72192 Beta3 CLONED HUMAN 125I-Pindolol 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
76032 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77824 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77572 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
74758 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
97030 Beta3 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
66312 Beta3 CLONED HUMAN I-125-Pindolol Finazine >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
77320 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
66570 Beta3 CLONED HUMAN I-125-Pindolol 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
75786 Beta3 CLONED HUMAN 125I-Pindolol 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
87562 Beta3 CLONED HUMAN 125I-Pindolol 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
99082 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99083 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
77068 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
99084 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
72973 Beta3 CLONED HUMAN 125I-Pindolol catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
66832 Beta3 CLONED HUMAN I-125-Pindolol N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
76816 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
74513 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75537 Beta3 CLONED HUMAN 125I-Pindolol propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
73235 Beta3 test test 125I-Pindolol N-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
76563 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
73493 Beta3 test test 125I-Pindolol 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
67094 Beta3 CLONED HUMAN I-125-Pindolol 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
68118 Beta3 UNDEFINED UNDEFINED 125I-CYP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
84247 Beta3 CLONED HUMAN 125I-Pindolol (±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 9057 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86039 Beta3 CLONED HUMAN 125I-Pindolol (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
102169 Beta3 CLONED HUMAN [3H]-CGP12177 NEMONAPRIDE >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
98843 Beta3 CLONED HUMAN 125I-Pindolol 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
75292 Beta3 CLONED HUMAN 125I-Pindolol Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
73757 Beta3 test test 125I-Pindolol {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
78621 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
84253 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 5751 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
101917 Beta3 CLONED HUMAN [3H]-CGP12177 Ziprasidone >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
74014 Beta3 test test 125I-Pindolol 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 1014 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
76318 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
69665 Beta3 CLONED HUMAN 125I-iodo-pindolol DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69666 Beta3 CLONED HUMAN 125I-iodo-pindolol 2-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
78370 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
69667 Beta3 CLONED HUMAN 125I-iodo-pindolol 3-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69668 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69669 Beta3 CLONED HUMAN 125I-iodo-pindolol 2-CI-DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
81189 Beta3 CLONED HUMAN 125I-Pindolol N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
64805 Beta3 CLONED HUMAN 125I-ICYP Salbutamol,(+/-) 4.62 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
74278 Beta3 test test 125I-Pindolol N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
75046 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
78118 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
64806 Beta3 CLONED HUMAN 125I-ICYP Salmeterol 5.58 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
72999 Beta3 CLONED HUMAN 125I-Pindolol Amentoflavone >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
96295 Beta3 CLONED HUMAN 125I-iodo-pindolol 4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
64807 Beta3 CLONED HUMAN 125I-ICYP Formoterol 5.49 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
64808 Beta3 CLONED HUMAN 125I-ICYP Indacaterol 5.48 Battram, C., et al., 2006 Jan 15, 2025 Jan 15, 2025
76073 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
96297 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
101673 Beta3 CLONED HUMAN [3H]-CGP12177 Perospirone >10000 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
77866 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
73003 Beta3 CLONED HUMAN 125I-Pindolol 2,3-dihydroamentoflavone >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
96299 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
73004 Beta3 CLONED HUMAN 125I-Pindolol tetrahydroamentoflavone >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
81708 Beta3 CLONED HUMAN 125I-iodo-pindolol trans-(3R, 6S)-6-benzhydryl-tetra-hydropyran-3-yl ester >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 28, 2025
96301 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
97069 Beta3 CLONED HUMAN [125I]Iodopindolol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
77614 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
74799 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
96303 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
60207 Beta3 CLONED HUMAN 125I-Pindolol MRS5698 1500 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
96305 Beta3 CLONED HUMAN 125I-iodo-pindolol 4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
77362 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
100146 Beta3 CLONED HUMAN 125I-Pindolol Brexpiprazole 1653 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
66355 Beta3 CLONED HUMAN I-125-Pindolol N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
75827 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
96307 Beta3 CLONED HUMAN 125I-iodo-pindolol 4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
66612 Beta3 CLONED HUMAN I-125-Pindolol N-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
81972 Beta3 CLONED HUMAN 125I-Pindolol [18F]MH.MZ >10000 Herth MM et al 2009 Jan 15, 2025 Jan 28, 2025
96309 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
77110 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
59702 Beta3 CLONED HUMAN 3H-CGP-12177 MH.MZ >10000 Herth, M. et. al., 2009 Jan 15, 2025 Jan 15, 2025
87607 Beta3 CLONED HUMAN 125I-Pindolol 3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
96311 Beta3 CLONED HUMAN 125I-iodo-pindolol 4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
60216 Beta3 CLONED HUMAN 125I-Pindolol MRS5676 2140 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
96313 Beta3 CLONED HUMAN 125I-iodo-pindolol 4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
72762 Beta3 CLONED HUMAN 125I-Pindolol dihydrobilobetin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
76858 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
96315 Beta3 CLONED HUMAN 125I-iodo-pindolol 3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
66876 Beta3 CLONED HUMAN I-125-Pindolol N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
71228 Beta3 CLONED HUMAN 125I-iodo-pindolol FEMPT 564 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
74556 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76604 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
89916 Beta3 CLONED HUMAN 125I-Pindolol 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
75581 Beta3 CLONED HUMAN 125I-Pindolol 3-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
73279 Beta3 test test 125I-Pindolol N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73535 Beta3 test test 125I-Pindolol N-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
67138 Beta3 CLONED HUMAN I-125-Pindolol {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
86084 Beta3 CLONED HUMAN 125I-Pindolol Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
75333 Beta3 CLONED HUMAN 125I-Pindolol ethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
68422 Beta3 CLONED HUMAN [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
70470 Beta3 CLONED HUMAN 125I-Pindolol MRP3200 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
76359 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
78663 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
95815 Beta3 CLONED HUMAN 125I-iodo-pindolol 6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
67400 Beta3 CLONED HUMAN I-125-Pindolol 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
73801 Beta3 test test 125I-Pindolol 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
95817 Beta3 CLONED HUMAN 125I-iodo-pindolol Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
74058 Beta3 test test 125I-Pindolol 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
95819 Beta3 CLONED HUMAN 125I-iodo-pindolol Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
58187 Beta3 CLONED HUMAN 3H-CGP-12177 (S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxy-5-phenylthiophene-3-yl-methylpyrimidine-2,4-dione >10000 Duncan GE, et at., 2012 Jan 15, 2025 Jan 15, 2025
78412 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
95821 Beta3 CLONED HUMAN 125I-iodo-pindolol 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
101966 Beta3 CLONED HUMAN [3H]-CGP12177 ILOPERIDONE >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
75087 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
95823 Beta3 CLONED HUMAN 125I-iodo-pindolol N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
78160 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
71761 Beta3 CLONED HUMAN 125I-Pindolol DKR-1677 >10000 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
95825 Beta3 CLONED HUMAN 125I-iodo-pindolol tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
74322 Beta3 test test 125I-Pindolol N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
76114 Beta3 CLONED HUMAN 125I-Pindolol 2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
97106 Beta3 CLONED HUMAN [125I]Iodopindolol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
98898 Beta3 CLONED HUMAN 125I-Pindolol 3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
95827 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
77908 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
80980 Beta3 CLONED HUMAN 125I-Pindolol 3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine >10000 Rajagopalan R et al 2014 Jan 15, 2025 Jan 28, 2025
101972 Beta3 CLONED HUMAN [3H]-CGP12177 ZOTEPINE >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
80981 Beta3 CLONED HUMAN 125I-Pindolol 3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine >10000 Rajagopalan R et al 2014 Jan 15, 2025 Jan 28, 2025
95829 Beta3 CLONED HUMAN 125I-iodo-pindolol 2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
80982 Beta3 CLONED HUMAN 125I-Pindolol 5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine >10000 Rajagopalan R et al 2014 Jan 15, 2025 Jan 28, 2025
74840 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77656 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
87385 Beta3 CLONED HUMAN 125I-Pindolol 1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide >10000 Huang XP et al 2016 Jan 15, 2025 Jan 28, 2025
101721 Beta3 CLONED HUMAN [3H]-CGP12177 CLOZAPINE >10000 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
75868 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77404 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
66398 Beta3 CLONED HUMAN I-125-Pindolol N-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
72799 Beta3 CLONED HUMAN 125I-Pindolol epigallocatechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
101471 Beta3 CLONED HUMAN [3H]QNB Amisulpride >10000 PDSP Certified Data Mar 20, 2025 Mar 20, 2025
66656 Beta3 CLONED HUMAN I-125-Pindolol 3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
77152 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
87650 Beta3 CLONED HUMAN 125I-Pindolol 3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
98915 Beta3 CLONED HUMAN 125I-Iodopindolol 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
76900 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
72037 Beta3 CLONED HUMAN 125I-Pindolol 1-methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g] quinoxalin-2(6H)-one HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
76645 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
89957 Beta3 CLONED HUMAN 125I-Pindolol 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
74598 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75622 Beta3 CLONED HUMAN 125I-Pindolol 2-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
66920 Beta3 CLONED HUMAN I-125-Pindolol N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
50537 Beta3 CLONED HUMAN 125I-ICYP Prucalopride >10000 Briejer MR, et al., 2001 Jan 15, 2025 Jan 15, 2025
73322 Beta3 test test 125I-Pindolol N-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73579 Beta3 test test 125I-Pindolol 3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
67181 Beta3 CLONED HUMAN I-125-Pindolol {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
75374 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
68463 Beta3 CLONED HUMAN 125I-Iodopindolol N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
71023 Beta3 CLONED HUMAN 125I-Pindolol N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
76399 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
78705 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
73842 Beta3 test test 125I-Pindolol {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
70515 Beta3 CLONED HUMAN 125I-iodo-pindolol MRP3201 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
86131 Beta3 CLONED HUMAN 125I-Pindolol 4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
78453 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
74102 Beta3 test test 125I-Pindolol 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
16247 Beta3 CLONED HUMAN 3H-CGP-12177 KUR-1246 >10000 Kobayashi M, et al., 2001 Jan 15, 2025 Jan 15, 2025
75128 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
34169 Beta3 CLONED HUMAN 125I-CYP NOREPINEPHRINE 4300 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
78202 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
97146 Beta3 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
34170 Beta3 CLONED HUMAN 125I-CYP EPINEPHRINE >10000 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
76155 Beta3 CLONED HUMAN 125I-Pindolol 2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
34171 Beta3 CLONED HUMAN 125I-CYP Isoproterenol-l 1570 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34172 Beta3 CLONED HUMAN 125I-CYP Fenoterol >10000 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
70781 Beta3 test test 3H-CGP12177 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
34173 Beta3 CLONED HUMAN 125I-CYP Salbutamol,(+/-) >10000 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
71806 Beta3 CLONED HUMAN 3H-CGP12177 SAS-0132 >10000 Yi B et al 2017 Jan 15, 2025 Jan 28, 2025
77950 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
34174 Beta3 CLONED HUMAN 125I-CYP Salmeterol 7180 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34175 Beta3 CLONED HUMAN 125I-CYP Formoterol 8090 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34176 Beta3 CLONED HUMAN 125I-CYP Terbutaline >10000 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
74881 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
34177 Beta3 CLONED HUMAN 125I-CYP BRL 37344 430 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
101761 Beta3 CLONED HUMAN [3H]-CGP12177 Remoxapride >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
77698 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
34178 Beta3 CLONED HUMAN 125I-CYP ALPRENOLOL 35 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
61826 Beta3 CLONED HUMAN 3H-CGP-12177 FECIMBI-36 >10000 Prabhakaran, Jaya et. al. 2015 Jan 15, 2025 Jan 15, 2025
34179 Beta3 CLONED HUMAN 125I-CYP PINDOLOL,(+/-) 44.1 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34180 Beta3 CLONED HUMAN 125I-CYP Carvedilol 247 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
75909 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
34181 Beta3 CLONED HUMAN 125I-CYP ATENOLOL >10000 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
59525 Beta3 CLONED HUMAN 3H-CGP-12177 Nantenin >10000 LeGendre, O. et. al., 2009 Jan 15, 2025 Jan 15, 2025
77446 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
34182 Beta3 CLONED HUMAN 125I-CYP Bisoprolol 9070 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34183 Beta3 CLONED HUMAN 125I-CYP metoprolol >10000 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34184 Beta3 CLONED HUMAN 125I-CYP PROPRANOLOL, l- 186 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
66441 Beta3 CLONED HUMAN I-125-Pindolol N-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
34185 Beta3 CLONED HUMAN 125I-CYP CGP 20712-A 2360 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
77194 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N,2-dibutyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
34186 Beta3 CLONED HUMAN 125I-CYP SR 59230A 122 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
34187 Beta3 CLONED HUMAN 125I-CYP CGP 12177 77.1 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
66700 Beta3 CLONED HUMAN I-125-Pindolol ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
72332 Beta3 CLONED HUMAN 3H-CGP-12177 2-Aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 28, 2025
72844 Beta3 CLONED HUMAN 125I-Pindolol isoginkgetin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
34188 Beta3 CLONED HUMAN 125I-CYP ICI 118,551 611 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
102028 Beta3 CLONED HUMAN [3H]-CGP12177 RS-(+/-)-Sulpriride >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
34189 Beta3 CLONED HUMAN 125I-CYP Broxaterol 3990 Hoffmann C, et al., 2004 Jan 15, 2025 Jan 15, 2025
76942 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
75663 Beta3 CLONED HUMAN 125I-Pindolol benzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76687 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
87695 Beta3 CLONED HUMAN 125I-Pindolol 3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
74640 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
91280 Beta3 CLONED HUMAN 125I-Pindolol 17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan >10000 Zheng Y et al 2018 Jan 15, 2025 Jan 28, 2025
87441 Beta3 CLONED HUMAN 125I-Pindolol 4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide >10000 Huang XP et al 2016 Jan 15, 2025 Jan 28, 2025
83858 Beta3 CLONED HUMAN 125I-Pindolol (±)-N-(((4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)methyl)aniline 1924 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84114 Beta3 CLONED HUMAN 125I-Pindolol (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-(trifluoromethyl)benzamide 7549 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
98962 Beta3 CLONED HUMAN 125I-Pindolol C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
83859 Beta3 CLONED HUMAN 125I-Pindolol (±)-4-chloro-N-(((4aS,8R,8aS)-2-benzyl-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)methyl)-3-(trifluoromethyl)aniline 1104 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
66964 Beta3 CLONED HUMAN I-125-Pindolol 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
71061 Beta3 CLONED HUMAN 125I-Pindolol N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
73365 Beta3 test test 125I-Pindolol N-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74390 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75414 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,2-dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d]- [1,3]dioxole-3b(3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
73623 Beta3 test test 125I-Pindolol ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
67224 Beta3 CLONED HUMAN I-125-Pindolol {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
76440 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
63128 Beta3 CLONED HUMAN I125- Pindolol Mitragynine >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
72089 Beta3 CLONED HUMAN 125I-Pindolol 2-methoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
78747 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
73884 Beta3 test test 125I-Pindolol {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
84126 Beta3 CLONED HUMAN 125I-Pindolol (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-methylbenzamide 6686 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
78495 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
86175 Beta3 CLONED HUMAN 125I-Pindolol 2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
70560 Beta3 CLONED HUMAN 125I-iodo-pindolol MRP3160 6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
75169 Beta3 CLONED HUMAN 125I-Pindolol methyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74146 Beta3 test test 125I-Pindolol naftopidil 250 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
97186 Beta3 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
70820 Beta3 CLONED HUMAN 125I-Iodopindolol D-578 2703 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
76196 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
78244 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
41381 Beta3 CLONED RAT 125I-Pindolol 2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione >10000 Kumar JS, et al., 2006 Jan 15, 2025 Jan 15, 2025
101798 Beta3 CLONED HUMAN [3H]-CGP12177 RISPERIDONE >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
83879 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aS,8S,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5066 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
77992 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
72361 Beta3 CLONED HUMAN 3H-CGP-12177 5-Methoxy-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 28, 2025
74922 Beta3 CLONED HUMAN 125I-Pindolol 1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
81066 Beta3 CLONED HUMAN 125I-Pindolol N-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
50602 Beta3 CLONED HUMAN 125I-Iodopindolol Amisulpride >10000 Abbas AI et.al., 2009 Jan 15, 2025 Jan 15, 2025
62379 Beta3 CLONED HUMAN 3H-CGP-12177 Diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
77740 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
62380 Beta3 CLONED HUMAN 3H-CGP-12177 2-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
62381 Beta3 CLONED HUMAN 3H-CGP-12177 3-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
75950 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
100014 Beta3 CLONED HUMAN 125I-Pindolol 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
62382 Beta3 CLONED HUMAN 3H-CGP-12177 4-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
100015 Beta3 CLONED HUMAN 125I-Pindolol 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
62383 Beta3 CLONED HUMAN 3H-CGP-12177 2-Cl-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63151 Beta3 CLONED HUMAN I125-Iodopindolol Mitragynine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
69552 Beta3 CLONED HUMAN 125I-iodo-pindolol Ephenidine >10000 Kang, H. et, al. 2017 Jan 15, 2025 Jan 28, 2025
77488 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
101552 Beta3 CLONED HUMAN [3H]-CGP12177 OLANZAPINE >10000 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
87474 Beta3 CLONED HUMAN 125I-Pindolol FK881 >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
66484 Beta3 CLONED HUMAN I-125-Pindolol N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
77236 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
91318 Beta3 CLONED HUMAN 125I-Pindolol 17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan >10000 Zheng Y et al 2018 Jan 15, 2025 Jan 28, 2025
94903 Beta3 CLONED HUMAN 125I-Pindolol 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
66744 Beta3 CLONED HUMAN I-125-Pindolol N-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
72888 Beta3 CLONED HUMAN 125I-Pindolol 2″-glucosylvitexin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
75704 Beta3 CLONED HUMAN 125I-Pindolol 2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76984 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
92600 Beta3 CLONED HUMAN 125I-Pindolol (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94904 Beta3 CLONED HUMAN 125I-Pindolol 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
76729 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
92601 Beta3 CLONED HUMAN 125I-Pindolol 9,13:15,16-diepoxylabdane-6b,15a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94905 Beta3 CLONED HUMAN 125I-Pindolol 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
74682 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
94906 Beta3 CLONED HUMAN 125I-Pindolol 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
94907 Beta3 CLONED HUMAN 125I-Pindolol 4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
92604 Beta3 CLONED HUMAN 125I-Pindolol 9,13:15,16-diepoxylabdane-6b,16b-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94908 Beta3 CLONED HUMAN 125I-Pindolol 4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
99004 Beta3 CLONED HUMAN 125I-Pindolol [[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
92605 Beta3 CLONED HUMAN 125I-Pindolol 9,13:15,16-diepoxylabdane-6b,16a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94909 Beta3 CLONED HUMAN 125I-Pindolol 4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
74430 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
94910 Beta3 CLONED HUMAN 125I-Pindolol 4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
67007 Beta3 CLONED HUMAN I-125-Pindolol [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
73407 Beta3 test test 125I-Pindolol N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
75455 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-4-(2-((5-bromothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
94911 Beta3 CLONED HUMAN 125I-Pindolol 4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
58303 Beta3 CLONED HUMAN 125I-Pindolol MRS3558 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
92608 Beta3 CLONED HUMAN 125I-Pindolol 9,13-epoxylabd-5-en-7-on-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94912 Beta3 CLONED HUMAN 125I-Pindolol 4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
58304 Beta3 CLONED HUMAN 125I-Pindolol MRS5202 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
76481 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
92609 Beta3 CLONED HUMAN 125I-Pindolol 15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94913 Beta3 CLONED HUMAN 125I-Pindolol 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
58305 Beta3 CLONED HUMAN 125I-Pindolol MRS5923 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
94914 Beta3 CLONED HUMAN 125I-Pindolol 2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate 1240 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
58306 Beta3 CLONED HUMAN 125I-Pindolol MRS5930 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
94915 Beta3 CLONED HUMAN 125I-Pindolol 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
58307 Beta3 CLONED HUMAN 125I-Pindolol MRS5474 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
67268 Beta3 CLONED HUMAN I-125-Pindolol 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
92612 Beta3 CLONED HUMAN 125I-Pindolol 9,13-epoxy-15,16-dihydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
94916 Beta3 CLONED HUMAN 3H-CGP-12177 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
102084 Beta3 CLONED HUMAN [3H]-CGP12177 Lurasidone HCl >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
73669 Beta3 test test 125I-Pindolol N-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
78789 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
92613 Beta3 CLONED HUMAN 125I-Pindolol 9,13-epoxylabd-5-ene-7 b,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
72390 Beta3 CLONED HUMAN 3H-CGP-12177 5-methoxy-6-methyl-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 28, 2025
73926 Beta3 test test 125I-Pindolol {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
92616 Beta3 CLONED HUMAN 125I-Pindolol (8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
78537 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
92617 Beta3 CLONED HUMAN 125I-Pindolol 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
102089 Beta3 CLONED HUMAN [3H]-CGP12177 GMC 1-116 >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
75210 Beta3 CLONED HUMAN 125I-Pindolol ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
101834 Beta3 CLONED HUMAN [3H]-CGP12177 SERTINDOLE >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
62922 Beta3 CLONED HUMAN 3H-CGP12177 Ketamine >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86219 Beta3 CLONED HUMAN 125I-Pindolol 4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
72140 Beta3 CLONED HUMAN 125I-Pindolol 2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
92620 Beta3 CLONED HUMAN 125I-Pindolol 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
76237 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
78286 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
74191 Beta3 test test 125I-Pindolol N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
84176 Beta3 CLONED HUMAN 125I-Pindolol (±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 4431 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85200 Beta3 recombinant HUMAN 125I-cyanopindolol Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 28, 2025
70610 Beta3 CLONED HUMAN 125I-iodo-pindolol MRP3172 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
78034 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
81106 Beta3 CLONED HUMAN 125I-Pindolol N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
96978 Beta3 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
74964 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77782 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
85974 Beta3 CLONED HUMAN 125I-Pindolol 1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
75991 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77530 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
72670 Beta3 CLONED HUMAN 125I-Pindolol 2,3-dihydrohinokiflavone >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
77278 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
66527 Beta3 CLONED HUMAN I-125-Pindolol N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
87519 Beta3 CLONED HUMAN 125I-Pindolol 1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 28, 2025
75745 Beta3 CLONED HUMAN 125I-Pindolol 3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
77026 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
72419 Beta3 CLONED HUMAN 3H-CGP-12177 5,6-methylenedioxy-2-aminoindan >10000 Halberstadt Adam L et al 2019 Jan 15, 2025 Jan 28, 2025
74723 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
84195 Beta3 CLONED HUMAN 125I-Pindolol (±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 5737 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
66788 Beta3 CLONED HUMAN I-125-Pindolol N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
76774 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
73191 Beta3 test test 125I-Pindolol 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74471 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
66024 Beta3 CLONED HUMAN I125- Iodopindolol Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
75496 Beta3 CLONED HUMAN 125I-Pindolol propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
73450 Beta3 test test 125I-Pindolol N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
76522 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
85994 Beta3 CLONED HUMAN 125I-Pindolol Delta9 -tetrahydrocannabinol (THC)) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
58602 Beta3 CLONED HUMAN 125I-Pindolol MRS5698 1450 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
67051 Beta3 CLONED HUMAN I-125-Pindolol {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
58603 Beta3 CLONED HUMAN 125I-Pindolol MRS5678 1560 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58604 Beta3 CLONED HUMAN 125I-Pindolol MRS5697 1170 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
98797 Beta3 CLONED HUMAN 125I-Pindolol 3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
58605 Beta3 CLONED HUMAN 125I-Pindolol MRS5676 2320 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58606 Beta3 CLONED HUMAN 125I-Pindolol MRS5755 2460 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
78831 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
73713 Beta3 test test 125I-Pindolol [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73970 Beta3 test test 125I-Pindolol 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
75251 Beta3 CLONED HUMAN 125I-Pindolol ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
78579 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
101619 Beta3 CLONED HUMAN [3H]-CGP12177 Paliperidone >10000 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
69877 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-(1-phenylcyclohexyl)morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
69878 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-[1-(3-methylphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
70646 Beta3 CLONED HUMAN 125I-iodo-pindolol MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
76278 Beta3 CLONED HUMAN 125I-Pindolol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
69879 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
101879 Beta3 CLONED HUMAN [3H]-CGP12177 S-(-)-Sulpride >10000 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
102135 Beta3 CLONED HUMAN [3H]-CGP12177 Melperone HCl >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
69880 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-[1-(4-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
78328 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
84216 Beta3 CLONED HUMAN 125I-Pindolol (±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 7503 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
69881 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
86265 Beta3 CLONED HUMAN 125I-Pindolol JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
100089 Beta3 CLONED HUMAN 125I-Pindolol Cariprazine 1882 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
69882 Beta3 CLONED HUMAN 125I-iodo-pindolol 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 15, 2025
74234 Beta3 test test 125I-Pindolol N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
81147 Beta3 CLONED HUMAN 125I-Pindolol N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
81915 Beta3 CLONED HUMAN 125I-Pindolol (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
78076 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
75005 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
256 5-HT1A CORTEX RAT 3H-8-OH-DPAT DHE 19 McCARTHY & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
512 5-HT1A HIPPOCAMPUS RAT 3H-SPIROXATRINE SPIPERONE 28.8 NELSON ET AL., 1987 Jan 15, 2025 Jan 15, 2025
69376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 1202 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
13312 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT CITALOPRAM >10000 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
80896 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
83200 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LSD 2.78 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85760 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide 230 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
20736 5-HT1A HIPPOCAMPUS RAT 3H-PAT QUIPAZINE 3388.44 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
27136 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CP-132,484 8410 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94208 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine 3300 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95488 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT 1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione 11 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
97280 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine BUSPIRONE 50 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
101632 5-HT1A CLONED HUMAN [3H]-8-OH-DPAT Perospirone 0.7 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
37632 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(1-Naphthalenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 0.6 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52224 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 11.2 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55040 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 19 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55552 5-HT1A UNDEFINED RAT UNDEFINED 4-[4-(4-Benzylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 2730 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
257 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DILTIAZEM >10000 PEROUTKA, 1988 Jan 15, 2025 Jan 15, 2025
67841 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
69377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPHENAZINE 145 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
71425 5-HT1A CLONED HUMAN WAY100635 4-acetoxy-N,N-diallyltryptamine 383 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71937 5-HT1A test test [3H] Way100635 8-(4-(Benzo[d]thiazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one 195 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
73217 5-HT1A test test [3H] Way100635 N-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride 371 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
76545 5-HT1A CLONED HUMAN 3H-WAY100635 (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
13313 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT INDALPINE 9120.1 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
82689 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
85761 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
20737 5-HT1A HIPPOCAMPUS RAT 3H-PAT CINANSERIN 1096.48 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
87041 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 2000 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 365 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24577 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 1.8 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
90881 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane 50.1187 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27137 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CP-132,484(4b) 287 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94209 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-benzyloxy-2,5-dimethoxyphenethylamine 2700 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95489 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT 7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione 1 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
101377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 22 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37633 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(4-Chloro-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 433 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52225 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 3.89 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55041 5-HT1A UNDEFINED HUMAN UNDEFINED 4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide 325 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55553 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 35 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
258 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DMT 119.51 PIERCE & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
514 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 32.76 HALL ET AL., 1985 Jan 15, 2025 Jan 15, 2025
69378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CHLORPROMAZINE 3115 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
73474 5-HT1A test test [3H] Way100635 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 476 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
13314 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT PAROXETINE >10000 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
20738 5-HT1A HIPPOCAMPUS RAT 3H-PAT PIZOTIFEN 2187.76 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
24578 5-HT1A FR. CORTEX RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 4.2 Borsini F, et al., 1995 Jan 15, 2025 Jan 15, 2025
27138 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N,N-dimethyl derivative 562 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94210 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-allyloxy-2,5-dimethoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95490 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT 7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione 5 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
37634 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[2-[4-(4-Methyl-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide 58.6 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52226 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 1.33 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55042 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 70 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55554 5-HT1A UNDEFINED RAT UNDEFINED 4-[3-(4-Phenylpiperazin-1-yl)propyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 294 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
63490 5-HT1A CLONED HUMAN 3H-WAY100635 bifeprunox 0.73 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
515 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 45.12 COSSERY ET AL.,1986 Jan 15, 2025 Jan 15, 2025
69379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RACLOPRIDE >10000 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
70403 5-HT1A CLONED HUMAN 3H-WAY100635 (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 328 Omran, A. et, al. 2018 Jan 15, 2025 Jan 15, 2025
13315 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT Femoxetine 3162.27 Wong DT, et al., 1991 Jan 15, 2025 Jan 15, 2025
20739 5-HT1A HIPPOCAMPUS RAT 3H-PAT CYPROHEPTADINE 977.237 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
27139 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95491 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT 7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride 433 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
37635 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[3-[4-(2,3-Dichlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 117 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52227 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(adamantan-1-ylamino)-3-(1H-indol-5-yloxy)-propan-2-ol 833 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55043 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 8.2 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55555 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 44 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
55811 5-HT1A UNDEFINED RAT UNDEFINED [C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline 54 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
59139 5-HT1A CLONED HUMAN 3H-WAY100635 CHLORPROMAZINE 3000 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
260 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT DMT 140.74 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
516 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 48.07 HOYER ET AL., 1985 Jan 15, 2025 Jan 15, 2025
67076 5-HT1A CLONED HUMAN 3H-WAY100635 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
69380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 427 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
70404 5-HT1A CLONED HUMAN 3H-WAY100635 MRP5063 5.7 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
80644 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
85508 5-HT1A test test [3H] Way100635 8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 103 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
20740 5-HT1A HIPPOCAMPUS RAT 3H-PAT METHIOTHEPIN 89.1251 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
86788 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide 590 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87044 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one 58.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
27140 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94212 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95492 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT 7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride 239 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
37636 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 123 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52228 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-5-yloxy)-3-(cyclohexylamino)propan-2-ol 3000 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55044 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide 13 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55556 5-HT1A UNDEFINED RAT UNDEFINED 4-[3-(4-Phenylpiperazin-1-yl)propyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 344 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
55812 5-HT1A UNDEFINED RAT UNDEFINED [C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline 1120 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
261 5-HT1A CORTEX RAT 3H-8-OH-DPAT DMT 245 TAYLOR ET AL,. 1987 Jan 15, 2025 Jan 15, 2025
517 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIPERONE 54 FOZARD ET AL., 1987 Jan 15, 2025 Jan 15, 2025
3333 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Amphetamine,(+) 6606 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 105 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
83205 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DMT 450 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
20741 5-HT1A HIPPOCAMPUS RAT 3H-PAT METHYSERGIDE 70.7946 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
86789 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide 325 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
90885 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 42.658 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27141 5-HT1A CLONED HUMAN 3H-8-OH-DPAT AL-37350A >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94213 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95493 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT 7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride 171 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
100101 5-HT1A CLONED HUMAN 3H-WAY100635 Quetiapine 267 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37637 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide 78.7 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52229 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-4-yloxy)-4-(cyclohexylamino)butan-2-ol 125 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55045 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide 139 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55557 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 27 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
55813 5-HT1A UNDEFINED RAT UNDEFINED [C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline 685 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
59141 5-HT1A CLONED HUMAN 3H-WAY100635 CYPROHEPTADINE 50 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
63493 5-HT1A CLONED HUMAN 3H-WAY100635 RISPERIDONE 420 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
262 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB 3770 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
67846 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3334 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SKF 82958 1781 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT OLANZAPINE 2063 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
83206 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOM >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85766 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide 495 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
20742 5-HT1A HIPPOCAMPUS RAT 3H-PAT METERGOLINE 34.6737 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
27142 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOI,(-) 3843 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
94214 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-isopropoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
95494 5-HT1A HIPPOCAMPUS RAT [3H]-8-OH-DPAT BUSPIRONE 20 Partyka A et al 2015 Jan 15, 2025 Jan 15, 2025
100870 5-HT1A CLONED HUMAN 3H-WAY100635 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1) 85.7 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 15, 2025
101382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 48 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37638 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 19.8 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52230 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(adamantan-1-ylamino)-4-(1H-indol-4-yloxy)-butan-2-ol 551 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55046 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide 161 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55558 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Pyridyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 200 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
55814 5-HT1A UNDEFINED RAT UNDEFINED [C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline 1990 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
59142 5-HT1A CLONED HUMAN 3H-WAY100635 HALOPERIDOL 3500 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
3335 5-HT1A CLONED HUMAN 3H-8-OH-DPAT APOMORPHINE 4929 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Quetiapine 431 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
71943 5-HT1A test test [3H] Way100635 8-(4-(5-Chlorobenzo[d]thiazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one 102 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
85767 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide 500 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
20743 5-HT1A HIPPOCAMPUS RAT 3H-PAT 5-MT 288.403 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
87047 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one 196.2 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
93191 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 410 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
94215 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,4,5-trimethoxyamphetamine >10000 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
31495 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) 1584.89 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
33287 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Acetylsalicylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37639 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 7.5 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52231 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(1H-indol-4-yloxy)-1-(cyclohexylamino)butan-2-ol 872 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55047 5-HT1A UNDEFINED HUMAN UNDEFINED N-Benzyl-4-(2-methylthiophenyl)-1-piperazinehexanamide 12 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55559 5-HT1A UNDEFINED RAT UNDEFINED 4-[3-(4-Phenylpiperazin-1-yl)propoxy]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 115 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
55815 5-HT1A UNDEFINED RAT UNDEFINED [C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline 50 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
264 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DOB 6326.73 PIERCE & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
520 5-HT1A CELLS C0S-7 3H-8-OH-DPAT SPIPERONE 63 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
66056 5-HT1A CLONED HUMAN 3H-WAY100635 Mellpaladine A 7500 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
3336 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BROMOCRIPTINE,(+) 25 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
80392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 3215 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
20744 5-HT1A HIPPOCAMPUS RAT 3H-PAT TRYPTAMINE 3715.35 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
89352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 3842 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89608 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 0.47863 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
94216 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-Bromo-2,5-dimethoxyphenethylamine 311 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
31496 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) 1000 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
37640 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide 4.5 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
39944 5-HT1A UNDEFINED RAT UNDEFINED BW-723C86 1258.93 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
52232 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(1H-indol-4-yloxy)-1-(isopropylamino)butan-2-ol 1772 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55048 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 40 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55560 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 80 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
55816 5-HT1A UNDEFINED RAT UNDEFINED [C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline 164 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
265 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB 3770 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
521 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 66.1 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
66057 5-HT1A CLONED HUMAN 3H-WAY100635 Mellpaladine B 652 Uchimasu, Hajime. et, al. 2016 Jan 15, 2025 Jan 15, 2025
67337 5-HT1A CLONED HUMAN 3H-WAY100635 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 58 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
3337 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CARBAMAZEPINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
72457 5-HT1A test test [3H] Way100635 2-(5-Iodo-1H-indol-3-yl)-N,N-dimethylethanamine 130 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
81161 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
20745 5-HT1A HIPPOCAMPUS RAT 3H-PAT alpha-M-5-HT 158.489 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
90889 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 20.4174 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
37641 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[3-[4-(4-Chlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide 850 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52233 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(adamantan-1-ylamino)-1-(1H-indol-4-yloxy)-butan-2-ol 76.1 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55049 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 3.7 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55561 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 37 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
59145 5-HT1A CLONED HUMAN 3H-WAY100635 KETANSERIN 1044 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
266 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB,R(-) 2332 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68106 5-HT1A UNDEFINED UNDEFINED 3H-8-OH-DPAT ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
3338 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CGS 12066B 44 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
75274 5-HT1A CLONED HUMAN 3H-WAY100635 Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
14602 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SB-277011-A 5011.87 Reavill C., et al., 2000 Jan 15, 2025 Jan 15, 2025
83722 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 9987 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
20746 5-HT1A HIPPOCAMPUS RAT 3H-PAT 5-M-N,N-DMT 39.8107 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
86794 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide 219 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87050 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 193.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
26890 5-HT1A CLONED HUMAN 3H-8-OH-DPAT xanomeline 63.0957 Watson J.,et. al.,1998 Jan 15, 2025 Jan 15, 2025
37642 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 397 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52234 5-HT1A UNDEFINED HUMAN UNDEFINED PINDOLOL,(+/-) 81.1 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55050 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 95 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55562 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 124 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
267 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOB,S(+) 4041 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
523 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 66.1 ENGEL ET AL, 1986 Jan 15, 2025 Jan 15, 2025
67851 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3339 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CHLORPROMAZINE 3115 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
70411 5-HT1A CLONED HUMAN 3H-WAY100635 MRP4268 5.6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
73739 5-HT1A test test [3H] Way100635 {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
78603 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
81675 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol >10000 Dutta AK et al 2011 Jan 15, 2025 Jan 15, 2025
83211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN 6510 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
18443 5-HT1A CLONED HUMAN 3H-5HT 1-NP 9.2 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
85515 5-HT1A test test [3H] Way100635 1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride 214 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
20747 5-HT1A HIPPOCAMPUS RAT 3H-PAT DMT,5-OH 21.3796 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
86795 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide 331 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
89355 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 802 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
100875 5-HT1A CLONED HUMAN 3H-WAY100635 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1) 24.6 Stephenson, K. et. al., 2008 Jan 15, 2025 Jan 15, 2025
101387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 35 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37643 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[5-[4-(4-Chlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide 850 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52235 5-HT1A UNDEFINED HUMAN UNDEFINED N-(3-(1H-indol-4-yloxy)propyl)cyclopentanamine 233 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55051 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2.04 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55563 5-HT1A UNDEFINED RAT UNDEFINED 4-[3-(4-Phenylpiperazin-1-yl)propoxy]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 616 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
59147 5-HT1A CLONED HUMAN 3H-WAY100635 METHYSERGIDE 25 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
268 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOBU 4178 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
524 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIPERONE 66.1 SCHLICKER ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3340 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOMIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
73996 5-HT1A test test [3H] Way100635 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 348 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
76300 5-HT1A CLONED HUMAN 3H-WAY100635 (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
80908 5-HT1A CLONED HUMAN 3H-WAY100635 3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine 630.957 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
82188 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one 62 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
83212 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ro 60-0175 6680 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
18444 5-HT1A CLONED HUMAN 3H-5HT 7-methoxy-1-naphthylpiperazine 2.8 Jorand-Lebrun C et al., 1997a Jan 15, 2025 Jan 15, 2025
85772 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
20748 5-HT1A HIPPOCAMPUS RAT 3H-PAT RU 24969 9.77237 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
31244 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PPP, S(-)-3 1730 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37644 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dimethylphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 268 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52236 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-4-yloxy)-3-(pentan-3-ylamino)propan-2-ol 49.8 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55052 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 3.2 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55564 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 331 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
269 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOET 3930 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3341 5-HT1A CLONED HUMAN 3H-8-OH-DPAT COCAINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71949 5-HT1A test test [3H] Way100635 8-(4-(Benzo[d]oxazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one 382 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
80909 5-HT1A CLONED HUMAN 3H-WAY100635 3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine 371.535 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
85773 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide 1000 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
20749 5-HT1A HIPPOCAMPUS RAT 3H-PAT 5-Hydroxy Tryptamine 6.76083 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
87053 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on 98 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89613 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 2.5704 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90893 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane 36.3078 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
25869 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27405 5-HT1A CLONED HUMAN 3H-8-OH-DPAT APOMORPHINE 117.49 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
37645 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(1-Naphthalenyl)piperazin-1-yl]butyl]-3-methoxybenzamide 0.43 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52237 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-4-yloxy)-3-(cycloheptylamino)propan-2-ol 11.3 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
55053 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 22 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55565 5-HT1A UNDEFINED RAT UNDEFINED 4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 92 Bojarski AJ et al., 2009 Jan 15, 2025 Jan 15, 2025
59149 5-HT1A CLONED HUMAN 3H-WAY100635 RISPERIDONE 427 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
63501 5-HT1A CLONED RAT 3H-WAY100635 Brexpiprazole 0.09 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
270 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT DOI 2355 TITELER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3342 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CYPROHEPTADINE 59 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
70414 5-HT1A CLONED HUMAN 3H-WAY100635 MRP4269 6.5 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
80910 5-HT1A CLONED HUMAN 3H-WAY100635 5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine >10000 Rajagopalan R et al 2014 Jan 15, 2025 Jan 15, 2025
20750 5-HT1A HIPPOCAMPUS RAT 3H-PAT Placeholder 3.01995 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
89614 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.86209 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27406 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BROMOCRIPTINE 12.8825 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
37646 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(1-Isoquinolyl)piperazin-1-yl]butyl]-3-methoxybenzamide 12.7 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52238 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-4-yloxy)-3-(cyclopentylamino)propan-2-ol 35.5 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53774 5-HT1A UNDEFINED HUMAN UNDEFINED CLOZAPINE 140 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
55054 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 124 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
271 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT GEPIRONE 70 GLENNON ET AL., 1988 Jan 15, 2025 Jan 15, 2025
3343 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DEPRENYL >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
27407 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Cabergoline 19.9526 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
93199 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 120 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
37647 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(1,2-Benzisoxazol-3-yl)piperazin-1-yl]butyl]-3-methoxybenzamide 7730 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52239 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 7.84 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53775 5-HT1A UNDEFINED HUMAN UNDEFINED HALOPERIDOL 3600 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
55055 5-HT1A UNDEFINED HUMAN UNDEFINED 2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 1.07 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
56591 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-((benzo[d][1,3]dioxol-5-yl)methyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate >10000 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
59151 5-HT1A CLONED HUMAN 3H-WAY100635 PROPANOLOL(-) 78 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
63503 5-HT1A CLONED RAT 3H-WAY100635 ARIPIPRAZOLE 1.2 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
67856 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3344 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DESIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78864 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-2,5-Dimethoxy-4-bromoamphetamine 2550 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80656 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
82448 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine 0.6 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
20752 5-HT1A HIPPOCAMPUS RAT 3H-PAT HALOPERIDOL 3548.13 Gozlan H et al., 1983 Jan 15, 2025 Jan 15, 2025
86800 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide 99.1 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87056 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one 69.1 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
27408 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LISURIDE 0.147911 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95248 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 192.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 482 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37648 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-bromo-1-methoxy-2-naphthalenecarboxamide 1000 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52240 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 9.83 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53776 5-HT1A UNDEFINED HUMAN UNDEFINED Quetiapine 230 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
55056 5-HT1A UNDEFINED HUMAN UNDEFINED 8-OH-DPAT 2.1 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
56592 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate >10000 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
273 5-HT1A CORTEX PIG 3H-8-OH-DPAT GEPIRONE 89.1 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
529 5-HT1A CELLS C0S-7 125I-NAPS SPIPERONE 66.2 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
3345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DHE 1.5 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78865 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-3,4-Methylenedioxyamphetamine 3762 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
83217 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SB242087 9300 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
86801 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide 100 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
88593 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 140 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
90897 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one 64.5654 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27409 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PERGOLIDE 1.90546 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95249 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 182 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37649 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-methoxy-2-naphthalenecarboxamide 575 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52241 5-HT1A UNDEFINED HUMAN UNDEFINED (R)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 29.9 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53777 5-HT1A UNDEFINED HUMAN UNDEFINED OLANZAPINE 2100 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56593 5-HT1A UNDEFINED RAT UNDEFINED ethyl 5-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate >10000 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
59153 5-HT1A CLONED HUMAN 3H-WAY100635 BROMOCRIPTINE 12.9 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
63505 5-HT1A CLONED RAT 3H-WAY100635 RISPERIDONE 250 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
274 5-HT1A CORTEX RAT 3H-WB4101 HALOPERIDOL 346.2 NORMAN ET AL., 1985 Jan 15, 2025 Jan 15, 2025
530 5-HT1A HIPPOCAMPUS HUMAN 3H-8-OH-DPAT SPIPERONE 100.92 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
72466 5-HT1A test test [3H] Way100635 ERGOTAMINE 0.17 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
78866 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-3,4-Methylenedioxymethamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
83218 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide 1.21 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
85522 5-HT1A test test [3H] Way100635 1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride 28.3 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
85778 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide 443 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
21778 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT CLOZAPINE 1700 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
89362 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 6631 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
27410 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piribedil 446.684 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
27666 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
95250 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 728.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37650 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-naphthalenecarboxamide 335 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52242 5-HT1A UNDEFINED HUMAN UNDEFINED (R)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 50.8 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53778 5-HT1A UNDEFINED HUMAN UNDEFINED Ziprasidone 2.5 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56594 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-(2-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate >10000 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
275 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT HALOPERIDOL 2761.11 GOZLAN ET AL., 1983 Jan 15, 2025 Jan 15, 2025
531 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 101 TITELER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
3347 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOPAMINE 8248 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71955 5-HT1A test test [3H] Way100635 8-(4-(1H-Indol-3-yl)butyl)-1-phenyl-1,3,8-triazaspiro[4.5] decan-4-one 376 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
78867 5-HT1A CLONED HUMAN 3H-WAY100635 3,4,5-Trimethoxyphenethylamine 1841 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85779 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide 52.7 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87059 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 82.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
21779 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT HALOPERIDOL 2500 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
89619 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1.25893 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27411 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Pramipexole 691.831 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95251 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 82.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37651 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-quinolinecarboxamide 88.5 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52243 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 24 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53779 5-HT1A UNDEFINED HUMAN UNDEFINED RISPERIDONE 210 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56595 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-(2-cyanophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate >10000 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
62227 5-HT1A CLONED HUMAN 3H-WAY100635 Tianeptine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
276 5-HT1A CORTEX HUMAN 3H-WB4101 HALOPERIDOL 2800 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
532 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIPERONE 120 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
3348 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 8-OH-DPAT 6.9 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
6164 5-HT1A UNDEFINED UNDEFINED UNDEFINED SB204070 1000 WARDLE KA, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
74260 5-HT1A test test [3H] Way100635 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 52 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
75028 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
78100 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78868 5-HT1A CLONED HUMAN 3H-WAY100635 4-Bromo-2,5-dimethoxyphenethylamine 240.8 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80404 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
21780 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT Amisulpride >10000 Schoemaker H et al., 1997 Jan 15, 2025 Jan 15, 2025
89620 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.562341 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27412 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Quinelorane >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95252 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 212.6 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31252 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PPP, R(+)-3 868.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
33556 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CELECOXIB >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
37652 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-(1,1'-biphenyl)-4-carboxamide 1000 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52244 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 4.65 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53780 5-HT1A UNDEFINED HUMAN UNDEFINED 4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one 2332 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56596 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-o-tolylpiperazin-1-yl)propoxy)-1H-indole-2-carboxylate >10000 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
277 5-HT1A CORTEX PIG 3H-8-OH-DPAT HALOPERIDOL 4790 HOYER, 1989 (J.R.R.) Jan 15, 2025 Jan 15, 2025
533 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT SPIPERONE 130.76 HOYER ET AL., 1986 Jan 15, 2025 Jan 15, 2025
67861 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 146 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
3349 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ETICLOPRIDE,S(-) 1790 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
77845 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78869 5-HT1A CLONED HUMAN 3H-WAY100635 DMT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
13845 5-HT1A BRAIN RAT 3H-8-OH-DPAT CLOZAPINE 150 Tang AH, et al., 1996 Jan 15, 2025 Jan 15, 2025
82709 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
89365 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 6064 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
90901 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one 323.594 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27413 5-HT1A CLONED HUMAN 3H-8-OH-DPAT QUINPIROLE 1698.24 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95253 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 2600 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101397 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 20 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37653 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-benzofurancarboxamide36 126 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
52245 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 6.68 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
53781 5-HT1A UNDEFINED HUMAN UNDEFINED 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one 117.4 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56597 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate 35.8 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
534 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIPERONE 140 SCHLEGEL & PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
3350 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPENTHIXOL, Alpha 8028 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78870 5-HT1A CLONED HUMAN 3H-WAY100635 4-Hydroxy-N,N-dimethyltryptamine 62.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86806 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide 9.19 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87062 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(3-(4-(6-fluoro benzo[d]isoxazol-3-yl)piperidin-1-yl)- 1-hydroxypropyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 19.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
27414 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ropinirole 288.403 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95254 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 158 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
33046 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT GBR-12909 3600 Andersen PH, et al., 1989 Jan 15, 2025 Jan 15, 2025
37654 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide 1660 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
53782 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one 30.5 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56598 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-(4-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate 14 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
63510 5-HT1A CLONED HUMAN 3H-WAY100635 Cariprazine 3 citrome, Leslie et. al, 2013 Jan 15, 2025 Jan 28, 2025
535 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIPERONE 148.4 HALL ET AL., 1986 Jan 15, 2025 Jan 15, 2025
3351 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPHENAZINE 2829 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
76055 5-HT1A CLONED HUMAN 3H-WAY100635 Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
78871 5-HT1A CLONED HUMAN 3H-WAY100635 DMT,5-MeO 1.9 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86807 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide 0.0113 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
27415 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Roxindole 0.114815 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95255 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 298 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37655 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indole-3-carboxamide 1110 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
50711 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT [11C]MMP 0.15 Kumar JS et al., 2007 Jan 15, 2025 Jan 15, 2025
53783 5-HT1A UNDEFINED HUMAN UNDEFINED 4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 831.5 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56599 5-HT1A UNDEFINED RAT UNDEFINED Ethyl 5-(3-(4-(3-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate 39 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
280 5-HT1A CELLS C0S-7 3H-8-OH-DPAT HISTAMINE 6011 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
536 5-HT1A HIPPOCAMPUS BOVINE 3H-8-OH-DPAT SPIPERONE 155.56 PEROUTKA, 1985 Jan 15, 2025 Jan 15, 2025
68376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT GBR-12909 4677 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78872 5-HT1A CLONED HUMAN 3H-WAY100635 4-Ethyl-2,5-dimethoxyphenethylamine 307.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14872 5-HT1A CLONED RAT UNDEFINED SERTINDOLE 2200 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
85784 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl)picolinamide 44.1 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
88600 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
89624 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 0.616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
27416 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Talipexole 1698.24 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95256 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 2500 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37656 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indazole-3-carboxamide 621 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
53784 5-HT1A UNDEFINED HUMAN UNDEFINED 4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 772.3 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
56600 5-HT1A UNDEFINED RAT UNDEFINED 8-OH-DPAT 0.8 Frecentese F et al., 2010 Jan 15, 2025 Jan 15, 2025
537 5-HT1A CORTEX HUMAN 3H-WB4101 SPIPERONE 320 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
68377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3353 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ondansetron HCl >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71961 5-HT1A test test [3H] Way100635 1-(1-(4-(Benzo[d]oxazol-2-yl)butyl)piperidin-4-yl)-5- chloro-1H-benzo[d]imidazol-2(3H)-one 611 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
78873 5-HT1A CLONED HUMAN 3H-WAY100635 4-Ethylthio-2,5-dimethoxyphenethylamine 381.2 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14873 5-HT1A CLONED RAT UNDEFINED CLOZAPINE 710 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
85785 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-OH-DPAT 0.8 Fiorino F et al 2017 Jan 15, 2025 Jan 15, 2025
87065 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 79.1 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89625 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90905 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 52.4807 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
27417 5-HT1A CLONED HUMAN 3H-8-OH-DPAT TERGURIDE 3.46737 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95257 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 196.3 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31257 5-HT1A C.H.O. HUMAN 3H-8-OH-DPAT Ropinirole 288.403 Millan MJ, et. al., 2004 Jan 15, 2025 Jan 15, 2025
32025 5-HT1A BRAIN RAT UNDEFINED RS-127445 3162.28 Bonhaus, DW et. al., 1999 Jan 15, 2025 Jan 15, 2025
99865 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride 138 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
37657 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide 5500 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
38937 5-HT1A CORTEX RAT 3H-8-OH-DPAT QUIPAZINE,8-Me 1700 Glennon RA, et al., 1989 Jan 15, 2025 Jan 15, 2025
53785 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(4-fluorophenyl)-4-(3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 414.4 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
538 5-HT1A HIPPOCAMPUS RAT 125I-BH-8-MeO-N-PA SPIPERONE 425.84 GOZLAN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
67866 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 66 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3354 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 5084 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
72474 5-HT1A test test [3H] Way100635 METHYSERGIDE 14 Ibrahim MA et al 2017 Jan 15, 2025 Jan 15, 2025
78874 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-4-Ethylthio-2,5-dimethoxyamphetamine 1674 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14874 5-HT1A CLONED RAT UNDEFINED OLANZAPINE 7100 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
17178 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METHYLPHENIDATE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27418 5-HT1A CLONED HUMAN 3H-8-OH-DPAT TL99 3801.89 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
95258 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 199.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101402 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 47 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
37658 5-HT1A Hippocampal RAT 3H-8-OH-DPAT N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-7-methoxy-2-benzofurancarboxamide 184 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
39194 5-HT1A CLONED HUMAN 125I-LSD ATC0065 62.9 Chaki S, et al., 2005 Jan 15, 2025 Jan 15, 2025
53786 5-HT1A UNDEFINED HUMAN UNDEFINED 1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 37.6 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
539 5-HT1A HIPPOCAMPUS RAT 125I-BH-8-MeO-N-PA SPIROXATRINE 1.51 GOZLAN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.25893 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3355 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IBOGAINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78875 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-2,5-Dimethoxy-4-ethoxyamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14875 5-HT1A CLONED RAT UNDEFINED RISPERIDONE 21 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
81947 5-HT1A CLONED HUMAN 3H-WAY100635 [18F]MH.MZ >10000 Herth MM et al 2009 Jan 15, 2025 Jan 15, 2025
83739 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 8590 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
95259 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 229.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
37659 5-HT1A Hippocampal RAT 3H-8-OH-DPAT 8-OH-DPAT 2.1 Leopoldo M, et al., 2002 Jan 15, 2025 Jan 15, 2025
39195 5-HT1A CLONED HUMAN 125I-LSD ATC0175 16.9 Chaki S, et al., 2005 Jan 15, 2025 Jan 15, 2025
53787 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 27.7 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54299 5-HT1A UNDEFINED RAT UNDEFINED 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 1000 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
540 5-HT1A CELLS C0S-7 3H-8-OH-DPAT SPIROXATRINE 1.8 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 6.60693 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3356 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ICS 205-930 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71196 5-HT1A CLONED HUMAN WAY100635 METHYSERGIDE 25 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
77596 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78876 5-HT1A CLONED HUMAN 3H-WAY100635 5-Methoxy-N-methyl-N-isopropyltryptamine 12.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14876 5-HT1A CLONED RAT UNDEFINED Quetiapine 830 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
80668 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
86812 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(furoyl)piperazin-1-yl)propyl)isonicotinamide 779 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87068 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 84.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89372 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 2630 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
93212 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 110 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
95260 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 365.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
96540 5-HT1A CLONED HUMAN [3H]-Way100635 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
101148 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone 272 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
53788 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one 90.9 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54300 5-HT1A UNDEFINED RAT UNDEFINED trans-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile 2863 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
541 5-HT1A CELLS C0S-7 125I-NAPS SPIROXATRINE 2.2 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3357 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IDAZOXAN 662 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71197 5-HT1A CLONED HUMAN WAY100635 SYA16263 1.1 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
74781 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
78877 5-HT1A CLONED HUMAN 3H-WAY100635 N,N-Diisopropyltryptamine 120.5 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14877 5-HT1A CLONED RAT UNDEFINED Ziprasidone 37 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
86813 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide 1000 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
88605 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
90909 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 26.9153 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
95261 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 210.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
99869 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride 7 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
101149 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone 350 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
54301 5-HT1A UNDEFINED RAT UNDEFINED cis-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile 5670 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
59677 5-HT1A CLONED HUMAN 3H-WAY100635 MH.MZ >10000 Herth, M. et. al., 2009 Jan 15, 2025 Jan 15, 2025
542 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT SPIROXATRINE 2.56 ALEXANDER & WOOD, 1988 Jan 15, 2025 Jan 15, 2025
68382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3358 5-HT1A CLONED HUMAN 3H-8-OH-DPAT IMIPRAMINE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71198 5-HT1A CLONED HUMAN WAY100635 SYA013 117.4 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
78878 5-HT1A CLONED HUMAN 3H-WAY100635 5-Methoxy-N,N-diisopropyltryptamine 132.4 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
13854 5-HT1A BRAIN RAT 3H-8-OH-DPAT PNU-96415E 134 Tang AH, et al., 1996 Jan 15, 2025 Jan 15, 2025
14878 5-HT1A CLONED RAT UNDEFINED AMPEROZIDE 3100 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
83486 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
89630 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0645654 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95262 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide 218 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
97054 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
99870 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride 22 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
54302 5-HT1A UNDEFINED RAT UNDEFINED 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 267 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
67871 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 91 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3359 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71199 5-HT1A CLONED HUMAN WAY100635 FEMPT 0.2 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71967 5-HT1A test test [3H] Way100635 1-(1-(4-(1H-Indol-3-yl)butyl)piperidin-4-yl)-5-chloro-1Hbenzo[d]imidazol-2(3H)-one >10000 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
78879 5-HT1A CLONED HUMAN 3H-WAY100635 N,N-Dipropyltryptamine 31.8 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14879 5-HT1A CLONED RAT UNDEFINED REMOXIPRIDE >10000 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
85535 5-HT1A test test [3H] Way100635 1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride 3.6 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
87071 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 81.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89375 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 1836 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89631 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0147911 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95263 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide 476 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
100127 5-HT1A CLONED HUMAN 3H-WAY100635 Brexpiprazole 1.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100639 5-HT1A CLONED HUMAN 3H-WAY100635 CYPROHEPTADINE 50 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
101407 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 28 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
54303 5-HT1A UNDEFINED RAT UNDEFINED 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile >10000 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
59423 5-HT1A CLONED HUMAN 3H-WAY100635 Desmethyldesipramine >10000 Deupree, J. et. al., 2007 Jan 15, 2025 Jan 15, 2025
68384 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3360 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDL 72222 >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
70432 5-HT1A CLONED HUMAN 3H-WAY100635 MRP3215 6 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
77344 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78880 5-HT1A CLONED HUMAN 3H-WAY100635 4-Ethylthio-2,5-dimethoxyphenylbutylamine 5339 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14880 5-HT1A CLONED RAT UNDEFINED HALOPERIDOL 2600 Arnt J and Skarsfeldt T Jan 15, 2025 Jan 15, 2025
80416 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (E)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
95264 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(3-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide 130 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31520 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(2-(1-(3,4-Dichloro-benzene sulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine 316.228 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
101152 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone >10000 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
54304 5-HT1A UNDEFINED RAT UNDEFINED 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 2530 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
545 5-HT1A CORTEX PIG 3H-8-OH-DPAT SPIROXATRINE 8.91 SCHOEFFTER AND HOYER,1988 Jan 15, 2025 Jan 15, 2025
66337 5-HT1A CLONED HUMAN 3H-WAY100635 N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
68385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 1.25893 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3361 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDA,R(-) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71457 5-HT1A CLONED HUMAN WAY100635 2-phenyl-N,N-diallyltryptamine 402 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
72737 5-HT1A CLONED HUMAN 3H-WAY100635 dihydrobilobetin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
75809 5-HT1A CLONED HUMAN 3H-WAY100635 Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
78881 5-HT1A CLONED HUMAN 3H-WAY100635 6-Fluoro-N,N-dimethyltryptamine 392.6 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
90913 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 37.1535 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
95265 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-[8-(4-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide 2000 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31521 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(2-(1-(3-bromo-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine 398.107 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
33057 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT BUPROPION >10000 Andersen PH, et al., 1989 Jan 15, 2025 Jan 15, 2025
101153 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone 33.5 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
38945 5-HT1A CORTEX RAT 3H-8-OH-DPAT QUIPAZINE 2000 Glennon RA, et al., 1989 Jan 15, 2025 Jan 15, 2025
58913 5-HT1A CLONED HUMAN 3H-WAY100635 (+)-SYA 09 722.3 Ablordeppey S, et al., 2006 Jan 15, 2025 Jan 15, 2025
66594 5-HT1A CLONED HUMAN 3H-WAY100635 N-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
68386 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 6.60693 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3362 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MDMA, R(-) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78882 5-HT1A CLONED HUMAN 3H-WAY100635 LISURIDE 0.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
82210 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one 20 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
86818 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide 0.13 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
87074 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile 473.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
25378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ARIPIPRAZOLE 5.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
25890 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Norephedrine, (+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
95266 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide 314.8 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
547 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIROXATRINE,(+) 21 NIKAM ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3363 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METHAMPHETAMINE (+) >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
78883 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-2,5-Dimethoxy-4-iodoamphetamine 2219 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
20259 5-HT1A CORTEX RAT 3H-8-OH-DPAT Benzamil 1900 Garritsen A et al., 1991 Jan 15, 2025 Jan 15, 2025
86819 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide 1060 Fiorino F et al 2016 Jan 15, 2025 Jan 15, 2025
89635 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0338844 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89891 5-HT1A CLONED HUMAN 3H-WAY100635 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
95267 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide 484.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
292 5-HT1A HIPPOCAMPUS BOVINE 3H-IPSAPIRONE HISTAMINE >10000 DOMPERT ET AL., 1985 Jan 15, 2025 Jan 15, 2025
67876 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 147 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68388 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piperazine 1.28825 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3364 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 5-HT,2-Me 3074 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
77092 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78884 5-HT1A CLONED HUMAN 3H-WAY100635 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane 147.1 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
82468 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-1-(Indolin-1-yl)-2-(2-((pyridin-3-yloxy)methyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
20260 5-HT1A CORTEX RAT 3H-8-OH-DPAT Amiloride >10000 Garritsen A et al., 1991 Jan 15, 2025 Jan 15, 2025
89636 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NLX-101 2.18776 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
93220 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 110 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
95268 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide 2300 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101156 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone 1684 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
101412 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 3569 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
293 5-HT1A CORTEX RAT 3H-8-OH-DPAT HISTAMINE >10000 PEROUTKA, 1986 Jan 15, 2025 Jan 15, 2025
549 5-HT1A CORTEX RAT 3H-8-OH-DPAT SPIROXATRINE,(-) 1.9 NIKAM ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68389 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 22.9087 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3365 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METHYLPHENIDATE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
71973 5-HT1A test test [3H] Way100635 2-(4-(4-(Bis(4-fluorophenyl)methyl)piperazin-1-yl)butyl) benzo[d]thiazole dihydrochloride >10000 Etukala JR et al 2016 Jan 15, 2025 Jan 15, 2025
12325 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 14489 0.61 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
78885 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-2,5-Dimethoxy-4-methylamphetamine 3656 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
86053 5-HT1A CLONED HUMAN 3H-WAY100635 Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
87077 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 54.6 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
90917 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane 69.1831 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
95269 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide 62.7 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
101157 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Phenyl-1-piperazinyl)-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone 81.8 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
101925 5-HT1A CLONED HUMAN [3H]8-OH-DPAT ZOTEPINE 131 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
550 5-HT1A CELLS C0S-7 3H-8-OH-DPAT SULPIRIDE 589 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
68390 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 0.831764 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3366 5-HT1A CLONED HUMAN 3H-8-OH-DPAT METOCLOPRAMIDE >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
12326 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 15535 1.77 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
78886 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-3,4,5-Trimethoxamphetamine 1678 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
85542 5-HT1A test test [3H] Way100635 1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride 7.3 Zhu XY et al 2012 Jan 15, 2025 Jan 15, 2025
87590 5-HT1A CLONED HUMAN 3H-WAY100635 3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
89382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 160 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
95270 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide 30.5 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
551 5-HT1A HIPPOCAMPUS RAT 125I-BH-8-MeO-N-PA SULPIRIDE,(-) >10000 GOZLAN ET AL., 1988 Jan 15, 2025 Jan 15, 2025
68391 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 4-hydroxy piperid-1-yl] 5-fluoroindan-1-01 1000 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3367 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MIANSERIN 2592 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11303 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 420 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12327 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT S 15931 1.51 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
78887 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-2,5-Dimethoxy-4-ethylamphetamine 14.4 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
88615 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 658 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
89639 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 8-OH-DPAT 0.812831 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95271 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 5-Hydroxy Tryptamine 9.4 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
40743 5-HT1A CLONED HUMAN 3H-8-OH-DPAT URB 597 >10000 Gobbi G, et al., 2005 Jan 15, 2025 Jan 15, 2025
296 5-HT1A CELLS C0S-7 3H-8-OH-DPAT ICS 205-930 1788 RAYMOND ET AL., 1989 Jan 15, 2025 Jan 15, 2025
552 5-HT1A CORTEX RAT 3H-5-MeO-DPAC SULPIRIDE,(-) >10000 COSSERY ET AL., 1987 Jan 15, 2025 Jan 15, 2025
68392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperid-1-yl] indan-1-01 0.707946 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3368 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NAN-190 3 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
11304 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 9-OH-risperidone 590 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
76840 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aR,8S,8aR)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
12328 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT Eltoprazine 9.33 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
78888 5-HT1A CLONED HUMAN 3H-WAY100635 (±)-2,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80680 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5E)-5-((4-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one 6927 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
85800 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT 2C-BI-1 542 Luethi D et al 2019 Jan 15, 2025 Jan 15, 2025
89640 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BUSPIRONE 5.01187 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
95272 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT DPAT 2.3 Stefanowicz J et al 2016a Jan 15, 2025 Jan 15, 2025
31016 5-HT1A CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
101160 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-(4-phenyl-1-piperazinyl)-1-propanone 1074 Intagliata S et al 2016 Jan 15, 2025 Jan 15, 2025
297 5-HT1A CORTEX PIG 3H-8-OH-DPAT ICS 205-930 >10000 MARKSTEIN ET AL, 1986 Jan 15, 2025 Jan 15, 2025
553 5-HT1A CORTEX RAT 3H-8-OH-DPAT SUMATRIPTAN 100 McCARTHY & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
67881 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 147 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68393 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piperidine 0.288403 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
3369 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NOMIFENSINE 1183 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
70441 5-HT1A CLONED HUMAN 3H-WAY100635 MRP3175 6.7 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
74537 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
11305 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 1500 Schotte A, et al., 1996 Jan 15, 2025 Jan 15, 2025
12329 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT MDL 73005 EF 1.25 Millan MJ, et al., 1993 Jan 15, 2025 Jan 15, 2025
78889 5-HT1A CLONED HUMAN 3H-WAY100635 LSD 7.3 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
82729 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
87081 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT 8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 53.9 Cao X et al 2018 Jan 15, 2025 Jan 15, 2025
89385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 152 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89641 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.51356 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
90921 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 24.5471 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025