The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 1-1,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
72192Beta3CLONEDHUMAN125I-Pindolol2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
76032Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77824Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77572Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
74758Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
97030Beta3CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
66312Beta3CLONEDHUMANI-125-PindololFinazine>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
77320Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
66570Beta3CLONEDHUMANI-125-Pindolol3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
75786Beta3CLONEDHUMAN125I-Pindolol1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
87562Beta3CLONEDHUMAN125I-Pindolol2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
99082Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99083Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
77068Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
99084Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
72973Beta3CLONEDHUMAN125I-Pindololcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
66832Beta3CLONEDHUMANI-125-PindololN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
76816Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
74513Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75537Beta3CLONEDHUMAN125I-Pindololpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
73235Beta3testtest125I-PindololN-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
76563Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
73493Beta3testtest125I-Pindolol3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
67094Beta3CLONEDHUMANI-125-Pindolol1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
68118Beta3UNDEFINEDUNDEFINED125I-CYPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
84247Beta3CLONEDHUMAN125I-Pindolol(±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide9057PDSP Certified DataJan 15, 2025Jan 28, 2025
86039Beta3CLONEDHUMAN125I-Pindolol(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
102169Beta3CLONEDHUMAN[3H]-CGP12177NEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
98843Beta3CLONEDHUMAN125I-Pindolol1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
75292Beta3CLONEDHUMAN125I-PindololEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
73757Beta3testtest125I-Pindolol{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
78621Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
84253Beta3CLONEDHUMAN125I-Pindolol(±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one5751PDSP Certified DataJan 15, 2025Jan 28, 2025
101917Beta3CLONEDHUMAN[3H]-CGP12177Ziprasidone>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
74014Beta3testtest125I-Pindolol1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride1014Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
76318Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
69665Beta3CLONEDHUMAN125I-iodo-pindololDPH>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
69666Beta3CLONEDHUMAN125I-iodo-pindolol2-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
78370Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
69667Beta3CLONEDHUMAN125I-iodo-pindolol3-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
69668Beta3CLONEDHUMAN125I-iodo-pindolol4-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
69669Beta3CLONEDHUMAN125I-iodo-pindolol2-CI-DPH>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
81189Beta3CLONEDHUMAN125I-PindololN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
64805Beta3CLONEDHUMAN125I-ICYPSalbutamol,(+/-)4.62Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
74278Beta3testtest125I-PindololN-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
75046Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
78118Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
64806Beta3CLONEDHUMAN125I-ICYPSalmeterol5.58Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
72999Beta3CLONEDHUMAN125I-PindololAmentoflavone>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
96295Beta3CLONEDHUMAN125I-iodo-pindolol4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
64807Beta3CLONEDHUMAN125I-ICYPFormoterol5.49Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
64808Beta3CLONEDHUMAN125I-ICYPIndacaterol5.48Battram, C., et al., 2006Jan 15, 2025Jan 15, 2025
76073Beta3CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
96297Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
101673Beta3CLONEDHUMAN[3H]-CGP12177Perospirone>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
77866Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
73003Beta3CLONEDHUMAN125I-Pindolol2,3-dihydroamentoflavone>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
96299Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
73004Beta3CLONEDHUMAN125I-Pindololtetrahydroamentoflavone>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
81708Beta3CLONEDHUMAN125I-iodo-pindololtrans-(3R, 6S)-6-benzhydryl-tetra-hydropyran-3-yl ester>10000Dutta AK et al 2011Jan 15, 2025Jan 28, 2025
96301Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
97069Beta3CLONEDHUMAN[125I]Iodopindolol3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
77614Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
74799Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
96303Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
60207Beta3CLONEDHUMAN125I-PindololMRS56981500Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
96305Beta3CLONEDHUMAN125I-iodo-pindolol4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
77362Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
100146Beta3CLONEDHUMAN125I-PindololBrexpiprazole1653PDSP Certified DataJan 15, 2025Jan 28, 2025
66355Beta3CLONEDHUMANI-125-PindololN-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
75827Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
96307Beta3CLONEDHUMAN125I-iodo-pindolol4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
66612Beta3CLONEDHUMANI-125-PindololN-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
81972Beta3CLONEDHUMAN125I-Pindolol[18F]MH.MZ>10000Herth MM et al 2009Jan 15, 2025Jan 28, 2025
96309Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
77110Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
59702Beta3CLONEDHUMAN3H-CGP-12177MH.MZ>10000Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
87607Beta3CLONEDHUMAN125I-Pindolol3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
96311Beta3CLONEDHUMAN125I-iodo-pindolol4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
60216Beta3CLONEDHUMAN125I-PindololMRS56762140Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
96313Beta3CLONEDHUMAN125I-iodo-pindolol4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
72762Beta3CLONEDHUMAN125I-Pindololdihydrobilobetin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
76858Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
96315Beta3CLONEDHUMAN125I-iodo-pindolol3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
66876Beta3CLONEDHUMANI-125-PindololN-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
71228Beta3CLONEDHUMAN125I-iodo-pindololFEMPT564Collier TL et al 2017Jan 15, 2025Jan 28, 2025
74556Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76604Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
89916Beta3CLONEDHUMAN125I-Pindolol5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
75581Beta3CLONEDHUMAN125I-Pindolol3-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
73279Beta3testtest125I-PindololN-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
73535Beta3testtest125I-PindololN-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
67138Beta3CLONEDHUMANI-125-Pindolol{2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
86084Beta3CLONEDHUMAN125I-PindololNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
75333Beta3CLONEDHUMAN125I-Pindololethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
68422Beta3CLONEDHUMAN[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
70470Beta3CLONEDHUMAN125I-PindololMRP3200>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
76359Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
78663Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
95815Beta3CLONEDHUMAN125I-iodo-pindolol6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
67400Beta3CLONEDHUMANI-125-Pindolol1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
73801Beta3testtest125I-Pindolol1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
95817Beta3CLONEDHUMAN125I-iodo-pindololTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
74058Beta3testtest125I-Pindolol1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
95819Beta3CLONEDHUMAN125I-iodo-pindololTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
58187Beta3CLONEDHUMAN3H-CGP-12177(S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxy-5-phenylthiophene-3-yl-methylpyrimidine-2,4-dione>10000Duncan GE, et at., 2012Jan 15, 2025Jan 15, 2025
78412Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
95821Beta3CLONEDHUMAN125I-iodo-pindolol6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
101966Beta3CLONEDHUMAN[3H]-CGP12177ILOPERIDONE>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
75087Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
95823Beta3CLONEDHUMAN125I-iodo-pindololN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
78160Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
71761Beta3CLONEDHUMAN125I-PindololDKR-1677>10000Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
95825Beta3CLONEDHUMAN125I-iodo-pindololtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
74322Beta3testtest125I-PindololN-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
76114Beta3CLONEDHUMAN125I-Pindolol2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
97106Beta3CLONEDHUMAN[125I]Iodopindolol4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
98898Beta3CLONEDHUMAN125I-Pindolol3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
95827Beta3CLONEDHUMAN125I-iodo-pindolol4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
77908Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
80980Beta3CLONEDHUMAN125I-Pindolol3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine>10000Rajagopalan R et al 2014Jan 15, 2025Jan 28, 2025
101972Beta3CLONEDHUMAN[3H]-CGP12177ZOTEPINE>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
80981Beta3CLONEDHUMAN125I-Pindolol3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine>10000Rajagopalan R et al 2014Jan 15, 2025Jan 28, 2025
95829Beta3CLONEDHUMAN125I-iodo-pindolol2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
80982Beta3CLONEDHUMAN125I-Pindolol5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine>10000Rajagopalan R et al 2014Jan 15, 2025Jan 28, 2025
74840Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77656Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
87385Beta3CLONEDHUMAN125I-Pindolol1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
101721Beta3CLONEDHUMAN[3H]-CGP12177CLOZAPINE>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
75868Beta3CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77404Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
66398Beta3CLONEDHUMANI-125-PindololN-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
72799Beta3CLONEDHUMAN125I-Pindololepigallocatechin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
101471Beta3CLONEDHUMAN[3H]QNBAmisulpride>10000PDSP Certified DataMar 20, 2025Mar 20, 2025
66656Beta3CLONEDHUMANI-125-Pindolol3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
77152Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
87650Beta3CLONEDHUMAN125I-Pindolol3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
98915Beta3CLONEDHUMAN125I-Iodopindolol1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
76900Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
72037Beta3CLONEDHUMAN125I-Pindolol1-methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g] quinoxalin-2(6H)-one HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
76645Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
89957Beta3CLONEDHUMAN125I-Pindolol3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
74598Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75622Beta3CLONEDHUMAN125I-Pindolol2-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
66920Beta3CLONEDHUMANI-125-PindololN-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
50537Beta3CLONEDHUMAN125I-ICYPPrucalopride>10000Briejer MR, et al., 2001Jan 15, 2025Jan 15, 2025
73322Beta3testtest125I-PindololN-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
73579Beta3testtest125I-Pindolol3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
67181Beta3CLONEDHUMANI-125-Pindolol{2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
75374Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
68463Beta3CLONEDHUMAN125I-IodopindololN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
71023Beta3CLONEDHUMAN125I-PindololN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
76399Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
78705Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
73842Beta3testtest125I-Pindolol{2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
70515Beta3CLONEDHUMAN125I-iodo-pindololMRP3201>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
86131Beta3CLONEDHUMAN125I-Pindolol4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
78453Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
74102Beta3testtest125I-Pindolol1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
16247Beta3CLONEDHUMAN3H-CGP-12177KUR-1246>10000Kobayashi M, et al., 2001Jan 15, 2025Jan 15, 2025
75128Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
34169Beta3CLONEDHUMAN125I-CYPNOREPINEPHRINE4300Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
78202Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
97146Beta3CLONEDHUMAN[125I]Iodopindolol2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
34170Beta3CLONEDHUMAN125I-CYPEPINEPHRINE>10000Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
76155Beta3CLONEDHUMAN125I-Pindolol2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
34171Beta3CLONEDHUMAN125I-CYPIsoproterenol-l1570Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34172Beta3CLONEDHUMAN125I-CYPFenoterol>10000Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
70781Beta3testtest3H-CGP121771-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
34173Beta3CLONEDHUMAN125I-CYPSalbutamol,(+/-)>10000Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
71806Beta3CLONEDHUMAN3H-CGP12177SAS-0132>10000Yi B et al 2017Jan 15, 2025Jan 28, 2025
77950Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
34174Beta3CLONEDHUMAN125I-CYPSalmeterol7180Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34175Beta3CLONEDHUMAN125I-CYPFormoterol8090Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34176Beta3CLONEDHUMAN125I-CYPTerbutaline>10000Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
74881Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
34177Beta3CLONEDHUMAN125I-CYPBRL 37344430Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
101761Beta3CLONEDHUMAN[3H]-CGP12177Remoxapride>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
77698Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
34178Beta3CLONEDHUMAN125I-CYPALPRENOLOL35Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
61826Beta3CLONEDHUMAN3H-CGP-12177FECIMBI-36>10000Prabhakaran, Jaya et. al. 2015Jan 15, 2025Jan 15, 2025
34179Beta3CLONEDHUMAN125I-CYPPINDOLOL,(+/-)44.1Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34180Beta3CLONEDHUMAN125I-CYPCarvedilol247Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
75909Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
34181Beta3CLONEDHUMAN125I-CYPATENOLOL>10000Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
59525Beta3CLONEDHUMAN3H-CGP-12177Nantenin>10000LeGendre, O. et. al., 2009Jan 15, 2025Jan 15, 2025
77446Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
34182Beta3CLONEDHUMAN125I-CYPBisoprolol9070Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34183Beta3CLONEDHUMAN125I-CYPmetoprolol>10000Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34184Beta3CLONEDHUMAN125I-CYPPROPRANOLOL, l-186Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
66441Beta3CLONEDHUMANI-125-PindololN-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
34185Beta3CLONEDHUMAN125I-CYPCGP 20712-A2360Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
77194Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N,2-dibutyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
34186Beta3CLONEDHUMAN125I-CYPSR 59230A122Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
34187Beta3CLONEDHUMAN125I-CYPCGP 1217777.1Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
66700Beta3CLONEDHUMANI-125-Pindololethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
72332Beta3CLONEDHUMAN3H-CGP-121772-Aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 28, 2025
72844Beta3CLONEDHUMAN125I-Pindololisoginkgetin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
34188Beta3CLONEDHUMAN125I-CYPICI 118,551611Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
102028Beta3CLONEDHUMAN[3H]-CGP12177RS-(+/-)-Sulpriride>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
34189Beta3CLONEDHUMAN125I-CYPBroxaterol3990Hoffmann C, et al., 2004Jan 15, 2025Jan 15, 2025
76942Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
75663Beta3CLONEDHUMAN125I-Pindololbenzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76687Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
87695Beta3CLONEDHUMAN125I-Pindolol3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
74640Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
91280Beta3CLONEDHUMAN125I-Pindolol17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
87441Beta3CLONEDHUMAN125I-Pindolol4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
83858Beta3CLONEDHUMAN125I-Pindolol(±)-N-(((4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)methyl)aniline1924PDSP Certified DataJan 15, 2025Jan 28, 2025
84114Beta3CLONEDHUMAN125I-Pindolol(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-(trifluoromethyl)benzamide7549PDSP Certified DataJan 15, 2025Jan 28, 2025
98962Beta3CLONEDHUMAN125I-PindololC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
83859Beta3CLONEDHUMAN125I-Pindolol(±)-4-chloro-N-(((4aS,8R,8aS)-2-benzyl-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)methyl)-3-(trifluoromethyl)aniline1104PDSP Certified DataJan 15, 2025Jan 28, 2025
66964Beta3CLONEDHUMANI-125-Pindolol3-(piperazin-1-yl)-N-(m-tolyl)propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
71061Beta3CLONEDHUMAN125I-PindololN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
73365Beta3testtest125I-PindololN-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
74390Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75414Beta3CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,2-dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d]- [1,3]dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
73623Beta3testtest125I-Pindololethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
67224Beta3CLONEDHUMANI-125-Pindolol{2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
76440Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
63128Beta3CLONEDHUMANI125- PindololMitragynine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
72089Beta3CLONEDHUMAN125I-Pindolol2-methoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
78747Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
73884Beta3testtest125I-Pindolol{2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
84126Beta3CLONEDHUMAN125I-Pindolol(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-methylbenzamide6686PDSP Certified DataJan 15, 2025Jan 28, 2025
78495Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
86175Beta3CLONEDHUMAN125I-Pindolol2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
70560Beta3CLONEDHUMAN125I-iodo-pindololMRP31606Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
75169Beta3CLONEDHUMAN125I-Pindololmethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
74146Beta3testtest125I-Pindololnaftopidil250Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
97186Beta3CLONEDHUMAN[125I]Iodopindolol3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
70820Beta3CLONEDHUMAN125I-IodopindololD-5782703Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
76196Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
78244Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
41381Beta3CLONEDRAT125I-Pindolol2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
101798Beta3CLONEDHUMAN[3H]-CGP12177RISPERIDONE>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
83879Beta3CLONEDHUMAN125I-Pindolol(±)-(4aS,8S,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5066PDSP Certified DataJan 15, 2025Jan 28, 2025
77992Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
72361Beta3CLONEDHUMAN3H-CGP-121775-Methoxy-2-aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 28, 2025
74922Beta3CLONEDHUMAN125I-Pindolol1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
81066Beta3CLONEDHUMAN125I-PindololN-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
50602Beta3CLONEDHUMAN125I-IodopindololAmisulpride>10000Abbas AI et.al., 2009Jan 15, 2025Jan 15, 2025
62379Beta3CLONEDHUMAN3H-CGP-12177Diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
77740Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
62380Beta3CLONEDHUMAN3H-CGP-121772-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
62381Beta3CLONEDHUMAN3H-CGP-121773-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
75950Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
100014Beta3CLONEDHUMAN125I-Pindolol5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
62382Beta3CLONEDHUMAN3H-CGP-121774-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
100015Beta3CLONEDHUMAN125I-Pindolol5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
62383Beta3CLONEDHUMAN3H-CGP-121772-Cl-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
63151Beta3CLONEDHUMANI125-IodopindololMitragynine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
69552Beta3CLONEDHUMAN125I-iodo-pindololEphenidine>10000Kang, H. et, al. 2017Jan 15, 2025Jan 28, 2025
77488Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
101552Beta3CLONEDHUMAN[3H]-CGP12177OLANZAPINE>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
87474Beta3CLONEDHUMAN125I-PindololFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
66484Beta3CLONEDHUMANI-125-PindololN-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
77236Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
91318Beta3CLONEDHUMAN125I-Pindolol17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
94903Beta3CLONEDHUMAN125I-Pindolol4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
66744Beta3CLONEDHUMANI-125-PindololN-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
72888Beta3CLONEDHUMAN125I-Pindolol2″-glucosylvitexin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
75704Beta3CLONEDHUMAN125I-Pindolol2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76984Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
92600Beta3CLONEDHUMAN125I-Pindolol(5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94904Beta3CLONEDHUMAN125I-Pindolol4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
76729Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
92601Beta3CLONEDHUMAN125I-Pindolol9,13:15,16-diepoxylabdane-6b,15a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94905Beta3CLONEDHUMAN125I-Pindolol4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
74682Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
94906Beta3CLONEDHUMAN125I-Pindolol5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94907Beta3CLONEDHUMAN125I-Pindolol4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
92604Beta3CLONEDHUMAN125I-Pindolol9,13:15,16-diepoxylabdane-6b,16b-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94908Beta3CLONEDHUMAN125I-Pindolol4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
99004Beta3CLONEDHUMAN125I-Pindolol[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
92605Beta3CLONEDHUMAN125I-Pindolol9,13:15,16-diepoxylabdane-6b,16a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94909Beta3CLONEDHUMAN125I-Pindolol4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
74430Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
94910Beta3CLONEDHUMAN125I-Pindolol4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
67007Beta3CLONEDHUMANI-125-Pindolol[2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
73407Beta3testtest125I-PindololN-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
75455Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(2-((5-bromothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
94911Beta3CLONEDHUMAN125I-Pindolol4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
58303Beta3CLONEDHUMAN125I-PindololMRS3558>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
92608Beta3CLONEDHUMAN125I-Pindolol9,13-epoxylabd-5-en-7-on-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94912Beta3CLONEDHUMAN125I-Pindolol4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
58304Beta3CLONEDHUMAN125I-PindololMRS5202>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
76481Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
92609Beta3CLONEDHUMAN125I-Pindolol15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94913Beta3CLONEDHUMAN125I-Pindolol4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
58305Beta3CLONEDHUMAN125I-PindololMRS5923>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
94914Beta3CLONEDHUMAN125I-Pindolol2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate1240Jung et al 2021Jan 15, 2025Jan 28, 2025
58306Beta3CLONEDHUMAN125I-PindololMRS5930>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
94915Beta3CLONEDHUMAN125I-Pindolol2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
58307Beta3CLONEDHUMAN125I-PindololMRS5474>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
67268Beta3CLONEDHUMANI-125-Pindolol1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
92612Beta3CLONEDHUMAN125I-Pindolol9,13-epoxy-15,16-dihydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
94916Beta3CLONEDHUMAN3H-CGP-121774-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
102084Beta3CLONEDHUMAN[3H]-CGP12177Lurasidone HCl>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
73669Beta3testtest125I-PindololN-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
78789Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
92613Beta3CLONEDHUMAN125I-Pindolol9,13-epoxylabd-5-ene-7 b,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
72390Beta3CLONEDHUMAN3H-CGP-121775-methoxy-6-methyl-2-aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 28, 2025
73926Beta3testtest125I-Pindolol{2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
92616Beta3CLONEDHUMAN125I-Pindolol(8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
78537Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
92617Beta3CLONEDHUMAN125I-Pindolol15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
102089Beta3CLONEDHUMAN[3H]-CGP12177GMC 1-116>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
75210Beta3CLONEDHUMAN125I-Pindololethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
101834Beta3CLONEDHUMAN[3H]-CGP12177SERTINDOLE>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
62922Beta3CLONEDHUMAN3H-CGP12177Ketamine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
86219Beta3CLONEDHUMAN125I-Pindolol4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
72140Beta3CLONEDHUMAN125I-Pindolol2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
92620Beta3CLONEDHUMAN125I-Pindolol9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
76237Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
78286Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
74191Beta3testtest125I-PindololN-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
84176Beta3CLONEDHUMAN125I-Pindolol(±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide4431PDSP Certified DataJan 15, 2025Jan 28, 2025
85200Beta3recombinantHUMAN125I-cyanopindololTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
70610Beta3CLONEDHUMAN125I-iodo-pindololMRP3172>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
78034Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
81106Beta3CLONEDHUMAN125I-PindololN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
96978Beta3CLONEDHUMAN[125I]Iodopindolol4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
74964Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77782Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
85974Beta3CLONEDHUMAN125I-Pindolol1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
75991Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77530Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
72670Beta3CLONEDHUMAN125I-Pindolol2,3-dihydrohinokiflavone>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
77278Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
66527Beta3CLONEDHUMANI-125-PindololN-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
87519Beta3CLONEDHUMAN125I-Pindolol1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
75745Beta3CLONEDHUMAN125I-Pindolol3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
77026Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
72419Beta3CLONEDHUMAN3H-CGP-121775,6-methylenedioxy-2-aminoindan>10000Halberstadt Adam L et al 2019Jan 15, 2025Jan 28, 2025
74723Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
84195Beta3CLONEDHUMAN125I-Pindolol(±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide5737PDSP Certified DataJan 15, 2025Jan 28, 2025
66788Beta3CLONEDHUMANI-125-PindololN-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
76774Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
73191Beta3testtest125I-Pindolol3-(piperazin-1-yl)-N-(m-tolyl)propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
74471Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
66024Beta3CLONEDHUMANI125- IodopindololOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
75496Beta3CLONEDHUMAN125I-Pindololpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
73450Beta3testtest125I-PindololN-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
76522Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
85994Beta3CLONEDHUMAN125I-PindololDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
58602Beta3CLONEDHUMAN125I-PindololMRS56981450Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
67051Beta3CLONEDHUMANI-125-Pindolol{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
58603Beta3CLONEDHUMAN125I-PindololMRS56781560Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58604Beta3CLONEDHUMAN125I-PindololMRS56971170Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
98797Beta3CLONEDHUMAN125I-Pindolol3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
58605Beta3CLONEDHUMAN125I-PindololMRS56762320Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58606Beta3CLONEDHUMAN125I-PindololMRS57552460Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
78831Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
73713Beta3testtest125I-Pindolol[2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
73970Beta3testtest125I-Pindolol1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
75251Beta3CLONEDHUMAN125I-Pindololethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
78579Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
101619Beta3CLONEDHUMAN[3H]-CGP12177Paliperidone>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
69877Beta3CLONEDHUMAN125I-iodo-pindolol4-(1-phenylcyclohexyl)morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
69878Beta3CLONEDHUMAN125I-iodo-pindolol4-[1-(3-methylphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
70646Beta3CLONEDHUMAN125I-iodo-pindololMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
76278Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
69879Beta3CLONEDHUMAN125I-iodo-pindolol4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
101879Beta3CLONEDHUMAN[3H]-CGP12177S-(-)-Sulpride>10000PDSP Certified DataMar 24, 2025Jul 28, 2026
102135Beta3CLONEDHUMAN[3H]-CGP12177Melperone HCl>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
69880Beta3CLONEDHUMAN125I-iodo-pindolol4-[1-(4-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
78328Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
84216Beta3CLONEDHUMAN125I-Pindolol(±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide7503PDSP Certified DataJan 15, 2025Jan 28, 2025
69881Beta3CLONEDHUMAN125I-iodo-pindolol4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
86265Beta3CLONEDHUMAN125I-PindololJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
100089Beta3CLONEDHUMAN125I-PindololCariprazine1882PDSP Certified DataJan 15, 2025Jan 28, 2025
69882Beta3CLONEDHUMAN125I-iodo-pindolol4-[1-(2-methoxyphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 15, 2025
74234Beta3testtest125I-PindololN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp AJ et al 2016Jan 15, 2025Jan 28, 2025
81147Beta3CLONEDHUMAN125I-PindololN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
81915Beta3CLONEDHUMAN125I-Pindolol(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
78076Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
75005Beta3CLONEDHUMAN125I-Pindolol(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
2565-HT1ACORTEXRAT3H-8-OH-DPATDHE19McCARTHY & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
5125-HT1AHIPPOCAMPUSRAT3H-SPIROXATRINESPIPERONE28.8NELSON ET AL., 1987Jan 15, 2025Jan 15, 2025
693765-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL1202Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
133125-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATCITALOPRAM>10000Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
808965-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
832005-HT1ACLONEDHUMAN3H-8-OH-DPATLSD2.78Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
857605-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide230Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
207365-HT1AHIPPOCAMPUSRAT3H-PATQUIPAZINE3388.44Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
271365-HT1ACLONEDHUMAN3H-8-OH-DPATCP-132,4848410May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942085-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine3300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
954885-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione11Partyka A et al 2015Jan 15, 2025Jan 15, 2025
972805-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamineBUSPIRONE50Perry CK et al 2020Jan 15, 2025Jan 15, 2025
1016325-HT1ACLONEDHUMAN[3H]-8-OH-DPATPerospirone0.7PDSP Certified DataMar 21, 2025Jul 28, 2026
376325-HT1AHippocampalRAT3H-8-OH-DPATN-[2-[4-(1-Naphthalenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide0.6Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
522245-HT1AUNDEFINEDHUMANUNDEFINED(S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol11.2Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
550405-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide19Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
555525-HT1AUNDEFINEDRATUNDEFINED4-[4-(4-Benzylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione2730Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
2575-HT1ACORTEXHUMAN3H-8-OH-DPATDILTIAZEM>10000PEROUTKA, 1988Jan 15, 2025Jan 15, 2025
678415-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
693775-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPHENAZINE145Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
714255-HT1ACLONEDHUMANWAY1006354-acetoxy-N,N-diallyltryptamine383Klein LM et al 2018Jan 15, 2025Jan 15, 2025
719375-HT1Atesttest[3H] Way1006358-(4-(Benzo[d]thiazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one195Etukala JR et al 2016Jan 15, 2025Jan 15, 2025
732175-HT1Atesttest[3H] Way100635N-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride371Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
765455-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
133135-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATINDALPINE9120.1Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
826895-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
857615-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
207375-HT1AHIPPOCAMPUSRAT3H-PATCINANSERIN1096.48Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
870415-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one2000Cao X et al 2018Jan 15, 2025Jan 15, 2025
893455-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide365Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
245775-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT5-Hydroxy Tryptamine1.8Borsini F, et al., 1995Jan 15, 2025Jan 15, 2025
908815-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane50.1187Franchini S et al 2014Jan 15, 2025Jan 15, 2025
271375-HT1ACLONEDHUMAN3H-8-OH-DPATCP-132,484(4b)287May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942095-HT1ACLONEDHUMAN3H-8-OH-DPAT4-benzyloxy-2,5-dimethoxyphenethylamine2700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
954895-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione1Partyka A et al 2015Jan 15, 2025Jan 15, 2025
1013775-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one22Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
376335-HT1AHippocampalRAT3H-8-OH-DPATN-[2-[4-(4-Chloro-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide433Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
522255-HT1AUNDEFINEDHUMANUNDEFINED(S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol3.89Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
550415-HT1AUNDEFINEDHUMANUNDEFINED4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide325Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
555535-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate35Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
2585-HT1ACORTEXHUMAN3H-8-OH-DPATDMT119.51PIERCE & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
5145-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSPIPERONE32.76HALL ET AL., 1985Jan 15, 2025Jan 15, 2025
693785-HT1ACLONEDHUMAN3H-8-OH-DPATCHLORPROMAZINE3115Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
734745-HT1Atesttest[3H] Way1006353-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride476Rennekamp AJ et al 2016Jan 15, 2025Jan 15, 2025
133145-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATPAROXETINE>10000Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
207385-HT1AHIPPOCAMPUSRAT3H-PATPIZOTIFEN2187.76Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
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271385-HT1ACLONEDHUMAN3H-8-OH-DPATN,N-dimethyl derivative562May JA, et al., 2003Jan 15, 2025Jan 15, 2025
942105-HT1ACLONEDHUMAN3H-8-OH-DPAT4-allyloxy-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
954905-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione5Partyka A et al 2015Jan 15, 2025Jan 15, 2025
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954915-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride433Partyka A et al 2015Jan 15, 2025Jan 15, 2025
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591395-HT1ACLONEDHUMAN3H-WAY100635CHLORPROMAZINE3000Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
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550495-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline3.7Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
555615-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate37Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
591455-HT1ACLONEDHUMAN3H-WAY100635KETANSERIN1044Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
2665-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOB,R(-)2332TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
681065-HT1AUNDEFINEDUNDEFINED3H-8-OH-DPATABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
33385-HT1ACLONEDHUMAN3H-8-OH-DPATCGS 12066B44TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
752745-HT1ACLONEDHUMAN3H-WAY100635Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
146025-HT1ACLONEDHUMAN3H-8-OH-DPATSB-277011-A5011.87Reavill C., et al., 2000Jan 15, 2025Jan 15, 2025
837225-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide9987PDSP Certified DataJan 15, 2025Jan 15, 2025
207465-HT1AHIPPOCAMPUSRAT3H-PAT5-M-N,N-DMT39.8107Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
867945-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide219Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
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268905-HT1ACLONEDHUMAN3H-8-OH-DPATxanomeline63.0957Watson J.,et. al.,1998Jan 15, 2025Jan 15, 2025
376425-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide397Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
522345-HT1AUNDEFINEDHUMANUNDEFINEDPINDOLOL,(+/-)81.1Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
550505-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline95Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
555625-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione124Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
2675-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOB,S(+)4041TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
5235-HT1ACORTEXPIG3H-8-OH-DPATSPIPERONE66.1ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
678515-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33395-HT1ACLONEDHUMAN3H-8-OH-DPATCHLORPROMAZINE3115TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
704115-HT1ACLONEDHUMAN3H-WAY100635MRP42685.6Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
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786035-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
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832115-HT1ACLONEDHUMAN3H-8-OH-DPATKETANSERIN6510Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
184435-HT1ACLONEDHUMAN3H-5HT1-NP9.2Jorand-Lebrun C et al., 1997aJan 15, 2025Jan 15, 2025
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207475-HT1AHIPPOCAMPUSRAT3H-PATDMT,5-OH21.3796Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
867955-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide331Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
893555-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide802Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
1008755-HT1ACLONEDHUMAN3H-WAY1006351-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)24.6Stephenson, K. et. al., 2008Jan 15, 2025Jan 15, 2025
1013875-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione35Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
376435-HT1AHippocampalRAT3H-8-OH-DPATN-[5-[4-(4-Chlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide850Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
522355-HT1AUNDEFINEDHUMANUNDEFINEDN-(3-(1H-indol-4-yloxy)propyl)cyclopentanamine233Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
550515-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline2.04Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
555635-HT1AUNDEFINEDRATUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propoxy]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione616Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
591475-HT1ACLONEDHUMAN3H-WAY100635METHYSERGIDE25Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
2685-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOBU4178TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
5245-HT1ACORTEXPIG3H-8-OH-DPATSPIPERONE66.1SCHLICKER ET AL., 1989Jan 15, 2025Jan 15, 2025
33405-HT1ACLONEDHUMAN3H-8-OH-DPATCLOMIPRAMINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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763005-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
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832125-HT1ACLONEDHUMAN3H-8-OH-DPATRo 60-01756680Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
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857725-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
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312445-HT1ACLONEDHUMAN3H-8-OH-DPATPPP, S(-)-31730PDSP Certified DataJan 15, 2025Jan 15, 2025
376445-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dimethylphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide268Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
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555645-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione331Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
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207495-HT1AHIPPOCAMPUSRAT3H-PAT5-Hydroxy Tryptamine6.76083Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
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258695-HT1ACLONEDHUMAN3H-8-OH-DPATPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
274055-HT1ACLONEDHUMAN3H-8-OH-DPATAPOMORPHINE117.49Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
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591495-HT1ACLONEDHUMAN3H-WAY100635RISPERIDONE427Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
635015-HT1ACLONEDRAT3H-WAY100635Brexpiprazole0.09Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
2705-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATDOI2355TITELER ET AL., 1988Jan 15, 2025Jan 15, 2025
33425-HT1ACLONEDHUMAN3H-8-OH-DPATCYPROHEPTADINE59TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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207505-HT1AHIPPOCAMPUSRAT3H-PATPlaceholder3.01995Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
896145-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1.86209Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274065-HT1ACLONEDHUMAN3H-8-OH-DPATBROMOCRIPTINE12.8825Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
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537745-HT1AUNDEFINEDHUMANUNDEFINEDCLOZAPINE140Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
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2715-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATGEPIRONE70GLENNON ET AL., 1988Jan 15, 2025Jan 15, 2025
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591515-HT1ACLONEDHUMAN3H-WAY100635PROPANOLOL(-)78Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
635035-HT1ACLONEDRAT3H-WAY100635ARIPIPRAZOLE1.2Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
678565-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
33445-HT1ACLONEDHUMAN3H-8-OH-DPATDESIPRAMINE>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
783525-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788645-HT1ACLONEDHUMAN3H-WAY100635(±)-2,5-Dimethoxy-4-bromoamphetamine2550Ray TS 2010 Jan 15, 2025Jan 15, 2025
806565-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
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207525-HT1AHIPPOCAMPUSRAT3H-PATHALOPERIDOL3548.13Gozlan H et al., 1983Jan 15, 2025Jan 15, 2025
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274085-HT1ACLONEDHUMAN3H-8-OH-DPATLISURIDE0.147911Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952485-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide192.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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522405-HT1AUNDEFINEDHUMANUNDEFINED1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol9.83Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
537765-HT1AUNDEFINEDHUMANUNDEFINEDQuetiapine230Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
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2735-HT1ACORTEXPIG3H-8-OH-DPATGEPIRONE89.1HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
5295-HT1ACELLSC0S-7125I-NAPSSPIPERONE66.2RAYMOND ET AL., 1989Jan 15, 2025Jan 15, 2025
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788655-HT1ACLONEDHUMAN3H-WAY100635(±)-3,4-Methylenedioxyamphetamine3762Ray TS 2010 Jan 15, 2025Jan 15, 2025
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868015-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide100Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
885935-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE140Peprah K et al 2012Jan 15, 2025Jan 15, 2025
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274095-HT1ACLONEDHUMAN3H-8-OH-DPATPERGOLIDE1.90546Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952495-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide182Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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537775-HT1AUNDEFINEDHUMANUNDEFINEDOLANZAPINE2100Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
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591535-HT1ACLONEDHUMAN3H-WAY100635BROMOCRIPTINE12.9Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
635055-HT1ACLONEDRAT3H-WAY100635RISPERIDONE250Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
2745-HT1ACORTEXRAT3H-WB4101HALOPERIDOL346.2NORMAN ET AL., 1985Jan 15, 2025Jan 15, 2025
5305-HT1AHIPPOCAMPUSHUMAN3H-8-OH-DPATSPIPERONE100.92HOYER ET AL., 1986Jan 15, 2025Jan 15, 2025
724665-HT1Atesttest[3H] Way100635ERGOTAMINE0.17Ibrahim MA et al 2017Jan 15, 2025Jan 15, 2025
788665-HT1ACLONEDHUMAN3H-WAY100635(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
832185-HT1ACLONEDHUMAN3H-8-OH-DPATCyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide1.21Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
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217785-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATCLOZAPINE1700Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
893625-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide6631Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
274105-HT1ACLONEDHUMAN3H-8-OH-DPATPiribedil446.684Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
276665-HT1ACLONEDHUMAN3H-8-OH-DPATMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
952505-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide728.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
376505-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-naphthalenecarboxamide335Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
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537785-HT1AUNDEFINEDHUMANUNDEFINEDZiprasidone2.5Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
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2755-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATHALOPERIDOL2761.11GOZLAN ET AL., 1983Jan 15, 2025Jan 15, 2025
5315-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATSPIPERONE101TITELER ET AL., 1987Jan 15, 2025Jan 15, 2025
33475-HT1ACLONEDHUMAN3H-8-OH-DPATDOPAMINE8248TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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788675-HT1ACLONEDHUMAN3H-WAY1006353,4,5-Trimethoxyphenethylamine1841Ray TS 2010 Jan 15, 2025Jan 15, 2025
857795-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide52.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
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217795-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATHALOPERIDOL2500Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
896195-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1.25893Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274115-HT1ACLONEDHUMAN3H-8-OH-DPATPramipexole691.831Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952515-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide82.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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537795-HT1AUNDEFINEDHUMANUNDEFINEDRISPERIDONE210Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
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622275-HT1ACLONEDHUMAN3H-WAY100635Tianeptine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
2765-HT1ACORTEXHUMAN3H-WB4101HALOPERIDOL2800WANDER ET AL., 1987Jan 15, 2025Jan 15, 2025
5325-HT1ACORTEXRAT3H-8-OH-DPATSPIPERONE120PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
33485-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT6.9TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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750285-HT1ACLONEDHUMAN3H-WAY100635(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
781005-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788685-HT1ACLONEDHUMAN3H-WAY1006354-Bromo-2,5-dimethoxyphenethylamine240.8Ray TS 2010 Jan 15, 2025Jan 15, 2025
804045-HT1ACLONEDHUMAN3H-8-OH-DPAT(E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
217805-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATAmisulpride>10000Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
896205-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone0.562341Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274125-HT1ACLONEDHUMAN3H-8-OH-DPATQuinelorane>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952525-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide212.6Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
312525-HT1ACLONEDHUMAN3H-8-OH-DPATPPP, R(+)-3868.9PDSP Certified DataJan 15, 2025Jan 15, 2025
335565-HT1ACLONEDHUMAN3H-8-OH-DPATCELECOXIB>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
376525-HT1AHippocampalRAT3H-8-OH-DPATN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-(1,1'-biphenyl)-4-carboxamide1000Leopoldo M, et al., 2002Jan 15, 2025Jan 15, 2025
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537805-HT1AUNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one2332Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
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2775-HT1ACORTEXPIG3H-8-OH-DPATHALOPERIDOL4790HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
5335-HT1ACORTEXHUMAN3H-8-OH-DPATSPIPERONE130.76HOYER ET AL., 1986Jan 15, 2025Jan 15, 2025
678615-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)146Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
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778455-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
788695-HT1ACLONEDHUMAN3H-WAY100635DMT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
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827095-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
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5345-HT1ACORTEXRAT3H-8-OH-DPATSPIPERONE140SCHLEGEL & PEROUTKA, 1986Jan 15, 2025Jan 15, 2025
33505-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPENTHIXOL, Alpha8028TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
788705-HT1ACLONEDHUMAN3H-WAY1006354-Hydroxy-N,N-dimethyltryptamine62.6Ray TS 2010 Jan 15, 2025Jan 15, 2025
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274145-HT1ACLONEDHUMAN3H-8-OH-DPATRopinirole288.403Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
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33515-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPHENAZINE2829TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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952555-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide298Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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5365-HT1AHIPPOCAMPUSBOVINE3H-8-OH-DPATSPIPERONE155.56PEROUTKA, 1985Jan 15, 2025Jan 15, 2025
683765-HT1ACLONEDHUMAN3H-8-OH-DPATcis 1-hydroxyindane67.6083Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33525-HT1ACLONEDHUMAN3H-8-OH-DPATGBR-129094677TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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896245-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone0.616595Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
274165-HT1ACLONEDHUMAN3H-8-OH-DPATTalipexole1698.24Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
952565-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide2500Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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566005-HT1AUNDEFINEDRATUNDEFINED8-OH-DPAT0.8Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
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683775-HT1ACLONEDHUMAN3H-8-OH-DPATtrans 1-hydroxyindane1.62181Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33535-HT1ACLONEDHUMAN3H-8-OH-DPATOndansetron HCl>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
719615-HT1Atesttest[3H] Way1006351-(1-(4-(Benzo[d]oxazol-2-yl)butyl)piperidin-4-yl)-5- chloro-1H-benzo[d]imidazol-2(3H)-one611Etukala JR et al 2016Jan 15, 2025Jan 15, 2025
788735-HT1ACLONEDHUMAN3H-WAY1006354-Ethylthio-2,5-dimethoxyphenethylamine381.2Ray TS 2010 Jan 15, 2025Jan 15, 2025
148735-HT1ACLONEDRATUNDEFINEDCLOZAPINE710Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
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896255-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0616595Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
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274175-HT1ACLONEDHUMAN3H-8-OH-DPATTERGURIDE3.46737Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
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312575-HT1AC.H.O.HUMAN3H-8-OH-DPATRopinirole288.403Millan MJ, et. al., 2004Jan 15, 2025Jan 15, 2025
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5385-HT1AHIPPOCAMPUSRAT125I-BH-8-MeO-N-PASPIPERONE425.84GOZLAN ET AL., 1988Jan 15, 2025Jan 15, 2025
678665-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline66Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
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33545-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL5084TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
724745-HT1Atesttest[3H] Way100635METHYSERGIDE14Ibrahim MA et al 2017Jan 15, 2025Jan 15, 2025
788745-HT1ACLONEDHUMAN3H-WAY100635(±)-4-Ethylthio-2,5-dimethoxyamphetamine1674Ray TS 2010 Jan 15, 2025Jan 15, 2025
148745-HT1ACLONEDRATUNDEFINEDOLANZAPINE7100Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
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952585-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide199.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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788755-HT1ACLONEDHUMAN3H-WAY100635(±)-2,5-Dimethoxy-4-ethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
148755-HT1ACLONEDRATUNDEFINEDRISPERIDONE21Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
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837395-HT1ACLONEDHUMAN3H-8-OH-DPAT(±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one8590PDSP Certified DataJan 15, 2025Jan 15, 2025
952595-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide229.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
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683815-HT1ACLONEDHUMAN3H-8-OH-DPAT(-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol1.02329Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33575-HT1ACLONEDHUMAN3H-8-OH-DPATIDAZOXAN662TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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788775-HT1ACLONEDHUMAN3H-WAY100635N,N-Diisopropyltryptamine120.5Ray TS 2010 Jan 15, 2025Jan 15, 2025
148775-HT1ACLONEDRATUNDEFINEDZiprasidone37Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
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596775-HT1ACLONEDHUMAN3H-WAY100635MH.MZ>10000Herth, M. et. al., 2009Jan 15, 2025Jan 15, 2025
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683825-HT1ACLONEDHUMAN3H-8-OH-DPAT1-hydroxyindane67.6083Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
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788795-HT1ACLONEDHUMAN3H-WAY100635N,N-Dipropyltryptamine31.8Ray TS 2010 Jan 15, 2025Jan 15, 2025
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893755-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1836Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
896315-HT1ACLONEDHUMAN3H-8-OH-DPAT(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0147911Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
952635-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide476Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
1001275-HT1ACLONEDHUMAN3H-WAY100635Brexpiprazole1.1PDSP Certified DataJan 15, 2025Jan 15, 2025
1006395-HT1ACLONEDHUMAN3H-WAY100635CYPROHEPTADINE50Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1014075-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione28Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
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788805-HT1ACLONEDHUMAN3H-WAY1006354-Ethylthio-2,5-dimethoxyphenylbutylamine5339Ray TS 2010 Jan 15, 2025Jan 15, 2025
148805-HT1ACLONEDRATUNDEFINEDHALOPERIDOL2600Arnt J and Skarsfeldt TJan 15, 2025Jan 15, 2025
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315205-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-1-(2-(1-(3,4-Dichloro-benzene sulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine316.228Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
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543045-HT1AUNDEFINEDRATUNDEFINED3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile2530Funke U et al., 2008Jan 15, 2025Jan 15, 2025
5455-HT1ACORTEXPIG3H-8-OH-DPATSPIROXATRINE8.91SCHOEFFTER AND HOYER,1988Jan 15, 2025Jan 15, 2025
663375-HT1ACLONEDHUMAN3H-WAY100635N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
683855-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-011.25893Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33615-HT1ACLONEDHUMAN3H-8-OH-DPATMDA,R(-)>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
714575-HT1ACLONEDHUMANWAY1006352-phenyl-N,N-diallyltryptamine402Klein LM et al 2018Jan 15, 2025Jan 15, 2025
727375-HT1ACLONEDHUMAN3H-WAY100635dihydrobilobetin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
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389455-HT1ACORTEXRAT3H-8-OH-DPATQUIPAZINE2000Glennon RA, et al., 1989Jan 15, 2025Jan 15, 2025
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788825-HT1ACLONEDHUMAN3H-WAY100635LISURIDE0.3Ray TS 2010 Jan 15, 2025Jan 15, 2025
822105-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one20Besnard J et al 2012Jan 15, 2025Jan 15, 2025
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870745-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile473.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
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258905-HT1ACLONEDHUMAN3H-8-OH-DPATNorephedrine, (+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
952665-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide314.8Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
5475-HT1ACORTEXRAT3H-8-OH-DPATSPIROXATRINE,(+)21NIKAM ET AL., 1988Jan 15, 2025Jan 15, 2025
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788835-HT1ACLONEDHUMAN3H-WAY100635(±)-2,5-Dimethoxy-4-iodoamphetamine2219Ray TS 2010 Jan 15, 2025Jan 15, 2025
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683885-HT1ACLONEDHUMAN3H-8-OH-DPATPiperazine1.28825Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
33645-HT1ACLONEDHUMAN3H-8-OH-DPAT5-HT,2-Me3074TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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683895-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-0122.9087Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
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1019255-HT1ACLONEDHUMAN[3H]8-OH-DPATZOTEPINE131PDSP Certified DataMar 24, 2025Jul 28, 2026
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33675-HT1ACLONEDHUMAN3H-8-OH-DPATMIANSERIN2592TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
113035-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE420Schotte A, et al., 1996Jan 15, 2025Jan 15, 2025
123275-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATS 159311.51Millan MJ, et al., 1993Jan 15, 2025Jan 15, 2025
788875-HT1ACLONEDHUMAN3H-WAY100635(±)-2,5-Dimethoxy-4-ethylamphetamine14.4Ray TS 2010 Jan 15, 2025Jan 15, 2025
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33695-HT1ACLONEDHUMAN3H-8-OH-DPATNOMIFENSINE1183TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
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896415-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1.51356Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
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