71452 H1 CLONED HUMAN 3H-PYRILAMINE 4-acetoxy-N,N-diallyltryptamine 353 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
6172 D3 CLONED HUMAN 125I-IODOSULPRIDE SB204070 1000 WARDLE KA, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
7196 NK2 CLONED HUMAN 125I-[MePhe7]-NKB NKA 0.74 Sarau HM, et al., 1997 Jan 15, 2025 Jan 15, 2025
72732 MOR CLONED HUMAN 3H-DAMGO naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
72988 M1 CLONED HUMAN 3H-QNB catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7708 GABAA CLONED HUMAN 3H-MUSCIMOL Bicuculline 4466.83 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7964 GABAA CLONED HUMAN 3H-RO-15-1788 27 740 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8220 SST1 CLONED HUMAN 125I-LTT-SRIF28 CST14-Tyr10 2.75 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8476 SST3 CLONED HUMAN 125I-LTT-SRIF28 octreotide-Tyr3 144.54 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8732 SST2 CLONED HUMAN 125I-LTT-SRIF28 cortistatin14 1.77 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8988 SST3 CLONED HUMAN 125I-SRIF-28 CGP 23996 0.39 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
9500 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Chloro 0.22 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
75036 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75292 Beta3 CLONED HUMAN 125I-Pindolol Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10012 NET CLONED HUMAN 3H-Norepinephrine Nisoxetine Inhibitor 4.21 Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999 Jan 15, 2025 Jan 15, 2025
75804 Sigma 2 CLONED HUMAN 3H-DTG 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76060 5-HT2B CLONED HUMAN 3H-LSD Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76316 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
11036 H1 CLONED HUMAN 3H-MEPYRAMINE Cetirizine 6.3 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
76572 KOR CLONED HUMAN 3H-U69593 (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol 1120 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76828 M1 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11548 H1 BRAIN HUMAN 3H-PYRILAMINE NORTRYPTYLINE 6.3 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
77084 M5 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11804 FR. CORTEX HUMAN 3H-PRAZOSIN PHENTOLAMINE 15 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77340 Sigma 2 CLONED HUMAN 3H-DTG (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77596 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77852 5-HT2A CLONED HUMAN 3H-KETANSERIN (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78108 5-HT5A CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78364 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78620 Beta 1 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78876 5-HT1A CLONED HUMAN 3H-WAY100635 5-Methoxy-N-methyl-N-isopropyltryptamine 12.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79132 5-HT6 CLONED HUMAN 3H-LSD N,N-Diisopropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79388 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-2,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79644 CLONED HUMAN 3H-CLONIDINE (±)-2,5-Dimethoxy-4-ethylamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79900 M5 CLONED HUMAN 3H-QNB EMDT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80156 V2 CLONED HUMAN 3H-VASOPRESSIN 5-MeO-TMT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80412 5-HT4 CLONED HUMAN 3H-GR113808 (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80668 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15388 5-HT1B CLONED HUMAN 3H-5HT RAUWOLSCINE 46.77 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80924 5-HT2B CLONED HUMAN 3H-LSD 3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine 56.2341 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
81180 KOR CLONED HUMAN 3H-U69593 N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81436 H1 CLONED HUMAN 3H-PYRILAMINE 2-[4-[(2R)-2-(3,4-dimethylphenyl)-2-hydroxyethyl]piperazin-1-yl]pyridine-3-carbonitrile 2103 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
81692 Beta1 CLONED HUMAN 125I-iodo-pindolol (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81948 5-HT1B CLONED HUMAN 3H-5CT [18F]MH.MZ 1846 Herth MM et al 2009 Jan 15, 2025 Jan 15, 2025
16668 M3 CLONED HUMAN 3H-QNB SCOPOLAMINE 0.44 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82204 D5 CLONED HUMAN 3H-SCH23390 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82460 Alpha1A CLONED HUMAN 3H-PRAZOSIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine 2720 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
17180 5-HT1E CLONED HUMAN 3H-5HT METHYLPHENIDATE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
82716 5-HT3 CLONED HUMAN 3H-GR65630 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17692 CLONED HUMAN 125I-VIP VIP [D-Gln16] 1.1 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83228 5-HT2A CLONED HUMAN 125I-DOI KETANSERIN 4.1 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83484 DAT HEK293 cells HUMAN 3H-WIN 35,428 MDMA 6500 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83740 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 4693 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83996 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84252 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18972 H1 CLONED HUMAN 3H-MEPYRAMINE MEPYRAMINE 1.18 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84508 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19228 NB-OK-1 HUMAN 125-[AcHis1]Pacap PACAP(9-38) 50 Vandermeers A et al., 1992 Jan 15, 2025 Jan 15, 2025
84764 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85020 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19740 D2 CLONED HUMAN UNDEFINED MOLINDONE 6 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
85276 H1 recombinant HUMAN 3H-PYRILAMINE Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 28, 2025
86044 H3 CLONED HUMAN 3H-Alpha-methylhistamine (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
87324 Alpha1B placeholder HUMAN Placeholder Tamsulosin 0.13 Rak A et al 2016 Jan 15, 2025 Jan 28, 2025
87580 M5 CLONED HUMAN 3H-QNB 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
87836 A3 test HUMAN 3H-PSB-11 8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
22556 hERG CLONED HUMAN 3H-Methylspiperone SERTINDOLE 3 Kongsamut, S, et. al., 2002 Jan 15, 2025 Jan 15, 2025
88092 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
23068 MOR CLONED HUMAN 3H-Diprenorphine L-homocysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88604 M1 CLONED HUMAN 3H-QNB HALOPERIDOL 1600 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88860 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 23.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23580 NPFF2 CLONED HUMAN 125I-1DMe-Y8Fa RFRP-1 15 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
89116 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 40.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89372 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 2630 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24092 5-HT2A CLONED HUMAN 3H-SPIPERONE CLOZAPINE 5.2 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89628 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
24348 CORTEX HUMAN 3H-PRAZOSIN Fluoxetine-R-(-) 1528 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
89884 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
24604 ETB CLONED HUMAN UNDEFINED SR 144528 >10000 Rinaldi-Carmona, M et al., 1998 Jan 15, 2025 Jan 15, 2025
90140 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24860 SLC6A4 CLONED HUMAN 3H-CITALOPRAM CLOZAPINE 1624 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90396 A2B CLONED HUMAN 3H-PSB-603 N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
25116 CCR5 CLONED HUMAN 3H-Epibatidine Quetiapine >10000 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90652 A2B CLONED HUMAN 3H-PSB-603 N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25372 H4 CLONED HUMAN 3H-Histamine ARIPIPRAZOLE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90908 Alpha1D CHO cells HUMAN 3H-PRAZOSIN 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 10.7152 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
91164 A2A CLONED HUMAN 3H-CGS-21680 2-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine >10000 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
25884 H1 CLONED HUMAN 3H-PYRILAMINE Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91420 CB1 CLONED HUMAN 3H-CP55940 O-6659 109 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26140 KOR CLONED HUMAN 3H-Diprenorphine Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91932 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-(4-fluorophenyl) thiophen-3-yl)(4-chlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92188 D2 CLONED HUMAN 3H-RACLOPRIDE 4-Fluoro-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide 50 Zajdel P et al 2012 Jan 15, 2025 Jan 28, 2025
27164 5-HT1D CORTEX HUMAN 3H-5CT 1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride 1900 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92700 5-HT1D CLONED HUMAN 3H-Cimetidine 9,13-epoxylabd-5-ene-7 b,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27420 5-HT1D CLONED HUMAN 3H-GR-125743 APOMORPHINE 1230.27 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92956 5-HT6 CLONED HUMAN 3H-LSD OLANZAPINE 7 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
93724 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester 3.19 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28444 mGluR5 CLONED HUMAN 3H-Quisqualate (S)-4CPG >10000 Mutel V, et.al., 2000 Jan 15, 2025 Jan 28, 2025
93980 D2 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one 13 Ortega R et al 2011 Jan 15, 2025 Jan 29, 2025
28700 PKCα CLONED HUMAN 3H-PDBU ARIPIPRAZOLE >10000 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94236 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine 4200 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29212 SST3 CLONED HUMAN UNDEFINED BIM 23197 26.8 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94748 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
95004 D4 CLONED HUMAN 3H-Methylspiperone 2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
95516 5-HT6 CLONED HUMAN [3H]-LSD 7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride 68 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
95772 Alpha1D CLONED HUMAN 3H-PRAZOSIN Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
30492 M3 CLONED HUMAN 3H-QNB exo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 0.84 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
96284 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96540 5-HT1A CLONED HUMAN [3H]-Way100635 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31260 5-HT2A C.H.O. HUMAN 3H-KETANSERIN Ropinirole >10000 Millan MJ, et. al., 2004 Jan 15, 2025 Jan 15, 2025
96796 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 630 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31516 D2 CLONED HUMAN 125I-IODOSULPRIDE (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) 630.957 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97052 Sigma 1 CLONED HUMAN [3H]Pentazocine Fluorolintane (2-F-DPPy) 110 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97308 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 47.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
32028 5-HT2C CLONED HUMAN 3H-MESULERGINE RS-127445 398.107 Bonhaus, DW et. al., 1999 Jan 15, 2025 Jan 15, 2025
97564 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 402 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98076 CB1 CHO cells HUMAN 3H-CP-55940 CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate 0.6 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98332 D3 CLONED HUMAN [3H]-N-methylspiperone 2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline 2176 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98588 5-HT2C CLONED HUMAN [3H]-mesulergine 1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride 2976 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98844 Beta 2 CLONED HUMAN 3H-CGP-12177 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
99100 D3 CLONED HUMAN 3H-N-Methylspiperone (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99356 D3 CLONED HUMAN [3H]N-methylspiperone 1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2,3-dichlorophenyl)piperazine 14 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34076 P2X2, P2X3 CLONED HUMAN 3H-A-317491 AP3A 320 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99612 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1.62 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
100124 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) Quetiapine 413 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
34844 CB2 CLONED HUMAN 3H-CP-55940 Rinvanil >10000 Jan 15, 2025 Jan 15, 2025
100380 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Etoperidone >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
35356 D2 CLONED HUMAN 3H-SPIPERONE 10-[1,2,3,6-tetrahydro-1(2-propenyl)-4-pyridinyl]-5H-dibenzo[a,d]cycloheptene 83 Phillips ST, et. al., 1995 Jan 15, 2025 Jan 27, 2025
100892 BchE serum HUMAN Functional N-(3-{[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-methylamino}propyl)-3-(1H-indol-3-yl)propionamide 0.03 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 15, 2025
101148 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone 272 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
35868 SLC6A4 CLONED HUMAN 3H-PAROXETINE 3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 141 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101404 5-HT6 CLONED HUMAN 3H-LSD 2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 347 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36124 EP2 CHO (COX-1)cells HUMAN Functional Indomethacin 18 Riendeau D, et.al., 2001 Jan 15, 2025 Jan 15, 2025
36380 Platelets HUMAN 3H-SQ 29548 BM 573 1.3 Hanson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
101916 M5 CLONED HUMAN [3H]QNB Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36636 5-HT7 CLONED HUMAN 3H-5HT MIANSERIN 56 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102172 Alpha1D CLONED HUMAN [3H]prazosin NEMONAPRIDE 1802 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37916 CDK1 CLONED HUMAN Functional 4-[[3-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-5-yl]amino]-benzenesulfonamide 2100 Lin R, et al., 2005 Jan 15, 2025 Jan 15, 2025
38428 D3 CLONED HUMAN 3H-NEMONAPRIDE MCL-205 >10000 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
38684 UNDEFINED HUMAN 3H-hypoxanthine N-[(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-cyclohexylcarbamoyl-2-hydroxy-propyl]-2,4,6-trifluoro-benzamide 3600 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39196 MC4 CLONED HUMAN 125I-NDP-MSH alpha MSH 50.1 Nickolls SA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39708 5-HT2C CLONED HUMAN 3H-5HT mCPP 14.1254 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40476 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln-Thr-NH2 739 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40732 mGluR5 CLONED HUMAN Functional 9-Cyclopropylamino-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one >10000 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41244 CLONED HUMAN 125I-Chemokine C28H32NClO 5500 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41500 CLONED HUMAN 3H-dexamethasone dexamethasone 6.7 Belvisi MG, et al., 2005 Jan 15, 2025 Jan 15, 2025
42012 M2 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42268 CLONED HUMAN 125I-Motilin Delta 30C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42524 CLONED HUMAN Functional [ala1,leu13]pMOT(1-14) 588.844 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42780 Y1 CLONED HUMAN 125I-PYY PYY 2 Kakui N, et al., 2006 Jan 15, 2025 Jan 15, 2025
43036 MAPK8 CLONED HUMAN 3H-Staurosporine Gleevec 3200 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43292 DAPK2 CLONED HUMAN 3H-Staurosporine SU11248 470 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43548 PAK4 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43804 CaMK CLONED HUMAN 3H-Staurosporine BIRB-796 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44060 CaMK CLONED HUMAN 3H-Staurosporine Tarceva >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44316 INSR CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44572 NEK9 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44828 CLK4 CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45084 PKMYT1 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45596 NET CLONED HUMAN 3H-Nisoxetine IPRINDOLE 1262 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
46108 Alpha2B CLONED HUMAN 3H-CLONIDINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47132 CLONED HUMAN 3H-SUBSTANCE P Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47388 D2 CLONED HUMAN 3H-SPIPERONE N-(1-Benzylpiperidin-4-yl)-2-naphthamide 1000 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47644 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 1.5 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47900 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 66 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48668 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49692 5-HT5A CLONED HUMAN 3H-LSD Pramipexole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
50460 SLC6A3 CLONED HUMAN 3H-WIN 35,428 N,N-Dimethyl-5-(4-fluorobutoxy)-2-(2-amino-4-methylphenoxy)benzylamine 3604 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
51484 Alpha1A UNDEFINED HUMAN UNDEFINED 3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 0.73 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51740 AR UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline 290 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51996 DOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 5.38 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52252 A2B UNDEFINED HUMAN UNDEFINED 1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione >10000 Drabczyńska A et al., 2007 Jan 15, 2025 Jan 15, 2025
52508 Alpha2B UNDEFINED HUMAN UNDEFINED 2-((2-(2-fluorophenyl)-7-methoxybenzofuran-4-yl)methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline 299 Hagihara K et al., 2007 Jan 15, 2025 Jan 15, 2025
52764 D2 UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide 5 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
53020 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan 0.31 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
53532 SLC6A2 UNDEFINED HUMAN UNDEFINED 1-[1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 18 Mahaney PE et al., 2008 Jan 15, 2025 Jan 15, 2025
53788 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one 90.9 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54556 A1 UNDEFINED HUMAN UNDEFINED 8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 443 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54812 D3 UNDEFINED HUMAN UNDEFINED N-(4-Propylaminobutyl)-4-biphenylcarboxamide >10000 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55068 D2 UNDEFINED HUMAN UNDEFINED 4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 64 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55324 KOR UNDEFINED HUMAN UNDEFINED 8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 137 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55580 MOR UNDEFINED HUMAN UNDEFINED N-Cyclopropylmethyl-14beta-4'-methylcinnamoyloxy-7,8-dihydrocodeinone 4.2 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
56092 MOR UNDEFINED HUMAN UNDEFINED (1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide 0.3 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
56604 NR3C1 UNDEFINED HUMAN UNDEFINED Benzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol 1150 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
56860 SLC6A4 UNDEFINED HUMAN UNDEFINED (3S)-3-((3-( 6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one 15 Rotella DP et al., 2009 Jan 15, 2025 Jan 15, 2025
57628 SST3 UNDEFINED HUMAN UNDEFINED N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57884 Beta2 UNDEFINED HUMAN UNDEFINED (2S,3S,4S,5R,6S)-6-(5-((R)-2-(5,6-diethyl-2,3-dihydro-1H-inden-2-ylamino)-1-hydroxyethyl)-2-oxo-1,2-dihydroquinolin-8-yloxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid >10000 Baur F et al., 2010 Jan 15, 2025 Jan 28, 2025
58140 5-HT2C CLONED HUMAN 125I-DOI N-(3-Iodobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 1.05 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58396 D1 CLONED HUMAN 3H-SCH23390 MRS5474 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58652 D3 CLONED HUMAN 3H-N-Methylspiporone Benzquinamide 3592 Gregori-Puigjane E, et al., 2012 Jan 15, 2025 Jan 15, 2025
58908 nAChR CLONED HUMAN 3H-Epibatidine Camel Snus extract 17.6 Harris A, et al., 2015 Jan 15, 2025 Jan 27, 2025
59420 D4 CLONED HUMAN 3H-N-Methylspiporone N-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide 1.5 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
60188 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-((1H-Pyrazol-3-yl)ethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 2.23 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60444 GABAA CLONED HUMAN FNZ QH-II-090 17 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60700 GABAA CLONED HUMAN FNZ YCT-5 200 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60956 GABAA CLONED HUMAN FNZ YT-II 3.518 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61212 GABAA CLONED HUMAN FNZ RY-061 17 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61468 GABAA CLONED HUMAN FNZ RY-059 89 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61724 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(4-methoxyphenyl)propan-1-amine 206 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62236 5-HT6 CLONED HUMAN 3H-LSD Tianeptine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
63516 NET CLONED HUMAN 3H-Nisoxetine 3-methoxy-diphenidine 325 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
63772 CXCR3 PHA/IL-2 T cells HUMAN 125I-CXCL11 CXCL9 29.5 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
64540 CLONED HUMAN 3H-Estradiol Methyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate 1 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
65308 GABAA CLONED HUMAN [3H] Flunitrazepam MLT-II-18 >10000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65565 GABAA CLONED HUMAN [3H] Flunitrazepam Alprazolam 1.43 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65821 GABAA CLONED HUMAN [3H] Flunitrazepam CM-D45 C19H21N3O4 1.65 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66077 M1 CLONED HUMAN 3H-QNB Mellpaladine A 7200 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66589 DOR CLONED HUMAN 3H-DADLE 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 29, 2025
66845 H4 CLONED HUMAN 3H-Histamine N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67101 SERT CLONED HUMAN 3H-CITALOPRAM 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67357 D1 CLONED HUMAN 3H-SCH23390 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67613 5-HT2C KIDNEY HUMAN 3H-MESULERGINE Ethyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate 30 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2333 5-HT3 AMYGDALA HUMAN 3H-ZACOPRIDE HISTAMINE >10000 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67869 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline ) 97 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68637 recombinant HUMAN UNKNOWN N-(Indan-2-yl)-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
3357 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IDAZOXAN 662 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68893 SST1 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH2 0.501187 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69149 H4 CLONED HUMAN 3H-N-alpha-methylhistamine N-alpha-methylhistamine 316.228 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3869 D1 CLONED HUMAN 3H-SCH23390 RISPERIDONE 523 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69661 BZP CLONED HUMAN FNZ 2-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
69917 D5 CLONED HUMAN 3H-SCH23390 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4637 SLC6A3 CLONED HUMAN 3H-WIN 35,428 BINDING 5-Hydroxy Tryptamine >10000 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4893 5-HT2A CLONED HUMAN 125I-DOI LY 063518 137 BRYANT HU, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
70429 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) MRP3215 7.4 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5149 5-HT2C CLONED HUMAN 125I-DOI DOCN 1011 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70685 DOR CLONED HUMAN 3H-Diprenorphine Tapentadol >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 28, 2025
5405 5-HT2C Choroid Plexus HUMAN 3H-MESULERGINE KETANSERIN 50.11 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
70941 5-HT1D CLONED HUMAN 125I-aminopotentidine (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 546 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
71197 5-HT1A CLONED HUMAN WAY100635 SYA16263 1.1 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
5917 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE BAM 1303 5.28 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
71453 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
7197 NK2 CLONED HUMAN 125I-[MePhe7]-NKB Substance P 129 Sarau HM, et al., 1997 Jan 15, 2025 Jan 15, 2025
72733 NET CLONED HUMAN 3H-Nisoxetine naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
72989 M2 CLONED HUMAN 3H-QNB catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7709 GABAA CLONED HUMAN 3H-MUSCIMOL Thio-4-PIOL 446.68 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7965 GABAA CLONED HUMAN 3H-RO-15-1788 28 319 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8221 SST1 CLONED HUMAN 125I-LTT-SRIF28 seglitide >10000 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8477 SST3 CLONED HUMAN 125I-LTT-SRIF28 L-362,855 23.98 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8733 SST2 CLONED HUMAN 125I-LTT-SRIF28 BIM 23030 16.98 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8989 SST3 CLONED HUMAN 125I-SRIF-28 BIM 23052 1.99 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74525 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74781 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
9501 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Phenyl 0.15 Sugden D, Pickering H, Teh MT, Garratt PJ, 1997 Jan 15, 2025 Jan 15, 2025
75037 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75293 Beta 2 CLONED HUMAN 3H-CGP12177 Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10013 NET CLONED HUMAN 3H-Norepinephrine DESIPRAMINE 8.54 Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999 Jan 15, 2025 Jan 15, 2025
75549 M1 CLONED HUMAN 3H-QNB propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75805 SERT CLONED HUMAN 3H-CITALOPRAM 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76061 5-HT2C CLONED HUMAN 3H-MESULERGINE Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76317 Beta 1 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11037 H1 CLONED HUMAN 3H-MEPYRAMINE CHLORPHENIRAMINE 2.51 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
76573 MOR CLONED HUMAN 3H-DAMGO (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol 2670 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76829 M2 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11549 H1 BRAIN HUMAN 3H-PYRILAMINE PAROXETINE >10000 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
77085 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11805 FR. CORTEX HUMAN 3H-PRAZOSIN CLOZAPINE 160 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77341 DOR CLONED HUMAN 3H-DADLE (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77597 5-HT1B CLONED HUMAN 3H-5-CT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77853 5-HT2B CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78109 5-HT6 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78365 Alpha1D CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78621 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78877 5-HT1A CLONED HUMAN 3H-WAY100635 N,N-Diisopropyltryptamine 120.5 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
13597 OT Myometrium HUMAN 3H-Oxytocin L-365,209 8.7 Pettibone DJ, et al., 1991 Jan 15, 2025 Jan 15, 2025
79133 5-HT6 CLONED HUMAN 3H-LSD 5-Methoxy-N,N-diisopropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79389 Alpha1B CLONED HUMAN 3H-PRAZOSIN LYSERGIC ACID 8677 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79645 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-2,5-Dimethoxy-4-bromoamphetamine 2193 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79901 M5 CLONED HUMAN 3H-QNB Salvinorin A >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80157 CLONED HUMAN 3H-VASOPRESSIN (±)-2,5-Dimethoxy-4-bromoamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80413 5-HT5A CLONED HUMAN 3H-LSD (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80669 5-HT1B CLONED HUMAN 3H-5-CT (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15389 5-HT1B CLONED HUMAN 3H-5HT 8-OH-DPAT 2818.38 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80925 5-HT2B CLONED HUMAN 3H-LSD 5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine 104.713 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
81181 MOR CLONED HUMAN 3H-DAMGO N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81437 H1 CLONED HUMAN 3H-PYRILAMINE N-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide 2096 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
81693 Beta2 CLONED HUMAN 125I-iodo-pindolol (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81949 5-HT1E CLONED HUMAN 3H-5HT [18F]MH.MZ >10000 Herth MM et al 2009 Jan 15, 2025 Jan 15, 2025
16669 M3 CLONED HUMAN 3H-QNB Trihexyphenidyl 6.4 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82205 D2 CLONED HUMAN 3H-N-Methylspiperone 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one 585 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82461 Alpha1B CLONED HUMAN 3H-PRAZOSIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine 7211.1 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82717 5-HT4 CLONED HUMAN 3H-GR113808 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82973 A2A CHO cells HUMAN 3H-MSX-2 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 2440 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
17693 CLONED HUMAN 125I-VIP VIP [D-Asn28] 0.71 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83229 5-HT2A CLONED HUMAN 125I-DOI MDL 100907 0.67 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83485 SERT HEK293 cells HUMAN 3H-CITALOPRAM MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83741 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 8897 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83997 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 165 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84253 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 5751 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18973 CCK2 CLONED HUMAN 125I-BH-CCK-8 44 25.1189 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
84509 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19229 NB-OK-1 HUMAN 125-[AcHis1]Pacap PACAP(8-38) 30 Vandermeers A et al., 1992 Jan 15, 2025 Jan 15, 2025
84765 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85021 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19741 D2 CLONED HUMAN UNDEFINED MOPERONE 1.8 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
19997 Platelets HUMAN 3H-NECA ddCHA >10000 Lohse MJ et al., 1988a Jan 15, 2025 Jan 15, 2025
86045 H4 CLONED HUMAN 3H-Histamine (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
87325 Alpha1B placeholder HUMAN Placeholder Terazosin 1.73 Rak A et al 2016 Jan 15, 2025 Jan 28, 2025
87581 MOR CLONED HUMAN 3H-DAMGO 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
87837 A3 test HUMAN 3H-PSB-11 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
22557 hERG CLONED HUMAN 3H-Methylspiperone PIMOZIDE 18 Kongsamut, S, et. al., 2002 Jan 15, 2025 Jan 15, 2025
88093 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
23069 MOR CLONED HUMAN 3H-Diprenorphine L-cysteic acid >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88605 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88861 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 647 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23581 NPFF2 CLONED HUMAN 125I-1DMe-Y8Fa RFRP-3 55 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
89117 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 8.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89373 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 54 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24093 5-HT2A CLONED HUMAN 3H-SPIPERONE FLUPHENAZINE 5.8 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
24349 CORTEX HUMAN 3H-PRAZOSIN FLUOXETINE 3171 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
89885 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
24605 CLONED HUMAN UNDEFINED SR 144528 >10000 Rinaldi-Carmona, M et al., 1998 Jan 15, 2025 Jan 15, 2025
90141 D2 CLONED HUMAN 3H-SPIPERONE , 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24861 CCR5 CLONED HUMAN 3H-Epibatidine CLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90397 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
25117 nAChR7 CLONED HUMAN 3H-Epibatidine Quetiapine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90653 A2B CLONED HUMAN 3H-PSB-603 N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90909 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 26.9153 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
25629 Alpha1B CLONED HUMAN 125I-HEAT COCAINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91165 A1 CLONED HUMAN 3H-DPCPX 2-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine >10000 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
25885 SLC6A3 CLONED HUMAN 3H-GBR 12935 Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91421 CB1 CLONED HUMAN 3H-SR144528 O-6659 128 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
91933 A1 CLONED HUMAN 3H-DPCPX (2-Amino-5-(2,3-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92189 D2 CLONED HUMAN 3H-RACLOPRIDE 4-Fluoro-N-({1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl} methyl) benzenesulfonamide 46 Zajdel P et al 2012 Jan 15, 2025 Jan 28, 2025
27165 5-HT1D CORTEX HUMAN 3H-5CT AL-37350A >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92701 5-HT1D CLONED HUMAN 3H-Cimetidine (8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27421 5-HT1B CLONED HUMAN 3H-GR-125743 BROMOCRIPTINE 354.813 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92957 5-HT2A CLONED HUMAN 3H-KETANSERIN WA-13 1830 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
28189 H2 CLONED HUMAN 3H-TIOTIDINE METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93725 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 3.73 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28445 CLONED HUMAN 3H-Quisqualate AIDA >10000 Mutel V, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93981 D2 CLONED HUMAN 3H-SPIPERONE 2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile 22 Ortega R et al 2011 Jan 15, 2025 Jan 29, 2025
28701 PKCΓ CLONED HUMAN 3H-PDBU ARIPIPRAZOLE 8000 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94237 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine 1900 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29213 SST3 CLONED HUMAN UNDEFINED CH275 1000 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94749 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
95005 D4 CLONED HUMAN 3H-Methylspiperone 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
95517 5-HT6 CLONED HUMAN [3H]-LSD 7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride 1902 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
95773 Alpha1A CLONED HUMAN 3H-PRAZOSIN Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
30493 M4 CLONED HUMAN 3H-QNB exo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 0.27 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
96285 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
31005 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96541 5-HT1B CLONED HUMAN [3H]5-CT 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31261 5-HT2B C.H.O. HUMAN 3H-MESULERGINE Ropinirole 3801.89 Millan MJ, et. al., 2004 Jan 15, 2025 Jan 15, 2025
96797 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 6400 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31517 D3 CLONED HUMAN 125I-IODOSULPRIDE (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) 1000 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97309 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 1.05 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
32029 5-HT3 CLONED HUMAN UNDEFINED RS-127445 1000 Bonhaus, DW et. al., 1999 Jan 15, 2025 Jan 15, 2025
97565 A2B CLONED HUMAN [3H]DPCPX (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98077 CB2 CHO cells HUMAN 3H-CP-55940 CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate 1050 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98333 D3 CLONED HUMAN [3H]-N-methylspiperone 2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 31 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98589 5-HT2C CLONED HUMAN [3H]-mesulergine ARIPIPRAZOLE 76 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98845 DAT CLONED HUMAN 3H-WIN 35,428 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
33565 5-HT6 CLONED HUMAN 3H-LSD CELECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99101 D3 CLONED HUMAN 3H-N-Methylspiperone (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99357 D3 CLONED HUMAN [3H]N-methylspiperone 5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole 1.47 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34077 P2X2, P2X3 CLONED HUMAN 3H-A-317491 AP2A >10000 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99613 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine 1.91 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
100125 Sigma 2 CLONED HUMAN 3H-DTG Quetiapine 1566 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
34845 CB2 CLONED HUMAN 3H-CP-55940 Rinvanil, Acetyl >10000 Jan 15, 2025 Jan 15, 2025
100381 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
35357 D4 CLONED HUMAN 3H-SPIROPERIDOL CLOZAPINE 21 Phillips ST, et. al., 1995 Jan 15, 2025 Jan 15, 2025
100893 AChE BRAIN HUMAN Functional N-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide 2.9 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
101149 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone 350 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
35869 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 74 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101405 5-HT7 CLONED HUMAN 3H-5-CT 2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 371 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36125 CA2+ platelets HUMAN Functional Indomethacin 2 Riendeau D, et.al., 2001 Jan 15, 2025 Jan 15, 2025
101661 Alpha1B CLONED HUMAN [3H]-prazosin Perospirone 44 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
36381 Platelets HUMAN 3H-SQ 29548 BM 613 1.4 Hanson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
101917 Beta3 CLONED HUMAN [3H]-CGP12177 Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36637 5-HT2C CLONED HUMAN 3H-MESULERGINE (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 7.6 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102173 Sigma 2 CLONED HUMAN [3H]DTG NEMONAPRIDE 137 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37917 CDK1 CLONED HUMAN Functional 3-Amino-5-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carbothioamide 3.2 Lin R, et al., 2005 Jan 15, 2025 Jan 15, 2025
38429 D3 CLONED HUMAN 3H-NEMONAPRIDE SKF 82958 77.3 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
38685 UNDEFINED HUMAN 3H-hypoxanthine N-[(1S,2S)-3-Cyclohexylcarbamoyl-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl]-2,4,6-trifluoro-benzamide 4940 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39197 MC4 CLONED HUMAN 125I-NDP-MSH Beta MSH 18.6 Nickolls SA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39709 5-HT2C CLONED HUMAN 3H-5HT METHYLERGONOVINE 4.57088 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40477 STAT3 CLONED HUMAN Functional Ac-pTyr-Val-Pro-Gln-Thr-NH2 1540 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40733 mGluR5 CLONED HUMAN Functional 9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one 49 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41245 CLONED HUMAN 125I-Chemokine 4-(4-Chlorophenyl)-1-(4-phenyl-4-m-tolylbutyl)piperidin-4-ol Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
42013 M2 CLONED HUMAN 3H-QNB Femoxetine 150 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42269 CLONED HUMAN 125I-Motilin Delta 31-32 2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42525 CLONED HUMAN Functional [ala3,leu13]pMOT(1-14) 1.31826 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42781 Y2 CLONED HUMAN 125I-PYY FMS586 >10000 Kakui N, et al., 2006 Jan 15, 2025 Jan 15, 2025
43037 MAPK9 CLONED HUMAN 3H-Staurosporine Staurosporine 1100 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43293 DAPK2 CLONED HUMAN 3H-Staurosporine LY-333531 2600 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43549 PAK6 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43805 CaMK CLONED HUMAN 3H-Staurosporine BIRB-796 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44061 CaMK CLONED HUMAN 3H-Staurosporine Tarceva >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44317 MAPK8 CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44573 NTRK1 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44829 CSK CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45085 MAPK14 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45597 SLC6A3 CLONED HUMAN 3H-WIN 35,428 IPRINDOLE 6530 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
46109 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone 23.36 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47133 CLONED HUMAN 3H-SUBSTANCE P Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47389 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-Phenylethylpiperidin-4-yl)-2-naphthamide 139 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47645 GABAA CLONED HUMAN 3H-RO-15-1788 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.25 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47901 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 56 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48669 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49693 5-HT6 CLONED HUMAN 3H-LSD Pramipexole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
51485 Alpha1A UNDEFINED HUMAN UNDEFINED 3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3.5 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51741 AR UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline 346 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51997 DOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 8 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52253 A2B UNDEFINED HUMAN UNDEFINED 9-(2-(benzylamino)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione >10000 Drabczyńska A et al., 2007 Jan 15, 2025 Jan 15, 2025
52509 Alpha2B UNDEFINED HUMAN UNDEFINED 6,7-dimethoxy-2-((7-methoxy-2-(3-methoxyphenyl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 804 Hagihara K et al., 2007 Jan 15, 2025 Jan 15, 2025
52765 D2 UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide 15 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
53021 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan 0.26 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
53533 SLC6A2 UNDEFINED HUMAN UNDEFINED (-)-1-[(1S)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 14 Mahaney PE et al., 2008 Jan 15, 2025 Jan 15, 2025
53789 5-HT2A UNDEFINED HUMAN UNDEFINED CLOZAPINE 8.9 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54557 A1 UNDEFINED HUMAN UNDEFINED 8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-ethyl-3,7-dihydropurine-2,6-dione 1000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54813 D3 UNDEFINED HUMAN UNDEFINED N-(4-Dipropylaminobutyl)-4-biphenylcarboxamide 950 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55069 D2 UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide 226 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55325 KOR UNDEFINED HUMAN UNDEFINED 8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 150 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55581 MOR UNDEFINED HUMAN UNDEFINED N-Cyclopropylmethyl-14beta-4'-chlorocinnamoyloxy-7,8-dihydrocodeinone 3.5 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
56093 MOR UNDEFINED HUMAN UNDEFINED 6-desoxonaltrexone 0.24 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
56605 NR3C1 UNDEFINED HUMAN UNDEFINED Benzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol 7 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
56861 SLC6A4 UNDEFINED HUMAN UNDEFINED (3S)-3-((3-( 6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one 4 Rotella DP et al., 2009 Jan 15, 2025 Jan 15, 2025
57629 SST3 UNDEFINED HUMAN UNDEFINED N-(1-(3-ethoxy-4-fluorobenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57885 SLC6A3 UNDEFINED HUMAN UNDEFINED MAZINDOL 22.1 O'Neill DJ et al., 2010 Jan 15, 2025 Jan 15, 2025
58141 5-HT2C CLONED HUMAN 125I-DOI N-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 4.27 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58397 D2 CLONED HUMAN 3H-N-Methylspiporone MRS5698 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58653 D4 CLONED HUMAN 3H-N-Methylspiporone Benzquinamide 574 Gregori-Puigjane E, et al., 2012 Jan 15, 2025 Jan 15, 2025
58909 nAChR CLONED HUMAN 3H-Epibatidine Nicotine 22.2 Harris A, et al., 2015 Jan 15, 2025 Jan 27, 2025
59421 D2 CLONED HUMAN 3H-N-Methylspiporone N-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide 60 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59677 5-HT1A CLONED HUMAN 3H-WAY100635 MH.MZ >10000 Herth, M. et. al., 2009 Jan 15, 2025 Jan 15, 2025
60189 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(2-((1-methyl-1H-pyrazol-4-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)bicyclo[3.1.0]- hexane-1-carboxamide 2.34 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60445 GABAA CLONED HUMAN FNZ XLI-286 0.684 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60701 GABAA CLONED HUMAN FNZ YCT-5 >10000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60957 GABAA CLONED HUMAN FNZ YT-II 0.8712 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61213 GABAA CLONED HUMAN FNZ ZG-224 17.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61469 GABAA CLONED HUMAN FNZ RY-047 200 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61725 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2,5-dimethoxyphenyl)propan-1-amine 273 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
61981 CLONED HUMAN UNDEFINED IMIPRAMINE 3400 Teschemacher, AG et al., 1999 Jan 15, 2025 Jan 15, 2025
62237 5-HT7 CLONED HUMAN 3H-LSD Tianeptine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
62749 H1 Brain Frontal Cortex HUMAN 3H-doxepin DOXEPIN 0.24 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 28, 2025
63517 NET CLONED HUMAN 3H-Nisoxetine 4-methoxy-diphenidine 2700 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
63773 CXCR3 PHA/IL-2 T cells HUMAN 125I-CXCL11 CXCL10 21.9 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
64541 CLONED HUMAN 3H-Estradiol 1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 15 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
64797 Beta1 CLONED HUMAN 125I-ICYP Indacaterol 6.21 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
65309 GABAA CLONED HUMAN [3H] Flunitrazepam SHU-1-19 4 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65566 GABAA CLONED HUMAN [3H] Flunitrazepam Alprazolam 1.54 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65822 GABAA CLONED HUMAN [3H] Flunitrazepam CM-D45 C19H21N3O4 0.23 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66078 M1 CLONED HUMAN 3H-QNB Mellpaladine B 5172 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66846 M1 CLONED HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67102 NET CLONED HUMAN 3H-Nisoxetine 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67358 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67614 A1 KIDNEY HUMAN 3H-N6 -phenylisopropyladenosine Ethyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate 360 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2334 5-HT3 HIPPOCAMPUS HUMAN 3H-ZACOPRIDE HISTAMINE >10000 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67870 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68638 recombinant HUMAN UNKNOWN N-(Adamant-2-yl)-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
3358 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IMIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68894 SST2 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH2 1.25893 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69150 H4 CLONED HUMAN 3H-N-alpha-methylhistamine Alpha-Methylhistamine-R 251.189 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3870 D1 CLONED HUMAN 3H-SCH23390 CLOZAPINE 196 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69662 BZP CLONED HUMAN FNZ 3-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
69918 D5 CLONED HUMAN 3H-SCH23390 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4638 SLC6A3 CLONED HUMAN 3H-WIN 35,428 BINDING RESERPINE >10000 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4894 5-HT2A CLONED HUMAN 125I-DOI LY 314228 65 BRYANT HU, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
70430 5-HT7 CLONED HUMAN 3H-LSD MRP3215 5.9 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5150 5-HT2C CLONED HUMAN 125I-DOI DOPR 1.1 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70686 DOR CLONED HUMAN 3H-Diprenorphine Tramadol(+-) >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 28, 2025
70942 5-HT1D CLONED HUMAN 125I-aminopotentidine 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
71198 5-HT1A CLONED HUMAN WAY100635 SYA013 117.4 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
5918 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE OXYMETAZOLINE 754 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
6686 D2 CLONED HUMAN 3H-NEMONAPRIDE RISPERIDONE 27 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
7198 NK2 CLONED HUMAN 125I-[MePhe7]-NKB NKB [MePhe7] 1597 Sarau HM, et al., 1997 Jan 15, 2025 Jan 15, 2025
72734 SERT CLONED HUMAN 3H-CITALOPRAM naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
72990 M3 CLONED HUMAN 3H-QNB catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7710 GABAA CLONED HUMAN 3H-MUSCIMOL SR 95531 34.67 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7966 GABAA CLONED HUMAN 3H-RO-15-1788 29 >10000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8222 SST1 CLONED HUMAN 125I-LTT-SRIF28 CGP 23996 4.67 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8478 SST3 CLONED HUMAN 125I-LTT-SRIF28 L-363,301 457.08 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8734 SST2 CLONED HUMAN 125I-LTT-SRIF28 BIM 23056 467.73 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8990 SST3 CLONED HUMAN 125I-SRIF-28 BIM 23056 100 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74526 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74782 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75038 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10014 NET CLONED HUMAN 3H-Norepinephrine IMIPRAMINE 118 Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999 Jan 15, 2025 Jan 15, 2025
75550 M2 CLONED HUMAN 3H-QNB propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75806 NET CLONED HUMAN 3H-Nisoxetine 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76062 5-HT3 CLONED HUMAN 3H-GR-65630 Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76318 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
11038 H1 CLONED HUMAN 3H-MEPYRAMINE HISTAMINE 1258.92 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
76830 M3 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11550 H1 BRAIN HUMAN 3H-PYRILAMINE SERTRALINE >10000 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
77086 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
11806 FR. CORTEX HUMAN 3H-RAUWOLSCINE THIOTHIXENE,cis- 200 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77342 KOR CLONED HUMAN 3H-U69593 (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 1030 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77598 5-HT1D CLONED HUMAN 3H-5-CT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77854 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78110 5-HT7 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78366 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78622 Beta 2 CLONED HUMAN 3H-CGP12177 (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78878 5-HT1A CLONED HUMAN 3H-WAY100635 5-Methoxy-N,N-diisopropyltryptamine 132.4 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
13598 OT Myometrium HUMAN 3H-Oxytocin L-366,670 4.1 Pettibone DJ, et al., 1991 Jan 15, 2025 Jan 15, 2025
79134 5-HT6 CLONED HUMAN 3H-LSD N,N-Dipropyltryptamine 4543 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79390 Alpha1B CLONED HUMAN 3H-PRAZOSIN cis-2a >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79646 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 3,4,5-Trimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79902 H1 CLONED HUMAN 3H-PYRILAMINE (±)-2,5-Dimethoxy-4-bromoamphetamine 9120 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
80158 CLONED HUMAN 3H-VASOPRESSIN (±)-3,4-Methylenedioxymethamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80414 5-HT6 CLONED HUMAN 3H-LSD (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80670 5-HT1D CLONED HUMAN 3H-5-CT (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15390 5-HT1B CLONED HUMAN 3H-5HT 5-HT,2-Me 512.86 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80926 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine 10.4713 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
81182 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81438 D2 CLONED HUMAN 3H-N-Methylspiperone N-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
81950 5-HT2A CLONED HUMAN 125I-DOI [18F]MH.MZ 3 Herth MM et al 2009 Jan 15, 2025 Jan 15, 2025
16670 M3 CLONED HUMAN 3H-QNB Procyclidine 12.4 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82206 D3 CLONED HUMAN 3H-N-Methylspiperone 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one 32 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82462 Alpha1D CLONED HUMAN 3H-PRAZOSIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine 2307 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
17182 5-HT2B CLONED HUMAN 3H-5HT METHYLPHENIDATE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
82718 5-HT5A CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17694 PANC1 HUMAN 125I-VIP VIP [D-Gln16] 2.9 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83230 5-HT2A CLONED HUMAN 3H-KETANSERIN MDL 100907 0.048 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83486 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83742 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 5536 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83998 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5029 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84254 5-HT7 CLONED HUMAN 3H-LSD (±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 1205 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
18974 CCK2 CLONED HUMAN 125I-BH-CCK-8 43 776.247 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
84510 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19230 NB-OK-1 HUMAN 125-[AcHis1]Pacap PACAP(7-38) 8 Vandermeers A et al., 1992 Jan 15, 2025 Jan 15, 2025
84766 MOR CLONED HUMAN 3H-DAMGO ±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85022 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19742 D2 CLONED HUMAN UNDEFINED N-DESMETHYLCLOZAPINE 100 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
85278 5-HT1D recombinant HUMAN 125I-iodoaminopotentidine Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 28, 2025
19998 Platelets HUMAN 3H-NECA alpha-ddCHA >10000 Lohse MJ et al., 1988a Jan 15, 2025 Jan 15, 2025
85790 D1 CLONED HUMAN 3H-SCH23390 N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide >10000 Fiorino F et al 2017 Jan 15, 2025 Jan 28, 2025
86046 KOR CLONED HUMAN 3H-U69593 (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86302 A1 CLONED HUMAN 3H-CCPA 3-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 156 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
86558 A2B CLONED HUMAN 3H-PSB-603 1-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1000 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87326 Alpha1A placeholder HUMAN Placeholder Terazosin 51.89 Rak A et al 2016 Jan 15, 2025 Jan 28, 2025
87582 NET CLONED HUMAN 3H-Nisoxetine 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
88094 A1 CLONED HUMAN 3H-CCPA 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
23070 MOR CLONED HUMAN 3H-Diprenorphine D-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88606 5-HT2A CLONED HUMAN 3H-KETANSERIN HALOPERIDOL 120 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88862 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23582 NPFF2 CLONED HUMAN 125I-1DMe-Y8Fa FMRFamide 13 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
89118 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 12 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89374 5-HT7 CLONED HUMAN 3H-5-CT 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 32 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24094 5-HT2A CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 103 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89630 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0645654 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
24350 CORTEX HUMAN 3H-PRAZOSIN PAROXETINE 2741 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
89886 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
24606 M1 CLONED HUMAN UNDEFINED SR 144528 >10000 Rinaldi-Carmona, M et al., 1998 Jan 15, 2025 Jan 15, 2025
90142 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90398 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
25118 nAChR CLONED HUMAN 3H-Epibatidine Quetiapine >10000 Jensen NH, et al., 2008 Jan 15, 2025 Jan 27, 2025
90654 A2B CLONED HUMAN 3H-PSB-603 N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25374 D5 CLONED HUMAN 3H-SCH23390 ARIPIPRAZOLE 1676 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90910 Alpha1A CHO cells HUMAN 3H-PRAZOSIN 8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 6.45654 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
91166 A1 CLONED HUMAN 3H-DPCPX N-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide >10000 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
91422 5-HT2A CLONED HUMAN 125I-DOI 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate 0.54 Li P et al 2014 Jan 15, 2025 Jan 15, 2025
26142 5-HT5A CLONED HUMAN 3H-LSD Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91934 A1 CLONED HUMAN 3H-DPCPX (2-Amino-5-(2,4-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92190 D2 CLONED HUMAN 3H-RACLOPRIDE 4-Fluoro-N-({1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl}methyl) benzenesulfonamide 839 Zajdel P et al 2012 Jan 15, 2025 Jan 28, 2025
92702 5-HT1D CLONED HUMAN 3H-Cimetidine 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27422 5-HT1D CLONED HUMAN 3H-GR-125743 BROMOCRIPTINE 10.7152 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92958 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine 5047 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
28190 NET CLONED HUMAN 3H-Nisoxetine METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93726 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 18.6 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28446 mGluR5 CLONED HUMAN 3H-Quisqualate AIDA >10000 Mutel V, et.al., 2000 Jan 15, 2025 Jan 28, 2025
93982 D2 CLONED HUMAN 3H-SPIPERONE 3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 8.8 Ortega R et al 2011 Jan 15, 2025 Jan 29, 2025
94238 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-benzyloxy-2,5-dimethoxyphenethylamine 110 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29214 SST3 CLONED HUMAN UNDEFINED L-797,591 2240 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94750 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
95518 5-HT6 CLONED HUMAN [3H]-LSD 1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione >10000 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
95774 Alpha1B CLONED HUMAN 3H-PRAZOSIN Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
30494 M5 CLONED HUMAN 3H-QNB exo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 0.56 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
96286 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96542 5-HT1D CLONED HUMAN [3H]5-CT 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31262 5-HT2C C.H.O. HUMAN 3H-MESULERGINE Ropinirole >10000 Millan MJ, et. al., 2004 Jan 15, 2025 Jan 15, 2025
96798 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 3200 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31518 D3 CLONED HUMAN 125I-IODOSULPRIDE (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) 1258.93 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97054 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97310 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 10.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
32030 CB1 CLONED HUMAN UNDEFINED RS-127445 1000 Bonhaus, DW et. al., 1999 Jan 15, 2025 Jan 27, 2025
97566 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 8.1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98078 CB1 CHO cells HUMAN 3H-CP-55940 Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate 4 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98334 D3 CLONED HUMAN [3H]-N-methylspiperone 5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 447 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98590 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione >10000 Ofon E et al 2016a Jan 15, 2025 Jan 28, 2025
33310 Alpha1A CLONED HUMAN 3H-PRAZOSIN Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98846 NET CLONED HUMAN 3H-Nisoxetine 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
33566 5-HT7 CLONED HUMAN 3H-LSD CELECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99102 D3 CLONED HUMAN 3H-N-Methylspiperone (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99358 D3 CLONED HUMAN [3H]N-methylspiperone 6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline 1.35 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34078 P2X2, P2X3 CLONED HUMAN 3H-A-317491 A-317491 0.9 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99614 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2-oxo-ethoxy}-phenyl]-xanthine 3.51 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
100126 D1 CLONED HUMAN 3H-SCH23390 Quetiapine 381 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
34846 CB2 CLONED HUMAN 3H-CP-55940 PhAR 300 Jan 15, 2025 Jan 15, 2025
100382 NET CLONED HUMAN 3H-Nisoxetine Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
35358 D4 CLONED HUMAN 3H-SPIROPERIDOL 5-methyl-10-(4-methylpiperazino)-5H-dibenzo[a,d]cycloheptene 12 Phillips ST, et. al., 1995 Jan 15, 2025 Jan 15, 2025
100894 BchE serum HUMAN Functional N-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide 21.4 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 15, 2025
101150 5-HT7 CLONED HUMAN 3H-5-HT 1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone 197 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
35870 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 12 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101406 D2 CLONED HUMAN 3H-RACLOPRIDE 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 27 Zareba P, et al., 2019 Jan 15, 2025 Jan 28, 2025
36126 COX-2 purified HUMAN Functional Indomethacin 600 Riendeau D, et.al., 2001 Jan 15, 2025 Jan 15, 2025
101662 Alpha2B CLONED HUMAN [3H]-rauwolscine Perospirone 202 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
36382 CLONED HUMAN 3H-SQ 29548 BM 573 1.1 Hanson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
101918 BZP CLONED HUMAN [3H] Flunitrazepam Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36638 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL 5454 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102174 Sigma 1 CLONED HUMAN [3H]Pentazocine NEMONAPRIDE 7 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37918 CDK1 CLONED HUMAN Functional 4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 6 Lin R, et al., 2005 Jan 15, 2025 Jan 15, 2025
38430 D3 CLONED HUMAN 3H-NEMONAPRIDE MCL-211 356 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
38686 UNDEFINED HUMAN 3H-hypoxanthine Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(3-bromo-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcarbamoyl}-2-methyl-propyl)-amide 32 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39198 MC4 CLONED HUMAN 125I-NDP-MSH Gamma1-MSH 589 Nickolls SA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39710 5-HT2C CLONED HUMAN 3H-5HT MK 212 97.7237 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40478 STAT3 CLONED HUMAN Functional Ac-pTyr-Ile-Pro-Gln-Thr-NH2 1070 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40734 mGluR5 CLONED HUMAN Functional 9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one 2100 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41246 CLONED HUMAN 125I-Chemokine 4-(4-Chlorophenyl)-1-(4-phenyl-4-p-tolylbutyl)piperidin-4-ol Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
42014 M2 CLONED HUMAN 3H-QNB FLUOXETINE 2700 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42270 CLONED HUMAN 125I-Motilin Delta 33-36 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42526 CLONED HUMAN Functional [ala4,leu13]pMOT(1-14) 2570.4 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42782 Y2 CLONED HUMAN 125I-PYY L-152,804 >10000 Kakui N, et al., 2006 Jan 15, 2025 Jan 15, 2025
43038 MAPK9 CLONED HUMAN 3H-Staurosporine SB202190 120 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43294 DAPK3 CLONED HUMAN 3H-Staurosporine EKB-569 4100 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43550 PAK7 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43806 CaMK CLONED HUMAN 3H-Staurosporine BIRB-796 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44062 CaMK CLONED HUMAN 3H-Staurosporine Tarceva >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44318 MAPK9 CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44574 PAK1 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44830 CSNK1E CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45086 MAPK P38 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45598 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
46110 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47646 GABAA CLONED HUMAN 3H-RO-15-1788 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47902 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 21 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48670 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49694 D1 CLONED HUMAN 3H-SCH23390 Pramipexole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
51486 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide 1 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51742 AR UNDEFINED HUMAN UNDEFINED (Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline 110 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51998 DOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 6.53 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52254 A2B UNDEFINED HUMAN UNDEFINED 9-(2-(4-chlorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione >10000 Drabczyńska A et al., 2007 Jan 15, 2025 Jan 15, 2025
52510 Alpha2B UNDEFINED HUMAN UNDEFINED 6,7-dimethoxy-2-((7-methoxy-2-phenylbenzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 752 Hagihara K et al., 2007 Jan 15, 2025 Jan 15, 2025
52766 D2 UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide 22 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
53022 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan 0.21 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
53534 SLC6A2 UNDEFINED HUMAN UNDEFINED (+)-1-[(1R)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 187 Mahaney PE et al., 2008 Jan 15, 2025 Jan 15, 2025
53790 5-HT2A UNDEFINED HUMAN UNDEFINED HALOPERIDOL 120 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54558 A1 UNDEFINED HUMAN UNDEFINED 8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione >10000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54814 D3 UNDEFINED HUMAN UNDEFINED N-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide 140 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55070 D2 UNDEFINED HUMAN UNDEFINED N-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide 9.2 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55326 KOR UNDEFINED HUMAN UNDEFINED 8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 506 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55582 DOR UNDEFINED HUMAN UNDEFINED N-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone 180 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
56094 MOR UNDEFINED HUMAN UNDEFINED (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide 2.5 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
56606 NR3C1 UNDEFINED HUMAN UNDEFINED Benzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol 36 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
56862 SLC6A4 UNDEFINED HUMAN UNDEFINED (3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one 7 Rotella DP et al., 2009 Jan 15, 2025 Jan 15, 2025
57630 SST3 UNDEFINED HUMAN UNDEFINED N-(1-(3-ethoxy-4-(trifluoromethyl)benzyl)piperidin-4-yl)benzo[d]oxazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57886 SLC6A2 UNDEFINED HUMAN UNDEFINED DESIPRAMINE 3.4 O'Neill DJ et al., 2010 Jan 15, 2025 Jan 15, 2025
58142 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 28.2 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58398 D2 CLONED HUMAN 3H-N-Methylspiporone MRS5678 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58654 M1 CLONED HUMAN 3H-QNB Cyclobenzaprine 25 Gregori-Puigjane E, et al., 2012 Jan 15, 2025 Jan 15, 2025
58910 D2 CLONED HUMAN 3H-N-Methylspiporone (+)-SYA 09 51.1 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
59422 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide 160 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59678 5-HT1B CLONED HUMAN 3H-5CT MH.MZ 1846 Herth, M. et. al., 2009 Jan 15, 2025 Jan 15, 2025
60190 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-(Furan-2-ylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 0.62 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60446 GABAA CLONED HUMAN FNZ XLI-286 0.118 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60702 GABAA CLONED HUMAN FNZ TJH-IV-51 >10000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60958 GABAA CLONED HUMAN FNZ YT-II 6.932 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61214 GABAA CLONED HUMAN FNZ ZG-224 33.7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61470 GABAA CLONED HUMAN FNZ RY-047 124 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61726 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine 194 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
62238 Alpha1A CLONED HUMAN 3H-PRAZOSIN Tianeptine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
62750 H1 Brain Frontal Cortex HUMAN 3H-doxepin Trimipramine 0.27 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 28, 2025
63006 5-HT2B CLONED HUMAN 3H-5-HT Fenfluramine (+) 5099 Rothman RB, et al., 2003 Jan 15, 2025 Jan 15, 2025
63518 NET CLONED HUMAN 3H-Nisoxetine 2-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
63774 CXCR3 PHA/IL-2 T cells HUMAN 125I-CXCL11 CXCL11 0.05 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
64542 CLONED HUMAN 3H-Estradiol 17beta-Estradiol 2100 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
64798 Beta1 CLONED HUMAN 125I-ICYP Formoterol 6.12 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
65054 H1 FR. CORTEX HUMAN 3H-MEPYRAMINE IPRINDOLE 670 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
65310 GABAA CLONED HUMAN [3H] Flunitrazepam SHU-1-19 12 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65567 GABAA CLONED HUMAN [3H] Flunitrazepam Alprazolam >10000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65823 GABAA CLONED HUMAN [3H] Flunitrazepam YT-5 0.421 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66079 NET CLONED HUMAN 3H-Nisoxetine Mellpaladine B 1259 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
66847 M2 CLONED HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67103 DAT CLONED HUMAN 3H-WIN35428 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67359 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 425 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67615 A2A KIDNEY HUMAN 3H-2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine Ethyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate 1570 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67871 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 91 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
2847 5-HT2A CORTEX HUMAN 3H-KETANSERIN KETANSERIN 0.56 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
68383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68639 recombinant HUMAN UNKNOWN N-[(Naphth-2-yl)methyl]-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
3359 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68895 SST3 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH2 0.630957 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69151 H4 CLONED HUMAN 3H-N-alpha-methylhistamine Alpha-Methylhistamine-S 3981.07 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3871 D1 CLONED HUMAN 3H-SCH23390 OLANZAPINE 35 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69663 BZP CLONED HUMAN FNZ 4-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
69919 SLC6A3 CLONED HUMAN 3H-WIN35428 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
4639 SLC6A3 CLONED HUMAN 3H-WIN 35,428 BINDING KETANSERIN >10000 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4895 5-HT2A CLONED HUMAN 125I-DOI LY 320950 248 BRYANT HU, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
70431 5-HT2B CLONED HUMAN 3H-LSD MRP3215 6.6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5151 5-HT2C CLONED HUMAN 125I-DOI DOHx 0.7 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70687 KOR CLONED HUMAN 3H-Diprenorphine NALOXONE 270 Olson KM, et al., 2019 Jan 15, 2025 Jan 28, 2025
70943 KOR CLONED HUMAN 3H-U69593 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
71199 5-HT1A CLONED HUMAN WAY100635 FEMPT 0.2 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
5919 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE PHENTOLAMINE 6.8 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
6175 Beta1 CLONED HUMAN 125I-CYP SB204070 1000 WARDLE KA, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
6687 D4 CLONED HUMAN 3H-NEMONAPRIDE RISPERIDONE 45 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
7199 NK2 CLONED HUMAN 125I-[MePhe7]-NKB Senktide >10000 Sarau HM, et al., 1997 Jan 15, 2025 Jan 15, 2025
72735 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
72991 M4 CLONED HUMAN 3H-QNB catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7711 GABAA CLONED HUMAN 3H-MUSCIMOL Bicuculline >10000 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7967 GABAA CLONED HUMAN 3H-RO-15-1788 30 7000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8223 SST1 CLONED HUMAN 125I-LTT-SRIF28 octreotide 223.87 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8479 SST3 CLONED HUMAN 125I-LTT-SRIF28 RC 160 42.65 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8735 SST2 CLONED HUMAN 125I-LTT-SRIF28 cycloantagonist SA 3981.07 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8991 SST3 CLONED HUMAN 125I-SRIF-28 SA 398.1 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74527 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74783 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75039 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9759 MT1 CLONED HUMAN 125I-Iodomelatonin Luzindole,5-Methoxy 32.7 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75295 D1 CLONED HUMAN 3H-SCH23390 Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
10015 NET CLONED HUMAN 3H-Norepinephrine COCAINE 217 Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999 Jan 15, 2025 Jan 15, 2025
75551 M3 CLONED HUMAN 3H-QNB propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75807 NOP CLONED HUMAN 3H-Nociceptin 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
76063 5-HT5A CLONED HUMAN 3H-LSD Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76319 Beta 2 CLONED HUMAN 3H-CGP12177 (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11039 H1 CLONED HUMAN 3H-MEPYRAMINE RANITIDINE >10000 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
76575 M1 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76831 M4 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11551 H1 BRAIN HUMAN 3H-PYRILAMINE TRAZODONE 1100 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
77087 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
11807 FR. CORTEX HUMAN 3H-RAUWOLSCINE d-Butaclamol 310 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77343 MOR CLONED HUMAN 3H-DAMGO (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77599 5-HT1E CLONED HUMAN 3H-5-HT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77855 5-HT3 CLONED HUMAN 3H-GR-65630 (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78111 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78367 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78623 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78879 5-HT1A CLONED HUMAN 3H-WAY100635 N,N-Dipropyltryptamine 31.8 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
13599 OT Myometrium HUMAN 3H-Oxytocin L-366,682 9.4 Pettibone DJ, et al., 1991 Jan 15, 2025 Jan 15, 2025
79135 5-HT6 CLONED HUMAN 3H-LSD 4-Ethylthio-2,5-dimethoxyphenylbutylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79391 Alpha1B CLONED HUMAN 3H-PRAZOSIN R,R-2b >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79647 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-Bromo-2,5-dimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79903 H1 CLONED HUMAN 3H-PYRILAMINE (±)-3,4-Methylenedioxymethamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
80159 CLONED HUMAN 3H-VASOPRESSIN 3,4,5-Trimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80415 5-HT7 CLONED HUMAN 3H-LSD (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80671 5-HT1E CLONED HUMAN 3H-5-HT (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15391 5-HT1B CLONED HUMAN 3H-5HT Propanolol,(+/-) 2691.53 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80927 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine >10000 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
81183 Alpha1B CLONED HUMAN 3H-PRAZOSIN N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81439 5-HT2A CLONED HUMAN 3H-KETANSERIN N-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 15, 2025
81695 CLONED HUMAN 3H-Nitrendipine (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 15, 2025
81951 5-HT2B CLONED HUMAN 3H-LSD [18F]MH.MZ 299 Herth MM et al 2009 Jan 15, 2025 Jan 15, 2025
16671 M3 CLONED HUMAN 3H-QNB PIRENZEPINE 150 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82207 D4 CLONED HUMAN 3H-N-Methylspiperone 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one 925 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82463 D1 CLONED HUMAN 3H-SCH23390 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine 1353 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82719 5-HT6 CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82975 A2B CHO cells HUMAN 3H-PSB-603 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
17695 PANC1 HUMAN 125I-VIP VIP [D-Met17] 29.5 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83231 5-HT2A CLONED HUMAN 3H-KETANSERIN KETANSERIN 0.77 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83487 5-HT2A HEK293 cells HUMAN 3H-KETANSERIN MDMA 7800 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83743 5-HT1D CLONED HUMAN 3H-5-CT (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 3230 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
18463 5-HT1B CLONED HUMAN 3H-5HT 1-NP 10.1 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
83999 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 180 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18975 CCK2 CLONED HUMAN 125I-BH-CCK-8 42 724.436 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
84511 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(2,6-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19231 NB-OK-1 HUMAN 125-[AcHis1]Pacap PACAP(6-38) 1.5 Vandermeers A et al., 1992 Jan 15, 2025 Jan 15, 2025
84767 DOR CLONED HUMAN 3H-DADLE ±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85023 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19743 D2 CLONED HUMAN 3H-Olanzapine OLANZAPINE 3 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
85279 H3 recombinant HUMAN 3H-NAMH Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 28, 2025
85791 D2 CLONED HUMAN 3H-N-Methylspiperone N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide 2300 Fiorino F et al 2017 Jan 15, 2025 Jan 28, 2025
86047 MOR CLONED HUMAN 3H-DAMGO (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86303 A2A CLONED HUMAN 3H-MSX-2 3-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1780 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
86559 A3 CLONED HUMAN 3H-PSB-11 1-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione >10000 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87327 Alpha1A placeholder HUMAN Placeholder Phenylephrine,(+/-) 55.99 Rak A et al 2016 Jan 15, 2025 Jan 28, 2025
88095 A1 CLONED HUMAN 3H-CCPA compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
23071 MOR CLONED HUMAN 3H-Diprenorphine L-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88607 D1 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 120 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88863 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23583 NPFF2 CLONED HUMAN 125I-1DMe-Y8Fa PrRP24-31 32 Engstrom M, et al., 2003 Jan 15, 2025 Jan 15, 2025
89119 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23839 CRF1 CLONED HUMAN 3H-SN003 DMP696 1.8 Zhang, GE. et al., 2003 Jan 15, 2025 Jan 15, 2025
89375 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 1836 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24095 5-HT2A CLONED HUMAN 3H-SPIPERONE LOXAPINE 2.5 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89631 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0147911 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
24351 CORTEX HUMAN 3H-PRAZOSIN SERTRALINE 188 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
24607 M2 CLONED HUMAN UNDEFINED SR 144528 >10000 Rinaldi-Carmona, M et al., 1998 Jan 15, 2025 Jan 15, 2025
90143 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 870 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24863 H1 CLONED HUMAN 3H-PYRILAMINE CLOZAPINE 2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90399 A2B CLONED HUMAN 3H-PSB-603 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 215 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
25119 EP3 CLONED HUMAN 3H-PGE2 Quetiapine >10000 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90655 A2B CLONED HUMAN 3H-PSB-603 N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide 547 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25375 D2 CLONED HUMAN 3H-NMSP ARIPIPRAZOLE 0.95 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90911 Alpha1B CHO cells HUMAN 3H-PRAZOSIN 8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 69.1831 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
25631 H2 CLONED HUMAN 3H-TIOTIDINE COCAINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91167 A2A CLONED HUMAN 3H-CGS21680 N-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide >10000 Kolb P et al 2012 Jan 15, 2025 Jan 15, 2025
91423 5-HT2A CLONED HUMAN 125I-DOI 4-((6bR,10aS)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone 0.94 Li P et al 2014 Jan 15, 2025 Jan 15, 2025
26143 MOR CLONED HUMAN 3H-Diprenorphine Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91935 A1 CLONED HUMAN 3H-DPCPX (2-Amino-5-(2,5-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92191 D2 CLONED HUMAN 3H-RACLOPRIDE 3-Chloro-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide 66 Zajdel P et al 2012 Jan 15, 2025 Jan 28, 2025
92703 5-HT1D CLONED HUMAN 3H-Cimetidine 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27423 5-HT1D CLONED HUMAN 3H-GR-125743 Cabergoline 8.70964 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92959 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 268 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
28191 nAChR7 CLONED HUMAN 3H-Epibatidine METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93727 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 23.4 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28447 CLONED HUMAN 3H-Quisqualate DCG-IV >10000 Mutel V, et.al., 2000 Jan 15, 2025 Jan 15, 2025
93983 D3 CLONED HUMAN 3H-SPIPERONE compound 42 1.7 Ortega R et al 2011 Jan 15, 2025 Jan 28, 2025
28703 Alpha1A CLONED HUMAN 3H-PRAZOSIN ARIPIPRAZOLE 25.7 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94239 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,5-dimethoxy-4-methallyloxyamphetamine 290 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29215 SST3 CLONED HUMAN UNDEFINED L-779,976 729 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94751 5-HT2C CLONED HUMAN 3H-MESULERGINE 4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
29727 D2 CLONED HUMAN 3H-SPIPERONE GMC1-169 140 Liao Y, et.al., 1999 Jan 15, 2025 Jan 15, 2025
95519 5-HT6 CLONED HUMAN [3H]-LSD 7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione 8987 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
95775 Alpha1D CLONED HUMAN 3H-PRAZOSIN Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
30495 M1 CLONED HUMAN 3H-QNB endo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 6.6 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
96031 MOR CLONED HUMAN 3H-DAMGO 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96287 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
31007 V2 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96543 5-HT1E CLONED HUMAN [3H]5-HT 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
96799 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31519 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 5011.87 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97055 5-HT1B CLONED HUMAN [3H]GR127543 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97311 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 66.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
32031 5-HT6 CLONED HUMAN UNDEFINED RS-127445 1000 Bonhaus, DW et. al., 1999 Jan 15, 2025 Jan 15, 2025
97567 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 43.41 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98079 CB2 CHO cells HUMAN 3H-CP-55940 Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate 710 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
32799 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 1 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
98335 D3 CLONED HUMAN [3H]-N-methylspiperone 5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 91 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98591 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione >10000 Ofon E et al 2016a Jan 15, 2025 Jan 28, 2025
33311 Alpha1B CLONED HUMAN 3H-PRAZOSIN Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98847 SERT CLONED HUMAN 3H-Cimetidine 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33567 D1 CLONED HUMAN 3H-SCH23390 CELECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99103 D4 CLONED HUMAN 3H-N-Methylspiperone (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99359 D3 CLONED HUMAN [3H]N-methylspiperone 1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine 8.32 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34079 P2X2, P2X3 CLONED HUMAN 3H-A-317491 ATP,TNP 14.5 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99615 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine 3.64 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
100127 5-HT1A CLONED HUMAN 3H-WAY100635 Brexpiprazole 1.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
34847 CB2 CLONED HUMAN 3H-CP-55940 PhAR, ent 400 Jan 15, 2025 Jan 15, 2025
100383 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100639 5-HT1A CLONED HUMAN 3H-WAY100635 CYPROHEPTADINE 50 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
35359 D4 CLONED HUMAN 3H-SPIROPERIDOL 5-methyl-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 320 Phillips ST, et. al., 1995 Jan 15, 2025 Jan 15, 2025
100895 AChE BRAIN HUMAN Functional N-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(5-cyano-1H-indol-3-yl)propionamide 0.7 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
101151 5-HT7 CLONED HUMAN 3H-5-HT 1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone 52 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
35871 SLC6A4 CLONED HUMAN 3H-PAROXETINE 7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 1.5 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101407 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 28 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36127 COX-2 purified w/detergent HUMAN Functional Indomethacin 400 Riendeau D, et.al., 2001 Jan 15, 2025 Jan 15, 2025
101663 Alpha2C CLONED HUMAN [3H]rauwolscine Perospirone 98 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
36383 CLONED HUMAN 3H-SQ 29548 BM 613 2.1 Hanson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
101919 PBR CLONED HUMAN [3H]PK11195 Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36639 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 21 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
37919 CDK2 CLONED HUMAN Functional 4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 2 Lin R, et al., 2005 Jan 15, 2025 Jan 15, 2025
38431 D3 CLONED HUMAN 3H-NEMONAPRIDE MCL-212 >10000 Neumeyer JL, et al., 2003a Jan 15, 2025 Jan 15, 2025
38687 UNDEFINED HUMAN 3H-hypoxanthine Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(biphenyl-3-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcarbamoyl}-2-methyl-propyl)-amide 3.9 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39199 MC4 CLONED HUMAN 125I-NDP-MSH desacetyl-alpha-MSH 30.2 Nickolls SA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39455 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-Methylpsilocybin >10000 Sard H, et al., 2005 Jan 15, 2025 Jan 15, 2025
39711 5-HT2C CLONED HUMAN 3H-5HT ORG-12962 14.7911 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40479 STAT3 CLONED HUMAN Functional Ac-pTyr-Phe-Pro-Gln-Thr-NH2 1890 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40735 mGluR5 CLONED HUMAN Functional 9-(2',2',2'-Trifluoroethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 99 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41247 CLONED HUMAN 125I-Chemokine 1-(4-Biphenyl-4-y)-4-(4-chlorophenyl)butyl]-4-(4-chlorophenyl)piperidin-4-ol >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
42015 M2 CLONED HUMAN 3H-QNB IMIPRAMINE 88 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42271 CLONED HUMAN 125I-Motilin Delta 103-104 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42527 CLONED HUMAN Functional [ala5,leu13]pMOT(1-14) 28.8403 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42783 Y2 CLONED HUMAN 125I-PYY PYY 2.1 Kakui N, et al., 2006 Jan 15, 2025 Jan 15, 2025
43039 MAPK9 CLONED HUMAN 3H-Staurosporine SB203580 95 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43295 DAPK3 CLONED HUMAN 3H-Staurosporine SU11248 300 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43551 PCTK1 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43807 CDK2 CLONED HUMAN 3H-Staurosporine BIRB-796 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44063 CaMK CLONED HUMAN 3H-Staurosporine Tarceva >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44319 MAPK10 CLONED HUMAN 3H-Staurosporine EKB-569 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44575 PAK3 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44831 CSNK1G1 CLONED HUMAN 3H-Staurosporine BAY-43-9006 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45087 MAPK12 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45599 NET CLONED HUMAN 3H-Nisoxetine Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
46111 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47391 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide 29 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47647 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.73 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47903 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48671 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49695 D5 CLONED HUMAN 3H-SCH23390 Pramipexole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
51487 Alpha1A UNDEFINED HUMAN UNDEFINED N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide 6.3 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51743 AR UNDEFINED HUMAN UNDEFINED (+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline 1530 Hudson AR et al., 2007 Jan 15, 2025 Jan 15, 2025
51999 DOR UNDEFINED HUMAN UNDEFINED 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7.59 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52255 A2B UNDEFINED HUMAN UNDEFINED 9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 590 Drabczyńska A et al., 2007 Jan 15, 2025 Jan 15, 2025
52511 Alpha2B UNDEFINED HUMAN UNDEFINED 6,7-dimethoxy-2-((7-methoxy-2-(pyridin-2-yl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 330 Hagihara K et al., 2007 Jan 15, 2025 Jan 15, 2025
52767 D2 UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide 67 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
53023 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan 0.21 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
53535 SLC6A2 UNDEFINED HUMAN UNDEFINED 1-[1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 46 Mahaney PE et al., 2008 Jan 15, 2025 Jan 15, 2025
53791 5-HT2A UNDEFINED HUMAN UNDEFINED Quetiapine 220 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54559 A1 UNDEFINED HUMAN UNDEFINED 8-(4-(4-(4-Methoxyphenyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione >10000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54815 D3 UNDEFINED HUMAN UNDEFINED Biphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide 0.2 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55071 D2 UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide 503 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55327 KOR UNDEFINED HUMAN UNDEFINED 8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one 1342 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55583 DOR UNDEFINED HUMAN UNDEFINED 14-O-phenylpropylnaltrexone 0.48 Moynihan H et al., 2009 Jan 15, 2025 Jan 15, 2025
56095 MOR UNDEFINED HUMAN UNDEFINED (1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide 0.16 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
56607 NR3C1 UNDEFINED HUMAN UNDEFINED (4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol 25 Xiao HY et al., 2010 Jan 15, 2025 Jan 15, 2025
56863 SLC6A4 UNDEFINED HUMAN UNDEFINED (3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one 1 Rotella DP et al., 2009 Jan 15, 2025 Jan 15, 2025
57631 SST3 UNDEFINED HUMAN UNDEFINED N-(1-(4-cyclopropoxy-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57887 SLC6A2 UNDEFINED HUMAN UNDEFINED DESIPRAMINE 2.1 O'Neill DJ et al., 2010 Jan 15, 2025 Jan 15, 2025
58143 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 47.9 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58399 D2 CLONED HUMAN 3H-N-Methylspiporone MRS5697 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58655 M2 CLONED HUMAN 3H-QNB Cyclobenzaprine 60 Gregori-Puigjane E, et al., 2012 Jan 15, 2025 Jan 15, 2025
58911 D3 CLONED HUMAN 3H-N-Methylspiporone (+)-SYA 09 1069 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
59423 5-HT1A CLONED HUMAN 3H-WAY100635 Desmethyldesipramine >10000 Deupree, J. et. al., 2007 Jan 15, 2025 Jan 15, 2025
59679 5-HT1E CLONED HUMAN 3H-5HT MH.MZ >10000 Herth, M. et. al., 2009 Jan 15, 2025 Jan 15, 2025
60191 A3 CLONED HUMAN [125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide (1S,2R,3S,4R,5S)-4-(2-((4,5-Dimethylfuran-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide 1.45 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60447 GABAA CLONED HUMAN FNZ XLI-286 0.064 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60703 GABAA CLONED HUMAN FNZ TJH-IV-51 316 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60959 GABAA CLONED HUMAN FNZ SVO-8-67 7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61215 GABAA CLONED HUMAN FNZ ZG-224 50 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61471 GABAA CLONED HUMAN FNZ RY-047 79 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61727 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine 103 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
61983 CLONED HUMAN UNDEFINED grepafloxacin >10000 Bischoff ,U et al., 2000 Jan 15, 2025 Jan 15, 2025
62239 Alpha1B CLONED HUMAN 3H-PRAZOSIN Tianeptine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
62751 H1 Brain Frontal Cortex HUMAN 3H-doxepin MIANSERIN 0.4 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 28, 2025
63007 5-HT2B CLONED HUMAN 3H-5-HT Fenfluramine (-) 5713 Rothman RB, et al., 2003 Jan 15, 2025 Jan 15, 2025
63519 NET CLONED HUMAN 3H-Nisoxetine 2-Cl-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
63775 CXCR3 PHA/IL-2 T cells HUMAN 125I-CXCL11 NBI-74330 15.8 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
64543 CLONED HUMAN 3H-Estradiol 4-hydroxytamoxifen 100 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
64799 Beta1 CLONED HUMAN 125I-ICYP Salmeterol 6.11 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
65311 GABAA CLONED HUMAN [3H] Flunitrazepam SHU-1-19 7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65568 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-082 1.7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65824 GABAA CLONED HUMAN [3H] Flunitrazepam YT-5 0.6034 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66080 H1 CLONED HUMAN 3H-PYRILAMINE Terfenadine 58 Pearlstein, Robert. et, al. 2003 Jan 15, 2025 Jan 28, 2025
66848 M3 CLONED HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67104 H1 CLONED HUMAN 3H-PYRILAMINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67360 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 222 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
2080 5-HT1D CAUDATE HUMAN 3H-5HT SDZ 21-009 646 WAEBER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
67616 A3 KIDNEY HUMAN I-125-N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamide Ethyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate 236 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67872 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 1150 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68384 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68640 recombinant HUMAN UNKNOWN N-Benzyl-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
3360 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDL 72222 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68896 SST4 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH2 0.630957 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69152 H4 CLONED HUMAN 3H-N-alpha-methylhistamine homohistamine 31.6228 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
3872 D1 CLONED HUMAN 3H-SCH23390 Quetiapine 1277 KONGSAMUT S, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69664 BZP CLONED HUMAN FNZ 2-CI-DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
69920 SLC6A3 CLONED HUMAN 3H-WIN35428 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
4640 SLC6A3 CLONED HUMAN 3H-WIN 35,428 BINDING BUDIPINE >10000 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4896 5-HT2A CLONED HUMAN 125I-DOI LY 320951 839 BRYANT HU, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
70432 5-HT1A CLONED HUMAN 3H-WAY100635 MRP3215 6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5152 5-HT2C CLONED HUMAN 125I-DOI DOTB 2.2 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70688 KOR CLONED HUMAN 3H-Diprenorphine BUPRENORPHINE 27 Olson KM, et al., 2019 Jan 15, 2025 Jan 28, 2025
70944 KOR CLONED HUMAN 3H-U69593 (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
71200 5-HT1B CLONED HUMAN 3H-5-CT FEMPT 122.5 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
5920 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE SPIROXATRINE 0.19 BYLUND DB, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
6176 Beta2 CLONED HUMAN 125I-CYP SB204070 1000 WARDLE KA, ET AL., 1994 Jan 15, 2025 Jan 28, 2025
6688 D2 CLONED HUMAN 3H-NEMONAPRIDE Quetiapine 1000 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
7200 NK2 CLONED HUMAN 125I-[MePhe7]-NKB SB 223412 144 Sarau HM, et al., 1997 Jan 15, 2025 Jan 15, 2025
72736 Sigma 2 CLONED HUMAN 3H-Pentazocine(+) naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
72992 M5 CLONED HUMAN 3H-QNB catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7712 GABAA CLONED HUMAN 3H-MUSCIMOL Thio-4-PIOL 1778.27 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7968 GABAA CLONED HUMAN 3H-RO-15-1788 31 7000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8224 SST1 CLONED HUMAN 125I-LTT-SRIF28 octreotide-Tyr3 2691.53 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8480 SST3 CLONED HUMAN 125I-LTT-SRIF28 BIM 23030 67.6 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8736 SST2 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.09 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8992 SST3 CLONED HUMAN 125I-SRIF-28 SMS 201-995 5.01 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74528 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74784 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75040 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9760 MT1 CLONED HUMAN 125I-Iodomelatonin GR 128107 90.4 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75296 D5 CLONED HUMAN 3H-SCH23390 Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75552 M4 CLONED HUMAN 3H-QNB propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76064 5-HT6 CLONED HUMAN 3H-LSD Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11040 H1 CLONED HUMAN 3H-MEPYRAMINE Thioperamide >10000 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
76576 M2 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76832 M5 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11552 H1 BRAIN HUMAN 3H-PYRILAMINE Venlafaxine >10000 Cusack, B et al., 1993 Jan 15, 2025 Jan 15, 2025
77088 Sigma 2 CLONED HUMAN 3H-DTG (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
11808 FR. CORTEX HUMAN 3H-RAUWOLSCINE PERPHENAZINE 510 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77344 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77600 5-HT2A CLONED HUMAN 3H-KETANSERIN (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77856 5-HT5A CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78112 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12832 Beta1 CLONED HUMAN 125I-ICYP TMQ, Racemic 10.47 Fraundorfer PF, et al., 1994 Jan 15, 2025 Jan 15, 2025
78368 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78624 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78880 5-HT1A CLONED HUMAN 3H-WAY100635 4-Ethylthio-2,5-dimethoxyphenylbutylamine 5339 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
13600 OT Myometrium HUMAN 3H-Oxytocin L-366,706 21 Pettibone DJ, et al., 1991 Jan 15, 2025 Jan 15, 2025
79136 5-HT6 CLONED HUMAN 3H-LSD 6-Fluoro-N,N-dimethyltryptamine 25.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79392 Alpha1B CLONED HUMAN 3H-PRAZOSIN S,S-2c >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
79648 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) DMT 5209 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79904 H1 CLONED HUMAN 3H-PYRILAMINE 3,4,5-Trimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
80160 CLONED HUMAN 3H-VASOPRESSIN 4-Bromo-2,5-dimethoxyphenethylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80416 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80672 5-HT2A CLONED HUMAN 3H-KETANSERIN (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15392 5-HT1B CLONED HUMAN 3H-5HT 5-CT 0.89 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
80928 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine >10000 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
81184 Alpha1D CLONED HUMAN 3H-PRAZOSIN N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81440 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-phenyl-4-[[4-(1,3-thiazol-2-yl)-1,4-diazepan-1-yl]methyl]-1,3-oxazole 3324 Weiss DR et al 2018 Jan 15, 2025 Jan 15, 2025
81696 DOR CLONED HUMAN 3H-DADLE (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
81952 5-HT2C CLONED HUMAN 3H-MESULERGINE [18F]MH.MZ 71 Herth MM et al 2009 Jan 15, 2025 Jan 15, 2025
16672 M3 CLONED HUMAN 3H-QNB Diphenhydramine 229 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
82208 5-HT1B CLONED HUMAN 3H-5-CT 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one 27 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82464 D5 CLONED HUMAN 3H-SCH23390 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
17184 5-HT3 CLONED HUMAN 3H-ZACOPRIDE METHYLPHENIDATE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
82720 5-HT7 CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82976 A3 CHO cells HUMAN 3H-PSB-11 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
17696 PANC1 HUMAN 125I-VIP VIP [D-Ala18] 15.4 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83232 5-HT2A CLONED HUMAN 3H-KETANSERIN DMT 175 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83488 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83744 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 561 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18464 5-HT1B CLONED HUMAN 3H-5HT 7-methoxy-1-naphthylpiperazine 2 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
84000 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-allyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84256 DOR CLONED HUMAN 3H-DADLE 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18976 CCK2 CLONED HUMAN 125I-BH-CCK-8 24 3630.78 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
84512 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(2,6-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19232 NB-OK-1 HUMAN 125-[AcHis1]Pacap PACAP(5-38) 5 Vandermeers A et al., 1992 Jan 15, 2025 Jan 15, 2025
84768 KOR CLONED HUMAN 3H-U69593 ±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025