63354 Y5 CLONED HUMAN 125I-PYY BIBP3226 0 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
63355 Y5 CLONED HUMAN 125I-PYY BIBP3226 0 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
63356 Y5 CLONED HUMAN 125I-PYY BIBO3304 0 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
63357 Y5 CLONED HUMAN 125I-PYY BIBO3304 0 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
63358 Y5 CLONED HUMAN 125I-PYY BIIE0246 0 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
63359 Y5 CLONED HUMAN 125I-PYY BIIE0246 0 Rodriguez, M et al., 2003 Jan 15, 2025 Jan 28, 2025
31228 D3 CLONED HUMAN 125I-IODOSULPRIDE L741,626 0 Millan MJ, et. al., 2004 Jan 15, 2025 Jan 15, 2025
22462 A3 CLONED HUMAN 125I-Aba 39 1.0E-6 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22368 A2A Striatal Membranes RAT 3H-CGS-21680 36 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22369 A2A Striatal Membranes RAT 3H-CGS-21680 37 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22370 A2A Striatal Membranes RAT 3H-CGS-21680 38 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22436 A2B CLONED HUMAN 3H-ZM241385 36 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22437 A2B CLONED HUMAN 3H-ZM241385 37 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22438 A2B CLONED HUMAN 3H-ZM241385 38 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22195 A2A Striatal Membranes RAT 3H-CGS-21680 9 1.0E-5 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
42603 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3',5'-trifluoromethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2.2E-5 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42597 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 3.1E-5 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42602 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 3.2E-5 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
22390 A1 BRAIN RAT 3H-R-PIA 36 0.0001 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
22391 A1 BRAIN RAT 3H-R-PIA 38 0.0001 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
56972 KOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-bromo)benzamido]morphinan-oxalate 0.0003 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
53384 CB1 UNDEFINED UNDEFINED UNDEFINED 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 0.00035 Wang H et al., 2008 Jan 15, 2025 Jan 15, 2025
55786 CB1 UNDEFINED UNDEFINED UNDEFINED 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 0.00035 Zhang Y et al., 2008 Jan 15, 2025 Jan 15, 2025
5628 5-HT4 CLONED RAT 3H-GR-113808 RS 100235 0.000398107 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
5619 5-HT4 CLONED RAT 3H-GR-113808 RS 100235 0.00047863 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
5641 5-HT4 CLONED HUMAN 3H-GR-113808 RS 100235 0.00057544 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
5614 5-HT4 CLONED HUMAN 3H-GR-113808 RS 100235 0.000630957 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
31365 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE 5-CT 0.000794328 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
5612 5-HT4 CLONED HUMAN 3H-GR-113808 GR 125487 0.000870964 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
5617 5-HT4 CLONED RAT 3H-GR-113808 GR 125487 0.000912011 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
50282 MOR CLONED RAT 3H-NALOXONE BCTC 0.00095 Valenzano KJ, et al., 2003 Jan 15, 2025 Jan 15, 2025
9223 SST2 CLONED MOUSE 125I-MK-678 BIM 23027 0.001 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9229 SST2 CLONED MOUSE 125I-MK-678 BIM 23023 0.001 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9032 SST4 CLONED RAT 125I-CGP23996 SRIF-[Des-Ala1,des-Gly2,His4,5,D-Trp8] 0.001 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
8593 SST2 CLONED MOUSE 125I-Tyr11-SRIF BIM 23027 0.001 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
8594 SST2 CLONED MOUSE 125I-Tyr11-SRIF BIM 23023 0.001 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
100929 AChE BRAIN HUMAN Functional N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-4-(1H-indol-3-yl)butyramide 0.0017 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
8660 SST5 CLONED RAT 125I-Tyr11-SRIF BIM 23003 0.00199526 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
8676 SST5 CLONED RAT 125I-Tyr11-SRIF BIM 23052 0.00199526 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
47874 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Aib29,D31,p34,F35]-h-alpha-CGRP 27-37 0.002 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
9230 SST2 CLONED MOUSE 125I-MK-678 NC4-28B 0.002 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9231 SST2 CLONED MOUSE 125I-MK-678 BIM 23034 0.002 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9031 SST4 CLONED RAT 125I-CGP23996 SRIF-D-Trp8 0.002 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
9033 SST4 CLONED RAT 125I-CGP23996 BIM 23003 0.002 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
9062 SST4 CLONED RAT 125I-CGP23996 BIM 23052 0.002 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
28900 SST4 CLONED RAT 125I-Tyr11-somatostatin BIM 23052 0.002 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
21500 CCR5 CLONED Xenopus 3H-Epibatidine NFEP 0.0024 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
48190 Y4 CLONED RAT 125I-hPP PP, rat 0.0027 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48189 Y4 CLONED RAT 125I-hPP PP, human 0.003 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
21487 nAChR CLONED Xenopus 3H-Epibatidine NEP 0.0031 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
21488 nAChR CLONED Xenopus 3H-Epibatidine NFEP 0.0038 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
31355 5-HT7 BRAIN RAT 3H-MESULERGINE 5-CT 0.00398107 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
21489 nAChR CLONED Xenopus 3H-Epibatidine NBEP 0.004 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
23388 NK1 BRAIN CORTEX HUMAN 3H-SUBSTANCE P SSR240600 0.0043 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
56975 KOR UNDEFINED UNDEFINED UNDEFINED Guanosine 5'-[gamma-thio]triphosphate tetralithium salt 0.0048 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
9220 SST2 CLONED MOUSE 125I-MK-678 SRIF-D-Trp8 0.005 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9222 SST2 CLONED MOUSE 125I-MK-678 BIM 23003 0.005 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
9058 SST4 CLONED RAT 125I-CGP23996 L-362,855 0.005 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
8588 SST2 CLONED MOUSE 125I-Tyr11-SRIF BIM 23003 0.00501187 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
8674 SST5 CLONED RAT 125I-Tyr11-SRIF L-362,855 0.00501187 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
5618 5-HT4 CLONED RAT 3H-GR-113808 SB 207266 0.00562341 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
47873 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Hyp29,D31,p34,F35]-h-alpha-CGRP 27-37 0.006 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
9221 SST2 CLONED MOUSE 125I-MK-678 SRIF-[Des-Ala1,des-Gly2,His4,5,D-Trp8] 0.006 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
48191 Y4 CLONED RAT 125I-hPP PP, BOVINE 0.006 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
4173 5-HT1B CLONED HUMAN 3H-5HT DHE 0.006 HAMBLIN MW, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
17396 NOP BRAIN MOUSE 125I-Tyr10-OFQ/N(1-11) OFQ/N,Iodo[Tyr14] 0.006 Mogil JS, Pasternak GW., 2001 Jan 15, 2025 Jan 15, 2025
23387 NK1 IM9 HUMAN 125I-Bolton Hunter SSR240600 0.0061 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
15404 5-HT1B CLONED HUMAN 3H-5HT DHE 0.00616595 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
60432 GABAA CLONED HUMAN FNZ WY-TSC-4 0.007 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65573 GABAA CLONED HUMAN [3H] Flunitrazepam WY-TSC-4 (WYS8) 0.007 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
48188 Y4 CLONED RAT 125I-hPP PP, guinea pig 0.007 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
17395 NOP BRAIN MOUSE 125I-Tyr10-OFQ/N(1-11) OFQ/N,[Tyr14] 0.007 Mogil JS, Pasternak GW., 2001 Jan 15, 2025 Jan 15, 2025
17397 NOP BRAIN MOUSE 125I-Tyr10-OFQ/N(1-11) OFQ/N 0.007 Mogil JS, Pasternak GW., 2001 Jan 15, 2025 Jan 15, 2025
8595 SST2 CLONED MOUSE 125I-Tyr11-SRIF BIM 23059 0.00794328 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
9232 SST2 CLONED MOUSE 125I-MK-678 BIM 23059 0.008 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
57371 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(3-nitrophenyl)epibatidine 0.008 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
63385 nAChR FOREBRAIN RAT 3H-Epibatidine Epibatidine, (+/-) 0.008 Gohlke, H et al., 2003 Jan 15, 2025 Jan 15, 2025
9895 nAChR BRAIN RAT 3H-Epibatidine Epibatidine 0.008 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
10357 BRAIN RAT 3H-Cytisine Epibatidine-(+) 0.0084 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
21511 nAChR CLONED Xenopus 3H-Epibatidine NEP 0.0085 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
5626 5-HT4 CLONED RAT 3H-GR-113808 GR 125487 0.00891251 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
53275 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(6-fluoro-5-(4-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.009 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
57376 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(3-Dimethylaminophenyl)epibatidine 0.009 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
100926 AChE BRAIN HUMAN Functional N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide 0.009 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
9876 BRAIN RAT 5-125I-Iodo-A-85380 Epibatidine-(-) 0.009 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
21510 nAChR CLONED Xenopus 3H-Epibatidine NFEP 0.0092 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
86754 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide 0.00956 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
22016 LHRH Pituitary RAT UNDEFINED 24 0.00977237 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
86805 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide 0.00985 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
10497 Olfactory bulbs MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10498 CEREBRAL CORTEX MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10499 STRIATUM MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10501 HYPOTHALAMUS MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
21509 nAChR CLONED Xenopus 3H-Epibatidine NBEP 0.01 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
10502 thalamus MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10503 Midbrain MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10505 Superior Colliculus MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10506 Inferior Colliculus MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10507 Hindbrain MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
10508 CEREBELLUM MOUSE 3H-Epibatidine Epibatidine 0.01 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
12304 AORTA Dog 3H-PRAZOSIN PRAZOSIN 0.01 Jones SB, et al., 1987 Jan 15, 2025 Jan 15, 2025
9233 SST2 CLONED MOUSE 125I-MK-678 BIM 23060 0.01 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
19731 D2 CLONED HUMAN UNDEFINED EPIDEPRIDE 0.01 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
12317 AORTA RAT 3H-PRAZOSIN PRAZOSIN 0.01 Jones SB, et al., 1987 Jan 15, 2025 Jan 15, 2025
6452 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 SB204070 0.01 HEGDE SS, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
52795 5-HT2A UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide 0.01 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
52796 5-HT2A UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide 0.01 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
6738 D2 CLONED HUMAN 3H-RACLOPRIDE NEMONAPRIDE 0.01 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
9811 MT2 CLONED HUMAN 125I-Iodomelatonin 4-P-PDOT 0.01 Nonno,Pannacci,Lucini, Angeloni,Fraschini,Stankov Jan 15, 2025 Jan 15, 2025
16222 D2 CLONED MOUSE 3H-SPIPERONE SPIPERONE 0.01 Neve KA, 1990 Jan 15, 2025 Jan 15, 2025
9830 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.01 Reppert SM, Weaver DR, Ebisawa, 1994 Jan 15, 2025 Jan 15, 2025
12393 BRAIN RAT 3H-5HT FK 1052 0.01 Nagakura Y, et al., 1993 Jan 15, 2025 Jan 15, 2025
12394 BRAIN RAT 3H-KETANSERIN FK 1052 0.01 Nagakura Y, et al., 1993 Jan 15, 2025 Jan 15, 2025
12395 D2 BRAIN RAT 3H-Spiperone + 40 nm Ketanserin FK 1052 0.01 Nagakura Y, et al., 1993 Jan 15, 2025 Jan 15, 2025
10370 nAChR M10 Cells Mammalian 3H-Epibatidine Epibatidine 0.01 Whiteaker P, Sharples CG, Wonnacott S, 1998 Jan 15, 2025 Jan 15, 2025
10384 nAChR M10 membranes Mammalian 3H-Epibatidine Epibatidine 0.01 Whiteaker P, Sharples CG, Wonnacott S, 1998 Jan 15, 2025 Jan 15, 2025
9877 BRAIN RAT 5-125I-Iodo-A-85380 A-85380,5-Iodo 0.01 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
34197 D2 Striatal Membranes RAT 125I-IABN SPIPERONE 0.01 Luedtke RR, et al., 2000 Jan 15, 2025 Jan 27, 2025
9878 BRAIN RAT 5-125I-Iodo-A-85380 A-85380 0.01 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
7333 DOR CLONED HUMAN 3H-Naltrindole BW373U86 0.01 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
7336 DOR CLONED HUMAN 3H-Naltrindole NTB 0.01 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
9898 nAChR BRAIN RAT 3H-Epibatidine A-85380 0.01 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
9899 nAChR BRAIN RAT 3H-Epibatidine A-85380,5-Iodo 0.01 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
8622 SST3 CLONED MOUSE 125I-Tyr11-SRIF BIM 23056 0.01 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
14269 Y1 KIDNEY RAT 125I-PYY 1229U91 0.01 Hegde SS, et al., 1995b Jan 15, 2025 Jan 15, 2025
50381 SST2 CLONED HUMAN 125I-LTT-SST-28 L-054,522 0.01 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
28888 SST2 CLONED RAT 125I-Tyr11-somatostatin NC8-12 0.01 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
26332 GAL1 CLONED RAT 125I-GALANIN M35 0.01 Howard AD, et al., 1997 Jan 15, 2025 Jan 15, 2025
7395 KOR CLONED HUMAN 3H-U69,593 DIPRENORPHINE-HCl 0.01 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
9444 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.01 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
5356 5-HT2A CLONED HUMAN 3H-KETANSERIN RITANSERIN 0.01 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
5613 5-HT4 CLONED HUMAN 3H-GR-113808 SB 207266 0.01 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
22005 LHRH Pituitary RAT UNDEFINED 13 0.01 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
11514 Beta2 CLONED HUMAN 125I-ICYP PROPRANOLOL 0.01 Schotte A, et al., 1996 Jan 15, 2025 Jan 28, 2025
35130 BRAIN RAT 3H-Cytisine 5-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 0.011 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
86807 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide 0.0113 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
55674 AChE UNDEFINED HUMAN UNDEFINED N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine 0.0118 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
57366 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(3-Fluorophenyl)epibatidine 0.012 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
60452 GABAA CLONED HUMAN FNZ QH-II-077 0.012 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
27020 nAChR CLONED HUMAN 3H-Epibatidine Epibatidine 0.012 Eaton JB, et.al.,2003 Jan 15, 2025 Jan 15, 2025
86733 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide 0.0126 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
57368 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(3-Chlorophenyl)epibatidine 0.013 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
48183 Y4 CLONED GUINEA PIG 125I-hPP PP, BOVINE 0.013 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
38278 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N-dimethyl-2-(2'-amino-4'-iodophenylthio)benzylamine 0.013 Jarkas N, et al., 2005 Jan 15, 2025 Jan 15, 2025
21492 CCR5 CLONED Xenopus 3H-Epibatidine NBEP 0.013 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
51209 CHRNA4 UNDEFINED RAT UNDEFINED (1R,4R)-2-(6-chloro-5-methyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane 0.014 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
100925 AChE BRAIN HUMAN Functional N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)propionamide 0.014 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
41807 CLONED HUMAN 3H-Estradiol Tamoxifen, 4-hydroxy 0.014 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
89631 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0147911 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
57370 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(4-Nitrophenyl)epibatidine 0.015 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
38966 nAChR BRAIN RAT 3H-Cytisine dechloroepibatidine-(-) 0.015 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
100927 AChE BRAIN HUMAN Functional N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-2-(1H-indol-3-yl)acetamide 0.015 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
55901 MOR UNDEFINED HUMAN UNDEFINED 6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 0.015 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
56970 KOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-methyl)benzamido]morphinan-oxalate 0.015 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
57369 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(3-Bromophenyl)epibatidine 0.016 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
36572 5-HT2A FR. CORTEX RAT 3H-KETANSERIN RISPERIDONE 0.016 Leysen JE, et.al., 1994 Jan 15, 2025 Jan 15, 2025
57365 CHRNA4 UNDEFINED RAT UNDEFINED (1R,2R,4S)-2-(6-chloro-5-(4-fluorophenyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane 0.017 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
57373 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(3-Aminophenyl)epibatidine 0.017 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
35123 BRAIN RAT 3H-Cytisine A-85380 0.017 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
99974 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 0.017 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
67731 Alpha1A CEREBRAL CORTEX RAT 3H-PRAZOSIN (+)Niguldipine 0.0177828 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
51203 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.018 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
51207 CHRNA4 UNDEFINED RAT UNDEFINED (1R,4R)-2-(5,6-dichloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.018 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
57362 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.018 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
51225 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane 0.018 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
37553 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.018 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
57375 CHRNA4 UNDEFINED RAT UNDEFINED (1R,2R,4S)-2-(6-chloro-5-(3-methoxyphenyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane 0.019 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
41772 CLONED HUMAN Functional 17beta-Estradiol 0.019 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
47680 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE PAROXETINE 0.019 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
22009 LHRH Pituitary RAT UNDEFINED 17 0.0194984 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
47872 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Tic29,D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
51202 CHRNA4 UNDEFINED RAT UNDEFINED 2-(3-pyridinyl)-2,5-diazabicyclo[2.2.2]octane 0.02 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
10500 HIPPOCAMPUS MOUSE 3H-Epibatidine Epibatidine 0.02 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
32007 D2 Striatal Membranes RAT 125I-Spectramide SPIPERONE 0.02 Sanchez-Roa, P.M., et al., 1989 Jan 15, 2025 Jan 15, 2025
10504 Interpeduncular n. MOUSE 3H-Epibatidine Epibatidine 0.02 Marks MJ, Smith KW, Collins AC, 1997 Jan 15, 2025 Jan 15, 2025
100882 AChE BRAIN HUMAN Functional N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)propionamide 0.02 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
12312 AORTA Dog 125I-HEAT PRAZOSIN 0.02 Jones SB, et al., 1987 Jan 15, 2025 Jan 15, 2025
4381 5-HT1B CLONED RAT 3H-5HT DHE 0.02 HAMBLIN MW, ET AL., 5/1992 Jan 15, 2025 Jan 15, 2025
12322 AORTA RAT 125I-HEAT PRAZOSIN 0.02 Jones SB, et al., 1987 Jan 15, 2025 Jan 15, 2025
53294 CHRNA4 UNDEFINED RAT UNDEFINED 2-Pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane 0.02 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
60463 GABAA CLONED HUMAN FNZ QH-II-085 0.02 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
8764 SST2 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.02 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
100928 AChE BRAIN HUMAN Functional 2-(5-Bromo-1H-indol-3-yl)-N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]acetamide 0.02 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
9819 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Bromo 0.02 Nonno,Lucini,Pannacci,Mazzucchelli,Angeloni 1998 Jan 15, 2025 Jan 15, 2025
9820 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Phenyl 0.02 Nonno,Lucini,Pannacci,Mazzucchelli,Angeloni 1998 Jan 15, 2025 Jan 15, 2025
15460 5-HT1B CLONED RAT 3H-5HT DHE 0.02 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
10876 D2 CLONED RAT 3H-YM 09151-2 YM-09151-2 0.02 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
50046 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-CONH2, [Aib15] 0.02 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
43144 SLK CLONED HUMAN 3H-Staurosporine Staurosporine 0.02 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
10893 D2 CLONED RAT 3H-SPIPERONE ETICLOPRIDE 0.02 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
3986 5-HT4 CLONED MOUSE 3H-GR-113808 GR 125487 0.02 CLAEYSEN S, ET AL., 1996 Jan 15, 2025 Jan 27, 2025
65429 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-085 0.02 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
54684 Alpha1A UNDEFINED UNDEFINED UNDEFINED mazapertine 0.02 Jain KS et al., 2008 Jan 15, 2025 Jan 15, 2025
9894 nAChR BRAIN RAT 3H-Epibatidine IPH 0.02 Mukhin, et al, 1999 Jan 15, 2025 Jan 15, 2025
7337 DOR CLONED HUMAN 3H-Naltrindole NALTRINDOLE 0.02 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
7873 GABAA CLONED HUMAN 3H-RO-15-1788 4 0.02 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
7381 KOR CLONED HUMAN 3H-U69,593 NOR-BNI (HCI)2 0.02 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
62679 SST2 COLON RAT UNKNOWN octreotide 0.02 Moore SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
28904 SST3 CLONED RAT 125I-Tyr11-somatostatin DC-25-20 0.02 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
5611 5-HT4 CLONED HUMAN 3H-GR-113808 GR 113808 0.02 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
5616 5-HT4 CLONED RAT 3H-GR-113808 GR 113808 0.02 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
47858 CLONED HUMAN 3H-CGRP 8-37 [D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
5622 5-HT4 CLONED HUMAN 3H-GR-113808 GR 125487 0.02 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
11513 Beta1 CLONED HUMAN 125I-ICYP PROPRANOLOL 0.02 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
9215 SST3 CLONED MOUSE 125I-CGP23996 BIM 23056 0.02 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
57364 CHRNA4 UNDEFINED RAT UNDEFINED (1R,2R,4S)-2-(6-chloro-5-phenylpyridin-3-yl)-7-azabicyclo[2.2.1]heptane 0.021 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
59703 5-HT1A CLONED HUMAN 3H-WAY100635 4-[3-[4-( o -Methoxyphenyl)piperazin-1-yl]propoxy]-4-aza-tricyclo- [5.2.1.02,6]dec-8-ene-3,5-dione 0.021 Herth, M. et. al., 2009 Jan 15, 2025 Jan 15, 2025
35129 BRAIN RAT 3H-Cytisine 5-Bromo-3-(2(S)-azetidinylmethoxy)pyridine 0.021 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
63729 nAChR BRAIN RAT 3H-NICOTINE Epibatidine, (+/-) 0.021 Wright, E et al., 1997 Jan 15, 2025 Jan 15, 2025
32659 NOP CLONED HUMAN 3H-N/OFQ OFQ/N UFP-102 0.0213796 Carra G, et al., 2004 Jan 15, 2025 Jan 15, 2025
63199 MOR FOREBRAIN RAT 3H-DAMGO Tyr-D-Ser-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) 0.0219 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
57374 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(4-Methoxylphenyl)epibatidine 0.022 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
85669 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide 0.0224 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
63188 KOR CEREBELLUM GUINEA PIG 3H-Bremazocine Dynorphin A (1-13) NH2 0.0228 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
29364 CCR5 CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.023 Jensen AA, et al., 2003 Jan 15, 2025 Jan 15, 2025
23707 MC1 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH alpha-MSH, [Nle4, D-Phe7] 0.0231 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
22487 MC1 CLONED HUMAN 125I-NDP-MSH NDP-MSH 0.0231 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
63198 MOR FOREBRAIN RAT 3H-DAMGO Tyr-D-Met-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) 0.0235 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
29192 SST2 CLONED HUMAN UNDEFINED NC8-12 0.024 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
29037 SST2 CLONED HUMAN 125I-LTT-SST-28 NC8-12 0.024 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
22007 LHRH Pituitary RAT UNDEFINED 15 0.0245471 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
56108 DOR UNDEFINED HUMAN UNDEFINED (1R,13S,14R)-24-(cyclopropylmethyl)-13,20-dihydroxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene-19-carboxamide 0.025 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
35128 BRAIN RAT 3H-Cytisine 5-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 0.025 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
35131 BRAIN RAT 3H-Cytisine 6-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 0.025 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
34917 CCR5 CLONED UNDEFINED 3H-Epibatidine Epibatidine 0.025 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
37550 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[2-[4-(4-Methylphenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.025 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
34488 CCR5 CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.025 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
30941 KOR CLONED HUMAN 35S-GTPGammaS TRK-820 0.025 Wang Y, et. al., 2004 Jan 15, 2025 Jan 15, 2025
28918 CCR5 CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.025 Wei ZL, et. al., 2003 Jan 15, 2025 Jan 15, 2025
57361 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.026 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
53271 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.026 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
29015 SST5 CLONED HUMAN 125I-LTT-SST-28 Leu8, D-Trp22, Tyr25 SST-28 0.026 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
52376 CHRNA4 UNDEFINED HUMAN UNDEFINED Epibatidine 0.026 Carroll FI et al., 2007 Jan 15, 2025 Jan 15, 2025
63196 MOR FOREBRAIN RAT 3H-DAMGO Tyr-D-Asn-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) 0.026 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
22020 LHRH Pituitary RAT UNDEFINED 28 0.0269153 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
19722 D2 CLONED HUMAN UNDEFINED BENPERIDOL 0.027 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
16654 M2 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.027 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
51217 CHRNA4 UNDEFINED RAT UNDEFINED (1R,4R)-2-(6-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.027 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
53293 CHRNA4 UNDEFINED RAT UNDEFINED 2-(6-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane 0.027 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
63046 MC5 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Hyp-DNal(2')Arg-Trp-Lys]-NH2 0.027 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
55945 KOR UNDEFINED HUMAN UNDEFINED norbinaltorphimine 0.027 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
67548 nAChR FOREBRAIN RAT 3H-Epibatidine N-methepibatidine 0.027 Gohlke, H et al., 2003 Jan 15, 2025 Jan 15, 2025
67549 nAChR FOREBRAIN RAT 3H-Epibatidine N-methylepibatidine 0.027 Gohlke, H et al., 2003 Jan 15, 2025 Jan 15, 2025
51223 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-fluoro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.028 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
56356 CHRNA4 UNDEFINED RAT UNDEFINED 5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine 0.028 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56369 CHRNA4 UNDEFINED RAT UNDEFINED (S)-2-chloro-5-((1-methylpyrrolidin-2-yl)methoxy)-3-(2-(pyridin-4-yl)vinyl)pyridine 0.028 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
29076 SST2 CLONED HUMAN 125I-LTT-SST-28 EC5-21 0.028 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
59292 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Fluoro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.028 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
21499 CCR5 CLONED Xenopus 3H-Epibatidine NEP 0.028 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
17381 Alpha1A CLONED HUMAN 3H-PRAZOSIN Tamsulosin 0.0288403 Hancock A, et al., 2001 Jan 15, 2025 Jan 15, 2025
53277 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(6-fluoro-5-(4-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.029 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
100608 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.03 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
48134 Y2 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 0.03 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
5644 Alpha2C CELLS OK 3H-RAUWOLSCINE L-657,743 0.03 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
4112 KOR CLONED HUMAN 3H-U69,593 BREMAZOCINE(-) 0.03 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
63762 CXCR3 CLONED HUMAN 125I-CXCL11 CXCL11 0.03 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
60439 GABAA CLONED HUMAN FNZ SH-TSC-2 0.03 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
100633 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.03 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100892 BchE serum HUMAN Functional N-(3-{[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-methylamino}propyl)-3-(1H-indol-3-yl)propionamide 0.03 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 15, 2025
4382 5-HT1B CLONED RAT 3H-5HT ERGOTAMINE 0.03 HAMBLIN MW, ET AL., 5/1992 Jan 15, 2025 Jan 15, 2025
42020 M2 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.03 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
60456 GABAA CLONED HUMAN FNZ QH-II-092 0.03 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
33843 D2 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.03 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
6453 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 GR 125487 0.03 HEGDE SS, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
35894 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7-(2-Methoxyethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ymethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.03 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
35127 BRAIN RAT 3H-Cytisine 5-Chloro-3-(2(S)-azetidinylmethoxy)pyridine 0.03 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
8762 SST2 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.03 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
22330 A1 BRAIN BOVINE 3H-DPCPX XAC 0.03 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
23358 A1 BRAIN BOVINE 3H-DPCPX R-PIA 0.03 Klotz KN et al., 1991 Jan 15, 2025 Jan 27, 2025
7235 ETA CLONED HUMAN 125I-ENDOTHELIN J-104132 0.03 Nishikibe M, et al., 1999 Jan 15, 2025 Jan 15, 2025
41797 CLONED HUMAN 3H-Estradiol raloxifene 0.03 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
6730 D2 CLONED HUMAN 3H-RACLOPRIDE EPIDEPRIDE 0.03 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
9806 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Phenyl 0.03 Nonno,Pannacci,Lucini, Angeloni,Fraschini,Stankov Jan 15, 2025 Jan 15, 2025
8527 5-HT4B CLONED HUMAN 3H-GR-113808 SB204070 0.03 Bender E, et al., 2000 Jan 15, 2025 Jan 27, 2025
29014 SST4 CLONED HUMAN 125I-LTT-SST-28 Leu8, D-Trp22, Tyr25 SST-28 0.03 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
6743 D2 ANTERIOR PITUITARY PIG 3H-RACLOPRIDE SPIPERONE 0.03 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
6744 D2 CLONED HUMAN 3H-RACLOPRIDE SPIPERONE 0.03 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
10073 MOR BRAIN MOUSE 125I-Endomorphin-1 Diprenorphine 0.03 Goldberg IE, et al, 1998 Jan 15, 2025 Jan 15, 2025
10332 nAChR BRAIN RAT 3H-Cytisine ABT-594 0.03 Bannon AW, et al., 1998 Jan 15, 2025 Jan 15, 2025
9824 CLONED Sheep 125I-Iodomelatonin Melatonin,2-Iodo 0.03 Reppert SM, Weaver DR, Ebisawa, 1994 Jan 15, 2025 Jan 15, 2025
15461 5-HT1B CLONED RAT 3H-5HT ERGOTAMINE 0.03 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
39034 D2 CLONED HUMAN R-SAT SPIPERONE 0.03 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
18557 CCK1 PANCREAS RAT 125I-BH-CCK-8 6 0.03 Pierson ME et al., 1997 Jan 15, 2025 Jan 15, 2025
18569 CCK1 PANCREAS RAT 125I-BH-CCK-8 9 0.03 Pierson ME et al., 1997 Jan 15, 2025 Jan 15, 2025
10894 D2 CLONED RAT 3H-YM 09151-2 YM-09151-2 0.03 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
3987 5-HT4 Colliculus Neurons MOUSE 3H-GR-113808 GR 125487 0.03 CLAEYSEN S, ET AL., 1996 Jan 15, 2025 Jan 27, 2025
10900 D4 CLONED HUMAN 3H-YM 09151-2 YM-09151-2 0.03 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
39061 D2 CLONED HUMAN R-SAT THIOTHIXENE 0.03 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
43158 STK10 CLONED HUMAN 3H-Staurosporine Staurosporine 0.03 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
65431 GABAA CLONED HUMAN [3H] Flunitrazepam SH-TSC-2 (BCCT) 0.03 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
10906 D4 CLONED HUMAN 3H-YM 09151-2 YM-09151-2 0.03 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
65436 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-092 0.03 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7843 GABAA CLONED HUMAN 3H-RO-15-1788 7 0.03 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
24489 CLONED RAT 3H-Quisqualate Quisqualate 0.03 Lavreysen, H, et al., 2003 Jan 15, 2025 Jan 15, 2025
8623 SST3 CLONED MOUSE 125I-Tyr11-SRIF BIM 23058 0.03 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
11963 H1 BRAIN GUINEA PIG 3H-Histamine Alpha-Dimethylhistane-alpha 0.03 Hill JA., 1992 Jan 15, 2025 Jan 15, 2025
11964 H1 BRAIN GUINEA PIG 3H-Histamine S-Beta-Dimethylhistamine-R-alpha 0.03 Hill JA., 1992 Jan 15, 2025 Jan 15, 2025
7379 KOR CLONED HUMAN 3H-U69,593 Spiradoline 0.03 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
4823 5-HT4 Colliculus Neurons MOUSE 3H-GR-113808 GR 125487 0.03 ANSANAY H, ET AL.,1996 Jan 15, 2025 Jan 15, 2025
47064 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-3P 0.03 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
28894 SST3 CLONED RAT 125I-Tyr11-somatostatin DC-25-12 0.03 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
10217 CLONED HUMAN 125I-HEAT PRAZOSIN 0.03 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
9452 MT2 CLONED HUMAN 125I-Iodomelatonin S 20098 0.03 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
9461 CEREBELLUM HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.03 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
5625 5-HT4 CLONED RAT 3H-GR-113808 GR 113808 0.03 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
9469 Colliculus Neurons GUINEA PIG 125I-Iodomelatonin Melatonin,2-Iodo 0.03 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
97843 5-HT2A Membranes HUMAN [3H]-ketanserin MDL 100907 0.0301995 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
22023 LHRH Pituitary RAT UNDEFINED 31 0.030903 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
48181 Y4 CLONED GUINEA PIG 125I-hPP PP, human 0.031 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48187 Y4 CLONED HUMAN 125I-hPP PP, BOVINE 0.031 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
63043 MC5 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Pro-DNal(2'Arg-Trp-Lys]-NH2 0.031 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
34494 CCR5 CLONED RAT 3H-Epibatidine A-85380-I 0.031 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
22025 LHRH Pituitary RAT UNDEFINED 33 0.0316228 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
50232 Y2 CLONED GUINEA PIG 125I-PYY PYY, porcine 0.032 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
59268 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-methyl-7-azabicyclo[2.2.1]heptane 0.032 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
22027 LHRH Pituitary RAT UNDEFINED 35 0.0323594 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
23709 MC1 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH alpha MSH 0.0334 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
22488 MC1 CLONED HUMAN 125I-NDP-MSH alpha MSH 0.0334 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
89635 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0338844 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
57372 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(4-Aminophenyl)epibatidine 0.034 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
16688 M4 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.034 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
62027 nAChR CLONED HUMAN 3H-Cytisine, (-) A 98593 0.034 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
59280 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methoxyphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.034 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
47829 KOR CLONED HUMAN 3H-U69,593 Cyclorphan 0.034 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
16645 M1 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.035 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
51214 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-[5-hydroxy-3-pyridinyl]-2,5-diazabicyclo[2.2.1]-heptane 0.035 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
56334 Chrna3 UNDEFINED RAT UNDEFINED Epibatidine 0.035 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
60437 GABAA CLONED HUMAN FNZ SH-TSC-2 0.035 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
55623 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(5-Ethoxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride 0.035 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
47730 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.035 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47731 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY,[leu31,Pro34], human 0.035 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
34941 nAChR CLONED UNDEFINED 3H-Epibatidine Epibatidine 0.035 Wei ZL, et al., 2005 Jan 15, 2025 Jan 27, 2025
65433 nAChR CLONED HUMAN [3H] Flunitrazepam SH-TSC-2 (BCCT) 0.035 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
59294 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Fluoro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.035 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
50115 SST2 CLONED HUMAN 125I-Tyr11-SRIF-14 Somatostatin-14 0.035 Poitout L., et.al., 2001 Jan 15, 2025 Jan 15, 2025
34514 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.035 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
28922 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.035 Wei ZL, et. al., 2003 Jan 15, 2025 Jan 27, 2025
60461 GABAA CLONED HUMAN FNZ JYI-57 0.036 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65470 nAChR CLONED HUMAN [3H] Flunitrazepam JYI-57 0.036 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
27501 5-HT1B FR. CORTEX RAT 3H-GR-125743 L694,247 0.0363078 Millan MJ, et al., 2002a Jan 15, 2025 Jan 15, 2025
62022 nAChR BRAIN RAT 3H-Cytisine, (-) ABT-594 0.037 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
42058 M4 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.037 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
59264 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-azabicyclo[2.2.1]heptane 0.037 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
63211 KOR CEREBELLUM GUINEA PIG 3H-Bremazocine Tyr-D-Asn-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) 0.0378 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
52386 CHRNA4 UNDEFINED HUMAN UNDEFINED N-methylepibatidine 0.038 Carroll FI et al., 2007 Jan 15, 2025 Jan 15, 2025
86796 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide 0.039 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
57367 CHRNA4 UNDEFINED RAT UNDEFINED 3'-(4-Chlorophenyl)epibatidine 0.039 Carroll FI et al., 2010 Jan 15, 2025 Jan 15, 2025
48185 Y4 CLONED HUMAN 125I-hPP PP, human 0.039 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
62023 nAChR BRAIN RAT 3H-Cytisine, (-) A 98593 0.039 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
59262 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-azabicyclo[2.2.1]heptane 0.039 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
59316 nAChR BRAIN CORTEX RAT 3H-Epibatidine 4-[5-(7-Azabicyclo[2.2.1]hept-2-yl)-2-fluoro-3-pyridinyl]benzonitrile 0.039 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
64727 H1 CLONED HUMAN 3H-PYRILAMINE KETOTIFEN 0.0398107 Appl, Heidrun. et. al, 2011 Jan 15, 2025 Jan 28, 2025
57091 D2 UNDEFINED HUMAN UNDEFINED Bifeprunox 0.04 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
9477 HYPOTHALAMUS GUINEA PIG 125I-Iodomelatonin Melatonin,2-Iodo 0.04 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
32008 D2 Striatal Membranes RAT 125I-Spectramide ETICLOPRIDE 0.04 Sanchez-Roa, P.M., et al., 1989 Jan 15, 2025 Jan 15, 2025
5642 Alpha2C CELLS OK 3H-RAUWOLSCINE RAUWOLSCINE 0.04 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
48139 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.04 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
63766 CXCR3 RBL HUMAN 125I-CXCL11 CXCL11 0.04 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
28964 SLC6A4 BRAIN RAT 3H-cyanoimipramine PAROXETINE 0.04 Beique JC, et.al, 1999 Jan 15, 2025 Jan 15, 2025
60455 GABAA CLONED HUMAN FNZ QH-II-092 0.04 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
15407 5-HT1B CLONED HUMAN 3H-5HT CGS 12066B 0.04 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
52786 5-HT2A UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2-phenylacetamide 0.04 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
6710 D2 CLONED HUMAN 3H-SPIPERONE NEMONAPRIDE 0.04 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
15934 CB2 CLONED MOUSE 3H-CP-55940 SR 144528 0.04 Iwamura H, et al., 2000 Jan 15, 2025 Jan 15, 2025
41796 CLONED HUMAN 3H-Estradiol OHT 0.04 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
4174 5-HT1B CLONED HUMAN 3H-5HT CGS 12066B 0.04 HAMBLIN MW, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
6737 D2 ANTERIOR PITUITARY PIG 3H-RACLOPRIDE NEMONAPRIDE 0.04 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
61271 GABAA CLONED HUMAN FNZ YT-II-76 0.04 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
10331 nAChR BRAIN RAT 3H-Cytisine Epibatidine 0.04 Bannon AW, et al., 1998 Jan 15, 2025 Jan 15, 2025
97628 SST2 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.04 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
23645 PDE4 CEREBRAL CORTEX RAT 3H-Rolipram Piclamilast 0.04 Zhao, Y et. al., 2003 Jan 15, 2025 Jan 15, 2025
4463 SLC6A4 BRAIN RAT 3H-IMIPRAMINE SERTRALINE 0.04 PALVIMAKI EP, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
99959 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.04 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
41344 CLONED HUMAN UNDEFINED 7-iodo-THIQ 0.04 Wu Q, et al., 2005 Jan 15, 2025 Jan 15, 2025
85648 nAChR CLONED HUMAN 3H-Epibatidine 3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 0.04 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
59282 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methoxyphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.04 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
65437 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-092 0.04 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
100771 PDE3a CLONED HUMAN Functional Trequinsin 0.04 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
65447 nAChR CLONED HUMAN [3H] Flunitrazepam YT-II-76 0.04 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
37545 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.04 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
37548 D4 CLONED HUMAN 3H-SPIROPERIDOL N-[2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.04 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
9901 nAChR ADRENAL RAT 3H-Epibatidine Epibatidine 0.04 Mukhin, et al, 1999 Jan 15, 2025 Jan 27, 2025
13494 CLONED OPOSSUM 3H-Yohimbine RAUWOLSCINE 0.04 Murphy TJ, et al., 1988 Jan 15, 2025 Jan 15, 2025
13503 CLONED OPOSSUM 3H-RAUWOLSCINE RAUWOLSCINE 0.04 Murphy TJ, et al., 1988 Jan 15, 2025 Jan 15, 2025
7876 GABAA CLONED HUMAN 3H-RO-15-1788 7 0.04 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
65990 nAChR BRAIN RAT 3H-Cytisine A-85380 0.04 Holladay MW et al., 1997 Jan 15, 2025 Jan 15, 2025
9443 MT1 CLONED HUMAN 125I-Iodomelatonin S 20098 0.04 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
27116 SLC6A4 BRAIN RAT 3H-IMIPRAMINE PAROXETINE 0.04 Beique JC, et.al.,1998 Jan 15, 2025 Jan 15, 2025
10478 BRAIN RAT 3H-Cytisine Epibatidine-(-) 0.04 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
31984 D2 HIPPOCAMPUS RAT 125I-Epidepride SPIPERONE 0.04 Kessler, R.M., et. al., 1993 Jan 15, 2025 Jan 15, 2025
10481 nAChR CLONED HUMAN 3H-Cytisine A-85380 0.04 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
50422 SST2 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.04 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
9208 SST3 CLONED MOUSE 125I-CGP23996 BIM 23058 0.04 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
11770 CAUDATE NUCLEUS HUMAN 3H-QNB Quinuclidinyl benzilate 0.04 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
49062 SST2 CLONED RAT 125I-Tyr11-SRIF Somatostatin-14 0.040738 Feniuk W, et.al., 2000 Jan 15, 2025 Jan 15, 2025
56338 Chrna3 UNDEFINED RAT UNDEFINED 5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine 0.041 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
55624 CHRNA4 UNDEFINED RAT UNDEFINED cis-3-(5-Propyloxy-3-pyridinyl)-3,7-diazabicyclo[3.3.0]octane Semifumarate 0.041 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
60438 GABAA CLONED HUMAN FNZ SH-TSC-2 0.0419 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65432 nAChR CLONED HUMAN [3H] Flunitrazepam SH-TSC-2 (BCCT) 0.0419 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
55095 H3 UNDEFINED HUMAN UNDEFINED 4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester 0.042 von Coburg Y et al., 2009 Jan 15, 2025 Jan 15, 2025
23397 NK1 ILEUM Gerbil 125I-Bolton Hunter Substance P 0.042 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
56969 KOR UNDEFINED UNDEFINED UNDEFINED Naltrexone 0.042 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
54122 TRPV1 UNDEFINED RAT UNDEFINED Resiniferatoxin 0.0426 Choi HK et al., 2009 Jan 15, 2025 Jan 15, 2025
22022 LHRH Pituitary RAT UNDEFINED 30 0.042658 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
16712 M5 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.043 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
62024 nAChR BRAIN RAT 3H-Cytisine, (-) Epibatidine, (+/-) 0.043 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
31062 BRAIN RAT 3H-Cytisine Epibatidine, (+/-) 0.043 Abreo MA, et al., 1996 Jan 15, 2025 Jan 15, 2025
47726 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY, porcine 0.043 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
52118 MOR UNDEFINED HUMAN UNDEFINED 3-((3R,4R)-1-((S)-3-cyclohexyl-3-hydroxypropyl)-3,4-dimethylpiperidin-4-yl)phenol 0.043 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
23710 MC1 CLONED HUMAN 125I-[Nle4,D-Phe7]Alpha-MSH desacetyl-alpha-MSH 0.0432 Schioth HB, et al., 1996 Jan 15, 2025 Jan 15, 2025
22489 MC1 CLONED HUMAN 125I-NDP-MSH desacetyl-alpha-MSH 0.0432 Schioth HB, et al., 1995 Jan 15, 2025 Jan 15, 2025
21504 nAChR CLONED Xenopus 3H-Epibatidine NBEP 0.044 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
42001 M1 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.044 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
53279 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(5-(4-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.044 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
48182 Y4 CLONED GUINEA PIG 125I-hPP PP, rat 0.044 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
62800 Brain caudate nucleus HUMAN 3H-QNB Quinuclidinyl benzilate 0.044 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 15, 2025
23401 NK1 IM9 HUMAN 125I-Bolton Hunter Substance P 0.044 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
59276 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.044 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
63734 nAChR BRAIN MICE 3H-NICOTINE Epibatidine-(+) 0.045 Damaj, MI et al., 1998 Jan 15, 2025 Jan 15, 2025
97844 5-HT2A Membranes HUMAN [3H]-ketanserin Eplivanserin 0.0457088 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
35122 BRAIN RAT 3H-Cytisine 2-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 0.046 Koren AO, et al., 1998 Jan 15, 2025 Jan 15, 2025
48180 Y4 CLONED GUINEA PIG 125I-hPP PP, guinea pig 0.046 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
29371 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.046 Jensen AA, et al., 2003 Jan 15, 2025 Jan 15, 2025
85707 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide 0.046 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
86736 5-HT2A FR. CORTEX RAT 3H-KETANSERIN N-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide 0.046 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
51201 CHRNA4 UNDEFINED RAT UNDEFINED 3-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane 0.047 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
51205 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.047 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
47681 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE SERTRALINE 0.047 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
55625 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.047 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
56184 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.047 Sippy KB et al., 2009 Jan 15, 2025 Jan 15, 2025
40156 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.047 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
83230 5-HT2A CLONED HUMAN 3H-KETANSERIN MDL 100907 0.048 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
47727 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY, porcine 0.048 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
56185 CHRNA4 UNDEFINED RAT UNDEFINED ABT-594 0.048 Sippy KB et al., 2009 Jan 15, 2025 Jan 15, 2025
97691 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-propylaminocarbonyl-4-quinolone 0.048 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
47843 KOR CLONED HUMAN 3H-U69,593 MCL-144 0.049 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
17920 CCK2 PANCREAS GUINEA PIG 125I-CCK CCK 0.05 Lotti VJ et al., 1988 Jan 15, 2025 Jan 15, 2025
100609 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-4-phenyl-2(2H)-oxoimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.05 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
8450 SST5 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.05 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
7428 MOR CLONED HUMAN 3H-DAMGO Naloxonazine 0.05 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
29188 SST2 CLONED HUMAN UNDEFINED L-779,976 0.05 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
9992 CB2 CLONED MOUSE 3H-CP-55940 SR 144528 0.05 Griffin G, Tao Q, Abood ME, 2000 Jan 15, 2025 Jan 15, 2025
19724 D2 CLONED HUMAN UNDEFINED BUTACLAMOL,(+) 0.05 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
5647 Alpha2C CELLS OK 3H-RAUWOLSCINE WIN 53024 0.05 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
60440 GABAA CLONED HUMAN FNZ QH-II-090 0.05 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
63774 CXCR3 PHA/IL-2 T cells HUMAN 125I-CXCL11 CXCL11 0.05 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
60451 GABAA CLONED HUMAN FNZ QH-II-077 0.05 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
53030 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan 0.05 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
32810 D2 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.05 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
22323 A1 BRAIN BOVINE 3H-DPCPX DPCPX 0.05 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
38963 nAChR BRAIN RAT 3H-Cytisine Epibatidine-(+) 0.05 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
6709 D2 ANTERIOR PITUITARY PIG 3H-SPIPERONE NEMONAPRIDE 0.05 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
29237 SST5 CLONED HUMAN UNDEFINED somatostatin-28 0.05 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
38968 nAChR BRAIN RAT 3H-Cytisine A-85380 0.05 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
8763 SST2 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.05 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
16957 5-HT4B CLONED HUMAN 3H-GR-113808 SB207710 0.05 Bach T, et al., 2001 Jan 15, 2025 Jan 15, 2025
8766 SST2 CLONED HUMAN 125I-Tyr3-octreotide RC 160 0.05 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
16958 5-HT4B CLONED HUMAN 3H-GR-113808 GR 113808 0.05 Bach T, et al., 2001 Jan 15, 2025 Jan 15, 2025
16959 5-HT4B CLONED HUMAN 3H-GR-113808 3H-GR113808 0.05 Bach T, et al., 2001 Jan 15, 2025 Jan 15, 2025
9536 SLC6A4 CLONED HUMAN 3H-CITALOPRAM CHLORIMIPRAMINE 0.05 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
13632 D2 HIPPOCAMPUS HUMAN 125I-Epidepride SPIPERONE 0.05 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
8774 SST5 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.05 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
9804 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.05 Nonno,Pannacci,Lucini, Angeloni,Fraschini,Stankov Jan 15, 2025 Jan 15, 2025
32849 D4 CLONED RAT 3H-SPIPERONE SPIPERONE 0.05 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
16226 D2 CLONED MOUSE 3H-SPIPERONE EPIDEPRIDE 0.05 Neve KA, 1990 Jan 15, 2025 Jan 15, 2025
97643 SST2 CLONED HUMAN 125I-LTT-SST-28 L-779,976 0.05 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
7802 GABAA CLONED HUMAN 3H-RO-15-1788 CGS 8216, 1 0.05 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
50044 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-CONH2, [Aib7] 0.05 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
97663 SST2 CLONED HUMAN Functional L-779,976 0.05 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
63360 nAChR CORTEX RAT 3H-Nicotine (-), S Epibatidine 0.05 Bencherif, M et al., 1998 Jan 15, 2025 Jan 15, 2025
50050 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-CONH2, [Aib7,Aib11] 0.05 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
10888 D3 CLONED RAT 3H-YM 09151-2 YM-09151-2 0.05 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
41866 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine 0.05 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
29835 nAChR UNDEFINED UNDEFINED 3H-NICOTINE Azabicyclo[2.2.1]heptane 0.05 Schmitt JD, et al., 1999 Jan 15, 2025 Jan 15, 2025
85652 nAChR CLONED HUMAN 3H-Epibatidine 3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 0.05 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
34198 D2 Striatal Membranes RAT 125I-IABN BUTACLAMOL,(+) 0.05 Luedtke RR, et al., 2000 Jan 15, 2025 Jan 27, 2025
42904 CaMK CLONED HUMAN 3H-Staurosporine Staurosporine 0.05 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
42905 CaMK CLONED HUMAN 3H-Staurosporine Staurosporine 0.05 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
47513 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PYY,[leu31,Pro34], human 0.05 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
5793 Alpha2A CELLS HT29 3H-RAUWOLSCINE WIN 53024 0.05 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
65441 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-077 0.05 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
100772 PDE3b CLONED HUMAN Functional Trequinsin 0.05 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
6821 Y4 CLONED HUMAN 125I-PYY PP, human 0.05 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
9639 SLC6A4 CORTEX RAT 3H-CITALOPRAM PAROXETINE 0.05 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
10408 FOREBRAIN RAT 3H-Epibatidine Epibatidine 0.05 Xiao,Meyer,Thompson,Surin,Wroblewski,Kellar, 1998 Jan 15, 2025 Jan 15, 2025
30893 BRAIN RAT 3H-Cytisine 3-(2(R)-Azetidinylmethoxy)pyridine Dihydrochloride 0.05 Abreo MA, et al., 1996 Jan 15, 2025 Jan 15, 2025
65457 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-090 (CGS-8216) 0.05 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
48060 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.05 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
7871 GABAA CLONED HUMAN 3H-RO-15-1788 2 0.05 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
9173 SST3 CLONED MOUSE 125I-CGP23996 SRIF-D-Trp8 0.05 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
40158 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.05 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
31976 D2 CORTEX RAT 125I-Epidepride SPIPERONE 0.05 Kessler, R.M., et. al., 1993 Jan 15, 2025 Jan 15, 2025
10476 BRAIN RAT 3H-Cytisine A-85380 0.05 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
9453 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.05 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
10477 BRAIN RAT 3H-Cytisine A-159470 0.05 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
10483 nAChR CLONED HUMAN 3H-Cytisine Epibatidine-(+) 0.05 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
8693 SST5 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.05 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
63733 nAChR BRAIN MICE 3H-NICOTINE Epibatidine-(-) 0.05 Damaj, MI et al., 1998 Jan 15, 2025 Jan 15, 2025
50427 SST2 CLONED HUMAN 125I-LTT-SST-28 MK 678 0.05 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
60448 GABAA CLONED HUMAN FNZ XLI-286 0.051 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
55626 CHRNA4 UNDEFINED RAT UNDEFINED cis-3-(5-Isopropyloxy-3-pyridinyl)-3,7-diazabicyclo[3.3.0]octane Semi(fumarate) 0.051 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
65453 GABAA CLONED HUMAN [3H] Flunitrazepam XLI-286 0.051 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
56104 MOR UNDEFINED HUMAN UNDEFINED CCDC 710249, HCl salt 0.052 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
31060 BRAIN RAT 3H-Cytisine A-85380 0.052 Abreo MA, et al., 1996 Jan 15, 2025 Jan 15, 2025
53274 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(6-fluoro-5-(3-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.053 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
32809 D2 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.053 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
23389 NK3 BRAIN CORTEX RAT 125I-BH Eledoisin NKB [MePhe7] 0.053 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
59270 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-methyl-7-azabicyclo[2.2.1]heptane 0.053 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
63625 KOR BRAIN GUINEA PIG 3H-U69,593 (3S)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-2-methyl-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide 0.053 Thomas JB, et al., 2003 Jan 15, 2025 Jan 28, 2025
23398 NK1 ILEUM RAT 125I-Bolton Hunter Substance P 0.054 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
27340 Alpha2A CLONED HUMAN 3H-RX821002 LISURIDE 0.0549541 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
56357 CHRNA4 UNDEFINED RAT UNDEFINED 2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine 0.055 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
62026 nAChR CLONED HUMAN 3H-Cytisine, (-) ABT-594 0.055 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
21494 nAChR CLONED Xenopus 3H-Epibatidine NBEP 0.055 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
61272 GABAA CLONED HUMAN FNZ YT-II-76 0.056 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
65446 nAChR CLONED HUMAN [3H] Flunitrazepam YT-II-76 0.056 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
63214 KOR CEREBELLUM GUINEA PIG 3H-Bremazocine Tyr-D-Ser-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) 0.0568 Story, S.C. et al., 1992 Jan 15, 2025 Jan 15, 2025
42457 D5 CLONED HUMAN 3H-SCH23390 4-chloro-3-hydroxy-dibenz[d,g]azecine 0.057 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
40154 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluoroacetic Acid Salt 0.057 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40174 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide 0.057 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
17383 Alpha1D CLONED HUMAN 3H-PRAZOSIN Tamsulosin 0.057544 Hancock A, et al., 2001 Jan 15, 2025 Jan 15, 2025
22013 LHRH Pituitary RAT UNDEFINED 21 0.057544 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
55627 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(5-(Benzyloxy)pyridin-3-yl)octahydropyrrolo[3,4-c]pyrrole 0.058 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
59274 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.058 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
34566 FOREBRAIN RAT 3H-Epibatidine Epibatidine, (+/-) 0.059 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
41773 CLONED HUMAN Functional (+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.059 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
49470 KOR CLONED HUMAN 3H-Diprenorphine Dynorphin A(1-11)-NH2 0.059 Schlechtingen, G et al., 2003 Jan 15, 2025 Jan 15, 2025
23396 NK1 ILEUM GUINEA PIG 125I-Bolton Hunter Substance P 0.059 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
34546 nAChR CLONED RAT 3H-Epibatidine A-85380-I 0.059 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
10758 D2 CLONED RAT 3H-LSD SPIPERONE 0.06 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
100614 CGRP SPLEEN marmoset 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.06 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
8455 SST5 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.06 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
48144 Y4 CLONED HUMAN 3H-Propionyl-NPY PP, human 0.06 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
10773 CLONED RAT 3H-LSD TIOSPERONE 0.06 ROTH ET AL., 1993 Jan 15, 2025 Jan 15, 2025
100885 AChE BRAIN HUMAN Functional N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide 0.06 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 29, 2025
53014 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(cinnamoylacetamido)morphinan 0.06 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
11034 H1 CLONED HUMAN 3H-MEPYRAMINE CYPROHEPTADINE 0.06 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
63770 CXCR3 H9 HUMAN 125I-CXCL11 CXCL11 0.06 Heise CE, et al., 2005 Jan 15, 2025 Jan 15, 2025
100638 CGRP SPLEEN marmoset Functional 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.06 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
60449 GABAA CLONED HUMAN FNZ QH-II-077 0.06 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
16165 D2 CLONED RAT 125I-IODOSULPRIDE SPIPERONE 0.06 Sokoloff P, et al., 1990 Jan 15, 2025 Jan 15, 2025
6702 D2 CLONED HUMAN 3H-SPIPERONE EPIDEPRIDE 0.06 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
4400 5-HT1D CLONED RAT 3H-5HT DHE 0.06 HAMBLIN MW, ET AL., 5/1992 Jan 15, 2025 Jan 15, 2025
60464 GABAA CLONED HUMAN FNZ QH-II-085 0.06 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
32817 D2 STRIATUM CANINE 3H-SPIPERONE YM-09151-2 0.06 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
20530 A1 myocardial membranes BOVINE 125I-HPIA DPCPX 0.06 Lohse MJ et al., 1987 Jan 15, 2025 Jan 15, 2025
6454 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 GR 113808 0.06 HEGDE SS, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
48184 Y4 CLONED HUMAN 125I-hPP PP, guinea pig 0.06 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
9529 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PAROXETINE 0.06 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
23867 D2 CLONED HUMAN UNDEFINED PIMOZIDE 0.06 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
6719 D2 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.06 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
9792 retina RABBIT 3H-Dopamine release Luzindole,5-Methoxy 0.06 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
9793 retina RABBIT 3H-Dopamine release GR 128107 0.06 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
11846 Alpha1A CLONED HUMAN 3H-PRAZOSIN PRAZOSIN 0.06 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
8775 SST5 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.06 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
11849 Alpha1B CLONED HUMAN 3H-PRAZOSIN PRAZOSIN 0.06 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
11852 Alpha1D CLONED HUMAN 3H-PRAZOSIN PRAZOSIN 0.06 Millan MJ, et al., 2000 Jan 15, 2025 Jan 15, 2025
55628 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(5-Bromopyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate 0.06 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
8535 5-HT4A CLONED HUMAN 3H-GR-113808 SB204070 0.06 Bender E, et al., 2000 Jan 15, 2025 Jan 15, 2025
53084 KOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan 0.06 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
63069 MC4 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-His-DNal(2')Arg-Trp-Lys]-NH2 0.06 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
8809 SST5 CLONED HUMAN 125I-CGP23996 seglitide 0.06 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
7803 GABAA CLONED HUMAN 3H-RO-15-1788 2 0.06 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
10875 D2 CLONED RAT 3H-SPIPERONE ETICLOPRIDE 0.06 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
47740 Y1 CLONED RAT [125I] - Peptide YY NPY, porcine 0.06 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
4478 D2 BRAIN RAT 3H-SPIPERONE SPIPERONE 0.06 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
15231 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 8-OH-DPAT 0.06 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
50049 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-CONH2,[MeAla15] 0.06 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
10882 D3 CLONED RAT 3H-YM 09151-2 YM-09151-2 0.06 Tang L, et al. 1994 Jan 15, 2025 Jan 15, 2025
55951 KOR UNDEFINED HUMAN UNDEFINED 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 0.06 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
65428 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-085 0.06 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
8342 SST2 CLONED HUMAN 125I-Tyr10-CST14 somatostatin-28 0.06 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
65439 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-077 0.06 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
7840 GABAA CLONED HUMAN 3H-RO-15-1788 4 0.06 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
5794 Alpha2A CELLS HT29 3H-RAUWOLSCINE BDF6143 0.06 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
172 5-HT1A CELLS C0S-7 3H-8-OH-DPAT 8-OH-DPAT 0.06 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
12720 Adrenal Membranes RAT 125I-Angiotensin II L-162,193 0.06 Beauchamp HT, et al., 1995 Jan 15, 2025 Jan 15, 2025
4541 5-HT2A BRAIN RAT 3H-SPIPERONE TIOSPERONE 0.06 ROTH BL, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
13757 D2 Putamen HUMAN 125I-Epidepride SPIPERONE 0.06 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
10432 FOREBRAIN RAT 3H-Epibatidine Low Epibatidine-(+) 0.06 Houghtling RA, Davila-Garcia MI, Kellar KJ, 1995 Jan 15, 2025 Jan 15, 2025
10433 FOREBRAIN RAT 3H-Epibatidine Low Epibatidine-(-) 0.06 Houghtling RA, Davila-Garcia MI, Kellar KJ, 1995 Jan 15, 2025 Jan 15, 2025
31695 D2 STRIATUM RAT 125I-Epidepride SPIPERONE 0.06 Kessler, R.M., et. al., 1993 Jan 15, 2025 Jan 15, 2025
17876 CCK1 Gallbladder GUINEA PIG 125I-CCK-8 FK480 0.06 Ito H et al., 1993 Jan 15, 2025 Jan 15, 2025
26324 GAL1 CLONED RAT 125I-GALANIN Galanin, Porcine 0.06 Howard AD, et al., 1997 Jan 15, 2025 Jan 15, 2025
4578 5-HT2A BRAIN RAT 3H-KETANSERIN TIOSPERONE 0.06 ROTH BL, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
9707 MT1 CLONED HUMAN 125I-Iodomelatonin Melatonin,2-Iodo 0.06 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
16363 Y2 jejunal crypt cells RAT [125I] - Peptide YY PYY, porcine 0.06 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
18155 NET FOREBRAIN RAT 3H-Nisoxetine DESIPRAMINE 0.06 Davids E et al., 2002 Jan 15, 2025 Jan 15, 2025
47856 CLONED HUMAN 3H-CGRP 8-37 h-alpha-CGRP 8-37 0.06 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
4082 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl NTB 0.06 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
8434 SST5 CLONED HUMAN 125I-CGP23996 CST17 0.06 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
10482 nAChR CLONED HUMAN 3H-Cytisine Epibatidine-(-) 0.06 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
8437 SST5 CLONED HUMAN 125I-CGP23996 seglitide 0.06 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
15349 5-HT1D CLONED RAT 3H-5HT DHE 0.06 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
8694 SST5 CLONED HUMAN 125I-Tyr3-octreotide seglitide 0.06 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
37623 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.06 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
9726 MT2 CLONED HUMAN 125I-Iodomelatonin S 20098 0.06 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
9982 CB2 CLONED RAT 3H-CP-55940 CP 55,940 0.06 Griffin G, Tao Q, Abood ME, 2000 Jan 15, 2025 Jan 15, 2025
56352 CHRNA4 UNDEFINED RAT UNDEFINED Epibatidine 0.061 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
99916 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 0.061 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
47744 Y1 CLONED RAT [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.061 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
34965 nAChR CLONED UNDEFINED 3H-Epibatidine Epibatidine 0.061 Wei ZL, et al., 2005 Jan 15, 2025 Jan 15, 2025
34540 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.061 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
28925 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.061 Wei ZL, et. al., 2003 Jan 15, 2025 Jan 15, 2025
89625 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
56355 CHRNA4 UNDEFINED RAT UNDEFINED 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine 0.062 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56359 CHRNA4 UNDEFINED RAT UNDEFINED (S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine 0.062 Gao Y et al., 2009 Jan 15, 2025 Jan 15, 2025
59304 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[5-(4-Chlorophenyl)-6-fluoro-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.062 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
47787 MOR CLONED HUMAN 3H-DAMGO Cyclorphan 0.062 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
21498 CCR5 CLONED Xenopus 3H-Epibatidine NNEP 0.062 Avalos M et al., 2002 Jan 15, 2025 Jan 15, 2025
91682 A1 CORTICAL MEMBRANES RAT 3H-DPCPX N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide 0.0628 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
99623 A2A CLONED HUMAN 3H-NECA 8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine 0.063 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
16949 5-HT4A CLONED HUMAN 3H-GR-113808 3H-GR113808 0.063 Bach T, et al., 2001 Jan 15, 2025 Jan 15, 2025
17325 Alpha1A CEREBRAL CORTEX PIG 3H-PRAZOSIN METHIOTHEPIN 0.0630957 Wikberg-Matsson A, et al., 1998 Jan 15, 2025 Jan 15, 2025
27088 MOR BRAIN MOUSE 3H-DAMGO Dmt-d-Arg-Phe-A2pr-NH2 0.0636 Zhao GM, et al., 2003 Jan 15, 2025 Jan 15, 2025
60447 GABAA CLONED HUMAN FNZ XLI-286 0.064 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
38965 nAChR BRAIN RAT 3H-Cytisine dechloroepibatidine-(+) 0.064 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
59306 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[5-(4-Chlorophenyl)-6-fluoro-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.064 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
65454 nAChR CLONED HUMAN [3H] Flunitrazepam XLI-286 0.064 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
89630 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0645654 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
51200 CHRNA4 UNDEFINED RAT UNDEFINED 6-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane 0.065 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
42077 M5 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.065 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
47728 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY, zebrafish 0.066 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
19837 D4 CLONED HUMAN UNDEFINED BENPERIDOL 0.066 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
59318 nAChR BRAIN CORTEX RAT 3H-Epibatidine 4-[5-(7-Azabicyclo[2.2.1]hept-2-yl)-2-fluoro-3-pyridinyl]benzonitrile 0.066 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
24733 Y1 CLONED HUMAN 125I-PYY NPY, porcine 0.0660693 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
42134 Alpha2C CLONED HUMAN 35S-GTPGammaS MK-912 0.0676083 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
49058 SST2 CLONED HUMAN 125I-Tyr11-SRIF Somatostatin-14 0.0676083 Feniuk W, et.al., 2000 Jan 15, 2025 Jan 15, 2025
49063 SST2 CLONED RAT 125I-Tyr11-SRIF Somatostatin-14 0.0676083 Feniuk W, et.al., 2000 Jan 15, 2025 Jan 15, 2025
32482 NOP CLONED HUMAN 35S-GTPGammaS OFQ/N UFP-102 0.0676083 Carra' G., et.al., 2004 Jan 15, 2025 Jan 15, 2025
17885 CCK2 BRAIN RAT 125I-CCK-8 YM022 0.068 Nishida A et al., 1994 Jan 15, 2025 Jan 15, 2025
32808 D2 CLONED RAT 3H-SPIPERONE SPIPERONE 0.069 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
97838 5-HT2A CLONED HUMAN Functional RITANSERIN 0.0691831 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
28764 SST2 CLONED HUMAN 125I-Tyr10-CST14 somatostatin-28 0.0691831 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
85185 MT2 CHO-K1 HUMAN 125I-Iodomelatonin Tasimelteon 0.0692 Lavedan C et al 2015 Jan 15, 2025 Jan 29, 2025
7432 MOR CLONED HUMAN 3H-DAMGO DIPRENORPHINE-HCl 0.07 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
8979 SST2 CLONED HUMAN 125I-SRIF-28 MK 678 0.07 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
8980 SST2 CLONED HUMAN 125I-SRIF-28 RC 160 0.07 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
87323 Alpha1A placeholder HUMAN Placeholder Tamsulosin 0.07 Rak A et al 2016 Jan 15, 2025 Jan 28, 2025
60457 GABAA CLONED HUMAN FNZ QH-II-092 0.07 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
34348 nAChR CORTEX RAT 3H-NICOTINE Epibatidine 0.07 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 15, 2025
5421 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 SB204070 0.07 Van den Wyngaert I, et al., 1997 Jan 15, 2025 Jan 15, 2025
8750 SST2 CORTEX HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.07 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
20526 A1 myocardial membranes BOVINE 3H-DPCPX DPCPX 0.07 Lohse MJ et al., 1987 Jan 15, 2025 Jan 15, 2025
4401 5-HT1D CLONED RAT 3H-5HT ERGOTAMINE 0.07 HAMBLIN MW, ET AL., 5/1992 Jan 15, 2025 Jan 15, 2025
54067 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-quinolyl)acetamido]morphinan 0.07 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
13620 D2 N. Accumbens HUMAN 125I-Epidepride SPIPERONE 0.07 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
13624 D2 FR. CORTEX HUMAN 125I-Epidepride SPIPERONE 0.07 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
62028 nAChR CLONED HUMAN 3H-Cytisine, (-) Epibatidine, (+/-) 0.07 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
29005 SST5 CLONED HUMAN 125I-LTT-SST-28 somatostatin-28 0.07 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
5467 5-HT4D CLONED HUMAN 3H-GR-113808 GR 113808 0.07 BLONDEL O, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
8808 SST5 CLONED HUMAN 125I-CGP23996 somatostatin-28 0.07 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
13672 nAChR CLONED HUMAN 3H-Cytisine, (-) Epibatidine, (+/-) 0.07 Gopalakrishnan M, et al., 1996 Jan 15, 2025 Jan 15, 2025
8554 SST2 CLONED MOUSE 125I-Tyr11-somatostatin-14 MK 678 0.07 Yasuda K, et al., 1992 Jan 15, 2025 Jan 15, 2025
37739 SST2 CLONED HUMAN UNDEFINED D-Trp8-SRIF-14 0.07 Neelamkavil S, et al., 2005 Jan 15, 2025 Jan 15, 2025
8560 SST1 CLONED HUMAN 125I-Tyr11-SRIF somatostatin-28 0.07 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
7808 GABAA CLONED HUMAN 3H-RO-15-1788 7 0.07 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
2690 5-HT2A CORTEX HUMAN 3H-SPIPERONE PRAZOSIN 0.07 ANDORN ET AL., 1984 Jan 15, 2025 Jan 15, 2025
45446 SLC6A4 CLONED HUMAN 3H-CITALOPRAM Duloxetine 0.07 Vaishnavi SN, et al., 2004 Jan 15, 2025 Jan 15, 2025
18571 CCK1 PANCREAS RAT 125I-BH-CCK-8 2 0.07 Pierson ME et al., 1997 Jan 15, 2025 Jan 15, 2025
55950 KOR UNDEFINED HUMAN UNDEFINED Cyclazocine 0.07 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
14225 D2 CLONED RAT 3H-Methylspiperone SPIPERONE 0.07 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 27, 2025
14229 D2 CLONED RAT 3H-Methylspiperone SPIPERONE 0.07 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 27, 2025
14232 D2 CLONED RAT 3H-Methylspiperone ETICLOPRIDE 0.07 Lawler C.P. et. Al., 1999 Jan 15, 2025 Jan 27, 2025
65435 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-092 0.07 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
8606 SST3 CLONED MOUSE 125I-Tyr11-SRIF Somatostatin-14 0.07 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
8607 SST3 CLONED MOUSE 125I-Tyr11-SRIF somatostatin-28 0.07 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
52127 MOR UNDEFINED HUMAN UNDEFINED 6-(4-((phenethylamino)methyl)phenoxy)nicotinamide 0.07 Takeuchi K et al., 2007 Jan 15, 2025 Jan 15, 2025
9125 SST1 CLONED HUMAN 125I-CGP23996 somatostatin-28 0.07 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
8359 SST2 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.07 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
6826 Y4 CLONED HUMAN 125I-PYY PP, BOVINE 0.07 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
8620 SST3 CLONED MOUSE 125I-Tyr11-SRIF L-362,823 0.07 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
10434 FOREBRAIN RAT 3H-Epibatidine Low Epibatidine 0.07 Houghtling RA, Davila-Garcia MI, Kellar KJ, 1995 Jan 15, 2025 Jan 15, 2025
12738 5-HT1A BRAIN RAT 3H-8-OH-DPAT LY 293284 0.07 Foreman MM, et al., 1994 Jan 15, 2025 Jan 15, 2025
65991 nAChR BRAIN RAT 3H-Cytisine Epibatidine, (+/-) 0.07 Holladay MW et al., 1997 Jan 15, 2025 Jan 15, 2025
93646 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 0.07 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
28879 SST3 CLONED RAT 125I-Tyr11-somatostatin Somatostatin-14 0.07 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
9172 SST3 CLONED MOUSE 125I-CGP23996 somatostatin-28 0.07 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
26325 GAL1 CLONED RAT 125I-GALANIN Galanin, Human 0.07 Howard AD, et al., 1997 Jan 15, 2025 Jan 15, 2025
8667 SST5 CLONED RAT 125I-Tyr11-SRIF BIM 23059 0.07 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
47838 KOR CLONED HUMAN 3H-U69,593 MCL-176 0.07 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
29154 SST2 CLONED HUMAN 125I-Tyr11-SRIF MK 678 0.07 Reisine T, et.al., 1995 Jan 15, 2025 Jan 15, 2025
11497 5-HT2A CLONED HUMAN 125I-R091150 BW501 0.07 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
10479 BRAIN RAT 3H-Cytisine Epibatidine-(+) 0.07 Sullivan, et al., 1996 Jan 15, 2025 Jan 15, 2025
8432 SST5 CLONED HUMAN 125I-CGP23996 somatostatin-28 0.07 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
10228 CLONED RAT 125I-HEAT PRAZOSIN 0.07 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
16372 Y2 jejunal crypt cells RAT [125I] - Peptide YY NPY, C2 0.07 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
15350 5-HT1D CLONED RAT 3H-5HT ERGOTAMINE 0.07 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
16636 Y4 CLONED HUMAN 125I-hPP PP, human 0.07 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
91681 A1 CORTICAL MEMBRANES RAT 3H-DPCPX 4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide 0.0709 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
48186 Y4 CLONED HUMAN 125I-hPP PP, rat 0.071 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
18717 CGRP1 CLONED PIG 125-h alpha-CGRP [N-benzol]h alpha-CGRP8-37 0.072 Rorabaugh BR et al., 2001 Jan 15, 2025 Jan 15, 2025
56099 MOR UNDEFINED HUMAN UNDEFINED (1R,9R,10S,13R)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide 0.072 Wentland MP et al., 2009 Jan 15, 2025 Jan 15, 2025
99958 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.072 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
29392 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.072 Jensen AA, et al., 2003 Jan 15, 2025 Jan 27, 2025
53278 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(5-(3-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.073 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
38964 nAChR BRAIN RAT 3H-Cytisine Epibatidine-(-) 0.073 Bisson WH, et al., 2005 Jan 15, 2025 Jan 15, 2025
54134 TRPV1 UNDEFINED RAT UNDEFINED [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1,10}.0^{2,6}.0^{11,15}]octadeca-3,8-dien-8-yl]methyl 2-(2-fluorophenyl)acetate 0.073 Choi HK et al., 2009 Jan 15, 2025 Jan 15, 2025
34493 CCR5 CLONED RAT 3H-Epibatidine A-85380 0.073 Xiao Y et al., 2004 Jan 15, 2025 Jan 15, 2025
22018 LHRH Pituitary RAT UNDEFINED 26 0.074131 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
69261 H3 CLONED RAT 3H-Alpha-Me-histamine GT 2331 0.074131 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
99649 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-oxo-ethoxy)-4-methoxy}-phenyl]-xanthine 0.075 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
30932 KOR CLONED HUMAN 3H-Diprenorphine TRK-820 0.075 Wang Y, et. al., 2004 Jan 15, 2025 Jan 15, 2025
32481 NOP CLONED HUMAN 35S-GTPGammaS OFQ/N UFP-102 0.0758578 Carra' G., et.al., 2004 Jan 15, 2025 Jan 15, 2025
60458 GABAA CLONED HUMAN FNZ JYI-57 0.076 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60459 GABAA CLONED HUMAN FNZ JYI-57 0.076 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
99652 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 0.076 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
65467 GABAA CLONED HUMAN [3H] Flunitrazepam JYI-57 0.076 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65468 nAChR CLONED HUMAN [3H] Flunitrazepam JYI-57 0.076 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
47839 KOR CLONED HUMAN 3H-U69,593 MCL-139 0.076 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
21486 nAChR CLONED Xenopus 3H-Epibatidine NNEP 0.077 Avalos M et al., 2002 Jan 15, 2025 Jan 27, 2025
69260 H3 CLONED RAT 3H-Alpha-Me-histamine Imetit 0.0776247 Krueger KM, et al., 2005 Jan 15, 2025 Jan 15, 2025
22011 LHRH Pituitary RAT UNDEFINED 19 0.0776247 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
59296 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Fluoro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.078 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
59310 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Fluoro-5-(4-fluorophenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.078 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
47845 KOR CLONED HUMAN 3H-U69,593 MCL-145 0.078 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
27884 mGluR2, mGluR3 BRAIN CORTEX RAT 3H-DCG IV LY341495 0.078 Mutel V, et.al., 1998a Jan 15, 2025 Jan 15, 2025
50949 KOR UNDEFINED HUMAN UNDEFINED 17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol 0.079 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
16947 5-HT4A CLONED HUMAN 3H-GR-113808 SB207710 0.079 Bach T, et al., 2001 Jan 15, 2025 Jan 15, 2025
16948 5-HT4A CLONED HUMAN 3H-GR-113808 GR 113808 0.079 Bach T, et al., 2001 Jan 15, 2025 Jan 15, 2025
16481 Beta2 CLONED HUMAN 125I-Pindolol Fluorocarazolol,(S) 0.079 Roth BL, et al., 2001 Jan 15, 2025 Jan 28, 2025
16998 M2 CLONED HUMAN 3H-NMS NNC 11-1585 0.079 Christopoulos A, et al., 2001 Jan 15, 2025 Jan 15, 2025
59312 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Fluoro-5-(4-fluorophenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.079 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
47830 KOR CLONED HUMAN 3H-U69,593 MCL-101 0.079 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
68899 SST2 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ala-Cys}-NH2 0.0794328 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
86599 5-HT4 CLONED HUMAN 3H-GR-113808 1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide 0.0794328 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
17326 Alpha1A CEREBRAL CORTEX PIG 3H-PRAZOSIN WB 4101 0.0794328 Wikberg-Matsson A, et al., 1998 Jan 15, 2025 Jan 15, 2025
68829 SST2 CLONED HUMAN 125I-SRIF RC 160 0.0794328 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
68834 SST2 CLONED HUMAN 125I-SRIF MK 678 0.0794328 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
17922 CCK2 PANCREAS GUINEA PIG 125I-CCK L-364,718 0.08 Lotti VJ et al., 1988 Jan 15, 2025 Jan 15, 2025
7430 MOR CLONED HUMAN 3H-DAMGO LEVORPHANOL-tartarate 0.08 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
5648 Alpha2C CELLS OK 3H-RAUWOLSCINE BDF6143 0.08 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
51989 DOR UNDEFINED HUMAN UNDEFINED 14beta-(2'-chlorocinnamoylamino)-7,8-dihydromorphinone 0.08 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
6680 D2 CLONED HUMAN 3H-NEMONAPRIDE NEMONAPRIDE 0.08 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
60441 GABAA CLONED HUMAN FNZ QH-II-090 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
30491 M2 CLONED HUMAN 3H-QNB exo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 0.08 Kim MG, et al., 2003 Jan 15, 2025 Jan 15, 2025
18716 CGRP1 CLONED PIG 125-h alpha-CGRP h alpha-CGRP 0.08 Rorabaugh BR et al., 2001 Jan 15, 2025 Jan 15, 2025
60450 GABAA CLONED HUMAN FNZ QH-II-077 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
52774 5-HT2A UNDEFINED HUMAN UNDEFINED Ziprasidone 0.08 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
60462 GABAA CLONED HUMAN FNZ QH-II-085 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
20527 A1 myocardial membranes BOVINE 3H-DPCPX XAC 0.08 Lohse MJ et al., 1987 Jan 15, 2025 Jan 15, 2025
52783 5-HT2A UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isoxazole-5-carboxamide 0.08 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
8752 SST2 CORTEX HUMAN 125I-Tyr3-octreotide seglitide 0.08 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
60465 GABAA CLONED HUMAN FNZ QH-II-085 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
42039 M3 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.08 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
8505 SST3 CLONED HUMAN 125I-CGP23996 LTT-SRIF28 0.08 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
13628 D2 Temp. Cortex HUMAN 125I-Epidepride SPIPERONE 0.08 Joyce JN, et al., 1991 Jan 15, 2025 Jan 15, 2025
6718 D2 ANTERIOR PITUITARY PIG 3H-SPIPERONE SPIPERONE 0.08 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
329 5-HT1A CORTEX RAT 3H-WB4101 LISURIDE 0.08 NORMAN ET AL., 1985 Jan 15, 2025 Jan 15, 2025
844 5-HT2C Choroid Plexus PIG 125I-LSD METERGOLINE 0.08 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
5711 Alpha2C KIDNEY OPOSSUM 3H-RAUWOLSCINE RAUWOLSCINE 0.08 BLAXALL H. ET AL., 1991 Jan 15, 2025 Jan 15, 2025
32850 D4 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.08 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
9047 SST4 CLONED RAT 125I-CGP23996 BIM 23059 0.08 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
8546 SST4 CLONED RAT 125I-Tyr11-SRIF somatostatin-28 0.08 O'Carroll AM, et al., 1993 Jan 15, 2025 Jan 15, 2025
8553 SST2 CLONED MOUSE 125I-Tyr11-somatostatin-14 Somatostatin-14 0.08 Yasuda K, et al., 1992 Jan 15, 2025 Jan 15, 2025
56697 MOR UNDEFINED HUMAN UNDEFINED (4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol 0.08 Hsin LW et al., 2010 Jan 15, 2025 Jan 15, 2025
7805 GABAA CLONED HUMAN 3H-RO-15-1788 4 0.08 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
19069 CLONED RAT 125-AcHis1-PACAP-27 PACAP(1-27) 0.08 Ciccarelli E et al., 1995 Jan 15, 2025 Jan 15, 2025
50045 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-CONH2, [Aib11] 0.08 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
41864 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-5-ylamine 0.08 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
9612 CORTEX RAT 3H-NMS ATR 0.08 Owens MJ, et al, 1997 Jan 15, 2025 Jan 15, 2025
6801 Y1 CLONED HUMAN 125I-PYY NPY, human 0.08 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
65427 GABAA CLONED HUMAN [3H] Flunitrazepam QH-II-085 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
8341 SST2 CLONED HUMAN 125I-Tyr10-CST14 Somatostatin-14 0.08 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
65430 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-085 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
47514 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PP, human 0.08 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
7837 GABAA CLONED HUMAN 3H-RO-15-1788 CGS 8216, 1 0.08 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
7838 GABAA CLONED HUMAN 3H-RO-15-1788 2 0.08 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
65440 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-077 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
6822 Y4 CLONED HUMAN 125I-PYY PP2-36, HUMAN 0.08 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
8361 SST2 CLONED HUMAN 125I-CGP23996 LTT-SRIF28 0.08 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
65458 nAChR CLONED HUMAN [3H] Flunitrazepam QH-II-090 (CGS-8216) 0.08 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
13510 D2 STRIATUM RAT 3H-S-Sulpiride SPIPERONE 0.08 Zahniser NR, et al., 1983 Jan 15, 2025 Jan 15, 2025
23752 BRAIN RAT 3H-Cytisine Epibatidine 0.08 Miller DK, et al., 2002 Jan 15, 2025 Jan 15, 2025
7376 KOR CLONED HUMAN 3H-U69,593 Bremazocine 0.08 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
9171 SST3 CLONED MOUSE 125I-CGP23996 Somatostatin-14 0.08 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
29146 SST2 CLONED HUMAN 125I-Tyr11-SRIF Somatostatin-14 0.08 Reisine T, et.al., 1995 Jan 15, 2025 Jan 15, 2025
13532 D2 STRIATUM RAT 3H-SPIPERONE SPIPERONE 0.08 Zahniser NR, et al., 1983 Jan 15, 2025 Jan 15, 2025
54751 SLC6A4 UNDEFINED HUMAN UNDEFINED PAROXETINE 0.08 Strappaghetti G et al., 2008 Jan 15, 2025 Jan 15, 2025
9441 MT1 CLONED HUMAN 125I-Iodomelatonin MELATONIN 0.08 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
7908 GABAA CLONED HUMAN 3H-RO-15-1788 4 0.08 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
7398 KOR CLONED HUMAN 3H-U69,593 Beta C N A 0.08 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
9192 SST3 CLONED MOUSE 125I-CGP23996 L-362,823 0.08 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
68074 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY, human 0.08 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68079 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY Leu31, Pro34, human 0.08 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
55629 CHRNA4 UNDEFINED RAT UNDEFINED cis-2-(5-Methoxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride 0.081 Bunnelle WH et al., 2009 Jan 15, 2025 Jan 15, 2025
23545 H3 BRAIN CORTEX Dog 3H-NAMH Clobenpropit 0.0812831 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
34371 MOR FOREBRAIN RAT 3H-DAMGO Naltrexone 0.0825 Codd EE et al, 1995 Jan 15, 2025 Jan 15, 2025
97837 5-HT2A Membranes HUMAN [3H]-ketanserin RITANSERIN 0.0831764 Vanover, K., et al., 2006 Jan 15, 2025 Jan 15, 2025
87876 A2B test HUMAN 3H-PSB-603 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.0835 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
55683 AChE UNDEFINED HUMAN UNDEFINED N-Allyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine 0.0847 Butini S et al., 2008 Jan 15, 2025 Jan 28, 2025
63506 D3 CLONED HUMAN 3H-N-Methylspiperone Cariprazine 0.085 citrome, Leslie et. al, 2013 Jan 15, 2025 Jan 15, 2025
22012 LHRH Pituitary RAT UNDEFINED 20 0.0851138 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
91680 A1 CORTICAL MEMBRANES RAT 3H-DPCPX N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide 0.0867 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
53276 CHRNA4 UNDEFINED RAT UNDEFINED rac-2-(6-fluoro-5-(3-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride 0.087 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
63042 MC4 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-Pro-DNal(2'Arg-Trp-Lys]-NH2 0.087 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
17098 H1 BRAIN HUMAN 3H-PYRILAMINE OLANZAPINE 0.087 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
28758 SST2 CLONED HUMAN 125I-Tyr10-CST14 Somatostatin-14 0.0870964 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
24732 Y1 CLONED HUMAN 125I-PYY NPY, human 0.0870964 GERALD C, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
50374 Y1 CLONED HUMAN 125I-PYY NPY, human 0.0870964 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
16664 M3 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.088 Bolden C, et al., 1992 Jan 15, 2025 Jan 15, 2025
27885 mGluR2, mGluR3 BRAIN CORTEX RAT 3H-DCG IV (+)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid 0.088 Mutel V, et.al., 1998a Jan 15, 2025 Jan 15, 2025
27502 5-HT1B STRIATUM GUINEA PIG 3H-GR-125743 L694,247 0.0891251 Millan MJ, et al., 2002a Jan 15, 2025 Jan 15, 2025
8708 SST2 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.09 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
9476 HYPOTHALAMUS GUINEA PIG 125I-Iodomelatonin S 20098 0.09 Beresford,Browning,Starkey, Brown, Foord, 1998 Jan 15, 2025 Jan 15, 2025
63501 5-HT1A CLONED RAT 3H-WAY100635 Brexpiprazole 0.09 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
34322 nAChR CLONED RAT 3H-NICOTINE A-85380 0.09 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 15, 2025
11803 FR. CORTEX HUMAN 3H-PRAZOSIN PRAZOSIN 0.09 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
29211 SST3 CLONED HUMAN UNDEFINED NC8-12 0.09 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
32795 D2 STRIATUM CANINE 3H-SPIPERONE ETICLOPRIDE 0.09 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
8736 SST2 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.09 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
60466 GABAA CLONED HUMAN FNZ XHE-II-024 0.09 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
33845 D2 CLONED HUMAN 3H-SPIPERONE YM-09151-2 0.09 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
22329 A1 BRAIN Sheep 3H-DPCPX XAC 0.09 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
60474 GABAA CLONED HUMAN FNZ PWZ-007A 0.09 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
52285 SLC6A4 UNDEFINED HUMAN UNDEFINED PAROXETINE 0.09 Gelmi ML et al., 2007 Jan 15, 2025 Jan 15, 2025
52797 5-HT2A UNDEFINED HUMAN UNDEFINED 6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-amine 0.09 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
6720 D4 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.09 SEBBEN M, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
53069 KOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan 0.09 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
32855 D4 STRIATUM CANINE 3H-SPIPERONE YM-09151-2 0.09 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
9048 SST4 CLONED RAT 125I-CGP23996 BIM 23060 0.09 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
23385 NK1 STTG1 HUMAN 125I-Bolton Hunter SSR240600 0.09 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
6747 D4 CLONED HUMAN 3H-SPIPERONE SPIPERONE 0.09 SEEMAN P, ET AL., 1995 Jan 15, 2025 Jan 27, 2025
63070 MC5 CLONED HUMAN 125I-[Tyr2][Nle,4DPhe7]alpha-MSH (125I-NDP-alpha-MSH), Ac-Nle-c[Asp-His-DNal(2')Arg-Trp-Lys]-NH2 0.09 Grieco, P et al., 2002 Jan 15, 2025 Jan 15, 2025
19816 D4 CLONED HUMAN UNDEFINED Perospirone 0.09 Seeman P, Tallerico T., 1998 Jan 15, 2025 Jan 15, 2025
29038 SST3 CLONED HUMAN 125I-LTT-SST-28 NC8-12 0.09 Patel YC, et.al., 1994 Jan 15, 2025 Jan 15, 2025
18570 CCK1 PANCREAS RAT 125I-BH-CCK-8 1 0.09 Pierson ME et al., 1997 Jan 15, 2025 Jan 15, 2025
7821 GABAA CLONED HUMAN 3H-RO-15-1788 20 0.09 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
6802 Y1 CLONED HUMAN 125I-PYY NPY, porcine 0.09 Gerald et al, 1995 Jan 15, 2025 Jan 15, 2025
8871 GABAA CLONED HUMAN 3H-15-4513 CGS 9895 0.09 Scholze P, et al., 1996 Jan 15, 2025 Jan 27, 2025
6825 Y4 CLONED HUMAN 125I-PYY I31,G34-PP,human 0.09 Bard JA, et. al., 1995 Jan 15, 2025 Jan 15, 2025
10410 FOREBRAIN RAT 3H-Epibatidine A-85380 0.09 Xiao,Meyer,Thompson,Surin,Wroblewski,Kellar, 1998 Jan 15, 2025 Jan 15, 2025
65450 nAChR CLONED HUMAN [3H] Flunitrazepam PWZ-007A 0.09 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
8377 SST2 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.09 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
47801 MOR CLONED HUMAN 3H-DAMGO MCL-144 0.09 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
48064 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.09 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
9414 MT1 CLONED HUMAN 125I-Mel Melatonin,2-Iodo 0.09 Reppert, Godson, Mahle, Weaver, Slaugenhaupt, 1995 Jan 15, 2025 Jan 15, 2025
7881 GABAA CLONED HUMAN 3H-RO-15-1788 12 0.09 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
65489 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-024 0.09 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
47063 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-3P 0.09 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47066 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-4P 0.09 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47069 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-MPM 0.09 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
8680 SST2 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.09 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
18923 H1 CLONED HUMAN 3H-trans-H2-PAT,(-) DOXEPIN 0.09 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
11503 D2 CLONED HUMAN 3H-SPIPERONE BUTACLAMOL,(+) 0.09 Schotte A, et al., 1996 Jan 15, 2025 Jan 27, 2025
34031 KOR CLONED RAT 3H-Diprenorphine Naltrindole G 0.09 Jones, RM et. al., 1998 Jan 15, 2025 Jan 15, 2025
4080 DOR BRAIN GUINEA PIG 3H-DPDPE-Cl NALTRINDOLE 0.09 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11504 D2 CLONED HUMAN 3H-SPIPERONE BUTACLAMOL,(+) 0.09 Schotte A, et al., 1996 Jan 15, 2025 Jan 27, 2025
5621 5-HT4 CLONED HUMAN 3H-GR-113808 GR 113808 0.09 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
16376 Y2 CLONED RAT [125I] - Peptide YY PYY, porcine 0.09 Goumain M, et al., 2001 Jan 15, 2025 Jan 15, 2025
251 5-HT1A CORTEX RAT 3H-WB4101 DIHYDROERGOCRYPTINE 0.09 NORMAN ET AL., 1985 Jan 15, 2025 Jan 15, 2025
100750 MT1 C.H.O. HUMAN 125I-Iodomelatonin MELATONIN 0.091 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
29378 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.091 Jensen AA, et al., 2003 Jan 15, 2025 Jan 27, 2025
50231 Y2 CLONED GUINEA PIG 125I-PYY NPY, porcine 0.092 Sharma P, et al., 1998 Jan 15, 2025 Jan 15, 2025
62827 Brain Frontal Cortex HUMAN 3H-PRAZOSIN PRAZOSIN 0.092 Richelson, Elliott et. al, 1984 Jan 15, 2025 Jan 15, 2025
21997 LHRH Pituitary RAT UNDEFINED 5 0.0933254 Haviv F et al., 1993 Jan 15, 2025 Jan 15, 2025
99653 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine 0.094 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
53829 5-HT1A UNDEFINED RAT UNDEFINED 2-[[4-[4-(2-Methoxyphenyl)-1-piperazinyl]butyl]thio]benzoxazole 0.094 Siracusa MA et al., 2008 Jan 15, 2025 Jan 15, 2025
60711 GABAA CLONED HUMAN FNZ YT-III-25 0.095 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
53295 CHRNA4 UNDEFINED RAT UNDEFINED rac-4-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride 0.095 Ivy Carroll F et al., 2008 Jan 15, 2025 Jan 15, 2025
34929 nAChR CLONED UNDEFINED 3H-Epibatidine Epibatidine 0.095 Wei ZL, et al., 2005 Jan 15, 2025 Jan 27, 2025
65204 GABAA CLONED HUMAN [3H] Flunitrazepam YT-III-25 0.095 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
34501 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.095 Xiao Y et al., 2004 Jan 15, 2025 Jan 27, 2025
28919 nAChR CLONED RAT 3H-Epibatidine Epibatidine, (+/-) 0.095 Wei ZL, et. al., 2003 Jan 15, 2025 Jan 27, 2025
34306 nAChR CLONED RAT 3H-Epibatidine Epibatidine 0.096 Grinevich VP, et al., 2004 Jan 15, 2025 Jan 28, 2025
17887 CCK2 BRAIN RAT 125I-CCK-8 CCK-8 0.097 Nishida A et al., 1994 Jan 15, 2025 Jan 15, 2025
41788 CLONED HUMAN Functional 17beta-Estradiol 0.098 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
86872 D1 Corpus Striatum RAT 3H-SCH23390 N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide 0.0983 Fiorino F et al 2016 Jan 15, 2025 Jan 28, 2025
55861 D3 UNDEFINED UNDEFINED UNDEFINED N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide 0.099 Butini S et al., 2009 Jan 15, 2025 Jan 15, 2025
48641 GNRHR CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48643 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48899 KOR BRAIN RAT 3H-DHM CAM 0.1 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
51204 CHRNA4 UNDEFINED RAT UNDEFINED (1S,4S)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane 0.1 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
8709 SST2 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.1 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
11525 CLONED HUMAN 3H-SUBSTANCE P Substance P 0.1 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
51206 CHRNA4 UNDEFINED RAT UNDEFINED (1R,4R)-2-(6-chloro-5-methoxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane 0.1 Bunnelle WH et al., 2007 Jan 15, 2025 Jan 15, 2025
48647 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48903 KOR BRAIN Frog 3H-DHM CAM 0.1 Benyhe S, et al., 1990 Jan 15, 2025 Jan 15, 2025
29194 SST2 CLONED HUMAN UNDEFINED seglitide 0.1 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
4111 KOR CLONED HUMAN 3H-U69,593 EKC(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
48655 CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
27152 5-HT2A BRAIN RAT 125I-DOI DOI,(-) 0.1 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
48656 GNRHR CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
56848 CB1 UNDEFINED HUMAN UNDEFINED 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-(1-(2-phenylpropan-2-yl)-1H-imidazol-4-yl)-1H-pyrazole 0.1 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
64528 CLONED HUMAN 3H-Estradiol (+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide 0.1 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
12049 H3 Striatal Membranes RAT 3H-RAMHA Imetit 0.1 Ligneau X, et al., 1994 Jan 15, 2025 Jan 15, 2025
8722 SST2 CLONED HUMAN 125I-LTT-SRIF28 Somatostatin-14 0.1 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8724 SST2 CLONED HUMAN 125I-LTT-SRIF28 seglitide 0.1 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
100884 BchE serum HUMAN Functional N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide 0.1 Munoz-Ruiz P, et al., 2005 Jan 15, 2025 Jan 15, 2025
35861 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 0.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
56853 CB1 UNDEFINED HUMAN UNDEFINED 1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-methyl-3-(1-(2-phenylpropan-2-yl)-1H-imidazol-4-yl)-1H-pyrazole 0.1 Dow RL et al., 2009 Jan 15, 2025 Jan 15, 2025
48664 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
4121 KOR CLONED HUMAN 3H-U69,593 CYCLAZOCINE (-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
48665 GNRHR CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
14619 H4 CORTEX GUINEA PIG 3H-Histamine R-alpha-methylhistamine 0.1 Zhu, Yand, et al., 2001 Jan 15, 2025 Jan 15, 2025
72478 5-HT2B test test 3H- LSD METHYSERGIDE 0.1 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
8737 SST2 CLONED HUMAN 125I-CGP23996 somatostatin-28 0.1 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
11042 H1 CEREBELLUM GUINEA PIG 3H-MEPYRAMINE CYPROHEPTADINE 0.1 Moguilevsky N et al, 1994 Jan 15, 2025 Jan 15, 2025
68901 SST4 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ala-Cys}-NH2 0.1 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
53029 MOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan 0.1 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
5414 5-HT4 CLONED HUMAN 3H-GR-113808 SB204070 0.1 Van den Wyngaert I, et al., 1997 Jan 15, 2025 Jan 15, 2025
99622 A2A CLONED HUMAN 3H-NECA 1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine 0.1 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
64550 CLONED HUMAN 3H-Estradiol (+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide 0.1 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
4138 KOR BRAIN GUINEA PIG 3H-U69,593 EKC(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
4139 KOR BRAIN GUINEA PIG 3H-U69,593 BREMAZOCINE(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
17963 CCK2 BRAIN RAT 125I-CCK-8 15c 0.1 Semple G et al., 1997 Jan 15, 2025 Jan 15, 2025
48686 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
38959 T47D HUMAN Functional 5-(4,4-diethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile 0.1 Fensome A, et al., 2005 Jan 15, 2025 Jan 15, 2025
4145 KOR BRAIN GUINEA PIG 3H-U69,593 DYNORPHIN(1-11)-OH 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
38961 T47D HUMAN Functional 5-(4-ethyl-4-methyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile 0.1 Fensome A, et al., 2005 Jan 15, 2025 Jan 15, 2025
67890 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 0.1 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
22322 A1 BRAIN Sheep 3H-DPCPX DPCPX 0.1 Klotz KN et al., 1991 Jan 15, 2025 Jan 15, 2025
35891 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7-Hydroxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
4149 KOR BRAIN GUINEA PIG 3H-U69,593 CYCLAZOCINE (-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
35893 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 7-(2-Methoxyethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ymethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
52789 5-HT2A UNDEFINED HUMAN UNDEFINED N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide 0.1 Graham JM et al., 2008 Jan 15, 2025 Jan 15, 2025
6455 5-HT4 STRIATUM GUINEA PIG 3H-GR-113808 RS 100235 0.1 HEGDE SS, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
11063 H3 CORTEX RAT 3H-methylhistamine Imetit 0.1 Lovenberg, TW et al., 2000 Jan 15, 2025 Jan 15, 2025
54071 MOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-isoquinolyl)acetamido]morphinan 0.1 Li G et al., 2009 Jan 15, 2025 Jan 15, 2025
85561 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate 0.1 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
81979 nAChR CLONED HUMAN 3H-Epibatidine 2-[(1R,2S)-2-(5-{[(2S)-azetidin-2-yl]methoxy}pyridin-3-yl)cyclopropyl]ethan-1-ol 0.1 Zhang HK et al 2012 Jan 15, 2025 Jan 29, 2025
60475 GABAA CLONED HUMAN FNZ PWZ-007A 0.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
85565 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate 0.1 Zhang HK et al 2013 Jan 15, 2025 Jan 29, 2025
35902 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 7-(2-Dimethylaminoethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
81983 nAChR CLONED HUMAN 3H-Epibatidine 2-[(1R,2S)-2-(5-{[(2S)-azetidin-2-yl]methoxy}pyridin-3-yl)cyclopropyl]ethan-1-ol 0.1 Zhang HK et al 2012 Jan 15, 2025 Jan 29, 2025
35903 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 7-(2-Dimethylaminoethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
9027 SST5 CLONED HUMAN 125I-SRIF-28 L-362,855 0.1 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
7236 ETB CLONED HUMAN 125I-ENDOTHELIN J-104132 0.1 Nishikibe M, et al., 1999 Jan 15, 2025 Jan 15, 2025
43076 MARK2 CLONED HUMAN 3H-Staurosporine Staurosporine 0.1 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
37703 DOR CLONED HUMAN 3H-Diprenorphine NTB 0.1 Tryoen-Toth P, et al., 2005 Jan 15, 2025 Jan 15, 2025
86603 5-HT4 CLONED HUMAN 3H-GR113808 1-Isopropyl-N-[[1-(2-pyridin-2-ylethyl)-4-piperidinyl]methyl]-1Hindazole-3-carboxamide 0.1 Furlotti G et al 2012 Jan 15, 2025 Jan 15, 2025
68942 SST5 CLONED HUMAN 125I-SRIF Cyclo[(N,N-dimethyldiaminoethylcarbamoyl)HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe 0.1 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
16208 D2 STRIATUM RAT 125I-Epidepride Spiroperidol 0.1 Neve KA, et al., 1990a Jan 15, 2025 Jan 15, 2025
18257 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Devazepide 0.1 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
9042 SST4 CLONED RAT 125I-CGP23996 BIM 23014 0.1 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
18259 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 sulfated CCK(26-33) 0.1 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
28755 SST2 CLONED HUMAN 125I-LTT-SRIF28 Somatostatin-14 0.1 Siehler S, et.al., 1998a Jan 15, 2025 Jan 15, 2025
82004 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2,2-difluoroethyl)-cyclopropyl]pyridine trifluoroacetate 0.1 Zhang HK et al 2012 Jan 15, 2025 Jan 29, 2025
68951 GABAA CLONED RAT 3H-Ro15-1788 3-(2,6-Difluorophenyl)-5-[4-fluoro-3-(3-fluoropyridin-2-yl)-phenyl]pyridazine 0.1 Lewis RT, et al., 2006 Jan 15, 2025 Jan 27, 2025
23386 NK1 U373MG HUMAN 125I-Bolton Hunter SSR240600 0.1 Emonds-Alt, X et. al., 2002 Jan 15, 2025 Jan 15, 2025
53085 KOR UNDEFINED HUMAN UNDEFINED 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan 0.1 Ghirmai S et al., 2008 Jan 15, 2025 Jan 15, 2025
8543 5-HT4B CLONED HUMAN 3H-GR-113808 SB204070 0.1 Bender E, et al., 2000 Jan 15, 2025 Jan 15, 2025
33121 SLC6A4 BRAIN RAT UNDEFINED WY-45655 0.1 Muth, EA et al., 1986 Jan 15, 2025 Jan 15, 2025
31843 M3 CLONED HUMAN 3H-Arachidonic Acid ATR 0.1 Bymaster F.P., et. al., 1999 Jan 15, 2025 Jan 15, 2025
13158 BRAIN RAT 3H-PRAZOSIN PRAZOSIN 0.1 Greengrass P, et al., 1979 Jan 15, 2025 Jan 15, 2025
56679 KOR UNDEFINED HUMAN UNDEFINED (4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol 0.1 Hsin LW et al., 2010 Jan 15, 2025 Jan 15, 2025
39016 D2 CLONED HUMAN R-SAT Ocaperidone 0.1 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
18795 M1 CLONED HUMAN 3H-NMS ml-toxin 3 0.1 Adem A and Karlsson E. 1997 Jan 15, 2025 Jan 15, 2025
8559 SST1 CLONED HUMAN 125I-Tyr11-SRIF Somatostatin-14 0.1 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
57715 NR3C1 UNDEFINED HUMAN UNDEFINED 4a-Benzyl-2-chloroethynyl-1,2,3,4,4a,9,10,10a-octahydro-phenanthrene-2,7-diol(CP-394531) 0.1 Onnis V et al., 2010 Jan 15, 2025 Jan 15, 2025
50038 NOP CLONED HUMAN 3H-Nociceptin Nociceptin-COOH, [Aib7] 0.1 Zhang C, et al., 2002 Jan 15, 2025 Jan 28, 2025
9080 SST5 CLONED HUMAN 125I-CGP23996 SRIF-[Des-Ala1,des-Gly2,His4,5,D-Trp8] 0.1 Raynor K, et al., 1993b Jan 15, 2025 Jan 15, 2025
57720 NR3C1 UNDEFINED HUMAN UNDEFINED 17-Hydroxy-13-methyl-10-(4-methyl-benzyl)-17-prop-1-ynyl-1,2,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-cyclopenta[a]phenanthren-3-one(RU-43044) 0.1 Onnis V et al., 2010 Jan 15, 2025 Jan 15, 2025
31866 M4 CLONED HUMAN 3H-QNB ATR 0.1 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
19070 CLONED RAT 125-AcHis1-PACAP-27 PACAP(1-27) 0.1 Ciccarelli E et al., 1995 Jan 15, 2025 Jan 15, 2025
47742 Y1 CLONED RAT [125I] - Peptide YY NPY, zebrafish 0.1 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
19071 CLONED RAT 125-AcHis1-PACAP-27 PACAP(1-38) 0.1 Ciccarelli E et al., 1995 Jan 15, 2025 Jan 15, 2025
8323 SST2 CLONED HUMAN 125I-LTT-SRIF28 Somatostatin-14 0.1 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
56963 DOR UNDEFINED UNDEFINED UNDEFINED 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-methyl)benzamido]morphinan-oxalate 0.1 Ghirmai S et al., 2009 Jan 15, 2025 Jan 15, 2025
31366 5-HT7 ILEUM GUINEA PIG 3H-MESULERGINE 5-Hydroxy Tryptamine 0.1 Hemedah M, et al., 1999 Jan 15, 2025 Jan 15, 2025
18055 CCK2 BRAIN GUINEA PIG 125I-BH-CCK-85 L-740,093 0.1 Patel S et al., 1994 Jan 15, 2025 Jan 15, 2025
8329 SST2 CLONED HUMAN 125I-LTT-SRIF28 seglitide 0.1 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
23692 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PAROXETINE 0.1 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
18573 CCK1 Acini RAT 125I-CCK-8 CCK-8 0.1 Akiyama T et al., 1996 Jan 15, 2025 Jan 15, 2025
8592 SST2 CLONED MOUSE 125I-Tyr11-SRIF RC 160 0.1 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
67729 Alpha1A, Alpha1B CEREBRAL CORTEX RAT 3H-PRAZOSIN PRAZOSIN 0.1 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
100756 PDE4b CLONED HUMAN Functional Roflumilast 0.1 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
42900 CaMK CLONED HUMAN 3H-Staurosporine Staurosporine 0.1 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
59284 nAChR BRAIN CORTEX RAT 3H-Epibatidine 2-[6-Chloro-5-(4-methoxyphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 0.1 Huang, Y. et. al., 2005 Jan 15, 2025 Jan 28, 2025
100758 PDE4d CLONED HUMAN Functional Roflumilast 0.1 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025
38043 CLONED RAT 3H-dexamethasone RU-486 0.1 Jacobson PB, et al., 2005 Jan 15, 2025 Jan 15, 2025
47519 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 0.1 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
55712 5-HT1B UNDEFINED HUMAN UNDEFINED N1,N13-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tridecanediamide 0.1 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
5026 5-HT2A CLONED HUMAN 3H-KETANSERIN METHIOTHEPIN 0.1 BONHAUS DW, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
9124 SST1 CLONED HUMAN 125I-CGP23996 Somatostatin-14 0.1 Raynor K, et al., 1993a Jan 15, 2025 Jan 15, 2025
55717 5-HT1B UNDEFINED HUMAN UNDEFINED 2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine 0.1 Choi SK et al., 2008 Jan 15, 2025 Jan 15, 2025
7848 GABAA CLONED HUMAN 3H-RO-15-1788 12 0.1 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8360 SST2 CLONED HUMAN 125I-CGP23996 somatostatin-28 0.1 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
35753 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 0.1 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
65449 nAChR CLONED HUMAN [3H] Flunitrazepam PWZ-007A 0.1 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
4782 5-HT1A test test 3H-DPAT WAY 100,635 0.1 HAMON M, ET AL., 1990 Jan 15, 2025 Jan 15, 2025
3762 MOR CLONED HUMAN 3H-DAMGO CYCLAZOCINE (-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
3765 MOR CLONED HUMAN 3H-DAMGO WIN 44,441(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
3258 D2 CLONED HUMAN 3H-YM 09151-2 ETICLOPRIDE,S(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
8378 SST2 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.1 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
48065 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.1 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
3779 MOR BRAIN GUINEA PIG 3H-DAMGO BREMAZOCINE(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
50116 SST3 CLONED HUMAN 125I-Tyr11-SRIF-14 Somatostatin-14 0.1 Poitout L., et.al., 2001 Jan 15, 2025 Jan 15, 2025
3787 MOR BRAIN GUINEA PIG 3H-DAMGO CYCLAZOCINE (-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
31947 M3 CLONED HUMAN 3H-Arachidonic Acid ATR 0.1 Bymaster F.P., et. al., 2003 Jan 15, 2025 Jan 15, 2025
28877 SST1 CLONED RAT 125I-Tyr11-somatostatin Somatostatin-14 0.1 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
3790 MOR BRAIN GUINEA PIG 3H-DAMGO WIN 44,441(-) 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
31694 D2 STRIATUM RAT 125I-Epidepride EPIDEPRIDE 0.1 Kessler, R.M., et. al., 1993 Jan 15, 2025 Jan 15, 2025
39123 D3 CLONED HUMAN R-SAT MOPERONE 0.1 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
30676 DOR CLONED HUMAN 3H-Diprenorphine SNC-80 0.1 Lecoq I et. al., 2004 Jan 15, 2025 Jan 15, 2025
28885 SST4 CLONED RAT 125I-Tyr11-somatostatin DC-25-100 0.1 Rossowski WJ, et.al. 1994 Jan 15, 2025 Jan 15, 2025
8662 SST5 CLONED RAT 125I-Tyr11-SRIF BIM 23014 0.1 Hoyer D, Lubbert H, Bruns Ch., 1994 Jan 15, 2025 Jan 15, 2025
4057 DOR CLONED HUMAN 3H-DPDPE-Cl NTB 0.1 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
39130 D3 CLONED HUMAN R-SAT 9-OH-risperidone 0.1 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
47067 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-4P 0.1 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025