96750 CORTEX RAT 3H-RAUWOLSCINE RISPERIDONE 28.2 Huang L et al 2020 Jan 15, 2025 Jul 30, 2025
96751 CORTEX RAT 3H-RAUWOLSCINE N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide 193 Huang L et al 2020 Jan 15, 2025 Jul 30, 2025
96752 H1 CEREBELLUM GUINEA PIG [3H]mepyramine N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 2143 Huang L et al 2020 Jan 15, 2025 Jan 28, 2025
96753 H1 CEREBELLUM GUINEA PIG [3H]mepyramine RISPERIDONE 49.3 Huang L et al 2020 Jan 15, 2025 Jan 28, 2025
96754 5-HT2C CORTEX RAT [3H]mesulergine N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 1987 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96755 5-HT2C CORTEX RAT [3H]mesulergine RISPERIDONE 39.1 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96756 5-HT2C CORTEX RAT [3H]mesulergine N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide 186 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96757 CORTEX RAT [3H]prazosin N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 3296 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96758 CORTEX RAT [3H]prazosin RISPERIDONE 21.9 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96759 CORTEX RAT [3H]prazosin N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide 195 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96760 D1 CLONED HUMAN [3H]SCH23390 ARIPIPRAZOLE 310 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96761 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96762 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96763 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96764 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96765 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96766 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 4800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96767 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 3800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96768 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96769 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96770 D1 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96771 D1 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96772 D1 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96773 D1 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96774 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96775 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96776 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96777 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 7700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96778 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96779 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 8800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96780 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96781 D2 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 0.52 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96782 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 1 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96783 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 1.1 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96784 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 5.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96785 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 3.4 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96786 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.6 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96787 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 0.91 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96788 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.98 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96789 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 29 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96790 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96791 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 5300 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96792 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 8300 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96793 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96794 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96795 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 780 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96796 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 630 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96797 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 6400 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96798 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 3200 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96799 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96800 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 120 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96801 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 360 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96802 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96803 D2 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 0.38 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96804 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 0.58 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96805 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 0.73 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96806 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96807 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 1.3 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96808 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.54 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96809 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 0.67 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96810 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.95 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96811 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 16 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96812 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.1 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96813 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1200 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96814 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1800 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96815 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 8900 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96816 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6000 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96817 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 250 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96818 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 200 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96819 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 3400 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96820 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 1500 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96821 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 480 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96822 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 35 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96823 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 5700 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96824 D3 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96825 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 2.3 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96826 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 1.2 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96827 D3 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 24 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96828 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96829 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96830 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 0.35 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96831 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.39 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96832 D3 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 30 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96833 D3 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 35 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96834 D3 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96835 D3 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 160 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96836 D3 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 510 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96837 D3 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 110 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96838 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 380 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96839 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 48 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96840 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 42 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96841 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 790 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96842 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 420 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96843 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 5.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96844 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 3.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96845 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 2800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96846 D4 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 63 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96847 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 41 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96848 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 10 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96849 D4 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 130 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96850 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 11 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96851 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 31 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96852 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2.3 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96853 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96854 D4 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 140 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96855 D4 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 62 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96856 D4 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 6100 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96857 D4 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 440 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96858 D4 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96859 D4 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96860 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 560 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96861 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 59 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96862 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 4900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96863 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 2600 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96864 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 7600 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96865 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 880 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96866 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 210 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96867 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96868 D5 CLONED HUMAN [3H]SCH23390 ARIPIPRAZOLE 1600 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96869 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96870 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 7700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96871 D5 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96872 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96873 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96874 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96875 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96876 D5 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96877 D5 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96878 D5 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96879 D5 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96880 D5 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96881 D5 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96882 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96883 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96884 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96885 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96886 D5 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96887 D5 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96888 D5 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96889 5-HT1A CLONED PIG [3H]WAY100635 ARIPIPRAZOLE 88 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96890 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 14 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96891 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 21 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96892 5-HT1A CLONED PIG [3H]WAY100635 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 4.7 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96893 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 13 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96894 5-HT1A CLONED HUMAN [3H]WAY100635 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 33 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96895 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 12 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96896 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 19 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96897 5-HT1A CLONED PIG [3H]WAY100635 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 23 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96898 5-HT1A CLONED PIG [3H]WAY100635 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 16 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96899 5-HT1A CLONED PIG [3H]WAY100635 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96900 5-HT1A CLONED PIG [3H]WAY100635 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 4500 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96901 5-HT1A CLONED PIG [3H]WAY100635 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96902 5-HT1A CLONED PIG [3H]WAY100635 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96903 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 620 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96904 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1700 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96905 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96906 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 1600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96907 5-HT1A CLONED PIG [3H]WAY100635 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96908 5-HT1A CLONED HUMAN [3H]WAY100635 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 180 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96909 5-HT1A CLONED PIG [3H]WAY100635 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96910 5-HT1A CLONED PIG [3H]WAY100635 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 5800 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96911 5-HT2A CLONED HUMAN [3H]ketanserin ARIPIPRAZOLE 3.6 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96912 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96913 5-HT2A CLONED HUMAN [3H]ketanserin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 1000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96914 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96915 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 5400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96916 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96917 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 880 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96918 5-HT2A CLONED HUMAN [3H]ketanserin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96919 5-HT2A CLONED HUMAN [3H]ketanserin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 980 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96920 5-HT2A CLONED HUMAN [3H]ketanserin 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96921 5-HT2A CLONED HUMAN [3H]ketanserin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96922 5-HT2A CLONED HUMAN [3H]ketanserin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96923 5-HT2A CLONED HUMAN [3H]ketanserin 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 3600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96924 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96925 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96926 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 6400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96927 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 2100 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96928 5-HT2A CLONED HUMAN [3H]ketanserin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96929 5-HT2A CLONED HUMAN [3H]ketanserin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 3700 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96930 5-HT2A CLONED HUMAN [3H]ketanserin 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96931 CLONED PIG [3H]prazosin ARIPIPRAZOLE 17 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96932 CLONED PIG [3H]prazosin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 49 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96933 CLONED PIG [3H]prazosin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 11 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96934 CLONED PIG [3H]prazosin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 160 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96935 CLONED PIG [3H]prazosin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 29 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96936 CLONED PIG [3H]prazosin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 39 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96937 CLONED PIG [3H]prazosin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 13 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96938 CLONED PIG [3H]prazosin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 17 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96939 CLONED PIG [3H]prazosin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 120 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96940 CLONED PIG [3H]prazosin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 89 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96941 CLONED PIG [3H]prazosin 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96942 CLONED PIG [3H]prazosin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 4200 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96943 CLONED PIG [3H]prazosin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96944 CLONED PIG [3H]prazosin 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 4200 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96945 CLONED PIG [3H]prazosin 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1500 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96946 CLONED PIG [3H]prazosin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1500 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96947 CLONED PIG [3H]prazosin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96948 CLONED PIG [3H]prazosin 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 2400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96949 CLONED PIG [3H]prazosin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96950 CLONED PIG [3H]prazosin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 160 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96951 CLONED PIG [3H]prazosin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 900 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96952 CLONED PIG [3H]prazosin 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96953 M2 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96954 M3 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96955 M4 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96956 M5 CLONED HUMAN [3H]QNB 3′′-F-DPPy 913 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96957 MOR CLONED HUMAN [3H]DAMGO 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96958 NET CLONED HUMAN [3H]Nisoxetine 3′′-F-DPPy 189 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96959 PBR CLONED HUMAN [3H]PK11195 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96960 SERT CLONED HUMAN [3H]Citalopram 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96961 Sigma 1 CLONED HUMAN [3H]Pentazocine 3′′-F-DPPy 124 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96962 Sigma 2 CLONED HUMAN [3H]DTG 3′′-F-DPPy 741 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96963 NMDA FOREBRAIN RAT [3H]MK-801 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96964 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96965 5-HT1B CLONED HUMAN [3H]GR127543 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96966 5-HT1D CLONED HUMAN [3H]GR127543 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96967 5-HT1E CLONED HUMAN [3H]5-HT 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96968 5-HT2A CLONED HUMAN [3H]ketanserin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96969 5-HT2C CLONED HUMAN [3H]mesulergine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96970 5-HT3 CLONED HUMAN [3H]LY278584 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96971 Alpha1A CLONED HUMAN [3H]prazosin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96972 Alpha1B CLONED HUMAN [3H]prazosin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96973 Alpha1D CLONED HUMAN [3H]prazosin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96974 Alpha2A CLONED HUMAN [3H]Clonidine 4′′-F-DPPy 86 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96975 Alpha2C CLONED HUMAN [3H]Clonidine 4′′-F-DPPy 101 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96976 Beta1 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96977 Beta2 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96978 Beta3 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96979 D1 CLONED HUMAN [3H]SCH23390 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96980 D2 CLONED HUMAN [3H]N-methylspiperone 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96981 D3 CLONED HUMAN [3H]N-methylspiperone 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96982 D4 CLONED HUMAN [3H]N-methylspiperone 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96983 D5 CLONED HUMAN [3H]SCH23390 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96984 DAT CLONED HUMAN [3H]WIN35428 4′′-F-DPPy 231 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96985 DOR CLONED HUMAN [3H]DADLE 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96986 GABAA BRAIN RAT [3H]-Muscimol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
96987 H1 CLONED HUMAN [3H]Pyrilamine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96988 5-HT1D CLONED HUMAN [3H]Tiotidine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96989 H3 CLONED HUMAN [3H]-alpha-methylhistamine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96990 H4 CLONED HUMAN [3H]Histamine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96991 KOR CLONED HUMAN [3H]U69593 4′′-F-DPPy 4460 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96992 M1 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96993 M2 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96994 M4 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96995 M5 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96996 MOR CLONED HUMAN [3H]DAMGO 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96997 NET CLONED HUMAN [3H]Nisoxetine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96998 PBR CLONED HUMAN [3H]PK11195 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96999 SERT CLONED HUMAN [3H]Citalopram 4′′-F-DPPy 352 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97000 Sigma 1 CLONED HUMAN [3H]Pentazocine 4′′-F-DPPy 139 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97001 Sigma 2 CLONED HUMAN [3H]DTG 4′′-F-DPPy 321 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97002 NMDA FOREBRAIN RAT [3H]MK-801 PCP 57.9 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97003 NMDA FOREBRAIN RAT [3H]MK-801 PCP 22.1 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97004 NMDA FOREBRAIN RAT [3H]MK-801 Diphenidine 18.2 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97005 NMDA FOREBRAIN RAT [3H]MK-801 Ketamine 323.9 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97006 NMDA FOREBRAIN RAT [3H]MK-801 (+)-MK-801 2.5 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97007 NMDA FOREBRAIN RAT [3H]MK-801 Memantine 378.4 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97008 NMDA FOREBRAIN RAT [3H]MK-801 DPPy 280 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97009 NMDA FOREBRAIN RAT [3H]MK-801 Fluorolintane (2-F-DPPy) 87.92 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97010 NMDA FOREBRAIN RAT [3H]MK-801 3-F-DPPy 632.64 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97011 NMDA FOREBRAIN RAT [3H]MK-801 4-F-DPPy 953.37 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97012 NMDA FOREBRAIN RAT [3H]MK-801 2′′-F-DPPy 609.74 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97013 NMDA FOREBRAIN RAT [3H]MK-801 3′′-F-DPPy 261.84 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97014 NMDA FOREBRAIN RAT [3H]MK-801 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97015 NMDA FOREBRAIN RAT [3H]MK-801 Fluorolintane (2-F-DPPy) 88 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97016 5-HT1A CLONED HUMAN [3H]8-OH-DPAT Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97017 5-HT1B CLONED HUMAN [3H]GR127543 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97018 5-HT1D CLONED HUMAN [3H]GR127543 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97019 5-HT1E CLONED HUMAN [3H]5-HT Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97020 5-HT2A CLONED HUMAN [3H]ketanserin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97021 5-HT2C CLONED HUMAN [3H]mesulergine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97022 5-HT3 CLONED HUMAN [3H]LY278584 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97023 Alpha1A CLONED HUMAN [3H]prazosin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97024 Alpha1B CLONED HUMAN [3H]prazosin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97025 Alpha2A CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) 829 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97026 Alpha2B CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) 388 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97027 Alpha2C CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97028 Beta1 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97029 Beta2 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97030 Beta3 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97031 D1 CLONED HUMAN [3H]SCH23390 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97032 D2 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97033 D3 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97034 D4 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97035 D5 CLONED HUMAN [3H]SCH23390 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97036 DAT CLONED HUMAN [3H]WIN35428 Fluorolintane (2-F-DPPy) 327 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97037 DOR CLONED HUMAN [3H]DADLE Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97038 GABAA BRAIN RAT [3H]-Muscimol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97039 H1 CLONED HUMAN [3H]Pyrilamine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97040 5-HT1D CLONED HUMAN [3H]Tiotidine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97041 H4 CLONED HUMAN [3H]Histamine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97042 KOR CLONED HUMAN [3H]U69593 Fluorolintane (2-F-DPPy) 1278 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97043 M1 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) 1597 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97044 M2 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97045 M3 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97046 M4 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97047 M5 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) 556 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97048 MOR CLONED HUMAN [3H]DAMGO Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97049 NET CLONED HUMAN [3H]Nisoxetine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97050 PBR CLONED HUMAN [3H]PK11195 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97051 SERT CLONED HUMAN [3H]Citalopram Fluorolintane (2-F-DPPy) 4115 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97052 Sigma 1 CLONED HUMAN [3H]Pentazocine Fluorolintane (2-F-DPPy) 110 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97053 NMDA FOREBRAIN RAT [3H]MK-801 3-F-DPPy 633 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97054 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97055 5-HT1B CLONED HUMAN [3H]GR127543 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97056 5-HT1D CLONED HUMAN [3H]GR127543 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97057 5-HT1E CLONED HUMAN [3H]5-HT 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97058 5-HT2A CLONED HUMAN [3H]ketanserin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97059 5-HT2C CLONED HUMAN [3H]mesulergine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97060 5-HT3 CLONED HUMAN [3H]LY278584 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97061 Alpha1A CLONED HUMAN [3H]prazosin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97062 Alpha1B CLONED HUMAN [3H]prazosin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97063 Alpha1D CLONED HUMAN [3H]prazosin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97064 Alpha2A CLONED HUMAN [3H]Clonidine 3-F-DPPy 732 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97065 Alpha2B CLONED HUMAN [3H]Clonidine 3-F-DPPy 129 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97066 Alpha2C CLONED HUMAN [3H]Clonidine 3-F-DPPy 333 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97067 Beta1 CLONED HUMAN [125I]Iodopindolol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97068 Beta2 CLONED HUMAN 3-F-DPPy [125I]Iodopindolol >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97069 Beta3 CLONED HUMAN [125I]Iodopindolol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97070 D1 CLONED HUMAN [3H]SCH23390 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97071 D2 CLONED HUMAN [3H]N-methylspiperone 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97072 D3 CLONED HUMAN [3H]N-methylspiperone 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97073 D4 CLONED HUMAN [3H]N-methylspiperone 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97074 D5 CLONED HUMAN [3H]SCH23390 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97075 DAT CLONED HUMAN [3H]WIN35428 3-F-DPPy 12 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97076 DOR CLONED HUMAN [3H]DADLE 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97077 GABAA BRAIN RAT [3H]-Muscimol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97078 H1 CLONED HUMAN [3H]Pyrilamine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97079 5-HT1D CLONED HUMAN [3H]Tiotidine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97080 H3 CLONED HUMAN [3H]-alpha-methylhistamine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97081 H4 CLONED HUMAN [3H]Histamine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97082 KOR CLONED HUMAN [3H]U69593 3-F-DPPy 1583 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97083 M1 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97084 M2 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97085 M3 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97086 M5 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97087 MOR CLONED HUMAN [3H]DAMGO 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97088 NET CLONED HUMAN [3H]Nisoxetine 3-F-DPPy 192 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97089 PBR CLONED HUMAN [3H]PK11195 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97090 SERT CLONED HUMAN [3H]Citalopram 3-F-DPPy 1202 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97091 Sigma 1 CLONED HUMAN [3H]Pentazocine 3-F-DPPy 193 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97092 Sigma 2 CLONED HUMAN [3H]DTG 3-F-DPPy 1934 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97093 NMDA FOREBRAIN RAT [3H]MK-801 4-F-DPPy 953 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97094 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97095 5-HT1B CLONED HUMAN [3H]GR127543 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97096 5-HT1D CLONED HUMAN [3H]GR127543 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97097 5-HT1E CLONED HUMAN [3H]5-HT 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97098 5-HT2C CLONED HUMAN [3H]mesulergine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97099 5-HT3 CLONED HUMAN [3H]LY278584 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97100 Alpha1A CLONED HUMAN [3H]prazosin 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97101 Alpha1B CLONED HUMAN [3H]prazosin 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97102 Alpha1D CLONED HUMAN [3H]prazosin 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97103 Alpha2A CLONED HUMAN [3H]Clonidine 4-F-DPPy 1401 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97104 Alpha2B CLONED HUMAN [3H]Clonidine 4-F-DPPy 1242 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97105 Beta2 CLONED HUMAN [125I]Iodopindolol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97106 Beta3 CLONED HUMAN [125I]Iodopindolol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97107 D1 CLONED HUMAN [3H]SCH23390 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97108 D2 CLONED HUMAN [3H]N-methylspiperone 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97109 D3 CLONED HUMAN [3H]N-methylspiperone 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97110 D4 CLONED HUMAN [3H]N-methylspiperone 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97111 D5 CLONED HUMAN [3H]SCH23390 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97112 DAT CLONED HUMAN [3H]WIN35428 4-F-DPPy 140 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97113 DOR CLONED HUMAN [3H]DADLE 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97114 GABAA BRAIN RAT [3H]-Muscimol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97115 H1 CLONED HUMAN [3H]Pyrilamine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97116 5-HT1D CLONED HUMAN [3H]Tiotidine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97117 H3 CLONED HUMAN [3H]-alpha-methylhistamine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97118 H4 CLONED HUMAN [3H]Histamine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97119 KOR CLONED HUMAN [3H]U69593 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97120 M1 CLONED HUMAN [3H]QNB 4-F-DPPy 1900 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97121 M2 CLONED HUMAN [3H]QNB 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97122 M3 CLONED HUMAN [3H]QNB 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97123 M5 CLONED HUMAN [3H]QNB 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97124 MOR CLONED HUMAN [3H]DAMGO 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97125 NET CLONED HUMAN [3H]Nisoxetine 4-F-DPPy 249 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97126 PBR CLONED HUMAN [3H]PK11195 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97127 SERT CLONED HUMAN [3H]Citalopram 4-F-DPPy 681 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97128 Sigma 1 CLONED HUMAN [3H]Pentazocine 4-F-DPPy 386 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97129 Sigma 2 CLONED HUMAN [3H]DTG 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97130 NMDA FOREBRAIN RAT [3H]MK-801 2′′-F-DPPy 610 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97131 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97132 5-HT1B CLONED HUMAN [3H]GR127543 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97133 5-HT1D CLONED HUMAN [3H]GR127543 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97134 5-HT1E CLONED HUMAN [3H]5-HT 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97135 5-HT2A CLONED HUMAN [3H]ketanserin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97136 5-HT2C CLONED HUMAN [3H]mesulergine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97137 5-HT3 CLONED HUMAN [3H]LY278584 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97138 Alpha1A CLONED HUMAN [3H]prazosin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97139 Alpha1B CLONED HUMAN [3H]prazosin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97140 Alpha1D CLONED HUMAN [3H]prazosin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97141 Alpha2A CLONED HUMAN [3H]Clonidine 2′′-F-DPPy 307 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97142 Alpha2B CLONED HUMAN [3H]Clonidine 2′′-F-DPPy 89 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97143 Alpha2C CLONED HUMAN [3H]Clonidine 2′′-F-DPPy 214 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97144 Beta1 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97145 Beta2 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97146 Beta3 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97147 D1 CLONED HUMAN [3H]SCH23390 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97148 D2 CLONED HUMAN [3H]N-methylspiperone 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97149 D3 CLONED HUMAN [3H]N-methylspiperone 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97150 D4 CLONED HUMAN [3H]N-methylspiperone 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97151 D5 CLONED HUMAN [3H]SCH23390 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97152 DAT CLONED HUMAN [3H]WIN35428 2′′-F-DPPy 85 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97153 DOR CLONED HUMAN [3H]DADLE 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97154 GABAA BRAIN RAT [3H]-Muscimol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97155 H1 CLONED HUMAN [3H]Pyrilamine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97156 5-HT1D CLONED HUMAN [3H]Tiotidine 2′′-F-DPPy 2194 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97157 H3 CLONED HUMAN [3H]-alpha-methylhistamine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97158 H4 CLONED HUMAN [3H]Histamine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97159 KOR CLONED HUMAN [3H]U69593 2′′-F-DPPy 642 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97160 M1 CLONED HUMAN [3H]QNB 2′′-F-DPPy 1660 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97161 M2 CLONED HUMAN [3H]QNB 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97162 M4 CLONED HUMAN [3H]QNB 2′′-F-DPPy 576 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97163 M5 CLONED HUMAN [3H]QNB 2′′-F-DPPy 489 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97164 MOR CLONED HUMAN [3H]DAMGO 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97165 NET CLONED HUMAN [3H]Nisoxetine 2′′-F-DPPy 215 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97166 PBR CLONED HUMAN [3H]PK11195 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97167 SERT CLONED HUMAN [3H]Citalopram 2′′-F-DPPy 661 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97168 Sigma 1 CLONED HUMAN [3H]Pentazocine 2′′-F-DPPy 146 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97169 Sigma 2 CLONED HUMAN [3H]DTG 2′′-F-DPPy 712 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97170 NMDA CLONED HUMAN [3H]MK-801 3′′-F-DPPy 262 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97171 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 3′′-F-DPPy 534 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97172 5-HT1B CLONED HUMAN [3H]GR127543 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97173 5-HT1D CLONED HUMAN [3H]GR127543 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97174 5-HT1E CLONED HUMAN [3H]5-HT 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97175 5-HT2A CLONED HUMAN [3H]ketanserin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97176 5-HT2C CLONED HUMAN [3H]mesulergine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97177 5-HT3 CLONED HUMAN [3H]LY278584 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97178 Alpha1A CLONED HUMAN [3H]prazosin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97179 Alpha1B CLONED HUMAN [3H]prazosin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97180 Alpha1D CLONED HUMAN [3H]prazosin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97181 Alpha2A CLONED HUMAN [3H]Clonidine 3′′-F-DPPy 915 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97182 Alpha2B CLONED HUMAN [3H]Clonidine 3′′-F-DPPy 307 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97183 Alpha2C CLONED HUMAN [3H]Clonidine 3′′-F-DPPy 1159 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97184 Beta1 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97185 Beta2 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97186 Beta3 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97187 D1 CLONED HUMAN [3H]SCH23390 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97188 D2 CLONED HUMAN 3′′-F-DPPy [3H]N-methylspiperone >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97189 D3 CLONED HUMAN [3H]N-methylspiperone 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97190 D4 CLONED HUMAN [3H]N-methylspiperone 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97191 D5 CLONED HUMAN [3H]SCH23390 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97192 DAT CLONED HUMAN [3H]WIN35428 3′′-F-DPPy 103 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97193 DOR CLONED HUMAN [3H]DADLE 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97194 GABAA BRAIN RAT [3H]-Muscimol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97195 H1 CLONED HUMAN [3H]Pyrilamine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97196 5-HT1D CLONED HUMAN [3H]Tiotidine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97197 H3 CLONED HUMAN [3H]-alpha-methylhistamine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97198 H4 CLONED HUMAN [3H]Histamine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97199 KOR CLONED HUMAN [3H]U69593 3′′-F-DPPy 1435 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97200 M1 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97201 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5200 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97202 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 9.5 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97203 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 740 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97204 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97205 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 4.2 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97206 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97207 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 18 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97208 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 26 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97209 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine  63 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97210 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-methoxyphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine  28 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97211 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 117 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97212 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 84 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97213 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 160 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97214 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl 16 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97215 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 180 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97216 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 400 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97217 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl >10000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97218 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 910 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97219 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 22 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97220 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 5.2 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97221 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 97 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97222 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 450 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97223 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 240 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97224 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 600 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97225 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 33 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97226 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 2600 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97227 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 71 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97228 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 180 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97229 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 17 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97230 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 390 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97231 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 5.9 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97232 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 190 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97233 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 34 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97234 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 740 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97235 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 5.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97236 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl 51 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97237 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine AS-19 12 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97238 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (R)-8-OH-DPAT 48 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97239 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (S)-8-OH-DPAT 1000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97240 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine BUSPIRONE 840 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97241 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1100 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97242 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 6.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97243 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97244 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 4 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97245 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 14 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97246 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 7.5 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97247 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 23 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97248 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 82 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97249 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine  180 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97250 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 73 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97251 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 30 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97252 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 19 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97253 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 190 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97254 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl 33 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97255 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 230 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97256 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 2200 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97257 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl >10000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97258 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 2230 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97259 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 130 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97260 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 64 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97261 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 650 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97262 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1400 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97263 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 98 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97264 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 550 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97265 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 24 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97266 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5600 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97267 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 33 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97268 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 150 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97269 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 4.5 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97270 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 130 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97271 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 0.64 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97272 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 210 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97273 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5.9 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97274 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 92 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97275 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 1.8 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97276 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl 1.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97277 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine AS-19 240 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97278 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (R)-8-OH-DPAT 7.1 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97279 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (S)-8-OH-DPAT 7.6 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97280 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine BUSPIRONE 50 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97281 MOR CLONED HUMAN [3H]diprenorphine SRI-22138 7.55 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97282 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 23.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97283 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 138 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97284 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 2.33 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97285 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 171 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97286 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 370 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97287 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 235 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97288 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 24.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97289 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 191 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97290 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97291 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 135 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97292 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 249 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97293 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 61.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97294 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 91.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97295 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 148 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97296 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 12.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97297 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.97 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97298 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 15.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97299 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 4.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97300 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol 56.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97301 MOR CLONED HUMAN [3H]diprenorphine N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 141 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97302 MOR CLONED HUMAN [3H]diprenorphine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 337 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97303 MOR CLONED HUMAN [3H]diprenorphine N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 159 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97304 MOR CLONED HUMAN [3H]diprenorphine NALOXONE 59.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97305 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 14.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97306 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 105 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97307 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 82.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97308 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 47.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97309 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 1.05 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97310 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 10.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97311 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 66.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97312 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 47.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97313 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 88.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97314 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 121 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97315 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 3.79 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97316 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 99.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97317 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.18 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97318 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.37 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97319 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 819 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97320 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 799 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97321 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.96 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97322 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.82 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97323 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 70.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97324 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 95.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97325 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.99 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97326 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 92.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97327 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol 499 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97328 DOR CLONED HUMAN [3H]diprenorphine SRI-22138 2.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97329 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 19.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97330 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 20.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97331 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.42 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97332 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 53.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97333 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 7.52 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97334 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 97.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97335 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 26.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97336 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 34.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97337 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.78 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97338 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 64.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97339 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 93.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97340 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97341 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 48 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97342 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 30.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97343 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 8.37 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97344 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 69.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97345 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 68.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97346 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 53.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97347 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol 14 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97348 DOR CLONED HUMAN [3H]diprenorphine N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 3333 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97349 DOR CLONED HUMAN [3H]diprenorphine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 3333 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97350 DOR CLONED HUMAN [3H]diprenorphine N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 394 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97351 DOR CLONED HUMAN [3H]diprenorphine NALOXONE 98.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97352 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 0.169 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97353 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 6.52 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97354 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 30.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97355 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.43 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97356 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 63.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97357 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97358 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 22.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97359 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.18 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97360 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 40.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97361 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 257 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97362 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 7.96 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97363 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 64.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97364 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 8.12 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97365 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.24 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97366 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 172 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97367 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 32.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97368 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.89 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97369 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97370 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 11 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97371 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 12.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97372 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 64.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97373 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 14.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97374 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol 7.48 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97375 KOR CLONED HUMAN [3H]diprenorphine SRI-22138 60.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97376 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 132 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97377 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 75.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97378 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.69 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97379 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 35.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97380 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 71.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97381 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 152 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97382 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 17.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97383 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 102 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97384 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 129 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97385 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 175 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97386 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 134 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97387 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 126 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97388 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 103 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97389 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 140 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97390 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 18.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97391 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 7.96 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97392 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 11.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97393 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.18 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97394 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol 22.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97395 KOR CLONED HUMAN [3H]diprenorphine N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 13.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97396 KOR CLONED HUMAN [3H]diprenorphine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 608 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97397 KOR CLONED HUMAN [3H]diprenorphine N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 15.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97398 KOR CLONED HUMAN [3H]diprenorphine U50,488 31.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97399 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 13.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97400 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 19.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97401 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 27.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97402 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 15.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97403 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 0.51 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97404 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.62 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97405 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 30.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97406 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 24.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97407 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 19.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97408 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97409 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 8.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97410 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 23.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97411 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 14.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97412 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 10.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97413 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 21.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97414 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 31 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97415 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97416 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 21.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97417 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 60.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97418 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 57.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97419 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 24.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97420 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 57.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97421 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol 252 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97422 A1 CLONED HUMAN [3H]DPCPX ISAM-141 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97423 A1 CLONED HUMAN [3H]DPCPX ISAM-142 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97424 A1 CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97425 A1 CLONED HUMAN [3H]DPCPX propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97426 A1 CLONED HUMAN [3H]DPCPX ISAM-134 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97427 A1 CLONED HUMAN [3H]DPCPX ISAM-140 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97428 A1 CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97429 A1 CLONED HUMAN [3H]DPCPX DPCPX 2.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97430 A1 CLONED HUMAN [3H]DPCPX ZM241385 683 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97431 A1 CLONED HUMAN [3H]DPCPX Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97432 A1 CLONED HUMAN [3H]DPCPX Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97433 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97434 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97435 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97436 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97437 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97438 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97439 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97440 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97441 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97442 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97443 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97444 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97445 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97446 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97447 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97448 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97449 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97450 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97451 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 14.8 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97452 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 8.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97453 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97454 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97455 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 20.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97456 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97457 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97458 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97459 A1 CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97460 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97461 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97462 A1 CLONED HUMAN [3H]DPCPX (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97463 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97464 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97465 A1 CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97466 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97467 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97468 A1 CLONED HUMAN [3H]DPCPX ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97469 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 233 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97470 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 301 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97471 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97472 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97473 A2A CLONED HUMAN [3H]ZM-241385 ISAM-141 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97474 A2A CLONED HUMAN [3H]ZM-241385 ISAM-142 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97475 A2A CLONED HUMAN [3H]ZM-241385 ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97476 A2A CLONED HUMAN [3H]ZM-241385 propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97477 A2A CLONED HUMAN [3H]ZM-241385 ISAM-134 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97478 A2A CLONED HUMAN [3H]ZM-241385 ISAM-140 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97479 A2A CLONED HUMAN [3H]ZM-241385 ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97480 A2A CLONED HUMAN Leucyl-3H-NC DPCPX 157 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97481 A2A CLONED HUMAN [3H]ZM-241385 ZM241385 1.9 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97482 A2A CLONED HUMAN [3H]ZM-241385 Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97483 A2A CLONED HUMAN [3H]ZM-241385 Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97484 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97485 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97486 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97487 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97488 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97489 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97490 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97491 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97492 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97493 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97494 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97495 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97496 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97497 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97498 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97499 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97500 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97501 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97502 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97503 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97504 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97505 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97506 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97507 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97508 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97509 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97510 A2A CLONED HUMAN [3H]ZM-241385 ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97511 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97512 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 5 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97513 A2A CLONED HUMAN [3H]ZM-241385 (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97514 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97515 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97516 A2A CLONED HUMAN [3H]ZM-241385 ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97517 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97518 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97519 A2A CLONED HUMAN [3H]ZM-241385 ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97520 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 282 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97521 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97522 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97523 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97524 A2B CLONED HUMAN [3H]DPCPX ISAM-141 20.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97525 A2B CLONED HUMAN [3H]DPCPX ISAM-142 11.4 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97526 A2B CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 29.71 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97527 A2B CLONED HUMAN [3H]DPCPX propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  29.34 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97528 A2B CLONED HUMAN [3H]DPCPX ISAM-134 12.03 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97529 A2B CLONED HUMAN [3H]DPCPX ISAM-140 3.49 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97530 A2B CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 484.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97531 A2B CLONED HUMAN [3H]DPCPX propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  371.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97532 A2B CLONED HUMAN [3H]DPCPX DPCPX 73.24 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97533 A2B CLONED HUMAN [3H]DPCPX ZM241385 65.7 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97534 A2B CLONED HUMAN [3H]DPCPX Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97535 A2B CLONED HUMAN [3H]DPCPX Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97536 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97537 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97538 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97539 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97540 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 449.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97541 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 517.1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97542 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 49.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97543 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 31.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97544 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97545 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97546 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 789 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97547 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 721 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97548 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 707 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97549 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1104 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97550 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 23.4 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97551 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 29.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97552 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97553 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 278 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97554 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 92.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97555 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 340 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97556 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 714 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97557 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1031 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97558 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 98.7 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97559 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 175 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97560 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 769 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97561 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 708 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97562 A2B CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 388 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97563 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 753 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97564 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 402 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97565 A2B CLONED HUMAN [3H]DPCPX (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97566 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 8.1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97567 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 43.41 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97568 A2B CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97569 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97570 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97571 A2B CLONED HUMAN [3H]DPCPX ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97572 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 508 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97573 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97574 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 215 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97575 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 68.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97576 A3 CLONED HUMAN [3H]NECA ISAM-141 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97577 A3 CLONED HUMAN [3H]NECA ISAM-142 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97578 A3 CLONED HUMAN [3H]NECA ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97579 A3 CLONED HUMAN [3H]NECA propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97580 A3 CLONED HUMAN [3H]NECA ISAM-134 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97581 A3 CLONED HUMAN [3H]NECA ISAM-140 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97582 A3 CLONED HUMAN [3H]NECA ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97583 A3 CLONED HUMAN [3H]NECA DPCPX 1722 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97584 A3 CLONED HUMAN [3H]NECA ZM241385 863 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97585 A3 CLONED HUMAN [3H]NECA Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97586 A3 CLONED HUMAN [3H]NECA Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97587 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97588 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97589 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97590 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97591 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97592 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97593 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97594 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97595 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97596 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97597 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97598 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97599 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97600 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97601 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97602 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97603 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97604 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97605 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97606 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97607 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97608 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97609 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97610 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97611 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97612 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97613 A3 CLONED HUMAN [3H]NECA ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97614 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97615 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97616 A3 CLONED HUMAN [3H]NECA (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97617 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97618 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97619 A3 CLONED HUMAN [3H]NECA ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97620 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97621 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97622 A3 CLONED HUMAN [3H]NECA ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97623 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 418 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97624 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97625 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97626 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97627 SST1 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97628 SST2 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.04 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97629 SST3 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97630 SST4 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 1.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97631 SST5 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97632 SST1 CLONED HUMAN 125I-LTT-SST-28 L-363,377 5664 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97633 SST2 CLONED HUMAN 125I-LTT-SST-28 L-363,377 0.5 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97634 SST3 CLONED HUMAN 125I-LTT-SST-28 L-363,377 3072 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97635 SST4 CLONED HUMAN 125I-LTT-SST-28 L-363,377 >10000 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97636 SST5 CLONED HUMAN 125I-LTT-SST-28 L-363,377 2009 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97637 SST1 CLONED HUMAN 125I-LTT-SST-28 L-797,591 1.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97638 SST2 CLONED HUMAN 125I-LTT-SST-28 L-797,591 1875 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97639 SST3 CLONED HUMAN 125I-LTT-SST-28 L-797,591 2240 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97640 SST4 CLONED HUMAN 125I-LTT-SST-28 L-797,591 170 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97641 SST5 CLONED HUMAN 125I-LTT-SST-28 L-797,591 3600 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97642 SST1 CLONED HUMAN 125I-LTT-SST-28 L-779,976 2760 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97643 SST2 CLONED HUMAN 125I-LTT-SST-28 L-779,976 0.05 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97644 SST3 CLONED HUMAN 125I-LTT-SST-28 L-779,976 729 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97645 SST4 CLONED HUMAN 125I-LTT-SST-28 L-779,976 310 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97646 SST5 CLONED HUMAN 125I-LTT-SST-28 L-779,976 4260 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97647 SST1 CLONED HUMAN 125I-LTT-SST-28 L-796,778 1255 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97648 SST2 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97649 SST3 CLONED HUMAN 125I-LTT-SST-28 L-796,778 24 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97650 SST4 CLONED HUMAN 125I-LTT-SST-28 L-796,778 8650 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97651 SST5 CLONED HUMAN 125I-LTT-SST-28 L-796,778 1200 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97652 SST1 CLONED HUMAN 125I-LTT-SST-28 L-803,087 199 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97653 SST2 CLONED HUMAN 125I-LTT-SST-28 L-803,087 4720 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97654 SST3 CLONED HUMAN 125I-LTT-SST-28 L-803,087 1280 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97655 SST4 CLONED HUMAN 125I-LTT-SST-28 L-803,087 0.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97656 SST5 CLONED HUMAN 125I-LTT-SST-28 L-803,087 3880 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97657 SST1 CLONED HUMAN 125I-LTT-SST-28 L-817,818 3.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97658 SST2 CLONED HUMAN 125I-LTT-SST-28 L-817,818 52 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97659 SST3 CLONED HUMAN 125I-LTT-SST-28 L-817,818 64 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97660 SST4 CLONED HUMAN 125I-LTT-SST-28 L-817,818 82 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97661 SST5 CLONED HUMAN 125I-LTT-SST-28 L-817,818 0.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97662 SST1 CLONED HUMAN Functional L-797,591 3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97663 SST2 CLONED HUMAN Functional L-779,976 0.05 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97664 SST4 CLONED HUMAN Functional L-803,087 0.2 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97665 SST5 CLONED HUMAN Functional L-817,818 1.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97666 SST3 CLONED HUMAN Functional L-796,778 18 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97667 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 4-quinolone 122 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97668 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-ethyl-4-quinolone 20 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97669 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-propoxycarbonyl-4-quinolone 1.8 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97670 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Butoxycarbonyl-6-ethyl-4-quinolone 13 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97671 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 28 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97672 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone 28 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97673 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-pentoxycarbonyl-4-quinolone 35 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97674 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone 92 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97675 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Cyclopentoxycarbonyl-6-ethyl-4-quinolone 19 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97676 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-i-propoxycarbonyl-4-quinolone 214 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97677 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(4-methyl-2-pentoxycarbonyl)-4-quinolone 295 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97678 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-pentoxycarbonyl)-4-quinolone 2600 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97679 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Carboxy-6-ethyl-4-quinolone 208 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97680 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-4-quinolone 78 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97681 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Butoxycarbonyl-4-quinolone 54 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97682 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-4-quinolone 16 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97683 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-propyl-4-quinolone 17 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97684 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-i-propyl-4-quinolone 15 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97685 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 1.4 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97686 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-propoxycarbonyl-4-quinolone 0.17 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97687 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone 6850 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97688 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-2-methyl-4-quinolone 4200 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97689 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-propylaminocarbonyl-4-quinolone 0.26 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97690 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Butylaminocarbonyl-6-ethyl-4-quinolone 0.54 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97691 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-propylaminocarbonyl-4-quinolone 0.048 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97692 KOR CORTICAL MEMBRANES RAT 3H-flumazenil Propyl 2-methyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate 870 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97693 KOR CORTICAL MEMBRANES RAT 3H-flumazenil Ethyl 7-Oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate >10000 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97694 KOR CORTICAL MEMBRANES RAT 3H-flumazenil Propyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate 7130 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97695 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 4.1 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97696 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 89 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97697 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-4-quinolone 26 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97698 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-4-quinolone 14 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97699 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 0.27 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97700 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 7.2 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97701 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil DIAZEPAM 12 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97702 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil DIAZEPAM 14 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97703 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil Zolpidem 1850 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97704 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil Zolpidem 53 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97705 L1210 cells MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 1800 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97706 L1210 cells MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 700 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97707 L1210 cells MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97708 L1210 cells MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97709 L1210 cells MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 1300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97710 L1210 cells MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97711 L1210 cells MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97712 L1210 + DFMO MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97713 L1210 + DFMO MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97714 L1210 + DFMO MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 700 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97715 L1210 + DFMO MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 150 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97716 L1210 + DFMO MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 200 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97717 L1210 + DFMO MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97718 L1210 + DFMO MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 1400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97719 L1210 cells MOUSE 14C-spermidine N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97720 L1210 cells MOUSE 14C-spermidine N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 2500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97721 L1210 cells MOUSE 14C-spermidine N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 6200 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97722 L1210 cells MOUSE 14C-spermidine N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 1800 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97723 L1210 cells MOUSE 14C-spermidine N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 5000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97724 L1210 cells MOUSE 14C-spermidine N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 1700 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97725 L1210 cells MOUSE 14C-spermidine N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97726 CHO-MG MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97727 C.H.O. MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97728 CHO-MG MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97729 C.H.O. MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 1500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97730 C.H.O. MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 4100 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97731 CHO-MG MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97732 CHO-MG MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97733 C.H.O. MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 450 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97734 C.H.O. MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97735 CHO-MG MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 9500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97736 CHO-MG MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 8800 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97737 C.H.O. MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 2500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97738 C.H.O. MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 1900 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97739 CHO-MG MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 3400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97740 Y5 CLONED HUMAN 125I-PYY FMS586 4.3 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97741 Y5 CLONED HUMAN 125I-PYY L-152,804 25 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97742 Y5 CLONED HUMAN 125I-PYY PYY 1 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97743 Y1 CLONED HUMAN 125I-PYY PYY 2 Kakui, N. et al., 2006 Jan 15, 2025 Jan 15, 2025
97744 Y1 CLONED HUMAN 125I-PYY L-152,804 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 15, 2025
97745 Y1 CLONED HUMAN 125I-PYY FMS586 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 15, 2025
97746 Y2 CLONED HUMAN 125I-PYY FMS586 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97747 Y2 CLONED HUMAN 125I-PYY L-152,804 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97748 Y2 CLONED HUMAN 125I-PYY PYY 2.1 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97749 H2 Sf9 HUMAN Functional HIS 1200 Xie, S. et. al., 2006 Jan 15, 2025 Jan 15, 2025