The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

If you desire to download the entire Ki database, you can do so by selecting the "Download Ki Database button below this message.

Showing 7,001-8,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
71452H1CLONEDHUMAN3H-PYRILAMINE4-acetoxy-N,N-diallyltryptamine353Klein LM et al 2018Jan 15, 2025Jan 28, 2025
6172D3CLONEDHUMAN125I-IODOSULPRIDESB2040701000WARDLE KA, ET AL., 1994Jan 15, 2025Jan 15, 2025
7196NK2CLONEDHUMAN125I-[MePhe7]-NKBNKA0.74Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72732MORCLONEDHUMAN3H-DAMGOnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
72988M1CLONEDHUMAN3H-QNBcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7708GABAACLONEDHUMAN3H-MUSCIMOLBicuculline4466.83Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7964GABAACLONEDHUMAN3H-RO-15-178827740He X, et al., 1999Jan 15, 2025Jan 27, 2025
8220SST1CLONEDHUMAN125I-LTT-SRIF28CST14-Tyr102.75Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8476SST3CLONEDHUMAN125I-LTT-SRIF28octreotide-Tyr3144.54Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8732SST2CLONEDHUMAN125I-LTT-SRIF28cortistatin141.77Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8988SST3CLONEDHUMAN125I-SRIF-28CGP 239960.39Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
9500MT2CLONEDHUMAN125I-IodomelatoninMelatonin,2-Chloro0.22Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
750365-HT5ACLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75292Beta3CLONEDHUMAN125I-PindololEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10012NETCLONEDHUMAN3H-NorepinephrineNisoxetine Inhibitor4.21Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
75804Sigma 2CLONEDHUMAN3H-DTG1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
760605-HT2BCLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76316Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
11036H1CLONEDHUMAN3H-MEPYRAMINECetirizine6.3Moguilevsky N et al, 1994Jan 15, 2025Jan 15, 2025
76572KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol1120Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76828M1CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11548H1BRAINHUMAN3H-PYRILAMINENORTRYPTYLINE6.3Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
77084M5CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11804FR. CORTEXHUMAN3H-PRAZOSINPHENTOLAMINE15Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77340Sigma 2CLONEDHUMAN3H-DTG(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
775965-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
778525-HT2ACLONEDHUMAN3H-KETANSERIN(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
781085-HT5ACLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78364Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78620Beta 1CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788765-HT1ACLONEDHUMAN3H-WAY1006355-Methoxy-N-methyl-N-isopropyltryptamine12.3Ray TS 2010 Jan 15, 2025Jan 15, 2025
791325-HT6CLONEDHUMAN3H-LSDN,N-Diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79388Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-2,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
79644CLONEDHUMAN3H-CLONIDINE(±)-2,5-Dimethoxy-4-ethylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79900M5CLONEDHUMAN3H-QNBEMDT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80156V2CLONEDHUMAN3H-VASOPRESSIN5-MeO-TMT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
804125-HT4CLONEDHUMAN3H-GR113808(E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806685-HT1ACLONEDHUMAN3H-8-OH-DPAT(5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153885-HT1BCLONEDHUMAN3H-5HTRAUWOLSCINE46.77BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809245-HT2BCLONEDHUMAN3H-LSD3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine56.2341Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
81180KORCLONEDHUMAN3H-U69593N-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
81436H1CLONEDHUMAN3H-PYRILAMINE2-[4-[(2R)-2-(3,4-dimethylphenyl)-2-hydroxyethyl]piperazin-1-yl]pyridine-3-carbonitrile2103Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
81692Beta1CLONEDHUMAN125I-iodo-pindolol(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
819485-HT1BCLONEDHUMAN3H-5CT[18F]MH.MZ1846Herth MM et al 2009Jan 15, 2025Jan 15, 2025
16668M3CLONEDHUMAN3H-QNBSCOPOLAMINE0.44Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82204D5CLONEDHUMAN3H-SCH233902-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82460Alpha1ACLONEDHUMAN3H-PRAZOSIN(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine2720Besnard J et al 2012Jan 15, 2025Jan 28, 2025
171805-HT1ECLONEDHUMAN3H-5HTMETHYLPHENIDATE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
827165-HT3CLONEDHUMAN3H-GR65630(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17692CLONEDHUMAN125I-VIPVIP [D-Gln16]1.1Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832285-HT2ACLONEDHUMAN125I-DOIKETANSERIN4.1Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83484DATHEK293 cellsHUMAN3H-WIN 35,428MDMA6500Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
83740DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one4693PDSP Certified DataJan 15, 2025Jan 28, 2025
83996KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84252MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
18972H1CLONEDHUMAN3H-MEPYRAMINEMEPYRAMINE1.18Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84508MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19228NB-OK-1HUMAN125-[AcHis1]PacapPACAP(9-38)50Vandermeers A et al., 1992Jan 15, 2025Jan 15, 2025
84764DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85020DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19740D2CLONEDHUMANUNDEFINEDMOLINDONE6Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
85276H1recombinantHUMAN3H-PYRILAMINETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
86044H3CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
87324Alpha1BplaceholderHUMANPlaceholderTamsulosin0.13Rak A et al 2016Jan 15, 2025Jan 28, 2025
87580M5CLONEDHUMAN3H-QNB2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87836A3testHUMAN3H-PSB-118-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
22556hERGCLONEDHUMAN3H-MethylspiperoneSERTINDOLE3Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88092A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
23068MORCLONEDHUMAN3H-DiprenorphineL-homocysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88604M1CLONEDHUMAN3H-QNBHALOPERIDOL1600Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88860A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide23.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23580NPFF2CLONEDHUMAN125I-1DMe-Y8FaRFRP-115Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
89116A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide40.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893725-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide2630Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240925-HT2ACLONEDHUMAN3H-SPIPERONECLOZAPINE5.2Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89628D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
24348CORTEXHUMAN3H-PRAZOSINFluoxetine-R-(-)1528Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89884nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
24604ETBCLONEDHUMANUNDEFINEDSR 144528>10000Rinaldi-Carmona, M et al., 1998Jan 15, 2025Jan 15, 2025
90140D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24860SLC6A4CLONEDHUMAN3H-CITALOPRAMCLOZAPINE1624PDSP Certified DataJan 15, 2025Jan 15, 2025
90396A2BCLONEDHUMAN3H-PSB-603N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25116CCR5CLONEDHUMAN3H-EpibatidineQuetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90652A2BCLONEDHUMAN3H-PSB-603N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25372H4CLONEDHUMAN3H-HistamineARIPIPRAZOLE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
90908Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane10.7152Franchini S et al 2014Jan 15, 2025Jan 28, 2025
91164A2ACLONEDHUMAN3H-CGS-216802-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25884H1CLONEDHUMAN3H-PYRILAMINEPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91420CB1CLONEDHUMAN3H-CP55940O-6659109Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26140KORCLONEDHUMAN3H-DiprenorphinePseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91932A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-(4-fluorophenyl) thiophen-3-yl)(4-chlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
92188D2CLONEDHUMAN3H-RACLOPRIDE4-Fluoro-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide50Zajdel P et al 2012Jan 15, 2025Jan 28, 2025
271645-HT1DCORTEXHUMAN3H-5CT1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride1900May JA, et al., 2003Jan 15, 2025Jan 15, 2025
927005-HT1DCLONEDHUMAN3H-Cimetidine9,13-epoxylabd-5-ene-7 b,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274205-HT1DCLONEDHUMAN3H-GR-125743APOMORPHINE1230.27Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929565-HT6CLONEDHUMAN3H-LSDOLANZAPINE7Sudol S et al 2020Jan 15, 2025Jan 15, 2025
93724A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester3.19Federico S et al 2018Jan 15, 2025Jan 15, 2025
28444mGluR5CLONEDHUMAN3H-Quisqualate(S)-4CPG>10000Mutel V, et.al., 2000Jan 15, 2025Jan 28, 2025
93980D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one13Ortega R et al 2011Jan 15, 2025Jan 29, 2025
28700PKCαCLONEDHUMAN3H-PDBUARIPIPRAZOLE>10000Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942365-HT2CCLONEDHUMAN3H-MESULERGINE4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine4200Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29212SST3CLONEDHUMANUNDEFINEDBIM 2319726.8Patel YC, 1999Jan 15, 2025Jan 15, 2025
947485-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95004D4CLONEDHUMAN3H-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
955165-HT6CLONEDHUMAN[3H]-LSD7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride68Partyka A et al 2015Jan 15, 2025Jan 15, 2025
95772Alpha1DCLONEDHUMAN3H-PRAZOSINTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
30492M3CLONEDHUMAN3H-QNBexo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene0.84Kim MG, et al., 2003Jan 15, 2025Jan 15, 2025
96284Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
965405-HT1ACLONEDHUMAN[3H]-Way1006351-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
312605-HT2AC.H.O.HUMAN3H-KETANSERINRopinirole>10000Millan MJ, et. al., 2004Jan 15, 2025Jan 15, 2025
96796D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA630Mannel B et al 2017Jan 15, 2025Jan 28, 2025
31516D2CLONEDHUMAN125I-IODOSULPRIDE(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)630.957Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97052Sigma 1CLONEDHUMAN[3H]PentazocineFluorolintane (2-F-DPPy)110Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97308MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol47.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
320285-HT2CCLONEDHUMAN3H-MESULERGINERS-127445398.107Bonhaus, DW et. al., 1999Jan 15, 2025Jan 15, 2025
97564A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate402Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98076CB1CHO cellsHUMAN3H-CP-55940CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate0.6Amato G et al 2019Jan 15, 2025Jan 28, 2025
98332D3CLONEDHUMAN[3H]-N-methylspiperone2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline2176Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985885-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride2976Ofon E et al 2016aJan 15, 2025Jan 15, 2025
98844Beta 2CLONEDHUMAN3H-CGP-121771-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
99100D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99356D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2,3-dichlorophenyl)piperazine14Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34076P2X2, P2X3CLONEDHUMAN3H-A-317491AP3A320Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99612A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine1.62Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
100124Sigma 1CLONEDHUMAN3H-Pentazocine(+)Quetiapine413PDSP Certified DataJan 15, 2025Jan 28, 2025
34844CB2CLONEDHUMAN3H-CP-55940Rinvanil>10000Jan 15, 2025Jan 15, 2025
100380SLC6A3CLONEDHUMAN3H-WIN 35,428Etoperidone>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
35356D2CLONEDHUMAN3H-SPIPERONE10-[1,2,3,6-tetrahydro-1(2-propenyl)-4-pyridinyl]-5H-dibenzo[a,d]cycloheptene83Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
100892BchEserumHUMANFunctionalN-(3-{[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-methylamino}propyl)-3-(1H-indol-3-yl)propionamide0.03Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
1011485-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone272Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
35868SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole141Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1014045-HT6CLONEDHUMAN3H-LSD2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione347Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36124EP2CHO (COX-1)cellsHUMANFunctionalIndomethacin18Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36380PlateletsHUMAN3H-SQ 29548BM 5731.3Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
101916M5CLONEDHUMAN[3H]QNBZiprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
366365-HT7CLONEDHUMAN3H-5HTMIANSERIN56Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102172Alpha1DCLONEDHUMAN[3H]prazosinNEMONAPRIDE1802PDSP Certified DataMar 25, 2025Jul 28, 2026
37916CDK1CLONEDHUMANFunctional4-[[3-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-5-yl]amino]-benzenesulfonamide2100Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38428D3CLONEDHUMAN3H-NEMONAPRIDEMCL-205>10000Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
38684UNDEFINEDHUMAN3H-hypoxanthineN-[(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-cyclohexylcarbamoyl-2-hydroxy-propyl]-2,4,6-trifluoro-benzamide3600Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39196MC4CLONEDHUMAN125I-NDP-MSHalpha MSH50.1Nickolls SA, et al., 2005Jan 15, 2025Jan 15, 2025
397085-HT2CCLONEDHUMAN3H-5HTmCPP14.1254Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40476STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln-Thr-NH2739Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40732mGluR5CLONEDHUMANFunctional9-Cyclopropylamino-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41244CLONEDHUMAN125I-ChemokineC28H32NClO5500Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41500CLONEDHUMAN3H-dexamethasonedexamethasone6.7Belvisi MG, et al., 2005Jan 15, 2025Jan 15, 2025
42012M2CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42268CLONEDHUMAN125I-MotilinDelta 30C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42524CLONEDHUMANFunctional[ala1,leu13]pMOT(1-14)588.844Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42780Y1CLONEDHUMAN125I-PYYPYY2Kakui N, et al., 2006Jan 15, 2025Jan 15, 2025
43036MAPK8CLONEDHUMAN3H-StaurosporineGleevec3200Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43292DAPK2CLONEDHUMAN3H-StaurosporineSU11248470Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43548PAK4CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43804CaMKCLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44060CaMKCLONEDHUMAN3H-StaurosporineTarceva>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44316INSRCLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44572NEK9CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44828CLK4CLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45084PKMYT1CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45596NETCLONEDHUMAN3H-NisoxetineIPRINDOLE1262Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
46108Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47132CLONEDHUMAN3H-SUBSTANCE PIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47388D2CLONEDHUMAN3H-SPIPERONEN-(1-Benzylpiperidin-4-yl)-2-naphthamide1000Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47644GABAACLONEDHUMAN3H-RO-15-17883'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile1.5Russell MG, et al., 2006Jan 15, 2025Jan 27, 2025
47900GABAACLONEDHUMAN3H-RO-15-17886,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one66Chambers, MS et al., 2003Jan 15, 2025Jan 27, 2025
48668CLONEDHUMANFunctionalN-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
496925-HT5ACLONEDHUMAN3H-LSDPramipexole>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
50460SLC6A3CLONEDHUMAN3H-WIN 35,428N,N-Dimethyl-5-(4-fluorobutoxy)-2-(2-amino-4-methylphenoxy)benzylamine3604Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
51484Alpha1AUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide0.73Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51740ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline290Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51996DORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine5.38Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
52252A2BUNDEFINEDHUMANUNDEFINED1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione>10000Drabczyńska A et al., 2007Jan 15, 2025Jan 15, 2025
52508Alpha2BUNDEFINEDHUMANUNDEFINED2-((2-(2-fluorophenyl)-7-methoxybenzofuran-4-yl)methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline299Hagihara K et al., 2007Jan 15, 2025Jan 15, 2025
52764D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
53020MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan0.31Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53532SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride18Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
537885-HT1AUNDEFINEDHUMANUNDEFINED4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one90.9Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54556A1UNDEFINEDHUMANUNDEFINED8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione443Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54812D3UNDEFINEDHUMANUNDEFINEDN-(4-Propylaminobutyl)-4-biphenylcarboxamide>10000Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
55068D2UNDEFINEDHUMANUNDEFINED4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide64Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55324KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one137Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55580MORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-methylcinnamoyloxy-7,8-dihydrocodeinone4.2Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
56092MORUNDEFINEDHUMANUNDEFINED(1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56604NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol1150Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56860SLC6A4UNDEFINEDHUMANUNDEFINED(3S)-3-((3-( 6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one15Rotella DP et al., 2009Jan 15, 2025Jan 15, 2025
57628SST3UNDEFINEDHUMANUNDEFINEDN-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57884Beta2UNDEFINEDHUMANUNDEFINED(2S,3S,4S,5R,6S)-6-(5-((R)-2-(5,6-diethyl-2,3-dihydro-1H-inden-2-ylamino)-1-hydroxyethyl)-2-oxo-1,2-dihydroquinolin-8-yloxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid>10000Baur F et al., 2010Jan 15, 2025Jan 28, 2025
581405-HT2CCLONEDHUMAN125I-DOIN-(3-Iodobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate1.05Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58396D1CLONEDHUMAN3H-SCH23390MRS5474>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58652D3CLONEDHUMAN3H-N-MethylspiporoneBenzquinamide3592Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58908nAChRCLONEDHUMAN3H-EpibatidineCamel Snus extract17.6Harris A, et al., 2015Jan 15, 2025Jan 27, 2025
59420D4CLONEDHUMAN3H-N-MethylspiporoneN-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide1.5Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
60188A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-4-(2-((1H-Pyrazol-3-yl)ethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide2.23Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60444GABAACLONEDHUMANFNZQH-II-09017Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60700GABAACLONEDHUMANFNZYCT-5200Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60956GABAACLONEDHUMANFNZYT-II3.518Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61212GABAACLONEDHUMANFNZRY-06117Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61468GABAACLONEDHUMANFNZRY-05989Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617245-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(4-methoxyphenyl)propan-1-amine206Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
622365-HT6CLONEDHUMAN3H-LSDTianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
63516NETCLONEDHUMAN3H-Nisoxetine3-methoxy-diphenidine325Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63772CXCR3PHA/IL-2 T cellsHUMAN125I-CXCL11CXCL929.5Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64540CLONEDHUMAN3H-EstradiolMethyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate1Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
65308GABAACLONEDHUMAN[3H] FlunitrazepamMLT-II-18>10000Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65565GABAACLONEDHUMAN[3H] FlunitrazepamAlprazolam1.43Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65821GABAACLONEDHUMAN[3H] FlunitrazepamCM-D45 C19H21N3O41.65Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66077M1CLONEDHUMAN3H-QNBMellpaladine A7200Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66589DORCLONEDHUMAN3H-DADLE3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 29, 2025
66845H4CLONEDHUMAN3H-HistamineN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67101SERTCLONEDHUMAN3H-CITALOPRAM1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67357D1CLONEDHUMAN3H-SCH233901-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
676135-HT2CKIDNEYHUMAN3H-MESULERGINEEthyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate30Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
23335-HT3AMYGDALAHUMAN3H-ZACOPRIDEHISTAMINE>10000BARNES ET AL., 1989Jan 15, 2025Jan 15, 2025
678695-HT7CLONEDHUMAN3H-5-CT(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline )97Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
683815-HT1ACLONEDHUMAN3H-8-OH-DPAT(-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol1.02329Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
68637recombinantHUMANUNKNOWNN-(Indan-2-yl)-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
33575-HT1ACLONEDHUMAN3H-8-OH-DPATIDAZOXAN662TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68893SST1CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH20.501187Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69149H4CLONEDHUMAN3H-N-alpha-methylhistamineN-alpha-methylhistamine316.228Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
3869D1CLONEDHUMAN3H-SCH23390RISPERIDONE523KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69661BZPCLONEDHUMANFNZ2-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
69917D5CLONEDHUMAN3H-SCH233904-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4637SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDING5-Hydroxy Tryptamine>10000PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48935-HT2ACLONEDHUMAN125I-DOILY 063518137BRYANT HU, ET AL., 1996Jan 15, 2025Jan 15, 2025
70429Sigma 1CLONEDHUMAN3H-Pentazocine(+)MRP32157.4Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
51495-HT2CCLONEDHUMAN125I-DOIDOCN1011NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70685DORCLONEDHUMAN3H-DiprenorphineTapentadol>10000Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
54055-HT2CChoroid PlexusHUMAN3H-MESULERGINEKETANSERIN50.11BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
709415-HT1DCLONEDHUMAN125I-aminopotentidine(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione546Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
711975-HT1ACLONEDHUMANWAY100635SYA162631.1Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
5917Alpha2BCLONEDHUMAN3H-RAUWOLSCINEBAM 13035.28BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
714535-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
7197NK2CLONEDHUMAN125I-[MePhe7]-NKBSubstance P129Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72733NETCLONEDHUMAN3H-Nisoxetinenaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
72989M2CLONEDHUMAN3H-QNBcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7709GABAACLONEDHUMAN3H-MUSCIMOLThio-4-PIOL446.68Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7965GABAACLONEDHUMAN3H-RO-15-178828319He X, et al., 1999Jan 15, 2025Jan 27, 2025
8221SST1CLONEDHUMAN125I-LTT-SRIF28seglitide>10000Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8477SST3CLONEDHUMAN125I-LTT-SRIF28L-362,85523.98Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8733SST2CLONEDHUMAN125I-LTT-SRIF28BIM 2303016.98Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8989SST3CLONEDHUMAN125I-SRIF-28BIM 230521.99Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74525M1CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
747815-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
9501MT2CLONEDHUMAN125I-IodomelatoninMelatonin,2-Phenyl0.15Sugden D, Pickering H, Teh MT, Garratt PJ, 1997Jan 15, 2025Jan 15, 2025
750375-HT6CLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75293Beta 2CLONEDHUMAN3H-CGP12177Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10013NETCLONEDHUMAN3H-NorepinephrineDESIPRAMINE8.54Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
75549M1CLONEDHUMAN3H-QNBpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75805SERTCLONEDHUMAN3H-CITALOPRAM1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
760615-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76317Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
11037H1CLONEDHUMAN3H-MEPYRAMINECHLORPHENIRAMINE2.51Moguilevsky N et al, 1994Jan 15, 2025Jan 15, 2025
76573MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol2670Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76829M2CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11549H1BRAINHUMAN3H-PYRILAMINEPAROXETINE>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
77085NETCLONEDHUMAN3H-Nisoxetine(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11805FR. CORTEXHUMAN3H-PRAZOSINCLOZAPINE160Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77341DORCLONEDHUMAN3H-DADLE(±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
775975-HT1BCLONEDHUMAN3H-5-CT(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
778535-HT2BCLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
781095-HT6CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78365Alpha1DCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78621Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
788775-HT1ACLONEDHUMAN3H-WAY100635N,N-Diisopropyltryptamine120.5Ray TS 2010 Jan 15, 2025Jan 15, 2025
13597OTMyometriumHUMAN3H-OxytocinL-365,2098.7Pettibone DJ, et al., 1991Jan 15, 2025Jan 15, 2025
791335-HT6CLONEDHUMAN3H-LSD5-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79389Alpha1BCLONEDHUMAN3H-PRAZOSINLYSERGIC ACID8677Ray TS 2010 Jan 15, 2025Jan 28, 2025
79645Sigma 1CLONEDHUMAN3H-Pentazocine(+)(±)-2,5-Dimethoxy-4-bromoamphetamine2193Ray TS 2010 Jan 15, 2025Jan 15, 2025
79901M5CLONEDHUMAN3H-QNBSalvinorin A>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80157CLONEDHUMAN3H-VASOPRESSIN(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
804135-HT5ACLONEDHUMAN3H-LSD(E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806695-HT1BCLONEDHUMAN3H-5-CT(5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153895-HT1BCLONEDHUMAN3H-5HT8-OH-DPAT2818.38BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809255-HT2BCLONEDHUMAN3H-LSD5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine104.713Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
81181MORCLONEDHUMAN3H-DAMGON-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
81437H1CLONEDHUMAN3H-PYRILAMINEN-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide2096Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
81693Beta2CLONEDHUMAN125I-iodo-pindolol(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
819495-HT1ECLONEDHUMAN3H-5HT[18F]MH.MZ>10000Herth MM et al 2009Jan 15, 2025Jan 15, 2025
16669M3CLONEDHUMAN3H-QNBTrihexyphenidyl6.4Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82205D2CLONEDHUMAN3H-N-Methylspiperone2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one585Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82461Alpha1BCLONEDHUMAN3H-PRAZOSIN(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine7211.1Besnard J et al 2012Jan 15, 2025Jan 28, 2025
827175-HT4CLONEDHUMAN3H-GR113808(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82973A2ACHO cellsHUMAN3H-MSX-28-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione2440Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
17693CLONEDHUMAN125I-VIPVIP [D-Asn28]0.71Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832295-HT2ACLONEDHUMAN125I-DOIMDL 1009070.67Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83485SERTHEK293 cellsHUMAN3H-CITALOPRAMMDMA>10000Simmler LD et al 2013Jan 15, 2025Jan 28, 2025
83741KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one8897PDSP Certified DataJan 15, 2025Jan 28, 2025
83997KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide165PDSP Certified DataJan 15, 2025Jan 28, 2025
84253Beta3CLONEDHUMAN125I-Pindolol(±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one5751PDSP Certified DataJan 15, 2025Jan 28, 2025
18973CCK2CLONEDHUMAN125I-BH-CCK-84425.1189Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
84509MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19229NB-OK-1HUMAN125-[AcHis1]PacapPACAP(8-38)30Vandermeers A et al., 1992Jan 15, 2025Jan 15, 2025
84765MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85021DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19741D2CLONEDHUMANUNDEFINEDMOPERONE1.8Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
19997PlateletsHUMAN3H-NECAddCHA>10000Lohse MJ et al., 1988aJan 15, 2025Jan 15, 2025
86045H4CLONEDHUMAN3H-Histamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
87325Alpha1BplaceholderHUMANPlaceholderTerazosin1.73Rak A et al 2016Jan 15, 2025Jan 28, 2025
87581MORCLONEDHUMAN3H-DAMGO2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87837A3testHUMAN3H-PSB-118- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
22557hERGCLONEDHUMAN3H-MethylspiperonePIMOZIDE18Kongsamut, S, et. al., 2002Jan 15, 2025Jan 15, 2025
88093A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
23069MORCLONEDHUMAN3H-DiprenorphineL-cysteic acid>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
886055-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL3600Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88861A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide647Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23581NPFF2CLONEDHUMAN125I-1DMe-Y8FaRFRP-355Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
89117A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide8.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893735-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide54Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240935-HT2ACLONEDHUMAN3H-SPIPERONEFLUPHENAZINE5.8Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
24349CORTEXHUMAN3H-PRAZOSINFLUOXETINE3171Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89885nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
24605CLONEDHUMANUNDEFINEDSR 144528>10000Rinaldi-Carmona, M et al., 1998Jan 15, 2025Jan 15, 2025
90141D2CLONEDHUMAN3H-SPIPERONE, 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24861CCR5CLONEDHUMAN3H-EpibatidineCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
90397A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25117nAChR7CLONEDHUMAN3H-EpibatidineQuetiapine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
90653A2BCLONEDHUMAN3H-PSB-603N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
909095-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane26.9153Franchini S et al 2014Jan 15, 2025Jan 15, 2025
25629Alpha1BCLONEDHUMAN125I-HEATCOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91165A1CLONEDHUMAN3H-DPCPX2-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
25885SLC6A3CLONEDHUMAN3H-GBR 12935Pseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91421CB1CLONEDHUMAN3H-SR144528O-6659128Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91933A1CLONEDHUMAN3H-DPCPX(2-Amino-5-(2,3-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
92189D2CLONEDHUMAN3H-RACLOPRIDE4-Fluoro-N-({1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl} methyl) benzenesulfonamide46Zajdel P et al 2012Jan 15, 2025Jan 28, 2025
271655-HT1DCORTEXHUMAN3H-5CTAL-37350A>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
927015-HT1DCLONEDHUMAN3H-Cimetidine(8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274215-HT1BCLONEDHUMAN3H-GR-125743BROMOCRIPTINE354.813Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929575-HT2ACLONEDHUMAN3H-KETANSERINWA-131830Sudol S et al 2020Jan 15, 2025Jan 15, 2025
28189H2CLONEDHUMAN3H-TIOTIDINEMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93725A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide3.73Federico S et al 2018Jan 15, 2025Jan 15, 2025
28445CLONEDHUMAN3H-QuisqualateAIDA>10000Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93981D2CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile22Ortega R et al 2011Jan 15, 2025Jan 29, 2025
28701PKCΓCLONEDHUMAN3H-PDBUARIPIPRAZOLE8000Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942375-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine1900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29213SST3CLONEDHUMANUNDEFINEDCH2751000Patel YC, 1999Jan 15, 2025Jan 15, 2025
947495-HT2CCLONEDHUMAN3H-MESULERGINE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95005D4CLONEDHUMAN3H-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
955175-HT6CLONEDHUMAN[3H]-LSD7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride1902Partyka A et al 2015Jan 15, 2025Jan 15, 2025
95773Alpha1ACLONEDHUMAN3H-PRAZOSINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
30493M4CLONEDHUMAN3H-QNBexo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene0.27Kim MG, et al., 2003Jan 15, 2025Jan 15, 2025
96285Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
31005CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
965415-HT1BCLONEDHUMAN[3H]5-CT1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
312615-HT2BC.H.O.HUMAN3H-MESULERGINERopinirole3801.89Millan MJ, et. al., 2004Jan 15, 2025Jan 15, 2025
96797D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA6400Mannel B et al 2017Jan 15, 2025Jan 28, 2025
31517D3CLONEDHUMAN125I-IODOSULPRIDE(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5)1000Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97309MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol1.05Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
320295-HT3CLONEDHUMANUNDEFINEDRS-1274451000Bonhaus, DW et. al., 1999Jan 15, 2025Jan 15, 2025
97565A2BCLONEDHUMAN[3H]DPCPX(±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98077CB2CHO cellsHUMAN3H-CP-55940CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate1050Amato G et al 2019Jan 15, 2025Jan 28, 2025
98333D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride31Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985895-HT2CCLONEDHUMAN[3H]-mesulergineARIPIPRAZOLE76Ofon E et al 2016aJan 15, 2025Jan 15, 2025
98845DATCLONEDHUMAN3H-WIN 35,4281-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
335655-HT6CLONEDHUMAN3H-LSDCELECOXIB>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99101D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99357D3CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole1.47Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34077P2X2, P2X3CLONEDHUMAN3H-A-317491AP2A>10000Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99613A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine1.91Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
100125Sigma 2CLONEDHUMAN3H-DTGQuetiapine1566PDSP Certified DataJan 15, 2025Jan 28, 2025
34845CB2CLONEDHUMAN3H-CP-55940Rinvanil, Acetyl>10000Jan 15, 2025Jan 15, 2025
100381SLC6A4CLONEDHUMAN3H-IMIPRAMINEIproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
35357D4CLONEDHUMAN3H-SPIROPERIDOLCLOZAPINE21Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
100893AChEBRAINHUMANFunctionalN-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide2.9Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
1011495-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone350Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
35869Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole74Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1014055-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione371Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36125CA2+ plateletsHUMANFunctionalIndomethacin2Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
101661Alpha1BCLONEDHUMAN[3H]-prazosinPerospirone44PDSP Certified DataMar 21, 2025Jul 28, 2026
36381PlateletsHUMAN3H-SQ 29548BM 6131.4Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
101917Beta3CLONEDHUMAN[3H]-CGP12177Ziprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
366375-HT2CCLONEDHUMAN3H-MESULERGINE(2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin7.6Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102173Sigma 2CLONEDHUMAN[3H]DTGNEMONAPRIDE137PDSP Certified DataMar 25, 2025Jul 28, 2026
37917CDK1CLONEDHUMANFunctional3-Amino-5-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carbothioamide3.2Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38429D3CLONEDHUMAN3H-NEMONAPRIDESKF 8295877.3Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
38685UNDEFINEDHUMAN3H-hypoxanthineN-[(1S,2S)-3-Cyclohexylcarbamoyl-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl]-2,4,6-trifluoro-benzamide4940Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39197MC4CLONEDHUMAN125I-NDP-MSHBeta MSH18.6Nickolls SA, et al., 2005Jan 15, 2025Jan 15, 2025
397095-HT2CCLONEDHUMAN3H-5HTMETHYLERGONOVINE4.57088Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40477STAT3CLONEDHUMANFunctionalAc-pTyr-Val-Pro-Gln-Thr-NH21540Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40733mGluR5CLONEDHUMANFunctional9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one49Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41245CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-phenyl-4-m-tolylbutyl)piperidin-4-ol Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42013M2CLONEDHUMAN3H-QNBFemoxetine150Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42269CLONEDHUMAN125I-MotilinDelta 31-322Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42525CLONEDHUMANFunctional[ala3,leu13]pMOT(1-14)1.31826Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42781Y2CLONEDHUMAN125I-PYYFMS586>10000Kakui N, et al., 2006Jan 15, 2025Jan 15, 2025
43037MAPK9CLONEDHUMAN3H-StaurosporineStaurosporine1100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43293DAPK2CLONEDHUMAN3H-StaurosporineLY-3335312600Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43549PAK6CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43805CaMKCLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44061CaMKCLONEDHUMAN3H-StaurosporineTarceva>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44317MAPK8CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44573NTRK1CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44829CSKCLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45085MAPK14CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45597SLC6A3CLONEDHUMAN3H-WIN 35,428IPRINDOLE6530Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
46109Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone23.36Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47133CLONEDHUMAN3H-SUBSTANCE PThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47389D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-Phenylethylpiperidin-4-yl)-2-naphthamide139Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47645GABAACLONEDHUMAN3H-RO-15-17882',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile0.25Russell MG, et al., 2006Jan 15, 2025Jan 27, 2025
47901GABAACLONEDHUMAN3H-RO-15-17886,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one56Chambers, MS et al., 2003Jan 15, 2025Jan 27, 2025
48669GNRHRCLONEDHUMANFunctionalN-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide0.5Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
496935-HT6CLONEDHUMAN3H-LSDPramipexole>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
51485Alpha1AUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide3.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51741ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline346Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51997DORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine8Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
52253A2BUNDEFINEDHUMANUNDEFINED9-(2-(benzylamino)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione>10000Drabczyńska A et al., 2007Jan 15, 2025Jan 15, 2025
52509Alpha2BUNDEFINEDHUMANUNDEFINED6,7-dimethoxy-2-((7-methoxy-2-(3-methoxyphenyl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline804Hagihara K et al., 2007Jan 15, 2025Jan 15, 2025
52765D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide15Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
53021MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan0.26Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53533SLC6A2UNDEFINEDHUMANUNDEFINED(-)-1-[(1S)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride14Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
537895-HT2AUNDEFINEDHUMANUNDEFINEDCLOZAPINE8.9Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54557A1UNDEFINEDHUMANUNDEFINED8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-ethyl-3,7-dihydropurine-2,6-dione1000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54813D3UNDEFINEDHUMANUNDEFINEDN-(4-Dipropylaminobutyl)-4-biphenylcarboxamide950Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
55069D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide226Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55325KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one150Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55581MORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-chlorocinnamoyloxy-7,8-dihydrocodeinone3.5Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
56093MORUNDEFINEDHUMANUNDEFINED6-desoxonaltrexone0.24Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56605NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol7Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56861SLC6A4UNDEFINEDHUMANUNDEFINED(3S)-3-((3-( 6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one4Rotella DP et al., 2009Jan 15, 2025Jan 15, 2025
57629SST3UNDEFINEDHUMANUNDEFINEDN-(1-(3-ethoxy-4-fluorobenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57885SLC6A3UNDEFINEDHUMANUNDEFINEDMAZINDOL22.1O'Neill DJ et al., 2010Jan 15, 2025Jan 15, 2025
581415-HT2CCLONEDHUMAN125I-DOIN-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate4.27Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58397D2CLONEDHUMAN3H-N-MethylspiporoneMRS5698>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58653D4CLONEDHUMAN3H-N-MethylspiporoneBenzquinamide574Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58909nAChRCLONEDHUMAN3H-EpibatidineNicotine22.2Harris A, et al., 2015Jan 15, 2025Jan 27, 2025
59421D2CLONEDHUMAN3H-N-MethylspiporoneN-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide60Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
596775-HT1ACLONEDHUMAN3H-WAY100635MH.MZ>10000Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
60189A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(2-((1-methyl-1H-pyrazol-4-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)bicyclo[3.1.0]- hexane-1-carboxamide2.34Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60445GABAACLONEDHUMANFNZXLI-2860.684Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60701GABAACLONEDHUMANFNZYCT-5>10000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60957GABAACLONEDHUMANFNZYT-II0.8712Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61213GABAACLONEDHUMANFNZZG-22417.1Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61469GABAACLONEDHUMANFNZRY-047200Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617255-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2,5-dimethoxyphenyl)propan-1-amine273Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
61981CLONEDHUMANUNDEFINEDIMIPRAMINE3400Teschemacher, AG et al., 1999Jan 15, 2025Jan 15, 2025
622375-HT7CLONEDHUMAN3H-LSDTianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
62749H1Brain Frontal CortexHUMAN3H-doxepinDOXEPIN0.24Richelson, Elliott et. al, 1984Jan 15, 2025Jan 28, 2025
63517NETCLONEDHUMAN3H-Nisoxetine4-methoxy-diphenidine2700Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63773CXCR3PHA/IL-2 T cellsHUMAN125I-CXCL11CXCL1021.9Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64541CLONEDHUMAN3H-Estradiol1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol15Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
64797Beta1CLONEDHUMAN125I-ICYPIndacaterol6.21Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
65309GABAACLONEDHUMAN[3H] FlunitrazepamSHU-1-194Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65566GABAACLONEDHUMAN[3H] FlunitrazepamAlprazolam1.54Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65822GABAACLONEDHUMAN[3H] FlunitrazepamCM-D45 C19H21N3O40.23Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66078M1CLONEDHUMAN3H-QNBMellpaladine B5172Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66846M1CLONEDHUMAN3H-QNBN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67102NETCLONEDHUMAN3H-Nisoxetine1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67358D2CLONEDHUMAN3H-N-Methylspiperone1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67614A1KIDNEYHUMAN3H-N6 -phenylisopropyladenosineEthyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate360Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
23345-HT3HIPPOCAMPUSHUMAN3H-ZACOPRIDEHISTAMINE>10000BARNES ET AL., 1989Jan 15, 2025Jan 15, 2025
67870D2CLONEDHUMAN3H-RACLOPRIDE(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
683825-HT1ACLONEDHUMAN3H-8-OH-DPAT1-hydroxyindane67.6083Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
68638recombinantHUMANUNKNOWNN-(Adamant-2-yl)-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
33585-HT1ACLONEDHUMAN3H-8-OH-DPATIMIPRAMINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68894SST2CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH21.25893Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69150H4CLONEDHUMAN3H-N-alpha-methylhistamineAlpha-Methylhistamine-R251.189Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
3870D1CLONEDHUMAN3H-SCH23390CLOZAPINE196KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69662BZPCLONEDHUMANFNZ3-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
69918D5CLONEDHUMAN3H-SCH233904-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4638SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDINGRESERPINE>10000PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48945-HT2ACLONEDHUMAN125I-DOILY 31422865BRYANT HU, ET AL., 1996Jan 15, 2025Jan 15, 2025
704305-HT7CLONEDHUMAN3H-LSDMRP32155.9Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51505-HT2CCLONEDHUMAN125I-DOIDOPR1.1NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70686DORCLONEDHUMAN3H-DiprenorphineTramadol(+-)>10000Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
709425-HT1DCLONEDHUMAN125I-aminopotentidine4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
711985-HT1ACLONEDHUMANWAY100635SYA013117.4Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
5918Alpha2BCLONEDHUMAN3H-RAUWOLSCINEOXYMETAZOLINE754BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
6686D2CLONEDHUMAN3H-NEMONAPRIDERISPERIDONE27SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
7198NK2CLONEDHUMAN125I-[MePhe7]-NKBNKB [MePhe7]1597Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72734SERTCLONEDHUMAN3H-CITALOPRAMnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
72990M3CLONEDHUMAN3H-QNBcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7710GABAACLONEDHUMAN3H-MUSCIMOLSR 9553134.67Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7966GABAACLONEDHUMAN3H-RO-15-178829>10000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8222SST1CLONEDHUMAN125I-LTT-SRIF28CGP 239964.67Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8478SST3CLONEDHUMAN125I-LTT-SRIF28L-363,301457.08Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8734SST2CLONEDHUMAN125I-LTT-SRIF28BIM 23056467.73Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8990SST3CLONEDHUMAN125I-SRIF-28BIM 23056100Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74526M2CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
747825-HT1BCLONEDHUMAN3H-5-CT(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
750385-HT7CLONEDHUMAN3H-LSD(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10014NETCLONEDHUMAN3H-NorepinephrineIMIPRAMINE118Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
75550M2CLONEDHUMAN3H-QNBpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75806NETCLONEDHUMAN3H-Nisoxetine1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760625-HT3CLONEDHUMAN3H-GR-65630Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76318Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
11038H1CLONEDHUMAN3H-MEPYRAMINEHISTAMINE1258.92Moguilevsky N et al, 1994Jan 15, 2025Jan 15, 2025
76830M3CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11550H1BRAINHUMAN3H-PYRILAMINESERTRALINE>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
77086SERTCLONEDHUMAN3H-CITALOPRAM(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
11806FR. CORTEXHUMAN3H-RAUWOLSCINETHIOTHIXENE,cis-200Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77342KORCLONEDHUMAN3H-U69593(±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide1030Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
775985-HT1DCLONEDHUMAN3H-5-CT(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
778545-HT2CCLONEDHUMAN3H-MESULERGINE(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
781105-HT7CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78366Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78622Beta 2CLONEDHUMAN3H-CGP12177(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788785-HT1ACLONEDHUMAN3H-WAY1006355-Methoxy-N,N-diisopropyltryptamine132.4Ray TS 2010 Jan 15, 2025Jan 15, 2025
13598OTMyometriumHUMAN3H-OxytocinL-366,6704.1Pettibone DJ, et al., 1991Jan 15, 2025Jan 15, 2025
791345-HT6CLONEDHUMAN3H-LSDN,N-Dipropyltryptamine4543Ray TS 2010 Jan 15, 2025Jan 15, 2025
79390Alpha1BCLONEDHUMAN3H-PRAZOSINcis-2a>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
79646Sigma 1CLONEDHUMAN3H-Pentazocine(+)3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79902H1CLONEDHUMAN3H-PYRILAMINE(±)-2,5-Dimethoxy-4-bromoamphetamine9120Ray TS 2010 Jan 15, 2025Jan 28, 2025
80158CLONEDHUMAN3H-VASOPRESSIN(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
804145-HT6CLONEDHUMAN3H-LSD(E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806705-HT1DCLONEDHUMAN3H-5-CT(5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153905-HT1BCLONEDHUMAN3H-5HT5-HT,2-Me512.86BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809265-HT2CCLONEDHUMAN3H-MESULERGINE3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine10.4713Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
81182Alpha1ACLONEDHUMAN3H-PRAZOSINN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
81438D2CLONEDHUMAN3H-N-MethylspiperoneN-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
819505-HT2ACLONEDHUMAN125I-DOI[18F]MH.MZ3Herth MM et al 2009Jan 15, 2025Jan 15, 2025
16670M3CLONEDHUMAN3H-QNBProcyclidine12.4Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82206D3CLONEDHUMAN3H-N-Methylspiperone2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one32Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82462Alpha1DCLONEDHUMAN3H-PRAZOSIN(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine2307Besnard J et al 2012Jan 15, 2025Jan 28, 2025
171825-HT2BCLONEDHUMAN3H-5HTMETHYLPHENIDATE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
827185-HT5ACLONEDHUMAN3H-LSD(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17694PANC1HUMAN125I-VIPVIP [D-Gln16]2.9Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832305-HT2ACLONEDHUMAN3H-KETANSERINMDL 1009070.048Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
834865-HT1AHEK293 cellsHUMAN3H-8-OH-DPATMDMA>10000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
83742MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one5536PDSP Certified DataJan 15, 2025Jan 28, 2025
83998MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5029PDSP Certified DataJan 15, 2025Jan 28, 2025
842545-HT7CLONEDHUMAN3H-LSD(±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one1205PDSP Certified DataJan 15, 2025Jan 15, 2025
18974CCK2CLONEDHUMAN125I-BH-CCK-843776.247Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
84510DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19230NB-OK-1HUMAN125-[AcHis1]PacapPACAP(7-38)8Vandermeers A et al., 1992Jan 15, 2025Jan 15, 2025
84766MORCLONEDHUMAN3H-DAMGO±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85022DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19742D2CLONEDHUMANUNDEFINEDN-DESMETHYLCLOZAPINE100Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
852785-HT1DrecombinantHUMAN125I-iodoaminopotentidineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
19998PlateletsHUMAN3H-NECAalpha-ddCHA>10000Lohse MJ et al., 1988aJan 15, 2025Jan 15, 2025
85790D1CLONEDHUMAN3H-SCH23390N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
86046KORCLONEDHUMAN3H-U69593(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86302A1CLONEDHUMAN3H-CCPA3-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione156Koch P et al 2018Jan 15, 2025Jan 15, 2025
86558A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
87326Alpha1AplaceholderHUMANPlaceholderTerazosin51.89Rak A et al 2016Jan 15, 2025Jan 28, 2025
87582NETCLONEDHUMAN3H-Nisoxetine2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
88094A1CLONEDHUMAN3H-CCPA10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
23070MORCLONEDHUMAN3H-DiprenorphineD-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
886065-HT2ACLONEDHUMAN3H-KETANSERINHALOPERIDOL120Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88862A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23582NPFF2CLONEDHUMAN125I-1DMe-Y8FaFMRFamide13Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
89118A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide12Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893745-HT7CLONEDHUMAN3H-5-CT3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide32Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240945-HT2ACLONEDHUMAN3H-SPIPERONEHALOPERIDOL103Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
896305-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone0.0645654Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
24350CORTEXHUMAN3H-PRAZOSINPAROXETINE2741Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89886nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
24606M1CLONEDHUMANUNDEFINEDSR 144528>10000Rinaldi-Carmona, M et al., 1998Jan 15, 2025Jan 15, 2025
90142D2CLONEDHUMAN3H-SPIPERONE2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90398A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25118nAChRCLONEDHUMAN3H-EpibatidineQuetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
90654A2BCLONEDHUMAN3H-PSB-603N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25374D5CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE1676PDSP Certified DataJan 15, 2025Jan 15, 2025
90910Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane6.45654Franchini S et al 2014Jan 15, 2025Jan 28, 2025
91166A1CLONEDHUMAN3H-DPCPXN-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
914225-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate0.54Li P et al 2014Jan 15, 2025Jan 15, 2025
261425-HT5ACLONEDHUMAN3H-LSDPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91934A1CLONEDHUMAN3H-DPCPX(2-Amino-5-(2,4-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
92190D2CLONEDHUMAN3H-RACLOPRIDE4-Fluoro-N-({1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl}methyl) benzenesulfonamide839Zajdel P et al 2012Jan 15, 2025Jan 28, 2025
927025-HT1DCLONEDHUMAN3H-Cimetidine15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274225-HT1DCLONEDHUMAN3H-GR-125743BROMOCRIPTINE10.7152Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929585-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine5047Sudol S et al 2020Jan 15, 2025Jan 15, 2025
28190NETCLONEDHUMAN3H-NisoxetineMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93726A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide18.6Federico S et al 2018Jan 15, 2025Jan 15, 2025
28446mGluR5CLONEDHUMAN3H-QuisqualateAIDA>10000Mutel V, et.al., 2000Jan 15, 2025Jan 28, 2025
93982D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one8.8Ortega R et al 2011Jan 15, 2025Jan 29, 2025
942385-HT2CCLONEDHUMAN3H-MESULERGINE4-benzyloxy-2,5-dimethoxyphenethylamine110Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29214SST3CLONEDHUMANUNDEFINEDL-797,5912240Patel YC, 1999Jan 15, 2025Jan 15, 2025
947505-HT2CCLONEDHUMAN3H-MESULERGINE5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
955185-HT6CLONEDHUMAN[3H]-LSD1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
95774Alpha1BCLONEDHUMAN3H-PRAZOSINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
30494M5CLONEDHUMAN3H-QNBexo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene0.56Kim MG, et al., 2003Jan 15, 2025Jan 15, 2025
96286Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
965425-HT1DCLONEDHUMAN[3H]5-CT1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
312625-HT2CC.H.O.HUMAN3H-MESULERGINERopinirole>10000Millan MJ, et. al., 2004Jan 15, 2025Jan 15, 2025
96798D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine3200Mannel B et al 2017Jan 15, 2025Jan 28, 2025
31518D3CLONEDHUMAN125I-IODOSULPRIDE(R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10)1258.93Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
970545-HT1ACLONEDHUMAN[3H]8-OH-DPAT3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97310MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol10.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
32030CB1CLONEDHUMANUNDEFINEDRS-1274451000Bonhaus, DW et. al., 1999Jan 15, 2025Jan 27, 2025
97566A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate8.1Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98078CB1CHO cellsHUMAN3H-CP-55940Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate4Amato G et al 2019Jan 15, 2025Jan 28, 2025
98334D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride447Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98590D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
33310Alpha1ACLONEDHUMAN3H-PRAZOSINAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98846NETCLONEDHUMAN3H-Nisoxetine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
335665-HT7CLONEDHUMAN3H-LSDCELECOXIB>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99102D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99358D3CLONEDHUMAN[3H]N-methylspiperone6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline1.35Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34078P2X2, P2X3CLONEDHUMAN3H-A-317491A-3174910.9Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99614A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2-oxo-ethoxy}-phenyl]-xanthine3.51Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
100126D1CLONEDHUMAN3H-SCH23390Quetiapine381PDSP Certified DataJan 15, 2025Jan 28, 2025
34846CB2CLONEDHUMAN3H-CP-55940PhAR300Jan 15, 2025Jan 15, 2025
100382NETCLONEDHUMAN3H-NisoxetineIproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
35358D4CLONEDHUMAN3H-SPIROPERIDOL5-methyl-10-(4-methylpiperazino)-5H-dibenzo[a,d]cycloheptene12Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
100894BchEserumHUMANFunctionalN-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide21.4Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
1011505-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone197Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
35870Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole12Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
101406D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione27Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
36126COX-2purifiedHUMANFunctionalIndomethacin600Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
101662Alpha2BCLONEDHUMAN[3H]-rauwolscinePerospirone202PDSP Certified DataMar 21, 2025Jul 28, 2026
36382CLONEDHUMAN3H-SQ 29548BM 5731.1Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
101918BZPCLONEDHUMAN[3H] FlunitrazepamZiprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
366385-HT2CCLONEDHUMAN3H-MESULERGINEHALOPERIDOL5454Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102174Sigma 1CLONEDHUMAN[3H]PentazocineNEMONAPRIDE7PDSP Certified DataMar 25, 2025Jul 28, 2026
37918CDK1CLONEDHUMANFunctional4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide6Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38430D3CLONEDHUMAN3H-NEMONAPRIDEMCL-211356Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
38686UNDEFINEDHUMAN3H-hypoxanthinePyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(3-bromo-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcarbamoyl}-2-methyl-propyl)-amide32Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39198MC4CLONEDHUMAN125I-NDP-MSHGamma1-MSH589Nickolls SA, et al., 2005Jan 15, 2025Jan 15, 2025
397105-HT2CCLONEDHUMAN3H-5HTMK 21297.7237Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40478STAT3CLONEDHUMANFunctionalAc-pTyr-Ile-Pro-Gln-Thr-NH21070Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40734mGluR5CLONEDHUMANFunctional9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one2100Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41246CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-phenyl-4-p-tolylbutyl)piperidin-4-ol Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42014M2CLONEDHUMAN3H-QNBFLUOXETINE2700Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42270CLONEDHUMAN125I-MotilinDelta 33-361000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42526CLONEDHUMANFunctional[ala4,leu13]pMOT(1-14)2570.4Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42782Y2CLONEDHUMAN125I-PYYL-152,804>10000Kakui N, et al., 2006Jan 15, 2025Jan 15, 2025
43038MAPK9CLONEDHUMAN3H-StaurosporineSB202190120Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43294DAPK3CLONEDHUMAN3H-StaurosporineEKB-5694100Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43550PAK7CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43806CaMKCLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44062CaMKCLONEDHUMAN3H-StaurosporineTarceva>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44318MAPK9CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44574PAK1CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44830CSNK1ECLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45086MAPK P38CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45598SLC6A4CLONEDHUMAN3H-IMIPRAMINEIproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
46110Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47646GABAACLONEDHUMAN3H-RO-15-17884,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile1.2Russell MG, et al., 2006Jan 15, 2025Jan 27, 2025
47902GABAACLONEDHUMAN3H-RO-15-17886,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one21Chambers, MS et al., 2003Jan 15, 2025Jan 27, 2025
48670CLONEDHUMANFunctionalN-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride>10000Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49694D1CLONEDHUMAN3H-SCH23390Pramipexole>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
51486Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51742ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline110Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51998DORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine6.53Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
52254A2BUNDEFINEDHUMANUNDEFINED9-(2-(4-chlorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione>10000Drabczyńska A et al., 2007Jan 15, 2025Jan 15, 2025
52510Alpha2BUNDEFINEDHUMANUNDEFINED6,7-dimethoxy-2-((7-methoxy-2-phenylbenzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline752Hagihara K et al., 2007Jan 15, 2025Jan 15, 2025
52766D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide22Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
53022MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan0.21Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53534SLC6A2UNDEFINEDHUMANUNDEFINED(+)-1-[(1R)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride187Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
537905-HT2AUNDEFINEDHUMANUNDEFINEDHALOPERIDOL120Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54558A1UNDEFINEDHUMANUNDEFINED8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione>10000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54814D3UNDEFINEDHUMANUNDEFINEDN-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide140Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
55070D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide9.2Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55326KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one506Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55582DORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone180Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
56094MORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide2.5Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56606NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol36Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56862SLC6A4UNDEFINEDHUMANUNDEFINED(3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one7Rotella DP et al., 2009Jan 15, 2025Jan 15, 2025
57630SST3UNDEFINEDHUMANUNDEFINEDN-(1-(3-ethoxy-4-(trifluoromethyl)benzyl)piperidin-4-yl)benzo[d]oxazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57886SLC6A2UNDEFINEDHUMANUNDEFINEDDESIPRAMINE3.4O'Neill DJ et al., 2010Jan 15, 2025Jan 15, 2025
581425-HT2CCLONEDHUMAN3H-MESULERGINEN-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate28.2Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58398D2CLONEDHUMAN3H-N-MethylspiporoneMRS5678>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58654M1CLONEDHUMAN3H-QNBCyclobenzaprine25Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58910D2CLONEDHUMAN3H-N-Methylspiporone(+)-SYA 0951.1Ablordeppey S, et al., 2006Jan 15, 2025Jan 15, 2025
59422Alpha1ACLONEDHUMAN3H-PRAZOSINN-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide160Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
596785-HT1BCLONEDHUMAN3H-5CTMH.MZ1846Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
60190A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-4-(2-(Furan-2-ylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide0.62Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60446GABAACLONEDHUMANFNZXLI-2860.118Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60702GABAACLONEDHUMANFNZTJH-IV-51>10000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60958GABAACLONEDHUMANFNZYT-II6.932Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61214GABAACLONEDHUMANFNZZG-22433.7Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61470GABAACLONEDHUMANFNZRY-047124Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617265-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine194Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
62238Alpha1ACLONEDHUMAN3H-PRAZOSINTianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
62750H1Brain Frontal CortexHUMAN3H-doxepinTrimipramine0.27Richelson, Elliott et. al, 1984Jan 15, 2025Jan 28, 2025
630065-HT2BCLONEDHUMAN3H-5-HTFenfluramine (+)5099Rothman RB, et al., 2003Jan 15, 2025Jan 15, 2025
63518NETCLONEDHUMAN3H-Nisoxetine2-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63774CXCR3PHA/IL-2 T cellsHUMAN125I-CXCL11CXCL110.05Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64542CLONEDHUMAN3H-Estradiol17beta-Estradiol2100Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
64798Beta1CLONEDHUMAN125I-ICYPFormoterol6.12Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
65054H1FR. CORTEXHUMAN3H-MEPYRAMINEIPRINDOLE670Chang, R et., 1978Jan 15, 2025Jan 15, 2025
65310GABAACLONEDHUMAN[3H] FlunitrazepamSHU-1-1912Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65567GABAACLONEDHUMAN[3H] FlunitrazepamAlprazolam>10000Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65823GABAACLONEDHUMAN[3H] FlunitrazepamYT-50.421Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66079NETCLONEDHUMAN3H-NisoxetineMellpaladine B1259Uchimasu, Hajime. et, al. 2016Jan 15, 2025Jan 15, 2025
66847M2CLONEDHUMAN3H-QNBN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67103DATCLONEDHUMAN3H-WIN354281-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67359D3CLONEDHUMAN3H-N-Methylspiperone1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride425Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67615A2AKIDNEYHUMAN3H-2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosineEthyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate1570Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
678715-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline91Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
28475-HT2ACORTEXHUMAN3H-KETANSERINKETANSERIN0.56WANDER ET AL., 1987Jan 15, 2025Jan 15, 2025
683835-HT1ACLONEDHUMAN3H-8-OH-DPAT1-hydroxyindane1.62181Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
68639recombinantHUMANUNKNOWNN-[(Naphth-2-yl)methyl]-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
33595-HT1ACLONEDHUMAN3H-8-OH-DPATKETANSERIN>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68895SST3CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH20.630957Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69151H4CLONEDHUMAN3H-N-alpha-methylhistamineAlpha-Methylhistamine-S3981.07Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
3871D1CLONEDHUMAN3H-SCH23390OLANZAPINE35KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69663BZPCLONEDHUMANFNZ4-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
69919SLC6A3CLONEDHUMAN3H-WIN354284-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
4639SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDINGKETANSERIN>10000PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48955-HT2ACLONEDHUMAN125I-DOILY 320950248BRYANT HU, ET AL., 1996Jan 15, 2025Jan 15, 2025
704315-HT2BCLONEDHUMAN3H-LSDMRP32156.6Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51515-HT2CCLONEDHUMAN125I-DOIDOHx0.7NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70687KORCLONEDHUMAN3H-DiprenorphineNALOXONE270Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
70943KORCLONEDHUMAN3H-U695934-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
711995-HT1ACLONEDHUMANWAY100635FEMPT0.2Collier TL et al 2017Jan 15, 2025Jan 15, 2025
5919Alpha2BCLONEDHUMAN3H-RAUWOLSCINEPHENTOLAMINE6.8BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
6175Beta1CLONEDHUMAN125I-CYPSB2040701000WARDLE KA, ET AL., 1994Jan 15, 2025Jan 15, 2025
6687D4CLONEDHUMAN3H-NEMONAPRIDERISPERIDONE45SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
7199NK2CLONEDHUMAN125I-[MePhe7]-NKBSenktide>10000Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72735Sigma 1CLONEDHUMAN3H-Pentazocine(+)naringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
72991M4CLONEDHUMAN3H-QNBcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7711GABAACLONEDHUMAN3H-MUSCIMOLBicuculline>10000Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7967GABAACLONEDHUMAN3H-RO-15-1788307000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8223SST1CLONEDHUMAN125I-LTT-SRIF28octreotide223.87Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8479SST3CLONEDHUMAN125I-LTT-SRIF28RC 16042.65Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8735SST2CLONEDHUMAN125I-LTT-SRIF28cycloantagonist SA3981.07Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8991SST3CLONEDHUMAN125I-SRIF-28SA398.1Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74527M3CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
747835-HT1DCLONEDHUMAN3H-5-CT(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75039Alpha1ACLONEDHUMAN3H-PRAZOSIN(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9759MT1CLONEDHUMAN125I-IodomelatoninLuzindole,5-Methoxy32.7Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75295D1CLONEDHUMAN3H-SCH23390Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
10015NETCLONEDHUMAN3H-NorepinephrineCOCAINE217Paczkowski,Bryan-Lluka,Porzgen,Bruss,Bonisch, 1999Jan 15, 2025Jan 15, 2025
75551M3CLONEDHUMAN3H-QNBpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75807NOPCLONEDHUMAN3H-Nociceptin1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
760635-HT5ACLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76319Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
11039H1CLONEDHUMAN3H-MEPYRAMINERANITIDINE>10000Moguilevsky N et al, 1994Jan 15, 2025Jan 15, 2025
76575M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76831M4CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11551H1BRAINHUMAN3H-PYRILAMINETRAZODONE1100Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
77087Sigma 1CLONEDHUMAN3H-Pentazocine(+)(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
11807FR. CORTEXHUMAN3H-RAUWOLSCINEd-Butaclamol310Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77343MORCLONEDHUMAN3H-DAMGO(±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
775995-HT1ECLONEDHUMAN3H-5-HT(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
778555-HT3CLONEDHUMAN3H-GR-65630(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78111Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78367Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78623D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
788795-HT1ACLONEDHUMAN3H-WAY100635N,N-Dipropyltryptamine31.8Ray TS 2010 Jan 15, 2025Jan 15, 2025
13599OTMyometriumHUMAN3H-OxytocinL-366,6829.4Pettibone DJ, et al., 1991Jan 15, 2025Jan 15, 2025
791355-HT6CLONEDHUMAN3H-LSD4-Ethylthio-2,5-dimethoxyphenylbutylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79391Alpha1BCLONEDHUMAN3H-PRAZOSINR,R-2b>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
79647Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79903H1CLONEDHUMAN3H-PYRILAMINE(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80159CLONEDHUMAN3H-VASOPRESSIN3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
804155-HT7CLONEDHUMAN3H-LSD(E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806715-HT1ECLONEDHUMAN3H-5-HT(5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153915-HT1BCLONEDHUMAN3H-5HTPropanolol,(+/-)2691.53BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809275-HT2CCLONEDHUMAN3H-MESULERGINE3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine>10000Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
81183Alpha1BCLONEDHUMAN3H-PRAZOSINN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
814395-HT2ACLONEDHUMAN3H-KETANSERINN-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide>10000Weiss DR et al 2018Jan 15, 2025Jan 15, 2025
81695CLONEDHUMAN3H-Nitrendipine(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 15, 2025
819515-HT2BCLONEDHUMAN3H-LSD[18F]MH.MZ299Herth MM et al 2009Jan 15, 2025Jan 15, 2025
16671M3CLONEDHUMAN3H-QNBPIRENZEPINE150Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
82207D4CLONEDHUMAN3H-N-Methylspiperone2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one925Besnard J et al 2012Jan 15, 2025Jan 28, 2025
82463D1CLONEDHUMAN3H-SCH23390(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine1353Besnard J et al 2012Jan 15, 2025Jan 28, 2025
827195-HT6CLONEDHUMAN3H-LSD(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82975A2BCHO cellsHUMAN3H-PSB-6038-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione300Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
17695PANC1HUMAN125I-VIPVIP [D-Met17]29.5Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832315-HT2ACLONEDHUMAN3H-KETANSERINKETANSERIN0.77Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
834875-HT2AHEK293 cellsHUMAN3H-KETANSERINMDMA7800Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
837435-HT1DCLONEDHUMAN3H-5-CT(±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one3230PDSP Certified DataJan 15, 2025Jan 15, 2025
184635-HT1BCLONEDHUMAN3H-5HT1-NP10.1Jorand-Lebrun C et al., 1997aJan 15, 2025Jan 15, 2025
83999KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide180PDSP Certified DataJan 15, 2025Jan 28, 2025
18975CCK2CLONEDHUMAN125I-BH-CCK-842724.436Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
84511DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(2,6-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19231NB-OK-1HUMAN125-[AcHis1]PacapPACAP(6-38)1.5Vandermeers A et al., 1992Jan 15, 2025Jan 15, 2025
84767DORCLONEDHUMAN3H-DADLE±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85023MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19743D2CLONEDHUMAN3H-OlanzapineOLANZAPINE3Seeman P, Tallerico T., 1998Jan 15, 2025Jan 15, 2025
85279H3recombinantHUMAN3H-NAMHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85791D2CLONEDHUMAN3H-N-MethylspiperoneN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide2300Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
86047MORCLONEDHUMAN3H-DAMGO(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86303A2ACLONEDHUMAN3H-MSX-23-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1780Koch P et al 2018Jan 15, 2025Jan 15, 2025
86559A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
87327Alpha1AplaceholderHUMANPlaceholderPhenylephrine,(+/-)55.99Rak A et al 2016Jan 15, 2025Jan 28, 2025
88095A1CLONEDHUMAN3H-CCPAcompound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
23071MORCLONEDHUMAN3H-DiprenorphineL-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88607D1CLONEDHUMAN3H-SCH23390HALOPERIDOL120Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88863A3HeLaHUMAN3H-NECAN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23583NPFF2CLONEDHUMAN125I-1DMe-Y8FaPrRP24-3132Engstrom M, et al., 2003Jan 15, 2025Jan 15, 2025
89119A3HeLaHUMAN3H-NECAN-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23839CRF1CLONEDHUMAN3H-SN003DMP6961.8Zhang, GE. et al., 2003Jan 15, 2025Jan 15, 2025
893755-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1836Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240955-HT2ACLONEDHUMAN3H-SPIPERONELOXAPINE2.5Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
896315-HT1ACLONEDHUMAN3H-8-OH-DPAT(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0147911Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
24351CORTEXHUMAN3H-PRAZOSINSERTRALINE188Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
24607M2CLONEDHUMANUNDEFINEDSR 144528>10000Rinaldi-Carmona, M et al., 1998Jan 15, 2025Jan 15, 2025
90143D2CLONEDHUMAN3H-SPIPERONE2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine870Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24863H1CLONEDHUMAN3H-PYRILAMINECLOZAPINE2PDSP Certified DataJan 15, 2025Jan 15, 2025
90399A2BCLONEDHUMAN3H-PSB-603N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide215Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
25119EP3CLONEDHUMAN3H-PGE2Quetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90655A2BCLONEDHUMAN3H-PSB-603N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide547 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25375D2CLONEDHUMAN3H-NMSPARIPIPRAZOLE0.95PDSP Certified DataJan 15, 2025Jan 15, 2025
90911Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane69.1831Franchini S et al 2014Jan 15, 2025Jan 28, 2025
25631H2CLONEDHUMAN3H-TIOTIDINECOCAINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91167A2ACLONEDHUMAN3H-CGS21680N-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
914235-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone0.94Li P et al 2014Jan 15, 2025Jan 15, 2025
26143MORCLONEDHUMAN3H-DiprenorphinePseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91935A1CLONEDHUMAN3H-DPCPX(2-Amino-5-(2,5-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
92191D2CLONEDHUMAN3H-RACLOPRIDE3-Chloro-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide66Zajdel P et al 2012Jan 15, 2025Jan 28, 2025
927035-HT1DCLONEDHUMAN3H-Cimetidine9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
274235-HT1DCLONEDHUMAN3H-GR-125743Cabergoline8.70964Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
929595-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine268Sudol S et al 2020Jan 15, 2025Jan 15, 2025
28191nAChR7CLONEDHUMAN3H-EpibatidineMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93727A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide23.4Federico S et al 2018Jan 15, 2025Jan 15, 2025
28447CLONEDHUMAN3H-QuisqualateDCG-IV>10000Mutel V, et.al., 2000Jan 15, 2025Jan 15, 2025
93983D3CLONEDHUMAN3H-SPIPERONEcompound 421.7Ortega R et al 2011Jan 15, 2025Jan 28, 2025
28703Alpha1ACLONEDHUMAN3H-PRAZOSINARIPIPRAZOLE25.7Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942395-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-methallyloxyamphetamine290Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29215SST3CLONEDHUMANUNDEFINEDL-779,976729Patel YC, 1999Jan 15, 2025Jan 15, 2025
947515-HT2CCLONEDHUMAN3H-MESULERGINE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
29727D2CLONEDHUMAN3H-SPIPERONEGMC1-169140Liao Y, et.al., 1999Jan 15, 2025Jan 15, 2025
955195-HT6CLONEDHUMAN[3H]-LSD7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione8987Partyka A et al 2015Jan 15, 2025Jan 15, 2025
95775Alpha1DCLONEDHUMAN3H-PRAZOSINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
30495M1CLONEDHUMAN3H-QNBendo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene6.6Kim MG, et al., 2003Jan 15, 2025Jan 15, 2025
96031MORCLONEDHUMAN3H-DAMGO4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96287Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
31007V2CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
965435-HT1ECLONEDHUMAN[3H]5-HT1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96799D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA1900Mannel B et al 2017Jan 15, 2025Jan 28, 2025
315195-HT2CCLONEDHUMAN3H-MESULERGINE(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)5011.87Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
970555-HT1BCLONEDHUMAN[3H]GR1275433-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97311MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol66.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
320315-HT6CLONEDHUMANUNDEFINEDRS-1274451000Bonhaus, DW et. al., 1999Jan 15, 2025Jan 15, 2025
97567A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate43.41Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98079CB2CHO cellsHUMAN3H-CP-55940Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate710Amato G et al 2019Jan 15, 2025Jan 28, 2025
32799D2CLONEDHUMAN3H-SPIPERONEHALOPERIDOL1Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
98335D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride91Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98591D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
33311Alpha1BCLONEDHUMAN3H-PRAZOSINAcetylsalicylic acid>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
98847SERTCLONEDHUMAN3H-Cimetidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33567D1CLONEDHUMAN3H-SCH23390CELECOXIB>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99103D4CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99359D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine8.32Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34079P2X2, P2X3CLONEDHUMAN3H-A-317491ATP,TNP14.5Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99615A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine3.64Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
1001275-HT1ACLONEDHUMAN3H-WAY100635Brexpiprazole1.1PDSP Certified DataJan 15, 2025Jan 15, 2025
34847CB2CLONEDHUMAN3H-CP-55940PhAR, ent400Jan 15, 2025Jan 15, 2025
100383SLC6A3CLONEDHUMAN3H-WIN 35,428Iproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
1006395-HT1ACLONEDHUMAN3H-WAY100635CYPROHEPTADINE50Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
35359D4CLONEDHUMAN3H-SPIROPERIDOL5-methyl-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene320Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
100895AChEBRAINHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(5-cyano-1H-indol-3-yl)propionamide0.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
1011515-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone52Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
35871SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1014075-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione28Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36127COX-2purified w/detergentHUMANFunctionalIndomethacin400Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
101663Alpha2CCLONEDHUMAN[3H]rauwolscinePerospirone98PDSP Certified DataMar 21, 2025Jul 28, 2026
36383CLONEDHUMAN3H-SQ 29548BM 6132.1Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
101919PBRCLONEDHUMAN[3H]PK11195Ziprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
366395-HT2CCLONEDHUMAN3H-MESULERGINECLOZAPINE21Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
37919CDK2CLONEDHUMANFunctional4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide2Lin R, et al., 2005Jan 15, 2025Jan 15, 2025
38431D3CLONEDHUMAN3H-NEMONAPRIDEMCL-212>10000Neumeyer JL, et al., 2003aJan 15, 2025Jan 15, 2025
38687UNDEFINEDHUMAN3H-hypoxanthinePyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(biphenyl-3-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcarbamoyl}-2-methyl-propyl)-amide3.9Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39199MC4CLONEDHUMAN125I-NDP-MSHdesacetyl-alpha-MSH30.2Nickolls SA, et al., 2005Jan 15, 2025Jan 15, 2025
394555-HT2ACLONEDHUMAN3H-KETANSERIN1-Methylpsilocybin>10000Sard H, et al., 2005Jan 15, 2025Jan 15, 2025
397115-HT2CCLONEDHUMAN3H-5HTORG-1296214.7911Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40479STAT3CLONEDHUMANFunctionalAc-pTyr-Phe-Pro-Gln-Thr-NH21890Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40735mGluR5CLONEDHUMANFunctional9-(2',2',2'-Trifluoroethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one99Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41247CLONEDHUMAN125I-Chemokine1-(4-Biphenyl-4-y)-4-(4-chlorophenyl)butyl]-4-(4-chlorophenyl)piperidin-4-ol>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
42015M2CLONEDHUMAN3H-QNBIMIPRAMINE88Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42271CLONEDHUMAN125I-MotilinDelta 103-1041000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42527CLONEDHUMANFunctional[ala5,leu13]pMOT(1-14)28.8403Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42783Y2CLONEDHUMAN125I-PYYPYY2.1Kakui N, et al., 2006Jan 15, 2025Jan 15, 2025
43039MAPK9CLONEDHUMAN3H-StaurosporineSB20358095Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43295DAPK3CLONEDHUMAN3H-StaurosporineSU11248300Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43551PCTK1CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43807CDK2CLONEDHUMAN3H-StaurosporineBIRB-796>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44063CaMKCLONEDHUMAN3H-StaurosporineTarceva>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44319MAPK10CLONEDHUMAN3H-StaurosporineEKB-569>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44575PAK3CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44831CSNK1G1CLONEDHUMAN3H-StaurosporineBAY-43-9006>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45087MAPK12CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45599NETCLONEDHUMAN3H-NisoxetineIproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
46111Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47391D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide29Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47647GABAACLONEDHUMAN3H-RO-15-17886,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile0.73Russell MG, et al., 2006Jan 15, 2025Jan 27, 2025
47903GABAACLONEDHUMAN3H-RO-15-17886,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one1.6Chambers, MS et al., 2003Jan 15, 2025Jan 27, 2025
48671CLONEDHUMANFunctionalN-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.5Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49695D5CLONEDHUMAN3H-SCH23390Pramipexole>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
51487Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide6.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51743ARUNDEFINEDHUMANUNDEFINED(+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1530Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51999DORUNDEFINEDHUMANUNDEFINED7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine7.59Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
52255A2BUNDEFINEDHUMANUNDEFINED9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione590Drabczyńska A et al., 2007Jan 15, 2025Jan 15, 2025
52511Alpha2BUNDEFINEDHUMANUNDEFINED6,7-dimethoxy-2-((7-methoxy-2-(pyridin-2-yl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline330Hagihara K et al., 2007Jan 15, 2025Jan 15, 2025
52767D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide67Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
53023MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan0.21Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53535SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride46Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
537915-HT2AUNDEFINEDHUMANUNDEFINEDQuetiapine220Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54559A1UNDEFINEDHUMANUNDEFINED8-(4-(4-(4-Methoxyphenyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione>10000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54815D3UNDEFINEDHUMANUNDEFINEDBiphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide0.2Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
55071D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide503Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55327KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one1342Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55583DORUNDEFINEDHUMANUNDEFINED14-O-phenylpropylnaltrexone0.48Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
56095MORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.16Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56607NR3C1UNDEFINEDHUMANUNDEFINED(4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol25Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56863SLC6A4UNDEFINEDHUMANUNDEFINED(3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one1Rotella DP et al., 2009Jan 15, 2025Jan 15, 2025
57631SST3UNDEFINEDHUMANUNDEFINEDN-(1-(4-cyclopropoxy-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57887SLC6A2UNDEFINEDHUMANUNDEFINEDDESIPRAMINE2.1O'Neill DJ et al., 2010Jan 15, 2025Jan 15, 2025
581435-HT2CCLONEDHUMAN3H-MESULERGINEN-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate47.9Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58399D2CLONEDHUMAN3H-N-MethylspiporoneMRS5697>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58655M2CLONEDHUMAN3H-QNBCyclobenzaprine60Gregori-Puigjane E, et al., 2012Jan 15, 2025Jan 15, 2025
58911D3CLONEDHUMAN3H-N-Methylspiporone(+)-SYA 091069Ablordeppey S, et al., 2006Jan 15, 2025Jan 15, 2025
594235-HT1ACLONEDHUMAN3H-WAY100635Desmethyldesipramine>10000Deupree, J. et. al., 2007Jan 15, 2025Jan 15, 2025
596795-HT1ECLONEDHUMAN3H-5HTMH.MZ>10000Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
60191A3CLONEDHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyl-uronamide(1S,2R,3S,4R,5S)-4-(2-((4,5-Dimethylfuran-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide1.45Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60447GABAACLONEDHUMANFNZXLI-2860.064Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60703GABAACLONEDHUMANFNZTJH-IV-51316Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60959GABAACLONEDHUMANFNZSVO-8-677Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61215GABAACLONEDHUMANFNZZG-22450Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61471GABAACLONEDHUMANFNZRY-04779Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
617275-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine103Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
61983CLONEDHUMANUNDEFINEDgrepafloxacin>10000Bischoff ,U et al., 2000Jan 15, 2025Jan 15, 2025
62239Alpha1BCLONEDHUMAN3H-PRAZOSINTianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
62751H1Brain Frontal CortexHUMAN3H-doxepinMIANSERIN0.4Richelson, Elliott et. al, 1984Jan 15, 2025Jan 28, 2025
630075-HT2BCLONEDHUMAN3H-5-HTFenfluramine (-)5713Rothman RB, et al., 2003Jan 15, 2025Jan 15, 2025
63519NETCLONEDHUMAN3H-Nisoxetine2-Cl-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
63775CXCR3PHA/IL-2 T cellsHUMAN125I-CXCL11NBI-7433015.8Heise CE, et al., 2005Jan 15, 2025Jan 15, 2025
64543CLONEDHUMAN3H-Estradiol4-hydroxytamoxifen100Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
64799Beta1CLONEDHUMAN125I-ICYPSalmeterol6.11Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
65311GABAACLONEDHUMAN[3H] FlunitrazepamSHU-1-197Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65568GABAACLONEDHUMAN[3H] FlunitrazepamQH-II-0821.7Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65824GABAACLONEDHUMAN[3H] FlunitrazepamYT-50.6034Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66080H1CLONEDHUMAN3H-PYRILAMINETerfenadine58Pearlstein, Robert. et, al. 2003Jan 15, 2025Jan 28, 2025
66848M3CLONEDHUMAN3H-QNBN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67104H1CLONEDHUMAN3H-PYRILAMINE1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67360D4CLONEDHUMAN3H-N-Methylspiperone1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride222Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
20805-HT1DCAUDATEHUMAN3H-5HTSDZ 21-009646WAEBER ET AL., 1988Jan 15, 2025Jan 15, 2025
67616A3KIDNEYHUMANI-125-N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamideEthyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate236Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
678725-HT2ACLONEDHUMAN3H-KETANSERIN(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline1150Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
683845-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-0123.4423Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
68640recombinantHUMANUNKNOWNN-Benzyl-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
33605-HT1ACLONEDHUMAN3H-8-OH-DPATMDL 72222>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68896SST4CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH20.630957Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69152H4CLONEDHUMAN3H-N-alpha-methylhistaminehomohistamine31.6228Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
3872D1CLONEDHUMAN3H-SCH23390Quetiapine1277KONGSAMUT S, ET AL., 1996Jan 15, 2025Jan 15, 2025
69664BZPCLONEDHUMANFNZ2-CI-DPH>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
69920SLC6A3CLONEDHUMAN3H-WIN354284-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
4640SLC6A3CLONEDHUMAN3H-WIN 35,428 BINDINGBUDIPINE>10000PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48965-HT2ACLONEDHUMAN125I-DOILY 320951839BRYANT HU, ET AL., 1996Jan 15, 2025Jan 15, 2025
704325-HT1ACLONEDHUMAN3H-WAY100635MRP32156Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
51525-HT2CCLONEDHUMAN125I-DOIDOTB2.2NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70688KORCLONEDHUMAN3H-DiprenorphineBUPRENORPHINE27Olson KM, et al., 2019Jan 15, 2025Jan 28, 2025
70944KORCLONEDHUMAN3H-U69593(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
712005-HT1BCLONEDHUMAN3H-5-CTFEMPT122.5Collier TL et al 2017Jan 15, 2025Jan 15, 2025
5920Alpha2BCLONEDHUMAN3H-RAUWOLSCINESPIROXATRINE0.19BYLUND DB, ET AL., 1992Jan 15, 2025Jan 15, 2025
6176Beta2CLONEDHUMAN125I-CYPSB2040701000WARDLE KA, ET AL., 1994Jan 15, 2025Jan 28, 2025
6688D2CLONEDHUMAN3H-NEMONAPRIDEQuetiapine1000SEEMAN P, ET AL., 1995Jan 15, 2025Jan 27, 2025
7200NK2CLONEDHUMAN125I-[MePhe7]-NKBSB 223412144Sarau HM, et al., 1997Jan 15, 2025Jan 15, 2025
72736Sigma 2CLONEDHUMAN3H-Pentazocine(+)naringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
72992M5CLONEDHUMAN3H-QNBcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7712GABAACLONEDHUMAN3H-MUSCIMOLThio-4-PIOL1778.27Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7968GABAACLONEDHUMAN3H-RO-15-1788317000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8224SST1CLONEDHUMAN125I-LTT-SRIF28octreotide-Tyr32691.53Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8480SST3CLONEDHUMAN125I-LTT-SRIF28BIM 2303067.6Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8736SST2CLONEDHUMAN125I-CGP23996Somatostatin-140.09Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8992SST3CLONEDHUMAN125I-SRIF-28SMS 201-9955.01Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
74528M4CLONEDHUMAN3H-QNB(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
747845-HT1ECLONEDHUMAN3H-5-HT(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75040Alpha1BCLONEDHUMAN3H-PRAZOSIN(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9760MT1CLONEDHUMAN125I-IodomelatoninGR 12810790.4Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75296D5CLONEDHUMAN3H-SCH23390Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75552M4CLONEDHUMAN3H-QNBpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760645-HT6CLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
11040H1CLONEDHUMAN3H-MEPYRAMINEThioperamide>10000Moguilevsky N et al, 1994Jan 15, 2025Jan 15, 2025
76576M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76832M5CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11552H1BRAINHUMAN3H-PYRILAMINEVenlafaxine>10000Cusack, B et al., 1993Jan 15, 2025Jan 15, 2025
77088Sigma 2CLONEDHUMAN3H-DTG(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
11808FR. CORTEXHUMAN3H-RAUWOLSCINEPERPHENAZINE510Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
773445-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
776005-HT2ACLONEDHUMAN3H-KETANSERIN(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
778565-HT5ACLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78112Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12832Beta1CLONEDHUMAN125I-ICYPTMQ, Racemic10.47Fraundorfer PF, et al., 1994Jan 15, 2025Jan 15, 2025
78368Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78624D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
788805-HT1ACLONEDHUMAN3H-WAY1006354-Ethylthio-2,5-dimethoxyphenylbutylamine5339Ray TS 2010 Jan 15, 2025Jan 15, 2025
13600OTMyometriumHUMAN3H-OxytocinL-366,70621Pettibone DJ, et al., 1991Jan 15, 2025Jan 15, 2025
791365-HT6CLONEDHUMAN3H-LSD6-Fluoro-N,N-dimethyltryptamine25.6Ray TS 2010 Jan 15, 2025Jan 15, 2025
79392Alpha1BCLONEDHUMAN3H-PRAZOSINS,S-2c>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
79648Sigma 1CLONEDHUMAN3H-Pentazocine(+)DMT5209Ray TS 2010 Jan 15, 2025Jan 15, 2025
79904H1CLONEDHUMAN3H-PYRILAMINE3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80160CLONEDHUMAN3H-VASOPRESSIN4-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
804165-HT1ACLONEDHUMAN3H-8-OH-DPAT(E)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
806725-HT2ACLONEDHUMAN3H-KETANSERIN(5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
153925-HT1BCLONEDHUMAN3H-5HT5-CT0.89BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
809285-HT2CCLONEDHUMAN3H-MESULERGINE5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine>10000Rajagopalan R et al 2014Jan 15, 2025Jan 15, 2025
81184Alpha1DCLONEDHUMAN3H-PRAZOSINN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
814405-HT2ACLONEDHUMAN3H-KETANSERIN2-phenyl-4-[[4-(1,3-thiazol-2-yl)-1,4-diazepan-1-yl]methyl]-1,3-oxazole3324Weiss DR et al 2018Jan 15, 2025Jan 15, 2025
81696DORCLONEDHUMAN3H-DADLE(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
819525-HT2CCLONEDHUMAN3H-MESULERGINE[18F]MH.MZ71Herth MM et al 2009Jan 15, 2025Jan 15, 2025
16672M3CLONEDHUMAN3H-QNBDiphenhydramine229Bolden C, et al., 1992Jan 15, 2025Jan 15, 2025
822085-HT1BCLONEDHUMAN3H-5-CT2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one27Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82464D5CLONEDHUMAN3H-SCH23390(S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 28, 2025
171845-HT3CLONEDHUMAN3H-ZACOPRIDEMETHYLPHENIDATE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
827205-HT7CLONEDHUMAN3H-LSD(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82976A3CHO cellsHUMAN3H-PSB-118-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
17696PANC1HUMAN125I-VIPVIP [D-Ala18]15.4Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832325-HT2ACLONEDHUMAN3H-KETANSERINDMT175Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
834885-HT2CHEK293 cellsHUMAN3H-MESULERGINEMDMA>10000Simmler LD et al 2013Jan 15, 2025Jan 15, 2025
83744KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide561PDSP Certified DataJan 15, 2025Jan 28, 2025
184645-HT1BCLONEDHUMAN3H-5HT7-methoxy-1-naphthylpiperazine2Jorand-Lebrun C et al., 1997aJan 15, 2025Jan 15, 2025
84000KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-allyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84256DORCLONEDHUMAN3H-DADLE2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
18976CCK2CLONEDHUMAN125I-BH-CCK-8243630.78Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
84512MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(2,6-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19232NB-OK-1HUMAN125-[AcHis1]PacapPACAP(5-38)5Vandermeers A et al., 1992Jan 15, 2025Jan 15, 2025
84768KORCLONEDHUMAN3H-U69593±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025