMAN 3H-N-Methylspiperone 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 264 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82443 D1 CLONED HUMAN 3H-SCH23390 (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82699 5-HT6 CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17675 CLONED HUMAN 125I-VIP VIP [D-Asn9] 1.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN 6510 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83467 M1 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 5.01187 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83723 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5904 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
18443 5-HT1A CLONED HUMAN 3H-5HT 1-NP 9.2 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
83979 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-cyclohexyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 6292 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84235 M2 CLONED HUMAN 3H-QNB (±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide 8259 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
18955 H1 CLONED GUINEA PIG 3H-MEPYRAMINE trans-H2-PAT(+) 23 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84491 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19211 CLONED RAT 125I-VIP VIP(2-28) 200 Ciccarelli E et al., 1994 Jan 15, 2025 Jan 15, 2025
84747 DOR CLONED HUMAN 3H-DADLE S-phenyl (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbothioate >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19467 GPR145 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Gly10 37 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
85003 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19723 D2 CLONED HUMAN UNDEFINED BROMOCRIPTINE 2 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
86027 M2 CLONED HUMAN 3H-QNB (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
86283 A2B CLONED HUMAN 3H-PSB-603 8-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1000 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
21003 CLONED RAT 3H-NECA 24 5600 Shamim MT et al., 1989 Jan 15, 2025 Jan 15, 2025
86539 A2A CLONED HUMAN 3H-MSX-2 1-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione 149 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87563 Beta 2 CLONED HUMAN 3H-CGP12177 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
22283 A1 CLONED HUMAN 125I-Aba 5 1660 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87819 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€4â€iodoâ€Nâ€(2â€phenylethyl)aniline 691 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
22539 D2 CLONED HUMAN 3H-Methylspiperone SERTINDOLE 6.55 Kongsamut, S, et. al., 2002 Jan 15, 2025 Jan 15, 2025
88075 A1 CLONED HUMAN 3H-CCPA 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3800 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
22795 H2 CLONED HUMAN 3H-TIOTIDINE D-homocysteine thiolactone >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
23051 nAChR CLONED HUMAN 3H-Epibatidine L-cysteine sulfinic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 27, 2025
88587 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 194.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
23563 GPR10 CLONED HUMAN 125I-PrRP20 NPY18-36 7400 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
89355 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 802 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24075 5-HT2A CLONED HUMAN UNDEFINED Trifluperazine 7.4 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89611 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89867 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 3400 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90123 D1 CLONED HUMAN 3H-SCH23390 LSD 310 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24843 M5 CLONED HUMAN 3H-QNB CLOZAPINE 94 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90379 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide 452 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
25099 H1 CLONED HUMAN 3H-PYRILAMINE Quetiapine 7.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90635 A2B CLONED HUMAN 3H-PSB-603 2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25355 5-HT2A CLONED RAT 3H-KETANSERIN ZOTEPINE 6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25611 5-HT3 CLONED HUMAN 3H-ZACOPRIDE COCAINE 1950 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91147 A3 CLONED HUMAN 125I-AB-MECA N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide >10000 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
25867 mGluR8 CLONED RAT Functional Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91403 CB1 CLONED HUMAN 3H-SR144528 O-6618 44 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26123 5-HT1B CLONED HUMAN 3H-GR-125743 Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91659 A3 CLONED HUMAN 3H-PSB-11 4-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 174 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26379 SLC6A3 CLONED BOVINE 3H-WIN 35,428 Amentoflavone 877.4 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91915 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (2,4-dichlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
26635 MOR CLONED HUMAN 3H-Diprenorphine Quercitrin >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
92171 5-HT6 CLONED HUMAN 3H-LSD 4-Fluoro-N-{1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 96 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
26891 5-HT1B CLONED HUMAN 3H-5HT xanomeline 50.1187 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
92427 KOR CLONED HUMAN 3H-U69593 9,13-epoxylabd-5-en-7-on-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92683 H1 CLONED HUMAN 3H-PYRILAMINE 9,13:15,16-diepoxylabdane-6b,15a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27403 Beta1 CLONED HUMAN 3H-CGP-12177 TL99 >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92939 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 6 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
27659 5-HT3 CLONED HUMAN 3H-ZACOPRIDE MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27915 5-HT2A CLONED HUMAN 3H-DOB DOI 3.1 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28171 D5 CLONED HUMAN 3H-SCH23390 METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93707 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester 4.88 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28427 CLONED HUMAN 3H-Quisqualate DHPG 900 Mutel V, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93963 D2 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one 38 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
28683 D3 CLONED HUMAN 3H-NMSP ARIPIPRAZOLE 9.7 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94219 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-allyloxy-2,5-dimethoxyphenethylamine 140 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29195 SST2 CLONED HUMAN UNDEFINED Vapreotide 5.4 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94731 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94987 D3 CLONED HUMAN 3H-N-Methylspiperone 4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29963 H4 CLONED HUMAN 3H-Histamine (1H-Indol-2-yl)-(4-phenethyl-piperazin-1-yl)-methanone 7000 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
30219 GABAA CLONED BOVINE UNDEFINED Venlafaxine 1000 Bymaster F.P., et. al., 2001 Jan 15, 2025 Jan 15, 2025
95755 5-HT5A CLONED HUMAN 3H-LSD N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
30475 CLONED Xenopus UNDEFINED (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-cyclohexylmethyl)amino]benzenepropaneamide bis(trifluoroacetate) 240 Kromann H, et. al., 2002a Jan 15, 2025 Jan 15, 2025
96011 NET CLONED HUMAN 3H-Nisoxetine 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
30731 NK1 CLONED RAT UNDEFINED Atomoxetine 1000 Bymaster F.P., et. al., 2002 Jan 15, 2025 Jan 15, 2025
96267 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30987 A1 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96523 Beta1 CLONED HUMAN [125I]-Pindolol 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 29, 2025
31243 H4 CLONED HUMAN 3H-Histamine MDL 100907 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96779 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 8800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31499 5-HT1D CLONED HUMAN 3H-5HT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) 501.187 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97035 D5 CLONED HUMAN [3H]SCH23390 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97291 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 135 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97547 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 721 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
32779 NK2 CLONED HUMAN 3H-NEUROKININ A SR 48968 0.4 Anthes, JC et al., 2002 Jan 15, 2025 Jan 15, 2025
98315 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline 5647 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98571 5-HT2B CLONED HUMAN [3H]-LSD 1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride 232 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33291 5-HT2B CLONED HUMAN 3H-LSD Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98827 M2 CLONED HUMAN 3H-QNB 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
33547 M2 CLONED HUMAN 3H-QNB Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99083 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99339 D2 CLONED HUMAN [3H]N-methylspiperone OMO5-057 321 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34059 P2X3 CLONED HUMAN 3H-A-317491 KN-62 >10000 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99595 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 2.43 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
34315 nAChR CLONED RAT 3H-Epibatidine GTS-21 1290 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 28, 2025
99851 D3 CLONED HUMAN [3H]N-methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
100107 5-HT6 CLONED HUMAN 3H-LSD Quetiapine 1777 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34827 CLONED RAT 3H-CP-55940 PhAR, Di-hydro >10000 Jan 15, 2025 Jan 15, 2025
100363 NET CLONED HUMAN 3H-Nisoxetine ILOPERIDONE 535 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100619 CGRP CLONED HUMAN Functional N2-[3,5-Dibromo-N-(4-phenyl-1-oxybutyl)-L-tyrosyl]-L-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100875 5-HT1A CLONED HUMAN 3H-WAY100635 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1) 24.6 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 15, 2025
35595 CLONED HUMAN 3H-SQ 29548 AH-23848 592 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35851 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 47 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 35 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
101643 NET CLONED HUMAN [3H] Nisoxetine Perospirone 303 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101899 KOR CLONED HUMAN [3H]U69593 Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36619 D3 CLONED HUMAN 125I-IODOSULPRIDE OLANZAPINE 43 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102155 H2 CLONED HUMAN [3H]Tiotidine NEMONAPRIDE 2108 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37899 MPP-9 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-iodo-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 10 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38155 CLONED RAT 3H-dexamethasone C54H76NO7 1000 von Geldern TW, et al, 2004 Jan 15, 2025 Jan 15, 2025
39435 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39691 5-HT2B CLONED HUMAN 3H-5HT QUIPAZINE 85.1138 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40459 mGluR5 CLONED RAT Functional (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40715 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-3-(4'-ethylphenyl)-3H-1,3,6-triazafluoren-4-one 1460 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41227 CLONED HUMAN 125I-Chemokine 5-(4-(4-Chlorophenyl)piperidin-1-yl)-2,2-diphenylpentanenitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41995 M1 CLONED HUMAN 3H-QNB FLUOXETINE 1030 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42251 CLONED HUMAN Functional K368,374C 0.3 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42507 CLONED RABBIT UNDEFINED erythromycin-A 190.546 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
43019 GAK CLONED HUMAN 3H-Staurosporine SB203580 39 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43275 CLK2 CLONED HUMAN 3H-Staurosporine EKB-569 700 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43531 INSR CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43787 MAPK12 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44043 TEK CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44299 CaMK CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44555 HCK CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44811 AURKC CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45067 SLK CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45323 CLONED HUMAN Functional alsterpaullone 110 Bain J, et al., 2003 Jan 15, 2025 Jan 15, 2025
45579 SLC6A3 CLONED HUMAN 3H-WIN 35,428 DOXEPIN >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45835 5-HT2B CLONED HUMAN 3H-LSD (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46091 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46603 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46859 M5 CLONED HUMAN 3H-QNB (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47115 M3 CLONED HUMAN 3H-NMS Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47371 Grik5 CLONED HUMAN 3H-Kainic acid LY 457691 1550 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47883 SST3 CLONED HUMAN 3H-thymidine BIM-23926 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
48139 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.04 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48651 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 12.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48907 Y1 CLONED Chicken [125I] - Peptide YY NPY, porcine 0.213796 Holmberg, SK et al., 2002 Jan 15, 2025 Jan 15, 2025
49163 CCK1 CLONED HUMAN 125I-CCK-8 TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-1-Adoc 840 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
49675 Y2 CLONED Chicken [125I] - Peptide YY NPY 3-36, porcine 0.74131 Salaneck E, et al., 2000 Jan 15, 2025 Jan 15, 2025
49931 mGluR6 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1996 Jan 15, 2025 Jan 15, 2025
50187 Kainate receptor CLONED UNDEFINED 3H-Kainic acid LY 382884 >10000 Bortolotto, Z., et al., 1999 Jan 15, 2025 Jan 28, 2025
50443 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N-Dimethyl-5-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine 7 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
58123 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 5.25 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58379 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5474 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58891 nAChR7 CLONED HUMAN 3H-Epibatidine Camel Snus extract 195.3 Harris A, et al., 2015 Jan 15, 2025 Jan 15, 2025
59147 5-HT1A CLONED HUMAN 3H-WAY100635 METHYSERGIDE 25 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025