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Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
76288KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
82944A1CORTICAL MEMBRANESRAT3H-CCPA1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione32.9Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
26880mGluR2CORTICAL MEMBRANESRAT3H-LY354740Ibotenate>10000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40448AMPACORTICAL MEMBRANESRAT3H-AMPA(5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
26881mGluR2CORTICAL MEMBRANESRAT3H-LY354740L-AP3>10000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40449AMPACORTICAL MEMBRANESRAT3H-AMPA(5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
72194BZPCORTICAL MEMBRANESRATFNZ2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl5789Magnus CJ et al 2019Jan 15, 2025Jan 29, 2025
76034BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
26882mGluR2CORTICAL MEMBRANESRAT3H-LY354740L-AP4>10000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40450KACORTICAL MEMBRANESRAT3H-Kainic acid(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
26883mGluR2CORTICAL MEMBRANESRAT3H-LY354740MCPG>10000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40451KACORTICAL MEMBRANESRAT3H-Kainic acid(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
81156KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 27, 2025
89348CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide1221Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
40452KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
82949A1CORTICAL MEMBRANESRAT3H-CCPA(R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
86277KORCORTICAL MEMBRANESRAT3H-MUSCIMOLJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
89349CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide310Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
40453KACORTICAL MEMBRANESRAT3H-Kainic acid(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
81926KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 27, 2025
84230BZPCORTICAL MEMBRANESRATFNZ(±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide293PDSP Certified DataJan 15, 2025Jan 29, 2025
86278BZPCORTICAL MEMBRANESRATFNZJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
40454KACORTICAL MEMBRANESRAT3H-Kainic acid(5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40455KACORTICAL MEMBRANESRAT3H-Kainic acid(5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
74760BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75016KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
40456KACORTICAL MEMBRANESRAT3H-Kainic acid(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
72713BZPCORTICAL MEMBRANESRATFNZnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 29, 2025
40457KACORTICAL MEMBRANESRAT3H-Kainic acid(5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
72202KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 27, 2025
82954A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione86.8Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
84234BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide299PDSP Certified DataJan 15, 2025Jan 29, 2025
40458KACORTICAL MEMBRANESRAT3H-Kainic acid(5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
76043KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75788BZPCORTICAL MEMBRANESRATFNZ1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
84237Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide1722PDSP Certified DataJan 15, 2025Jan 28, 2025
89358CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide471Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
41742AMPACORTICAL MEMBRANESRAT3H-AMPAAMPA23Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
72975BZPCORTICAL MEMBRANESRATFNZcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 29, 2025
89359CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide914Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
41743AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate94Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
82960A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione25.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
41744AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
72721KORCORTICAL MEMBRANESRAT3H-MUSCIMOLnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
74769KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
41745AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41746AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate1500Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
74515BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75539BZPCORTICAL MEMBRANESRATFNZpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
87571KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
41747AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate5800Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41748AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate700Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
75797KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76565BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
89877nAChRCORTICAL MEMBRANESRAT3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
41749AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
72982KORCORTICAL MEMBRANESRAT3H-MUSCIMOLcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
82966A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione33.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
41750AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41751AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate30Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
84248Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2567PDSP Certified DataJan 15, 2025Jan 28, 2025
89368CORTICAL MEMBRANESPIG3H-PRAZOSIN3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide263Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
41752KACORTICAL MEMBRANESRAT3H-Kainic acidAMPA>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
89369CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide156Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
41753KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate4900Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41754KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41755KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
74524KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75548KORCORTICAL MEMBRANESRAT3H-MUSCIMOLpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
82972A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione44.4Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
41756KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41757KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
75294BZPCORTICAL MEMBRANESRATFNZEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76574KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
81694BZPCORTICAL MEMBRANESRATFNZ(2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol>10000Dutta AK et al 2011Jan 15, 2025Jan 29, 2025
41758KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
84255Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one359PDSP Certified DataJan 15, 2025Jan 28, 2025
89887nAChRCORTICAL MEMBRANESRAT3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
91679A1CORTICAL MEMBRANESRAT3H-DPCPXN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide2.93Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
41759KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
76320BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
91680A1CORTICAL MEMBRANESRAT3H-DPCPXN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide0.0867Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
41760KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
91681A1CORTICAL MEMBRANESRAT3H-DPCPX4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide0.0709Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
41761KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
82978A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione14.1Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
89378CORTICAL MEMBRANESPIG3H-PRAZOSIN3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1369Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
91682A1CORTICAL MEMBRANESRAT3H-DPCPXN-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide0.0628Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
99874B1CORTICAL MEMBRANESRat brain3H-BRADYKININABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
41762NMDACORTICAL MEMBRANESRAT3H-CGP39653AMPA>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
86051KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
89379CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide5.9Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
99875ETACORTICAL MEMBRANESRat brain125I-ENDOTHELINABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
41763NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
12068H3CORTICAL MEMBRANESRAT3H-Alpha-Me-histamineGT 201643.8Tedford CE, et al., 1995Jan 15, 2025Jan 15, 2025
86052BZPCORTICAL MEMBRANESRATFNZ(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
87588BZPCORTICAL MEMBRANESRATFNZ2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
99876ETBCORTICAL MEMBRANESRat brain125I-ENDOTHELINABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
41764NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
12069H3CORTICAL MEMBRANESRAT3H-Alpha-Me-histamineThioperamide1.8Tedford CE, et al., 1995Jan 15, 2025Jan 15, 2025
87589BZPCORTICAL MEMBRANESRATFNZ3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
99877NK1CORTICAL MEMBRANESRat brain3H-Leu,4,5 Substance PABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
41765NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
99878CORTICAL MEMBRANESRat brain125I-NPYABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
41766NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
75303KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
81191BZPCORTICAL MEMBRANESRATFNZN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 29, 2025
99879CORTICAL MEMBRANESRat brain3H-NeurotensinABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39207AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-HIBO800Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
41767NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
75048BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
82984A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione351Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
99880CORTICAL MEMBRANESRat brain125I-VIPABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39208AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-(+)-Br-HIBO320Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
41768NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
76329KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
99881CORTICAL MEMBRANESRat brain125I-Omega-ConotoxinABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39209AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-(+)-Bu-HIBO480Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
41769NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
99882CORTICAL MEMBRANESRat brain3H-NitrendipineABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39210AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
41770NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
76075BZPCORTICAL MEMBRANESRATFNZEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
99883CORTICAL MEMBRANESRat brain3H-TBOBABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39211AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-(3-hydroxy-4-pentyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
41771NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
89388CORTICAL MEMBRANESPIG3H-PRAZOSINN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide53Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
99884CORTICAL MEMBRANESRat brain125I-ApaminABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39212AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
89389CORTICAL MEMBRANESPIG3H-PRAZOSIN4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide26Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
99885CORTICAL MEMBRANESRat brain3H-GlibenclamideABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39213AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-(+)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
81198KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 27, 2025
82990A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione238Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
99886CORTICAL MEMBRANESRat brain3H-CharybdotoxinABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39214AMPACORTICAL MEMBRANESRAT3H-AMPA(R)-(-)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
99887NETCORTICAL MEMBRANESRat brain3H-NisoxetineABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39215AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-(4-heptyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
99888SLC6A4CORTICAL MEMBRANESRat brain3H-CITALOPRAMABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39216AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
74801BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80177KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
99889CORTICAL MEMBRANESRat brain3H-GABAABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39217AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
72754BZPCORTICAL MEMBRANESRATFNZdihydrobilobetin5218Moawad A et al 2017Jan 15, 2025Jan 29, 2025
80178KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-3,4-Methylenedioxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
82994A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
99890CORTICAL MEMBRANESRat brain3H-Choline ChlorideABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39218AMPACORTICAL MEMBRANESRAT3H-AMPA(R)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
75059KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80179KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
99891SLC6A3CORTICAL MEMBRANESRat brain3H-WIN 35,428ABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
39219NMDACORTICAL MEMBRANESRAT3H-CPP(S)-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
76084KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80180KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
89908BZPCORTICAL MEMBRANESRATFNZ5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
99892AChECORTICAL MEMBRANESRat brainUNDEFINEDABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 28, 2025
39220NMDACORTICAL MEMBRANESRAT3H-CPP(S)-(+)-Br-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
75829BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80181KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
99893MOACORTICAL MEMBRANESRat brain14C-5-HTABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 29, 2025
39221NMDACORTICAL MEMBRANESRAT3H-CPP(S)-(+)-Bu-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
80182KORCORTICAL MEMBRANESRAT3H-MUSCIMOLDMT>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
89398CORTICAL MEMBRANESPIG3H-PRAZOSIN4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide53Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
99894MOACORTICAL MEMBRANESRat brain14C-PhenylethylamineABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 29, 2025
39222NMDACORTICAL MEMBRANESRAT3H-CPP(RS)-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
80183KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Hydroxy-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
82999A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione77.1Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
89399CORTICAL MEMBRANESPIG3H-PRAZOSINN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide30Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
39223NMDACORTICAL MEMBRANESRAT3H-CPP(RS)-2-Amino-3-(3-hydroxy-4-pentyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
80184KORCORTICAL MEMBRANESRAT3H-MUSCIMOLDMT,5-MeO>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
39224NMDACORTICAL MEMBRANESRAT3H-CPP(RS)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40248NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid210Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
80185KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Ethyl-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
87353BZPCORTICAL MEMBRANESRATFNZ4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide933Huang XP et al 2016Jan 15, 2025Jan 29, 2025
39225NMDACORTICAL MEMBRANESRAT3H-CPP(S)-(+)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40249AMPACORTICAL MEMBRANESRAT3H-AMPA(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
74810KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80186KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Ethylthio-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
39226NMDACORTICAL MEMBRANESRAT3H-CPP(R)-(-)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40250KACORTICAL MEMBRANESRAT3H-Kainic acid(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
80187KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-4-Ethylthio-2,5-dimethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
39227NMDACORTICAL MEMBRANESRAT3H-CPP(RS)-2-Amino-3-(4-heptyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40251NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid960Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
80188KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-2,5-Dimethoxy-4-ethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
83004A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione85.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
39228NMDACORTICAL MEMBRANESRAT3H-CPP(RS)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40252NMDACORTICAL MEMBRANESRAT3H-CGP39653(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
72765KORCORTICAL MEMBRANESRAT3H-MUSCIMOLdihydrobilobetin>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
80189KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN,N-Diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
39229NMDACORTICAL MEMBRANESRAT3H-CPP(S)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40253AMPACORTICAL MEMBRANESRAT3H-AMPA(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
74558BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75838KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76606BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80190KORCORTICAL MEMBRANESRAT3H-MUSCIMOL5-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
39230NMDACORTICAL MEMBRANESRAT3H-CPP(R)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 28, 2025
40254KACORTICAL MEMBRANESRAT3H-Kainic acid(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
75583BZPCORTICAL MEMBRANESRATFNZ3-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80191KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN,N-Dipropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90687Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine12Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39231KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40255NMDACORTICAL MEMBRANESRAT3H-CGP39653(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
80192KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Ethylthio-2,5-dimethoxyphenylbutylamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
83008A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
87616KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
89408CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide20Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
90688Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine5.7Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39232KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-(+)-Br-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40256AMPACORTICAL MEMBRANESRAT3H-AMPA(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
80193KORCORTICAL MEMBRANESRAT3H-MUSCIMOL6-Fluoro-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
89409CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-piperazinehexanamide4.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
90689Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine4.9Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39233KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-(+)-Bu-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40257NMDACORTICAL MEMBRANESRAT3H-CGP39653(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid370Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
80194KORCORTICAL MEMBRANESRAT3H-MUSCIMOLLISURIDE>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90690Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine2.3Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39234KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-HIBO>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40258NMDACORTICAL MEMBRANESRAT3H-D-APV(-)-2-aminoadipic acid>10000Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
80195KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-2,5-Dimethoxy-4-iodoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90691Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine183Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39235KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-(3-hydroxy-4-pentyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40259NMDACORTICAL MEMBRANESRAT3H-CPPCGS 1975595Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
80196KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90692Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine36Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39236KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40260AMPACORTICAL MEMBRANESRAT3H-AMPA(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
80197KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-2,5-Dimethoxy-4-methylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
83013A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione107Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90693Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine15Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39237KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-(+)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
40261KACORTICAL MEMBRANESRAT3H-Kainic acid(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
80198KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-3,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90694Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine8.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39238KACORTICAL MEMBRANESRAT3H-Kainic acid(R)-(-)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
74567KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75335BZPCORTICAL MEMBRANESRATFNZethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76615KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80199KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(±)-2,5-Dimethoxy-4-ethylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
89415CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide7.4Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
90695Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine19Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39239KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-(4-heptyl-3-hydroxy-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
75592KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80200KORCORTICAL MEMBRANESRAT3H-MUSCIMOLLYSERGIC ACID>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
89416CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide12.3Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
90696Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine5.8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39240KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
76361BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80201KORCORTICAL MEMBRANESRAT3H-MUSCIMOLcis-2a>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90697Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine3.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39241KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
80202KORCORTICAL MEMBRANESRAT3H-MUSCIMOLR,R-2b>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
83018A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90698Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine1.9Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
39242KACORTICAL MEMBRANESRAT3H-Kainic acid(R)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid>10000Madsen U, et al., 2001Jan 15, 2025Jan 15, 2025
80203KORCORTICAL MEMBRANESRAT3H-MUSCIMOLS,S-2c>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90699Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine19Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
80204KORCORTICAL MEMBRANESRAT3H-MUSCIMOLIBOGAINE>10000Ray TS 2010 Jan 15, 2025Jan 27, 2025
90700Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine20Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90701Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
72526BZPCORTICAL MEMBRANESRATFNZAmentoflavone22Moawad A et al 2017Jan 15, 2025Jan 29, 2025
90702Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine8.2Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
72527BZPCORTICAL MEMBRANESRATFNZtetrahydroamentoflavone196Moawad A et al 2017Jan 15, 2025Jan 29, 2025
83023A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione54.4Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90703Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine15Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
72528BZPCORTICAL MEMBRANESRATFNZA, 2, 3-dihydroamentoflavone295Moawad A et al 2017Jan 15, 2025Jan 29, 2025
75344KORCORTICAL MEMBRANESRAT3H-MUSCIMOLethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
86096KORCORTICAL MEMBRANESRAT3H-MUSCIMOLNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
90704Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine18Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
75089BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
86097BZPCORTICAL MEMBRANESRATFNZNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
89425CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide23Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
90705Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
76370KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
86098BZPCORTICAL MEMBRANESRATFNZ4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
89426CORTICAL MEMBRANESPIG3H-PRAZOSINN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide6.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
90706Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine3.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
86099KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
90707Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine262Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
76116BZPCORTICAL MEMBRANESRATFNZ2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
90708Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine50Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
83029A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione99.9Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90709Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine256Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90710Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine97Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90711Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)PENTAZOCINE (+)5.4Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90712Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)DTG71Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
74842BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75098KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
83035A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione95.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
89435CORTICAL MEMBRANESPIG3H-PRAZOSINN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide3.2Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89436CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide12.9Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
76125KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
89949BZPCORTICAL MEMBRANESRATFNZ3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
75870BZPCORTICAL MEMBRANESRATFNZEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
95838BZPCORTICAL MEMBRANESRATFNZ6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
83039A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
95839BZPCORTICAL MEMBRANESRATFNZTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95840BZPCORTICAL MEMBRANESRATFNZTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
72801BZPCORTICAL MEMBRANESRATFNZepigallocatechin>10000Moawad A et al 2017Jan 15, 2025Jan 29, 2025
95841BZPCORTICAL MEMBRANESRATFNZ6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95842BZPCORTICAL MEMBRANESRATFNZN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
74851KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
95843BZPCORTICAL MEMBRANESRATFNZtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
83044A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione28.9Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
95844BZPCORTICAL MEMBRANESRATFNZ4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
89445CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide17.8Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
95845BZPCORTICAL MEMBRANESRATFNZ2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
98917KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 27, 2025
100453Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine110Niso M et al 2013Jan 15, 2025Jan 28, 2025
87398KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 27, 2025
89446CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide46.4Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
100454Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine8.67Niso M et al 2013Jan 15, 2025Jan 28, 2025
72039BZPCORTICAL MEMBRANESRATFNZ1-methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g] quinoxalin-2(6H)-one HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 29, 2025
75879KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76647BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
89447D2CORTICAL MEMBRANESPIG3H-RACLOPRIDE(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide53Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
100455Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine373Niso M et al 2013Jan 15, 2025Jan 28, 2025
74600BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75624BZPCORTICAL MEMBRANESRATFNZ2-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
83816Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide5920PDSP Certified DataJan 15, 2025Jan 28, 2025
100456Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine35.9Niso M et al 2013Jan 15, 2025Jan 28, 2025
29289GABABCORTICAL MEMBRANESRAT3H-CGP-62349N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine20.893Urwyler S, et al., 2003Jan 15, 2025Jan 15, 2025
100457Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 7.43Niso M et al 2013Jan 15, 2025Jan 28, 2025
72810KORCORTICAL MEMBRANESRAT3H-MUSCIMOLepigallocatechin>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
83050A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione144Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
29290GABABCORTICAL MEMBRANESRAT3H-CGP-62349N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine32.3594Urwyler S, et al., 2003Jan 15, 2025Jan 15, 2025
100458Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine18.5Niso M et al 2013Jan 15, 2025Jan 28, 2025
87659KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
29291GABABCORTICAL MEMBRANESRAT3H-CGP-62349N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine2.75423Urwyler S, et al., 2003Jan 15, 2025Jan 15, 2025
100459Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine236Niso M et al 2013Jan 15, 2025Jan 28, 2025
100460Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 88.6Niso M et al 2013Jan 15, 2025Jan 28, 2025
72557KORCORTICAL MEMBRANESRAT3H-MUSCIMOLAmentoflavone>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
10862CORTICAL MEMBRANESRAT3H-KETANSERINKETANSERIN14.5Rinaldi-Carmona M., et al, 1992Jan 15, 2025Jan 15, 2025
72047KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1-methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g] quinoxalin-2(6H)-one HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 27, 2025
10863CORTICAL MEMBRANESRAT3H-KETANSERINRITANSERIN58.1Rinaldi-Carmona M., et al, 1992Jan 15, 2025Jan 15, 2025
89455CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide36.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
91247Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
75376BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
10864CORTICAL MEMBRANESRAT3H-KETANSERINSR 46349B5.8Rinaldi-Carmona M., et al, 1992Jan 15, 2025Jan 15, 2025
76656KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
83056A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione151Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
89456CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide36Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
74609KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75633KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76401BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
84081BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide1089PDSP Certified DataJan 15, 2025Jan 29, 2025
87409Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
84082BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide3617PDSP Certified DataJan 15, 2025Jan 29, 2025
83060A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
71797nAChR7CORTICAL MEMBRANESRAT3H-EpibatidineSAS-0132>10000Yi B et al 2017Jan 15, 2025Jan 29, 2025
100469Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-PentazocinePENTAZOCINE (+)4.1Niso M et al 2013Jan 15, 2025Jan 28, 2025
29815CB1CORTICAL MEMBRANESHUMAN3H-BAY 38-7271BAY 59-307448.3De Vry JM, et. al., 2004Jan 15, 2025Jan 15, 2025
83064A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
75385KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
84089Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3-chlorobenzamide2309PDSP Certified DataJan 15, 2025Jan 28, 2025
89465CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide22.1Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
75130BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76410KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
89466CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide11.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
29818CB1CORTICAL MEMBRANESHUMAN3H-BAY 38-7271CP 55,9400.51De Vry JM, et. al., 2004Jan 15, 2025Jan 15, 2025
84091BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3-chlorobenzamide3651PDSP Certified DataJan 15, 2025Jan 29, 2025
87676BZPCORTICAL MEMBRANESRATFNZ3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
76157BZPCORTICAL MEMBRANESRATFNZ2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
87677BZPCORTICAL MEMBRANESRATFNZ3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
29821CB1CORTICAL MEMBRANESHUMAN3H-BAY 38-7271THC, delta 913.7De Vry JM, et. al., 2004Jan 15, 2025Jan 15, 2025
83071A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
91263KORCORTICAL MEMBRANESRAT3H-MUSCIMOL17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 27, 2025
84097Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3,5-dichlorobenzamide3948PDSP Certified DataJan 15, 2025Jan 28, 2025
74883BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75139KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
89475CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide42.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
97667KORCORTICAL MEMBRANESRAT3H-flumazenil4-quinolone122Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
83076A1CORTICAL MEMBRANESRAT3H-CCPA8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione611Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
97668KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-ethyl-4-quinolone20Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97669KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-propoxycarbonyl-4-quinolone1.8Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
76166KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
97670KORCORTICAL MEMBRANESRAT3H-flumazenil3-Butoxycarbonyl-6-ethyl-4-quinolone13Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
75911BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
81031Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol1450Banister SD et al 2011Jan 15, 2025Jan 28, 2025
30599AMPACORTICAL MEMBRANESRAT3H-AMPAGlutamate500Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97671KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone28Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
81032Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol862Banister SD et al 2011Jan 15, 2025Jan 28, 2025
83080A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
30600AMPACORTICAL MEMBRANESRAT3H-AMPAKainate4000Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97672KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone28Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
81033Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(4-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol650Banister SD et al 2011Jan 15, 2025Jan 28, 2025
30601AMPACORTICAL MEMBRANESRAT3H-AMPAAMPA79Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97673KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-pentoxycarbonyl-4-quinolone35Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
71818KORCORTICAL MEMBRANESRAT3H-MethylspiperoneSAS-0132>10000Yi B et al 2017Jan 15, 2025Jan 27, 2025
81034Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(3-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol1950Banister SD et al 2011Jan 15, 2025Jan 28, 2025
84106BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-bromobenzamide7014PDSP Certified DataJan 15, 2025Jan 29, 2025
933225-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride39Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30602AMPACORTICAL MEMBRANESRAT3H-AMPAACPA20Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97674KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone92Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
81035Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(4-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol1240Banister SD et al 2011Jan 15, 2025Jan 28, 2025
933235-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride68Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30603KACORTICAL MEMBRANESRAT3H-Kainic acidGlutamate400Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97675KORCORTICAL MEMBRANESRAT3H-flumazenil3-Cyclopentoxycarbonyl-6-ethyl-4-quinolone19Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
74892KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
81036Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(3-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol234Banister SD et al 2011Jan 15, 2025Jan 28, 2025
83084A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
933245-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride20Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30604KACORTICAL MEMBRANESRAT3H-Kainic acidKainate16Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97676KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-i-propoxycarbonyl-4-quinolone214Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
72589BZPCORTICAL MEMBRANESRATFNZ2,3-dihydroamentoflavone295Moawad A et al 2017Jan 15, 2025Jan 29, 2025
81037Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(4-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol246Banister SD et al 2011Jan 15, 2025Jan 28, 2025
933255-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride4.3Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30605KACORTICAL MEMBRANESRAT3H-Kainic acidAMPA>10000Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97677KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(4-methyl-2-pentoxycarbonyl)-4-quinolone295Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
72846BZPCORTICAL MEMBRANESRATFNZisoginkgetin>10000Moawad A et al 2017Jan 15, 2025Jan 29, 2025
81038Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-Benzyl-2-azatricyclo[3.3.1.13,7]decane29Banister SD et al 2011Jan 15, 2025Jan 28, 2025
82830A1CORTICAL MEMBRANESRAT3H-CCPAIstradefylline230Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
933265-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride4.5Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30606KACORTICAL MEMBRANESRAT3H-Kainic acidACPA6300Madsen U et. al., 1992Jan 15, 2025Jan 15, 2025
97678KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-pentoxycarbonyl)-4-quinolone2600Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
81039Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane22Banister SD et al 2011Jan 15, 2025Jan 28, 2025
84111Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-(trifluoromethyl)benzamide1316PDSP Certified DataJan 15, 2025Jan 28, 2025
933275-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride4.5Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30607NMDACORTICAL MEMBRANESRAT3H-GLUTAMATEGlutamate200Madsen U et. al., 1992Jan 15, 2025Jan 28, 2025
97679KORCORTICAL MEMBRANESRAT3H-flumazenil3-Carboxy-6-ethyl-4-quinolone208Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
75920KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
81040Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(4-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane12Banister SD et al 2011Jan 15, 2025Jan 28, 2025
933285-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride25Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30608NMDACORTICAL MEMBRANESRAT3H-GLUTAMATEKainate>10000Madsen U et. al., 1992Jan 15, 2025Jan 28, 2025
97680KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-4-quinolone78Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
75665BZPCORTICAL MEMBRANESRATFNZbenzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76689BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
81041Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(3-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decane239Banister SD et al 2011Jan 15, 2025Jan 28, 2025
83089A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione23Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
91281BZPCORTICAL MEMBRANESRATFNZ17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
933295-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride66Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30609NMDACORTICAL MEMBRANESRAT3H-GLUTAMATEAMPA>10000Madsen U et. al., 1992Jan 15, 2025Jan 28, 2025
97681KORCORTICAL MEMBRANESRAT3H-flumazenil3-Butoxycarbonyl-4-quinolone54Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
71826NMDACORTICAL MEMBRANESRAT3H-MK-801SAS-0132>10000Yi B et al 2017Jan 15, 2025Jan 28, 2025
74642BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
81042Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(4-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decane12.4Banister SD et al 2011Jan 15, 2025Jan 28, 2025
933305-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride18Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
30610NMDACORTICAL MEMBRANESRAT3H-GLUTAMATEACPA>10000Madsen U et. al., 1992Jan 15, 2025Jan 28, 2025
97682KORCORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-4-quinolone16Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
80019NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
81043Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(3-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decane8.3Banister SD et al 2011Jan 15, 2025Jan 28, 2025
933315-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride204Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97683KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-propyl-4-quinolone17Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
80020NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
81044Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)N-(4-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decane12.8Banister SD et al 2011Jan 15, 2025Jan 28, 2025
82836A1CORTICAL MEMBRANESRAT3H-CCPACSC>10000Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
933325-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride146Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97684KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-i-propyl-4-quinolone15Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
72597KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2,3-dihydroamentoflavone>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
80021NMDACORTICAL MEMBRANESRAT3H-MK-8013,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
933335-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride488Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97685KORCORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-ethoxycarbonyl-4-quinolone1.4Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49045nAChRCORTICAL MEMBRANESRAT3H-NICOTINE(R)-SIB-1508Y75Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
72854KORCORTICAL MEMBRANESRAT3H-MUSCIMOLisoginkgetin>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
80022NMDACORTICAL MEMBRANESRAT3H-MK-8014-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
83094A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Fluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
933345-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride354Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97686KORCORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-propoxycarbonyl-4-quinolone0.17Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49046CORTICAL MEMBRANESRAT3H-QNB(R)-SIB-1508Y4500Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
71063KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 27, 2025
80023NMDACORTICAL MEMBRANESRAT3H-MK-8014-Ethyl-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80279BZPCORTICAL MEMBRANESRATFNZ(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
933355-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride56Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97687KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone6850Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49047nAChRCORTICAL MEMBRANESRAT3H-NICOTINENicotine4Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
74392BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75416BZPCORTICAL MEMBRANESRATFNZEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,2-dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d]- [1,3]dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80024NMDACORTICAL MEMBRANESRAT3H-MK-8014-Ethylthio-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80280BZPCORTICAL MEMBRANESRATFNZ(±)-3,4-Methylenedioxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
87704KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
91544A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide2.79Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
933365-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride104Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97688KORCORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-2-methyl-4-quinolone4200Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49048nAChRCORTICAL MEMBRANESRAT3H-NICOTINE5-Bromo-3-(1-methyl-2-pyrrolidinyl)pyridine19Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
80025NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-2,5-Dimethoxy-4-ethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80281BZPCORTICAL MEMBRANESRATFNZ(±)-3,4-Methylenedioxymethamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
91545A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide3.47Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
933375-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride70Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97689KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-propylaminocarbonyl-4-quinolone0.26Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49049nAChRCORTICAL MEMBRANESRAT3H-NICOTINESIB-1508Y4.6Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
75674KORCORTICAL MEMBRANESRAT3H-MUSCIMOLbenzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76442BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76698KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80026NMDACORTICAL MEMBRANESRAT3H-MK-8015-Methoxy-N-methyl-N-isopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80282BZPCORTICAL MEMBRANESRATFNZ3,4,5-Trimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
82842A1CORTICAL MEMBRANESRAT3H-CCPA8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione79.3Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
83098A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
933385-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride15Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97690KORCORTICAL MEMBRANESRAT3H-flumazenil3-Butylaminocarbonyl-6-ethyl-4-quinolone0.54Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49050nAChRCORTICAL MEMBRANESRAT3H-NICOTINE5-ethyl-3-(1-methyl-2-pyrrolidinyl)pyridine11Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
72091BZPCORTICAL MEMBRANESRATFNZ2-methoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 29, 2025
80027NMDACORTICAL MEMBRANESRAT3H-MK-801N,N-Diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80283BZPCORTICAL MEMBRANESRATFNZ4-Bromo-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
933395-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride20Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97691KORCORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-propylaminocarbonyl-4-quinolone0.048Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49051nAChRCORTICAL MEMBRANESRAT3H-NICOTINE(S)-SIB-1508Y3Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
80028NMDACORTICAL MEMBRANESRAT3H-MK-8015-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80284BZPCORTICAL MEMBRANESRATFNZDMT>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
91548A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide0.939Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
933405-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride133Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97692KORCORTICAL MEMBRANESRAT3H-flumazenilPropyl 2-methyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate870Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49052CORTICAL MEMBRANESRAT3H-QNBNicotine>10000Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
80029NMDACORTICAL MEMBRANESRAT3H-MK-801N,N-Dipropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80285BZPCORTICAL MEMBRANESRATFNZ4-Ethyl-2,5-dimethoxyphenethylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
91549A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
933415-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride899Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97693KORCORTICAL MEMBRANESRAT3H-flumazenilEthyl 7-Oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate>10000Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49053CORTICAL MEMBRANESRAT3H-QNB5-Bromo-3-(1-methyl-2-pyrrolidinyl)pyridine>10000Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
74398KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80030NMDACORTICAL MEMBRANESRAT3H-MK-8014-Ethylthio-2,5-dimethoxyphenylbutylamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80286BZPCORTICAL MEMBRANESRATFNZ4-Hydroxy-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
933425-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride230Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97694KORCORTICAL MEMBRANESRAT3H-flumazenilPropyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate7130Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49054CORTICAL MEMBRANESRAT3H-QNBSIB-1508Y>10000Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
80031NMDACORTICAL MEMBRANESRAT3H-MK-8016-Fluoro-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80287BZPCORTICAL MEMBRANESRATFNZDMT,5-MeO>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
83103A1CORTICAL MEMBRANESRAT3H-CCPA8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione36Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
933435-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride7.6Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97695GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone4.1Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
49055CORTICAL MEMBRANESRAT3H-QNB5-ethyl-3-(1-methyl-2-pyrrolidinyl)pyridine5800Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
80032NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-2,5-Dimethoxy-4-iodoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
80288BZPCORTICAL MEMBRANESRATFNZ(±)-4-Ethylthio-2,5-dimethoxyamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
82848A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione40.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
91552A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93088Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
933445-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride64Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97696GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone89Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
49056CORTICAL MEMBRANESRAT3H-QNB(S)-SIB-1508Y8900Cosford, N. D et al., 1996Jan 15, 2025Jan 15, 2025
75425KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,2-dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d]- [1,3]dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80033NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-2,5-Dimethoxy-4-methylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
83873Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(4aS,8R,8aS)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide6924PDSP Certified DataJan 15, 2025Jan 28, 2025
856655-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPATN-(2-(4-phenylpiperazin-1-yl)ethyl)picolinamide161Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
91553A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93089Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
933455-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride48Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
97697GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-4-quinolone26Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
80034NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-3,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
93090Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
933465-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride477Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
316505-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H28N2 dimaleate (37)21Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97698GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-4-quinolone14Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
71843nAChRCORTICAL MEMBRANESRAT3H-EpibatidineSAS-0132>10000Yi B et al 2017Jan 15, 2025Jan 29, 2025
72099KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-methoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 27, 2025
75171BZPCORTICAL MEMBRANESRATFNZmethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76451KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
80035NMDACORTICAL MEMBRANESRAT3H-MK-801(±)-2,5-Dimethoxy-4-ethylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
93091Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
933475-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride151Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
316515-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27ClN2 1.5maleate (38)3.2Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97699GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-ethoxycarbonyl-4-quinolone0.27Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
80036NMDACORTICAL MEMBRANESRAT3H-MK-801LYSERGIC ACID>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
83108A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
91556A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93092Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
933485-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride631Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
316525-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27ClN2 fumarate (38, -)4.4Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97700GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-ethoxycarbonyl-4-quinolone7.2Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
80037NMDACORTICAL MEMBRANESRAT3H-MK-801cis-2a>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
82853A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione42Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
91301KORCORTICAL MEMBRANESRAT3H-MUSCIMOL17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 27, 2025
91557A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide1.47Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93093Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
933495-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride34Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
316535-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27ClN2 fumarate (38, +)68Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97701GABAACORTICAL MEMBRANESRAT3H-flumazenilDIAZEPAM12Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
76198BZPCORTICAL MEMBRANESRATFNZ(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
80038NMDACORTICAL MEMBRANESRAT3H-MK-801R,R-2b>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
93094Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
316545-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27FN2 dimaleate (39)5.1Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97702GABAACORTICAL MEMBRANESRAT3H-flumazenilDIAZEPAM14Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
80039NMDACORTICAL MEMBRANESRAT3H-MK-801S,S-2c>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
93095Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
316555-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27FN2 fumarate (39, -)2.9Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97703GABAACORTICAL MEMBRANESRAT3H-flumazenilZolpidem1850Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
80040NMDACORTICAL MEMBRANESRAT3H-MK-801DMT,5-MeO>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
91560A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1.01Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93096Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
316565-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27FN2 fumarate (39, +)650Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
97704GABAACORTICAL MEMBRANESRAT3H-flumazenilZolpidem53Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
80041NMDACORTICAL MEMBRANESRAT3H-MK-801EMDT>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
91561A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide1.77Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93097Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine1400Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
316575-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26F2N2 dimaleate (40)3.6Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
80042NMDACORTICAL MEMBRANESRAT3H-MK-801IBOGAINE2001Ray TS 2010 Jan 15, 2025Jan 28, 2025
82858A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione54.2Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
83114A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione46Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
93098Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
316585-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26F2N2 fumarate (40, -)1.9Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
86187GABAACORTICAL MEMBRANESRAT3H-MUSCIMOL2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
316595-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26F2N2 fumarate (40, +)360Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
74924BZPCORTICAL MEMBRANESRATFNZ1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75180KORCORTICAL MEMBRANESRAT3H-MUSCIMOLmethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
81068BZPCORTICAL MEMBRANESRATFNZN-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 29, 2025
84140BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-2-methylbenzamide5311PDSP Certified DataJan 15, 2025Jan 29, 2025
316605-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC21H24ClFN2 hemifumarate (41)3.2Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
316615-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC21H24ClFN2 fumarate (41, -)3.7Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
83118A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,5-bis(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
91566A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
316625-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC21H24ClFN2 fumarate (41, +)3600Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
76207KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
82863A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione15.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
84143Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide4005PDSP Certified DataJan 15, 2025Jan 28, 2025
91567A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
316635-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26BrFN2 1.5fumarate (42)3Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
75952BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
316645-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H24F4N2 (43)7.5Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
84145BZPCORTICAL MEMBRANESRATFNZ±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide3438PDSP Certified DataJan 15, 2025Jan 29, 2025
316655-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC23H26F4N2 (44)4.5Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
81074KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 27, 2025
90546A1CORTICAL MEMBRANESRAT3H-CCPAPreladenant (SCH420814)68.7 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91570A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
316665-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H27FN2 (45)1.5Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
83123A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione134Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90547A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide422 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91571A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
316675-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC23H29FN2 (46)3.4Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
82868A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione61.9Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90548A1CORTICAL MEMBRANESRAT3H-CCPA3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide367 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
316685-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26ClFN2 dioxalate (47)29Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
74933KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
90549A1CORTICAL MEMBRANESRAT3H-CCPA3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
316695-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26ClFN2 (48)9.3Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
90550A1CORTICAL MEMBRANESRAT3H-CCPA3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91574A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide0.348Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
316705-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26ClFN2 1.3oxalate (49)31Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
84151Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-bromo-3-(trifluoromethyl)benzamide845PDSP Certified DataJan 15, 2025Jan 28, 2025
90551A1CORTICAL MEMBRANESRAT3H-CCPA3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91319BZPCORTICAL MEMBRANESRATFNZ17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91575A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide6.69Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93111NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316715-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26F2N2 oxalate (50)9.8Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
83128A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,4-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90552A1CORTICAL MEMBRANESRAT3H-CCPA2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93112NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316725-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26ClFN2 dimaleate (51)21Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
75961KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
82873A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90553A1CORTICAL MEMBRANESRAT3H-CCPA(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide205 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93113NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316735-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26ClFN2 dimaleate (52)26Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
72890BZPCORTICAL MEMBRANESRATFNZ2″-glucosylvitexin>10000Moawad A et al 2017Jan 15, 2025Jan 29, 2025
75706BZPCORTICAL MEMBRANESRATFNZ2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
90554A1CORTICAL MEMBRANESRAT3H-CCPA(E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91578A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93114NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine893Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316745-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC22H26Cl2N2 dioxalate 0.5H2O (53)32Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
76731BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
87483KORCORTICAL MEMBRANESRAT3H-MUSCIMOLFK881>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
90555A1CORTICAL MEMBRANESRAT3H-CCPA3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91579A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93115NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine413Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316755-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC19H23ClN2S dimaleate (54)1Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
74684BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
83132A1CORTICAL MEMBRANESRAT3H-CCPA8-(Benzo[d][1,3]dioxol-5-ylmethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90556A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide229 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93116NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine712Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316765-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC19H23ClN2S hemifumarate (54, -)1.9Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
11965H2CORTICAL MEMBRANESGUINEA PIG3H-HistamineHISTAMINE100Hill JA., 1992Jan 15, 2025Jan 15, 2025
90557A1CORTICAL MEMBRANESRAT3H-CCPA4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide22.5 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93117NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316775-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC19H23ClN2S hemifumarate (54, +)1100Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
11966H2CORTICAL MEMBRANESGUINEA PIG3H-HistamineAlpha-Methylhistane-R1Hill JA., 1992Jan 15, 2025Jan 15, 2025
82878A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione40.1Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
84158Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(4aS,8R,8aS)-8-amino-2-benzyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one521PDSP Certified DataJan 15, 2025Jan 28, 2025
90558A1CORTICAL MEMBRANESRAT3H-CCPA4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide898 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91582A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93118NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316785-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINC20H25ClN2S 2HCl 0.7H2O (55)1.7Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
11967H2CORTICAL MEMBRANESGUINEA PIG3H-HistamineBeta-Methylhistamine0.9Hill JA., 1992Jan 15, 2025Jan 15, 2025
90559A1CORTICAL MEMBRANESRAT3H-CCPA4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
91583A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
93119NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316795-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINCLOZAPINE7.8Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
74432BZPCORTICAL MEMBRANESRAT3H-CGP-12177(1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
11968H2CORTICAL MEMBRANESGUINEA PIG3H-HistamineAlpha-Dimethylhistane-alpha0.2Hill JA., 1992Jan 15, 2025Jan 15, 2025
83136A1CORTICAL MEMBRANESRAT3H-CCPA(R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1530Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90560A1CORTICAL MEMBRANESRAT3H-CCPA(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide53 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93120NMDACORTICAL MEMBRANESPIG3H-MK-801((±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
316805-HT2ACORTICAL MEMBRANESRAT3H-KETANSERINSCH 2339014Bogeso, K.P., et al., 1995Jan 15, 2025Jan 15, 2025
75457BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-4-(2-((5-bromothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
11969H2CORTICAL MEMBRANESGUINEA PIG3H-HistamineS-Beta-Dimethylhistamine-R-alpha0.2Hill JA., 1992Jan 15, 2025Jan 15, 2025
90561A1CORTICAL MEMBRANESRAT3H-CCPA(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide11.2 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93121NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
72898KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2″-glucosylvitexin>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
90562A1CORTICAL MEMBRANESRAT3H-CCPA(E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide11.4 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93122NMDACORTICAL MEMBRANESPIG3H-MK-801(S)-(+)-ketamine419Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
75715KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76483BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
90563A1CORTICAL MEMBRANESRAT3H-CCPA(E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide1500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93123NMDACORTICAL MEMBRANESPIG3H-MK-801PCP28Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
76740KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
82884A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione52.8Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
84164BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide84PDSP Certified DataJan 15, 2025Jan 29, 2025
90564A1CORTICAL MEMBRANESRAT3H-CCPAN-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide98.3 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93124NMDACORTICAL MEMBRANESPIG3H-MK-801Dexoxadrol19Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
74693KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
83141A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,4,5-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
84165BZPCORTICAL MEMBRANESRATFNZ(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide322PDSP Certified DataJan 15, 2025Jan 29, 2025
90565A1CORTICAL MEMBRANESRAT3H-CCPAN-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93125NMDACORTICAL MEMBRANESPIG3H-MK-801Etoxadrol22Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40133NMDACORTICAL MEMBRANESRAT3H-CPP(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
90566A1CORTICAL MEMBRANESRAT3H-CCPAN-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93126NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40134AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
90567A1CORTICAL MEMBRANESRAT3H-CCPAN-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93127NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40135KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
700885-HT3CORTICAL MEMBRANESRAT3H-GR-65630d^/-10-[(2-Methyl-lH-imidazol-l-yl)methyl]-5,6,8,9,10,llhexahydro-4i7-pyrido[3,2,l-/A]carbazol-ll-one0.25Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
90568A1CORTICAL MEMBRANESRAT3H-CCPAN-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide64.4 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93128NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40136NMDACORTICAL MEMBRANESRAT3H-CPP(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid490Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
700895-HT3CORTICAL MEMBRANESRAT3H-GR-656301.4Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
74441KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
82889A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
83145A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,4,6-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90569A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93129NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40137AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
700905-HT3CORTICAL MEMBRANESRAT3H-GR-656300-[(2-Methyl-lH-imidazol-l-yl)methyl]-5,6,8,9,10,llhexahydro-4H-pyrido[3^,l-ji]carbazol-1l-oneHydrochloride0.19Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
75466KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-4-(2-((5-bromothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
90570A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide35.2 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93130NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40138KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
700915-HT3CORTICAL MEMBRANESRAT3H-GR-65630l-(2,3-Dihydropyrrolo[l,2,3-de][l,4]benzothiazin-6-yl)-3-(5-methylimidazol-4-yl)propan-l-one Hydrochloride0.19Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
90571A1CORTICAL MEMBRANESRAT3H-CCPAN-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
93131NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40139NMDACORTICAL MEMBRANESRAT3H-CPP(+/-)-AP5290Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
700925-HT3CORTICAL MEMBRANESRAT3H-GR-65630ONDANSETRON1.6Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
75212BZPCORTICAL MEMBRANESRATFNZethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76492KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
84172BZPCORTICAL MEMBRANESRATFNZ(±)-3-chloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide661PDSP Certified DataJan 15, 2025Jan 29, 2025
93132NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40140NMDACORTICAL MEMBRANESRAT3H-CPP(R)-AP5880Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
700935-HT3CORTICAL MEMBRANESRAT3H-GR-65630GR 656300.28Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
84173Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-3-chloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide736PDSP Certified DataJan 15, 2025Jan 28, 2025
85965GABAACORTICAL MEMBRANESRAT3H-MUSCIMOL1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
93133NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40141NMDACORTICAL MEMBRANESRAT3H-CPP(S)-AP5>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
70094CORTICAL MEMBRANESRAT3H-PRAZOSINcilanseton5600Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
72142BZPCORTICAL MEMBRANESRATFNZ2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl5840Magnus CJ et al 2019Jan 15, 2025Jan 29, 2025
83150A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione73Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
93134NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
40142NMDACORTICAL MEMBRANESRAT3H-CPP(R)-CPPene40Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
70095CORTICAL MEMBRANESRAT3H-PRAZOSINONDANSETRON3400Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
76239BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
82895A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione25.5Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90831NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93135NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
70096CORTICAL MEMBRANESRAT3H-CLONIDINEONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
90832NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93136NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
70097CORTICAL MEMBRANESRAT3H-CLONIDINEcilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
90833NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93137NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
90834NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93138NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
94930BZPCORTICAL MEMBRANESRATFNZ4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
90835NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-Benzyl-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93139NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
94931BZPCORTICAL MEMBRANESRATFNZ4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
70100Beta 1CORTICAL MEMBRANESRAT3H-DHAONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
81108BZPCORTICAL MEMBRANESRATFNZN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 29, 2025
82900A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
83156A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione111Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
90836NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-Benzyl-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93140Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine155Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94932BZPCORTICAL MEMBRANESRATFNZ4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
66261GABAACORTICAL MEMBRANESBOVINE3H-flumazenilbenzylamine531Primofiore G, et al., 2006Jan 15, 2025Jan 15, 2025
70101Beta 1CORTICAL MEMBRANESRAT3H-DHAcilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
75221KORCORTICAL MEMBRANESRAT3H-MUSCIMOLethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
90837NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-Benzyl-3-methoxy-N-methyl-3,4-dihydrospiro-[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93141Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine542Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94933BZPCORTICAL MEMBRANESRATFNZ5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
66262GABAACORTICAL MEMBRANESBOVINE3H-flumazenilDIAZEPAM10Primofiore G, et al., 2006Jan 15, 2025Jan 15, 2025
70102D1CORTICAL MEMBRANESRAT3H-dopaminecilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
72150KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 27, 2025
74966BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
90838NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-Benzyl-3-methoxy-N-methyl-3,4-dihydrospiro-[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
93142Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine543Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94934BZPCORTICAL MEMBRANESRATFNZ4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
66263GABAACORTICAL MEMBRANESBOVINE3H-flumazenilflumazenil0.9Primofiore G, et al., 2006Jan 15, 2025Jan 15, 2025
70103D1CORTICAL MEMBRANESRAT3H-dopamineONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
86231KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
93143Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine607Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94935BZPCORTICAL MEMBRANESRATFNZ4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
70104D2CORTICAL MEMBRANESRAT3H-SPIPERONEONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
76248KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
86232BZPCORTICAL MEMBRANESRATFNZ4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
93144Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine1500Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94936BZPCORTICAL MEMBRANESRATFNZ4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
70105D2CORTICAL MEMBRANESRAT3H-SPIPERONEcilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
75993BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
82905A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione26Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
83161A1CORTICAL MEMBRANESRAT3H-CCPA8-(4,5-Difluoro-2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
93145Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine2700Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94937BZPCORTICAL MEMBRANESRATFNZ4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
70106D3CORTICAL MEMBRANESRAT3H-SPIPERONEcilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
81114KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol>10000Banister SD et al 2011Jan 15, 2025Jan 27, 2025
84186BZPCORTICAL MEMBRANESRATFNZ(±)-4-bromo-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide263PDSP Certified DataJan 15, 2025Jan 29, 2025
93146Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine4900Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94938BZPCORTICAL MEMBRANESRATFNZ4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
70107D3CORTICAL MEMBRANESRAT3H-SPIPERONEONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
70619KORCORTICAL MEMBRANESRAT3H-WIN 35,428MRP3172>10000Porter, MR et. al, 2019Jan 15, 2025Jan 27, 2025
93147Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine502Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94939BZPCORTICAL MEMBRANESRATFNZ4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
701085-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPATONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
11996H1CORTICAL MEMBRANESHUMAN3H-doxepinPYRILAMINE4Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
93148Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine192Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94940BZPCORTICAL MEMBRANESRATFNZ2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
701095-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPATcilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
11997H1CORTICAL MEMBRANESHUMAN3H-doxepind-Chlorpheniramine30Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
83165A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,3-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
93149Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine37Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
94941BZPCORTICAL MEMBRANESRATFNZ2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
701105-HT1BCORTICAL MEMBRANESRAT3H-Serotonincilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
11998H1CORTICAL MEMBRANESHUMAN3H-doxepinl-Chlorpheniramine1200Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
93150Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine7.37Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
701115-HT1BCORTICAL MEMBRANESRAT3H-SerotoninONDANSETRON3700Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
74975KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
11999H1CORTICAL MEMBRANESHUMAN3H-doxepinDiphenhydramine62Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
82911A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione74.4Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
93151Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine297Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
701125-HT2CCORTICAL MEMBRANESRAT3H-SerotoninONDANSETRON5000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
72672BZPCORTICAL MEMBRANESRATFNZ2,3-dihydrohinokiflavone1389Moawad A et al 2017Jan 15, 2025Jan 29, 2025
12000H1CORTICAL MEMBRANESHUMAN3H-doxepinMequitazine5.8Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
93152Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine314Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
701135-HT2CCORTICAL MEMBRANESRAT3H-Serotonincilansetron4900Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
12001H1CORTICAL MEMBRANESHUMAN3H-doxepinDOXEPIN0.49Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
83169A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,5-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
85985BZPCORTICAL MEMBRANESRATFNZ1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
93153Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine3000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
701145-HT1DCORTICAL MEMBRANESRAT3H-Serotonincilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
76002KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
12002H1CORTICAL MEMBRANESHUMAN3H-doxepinAMITRIPTYLINE0.67Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
84194Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2220PDSP Certified DataJan 15, 2025Jan 28, 2025
85986BZPCORTICAL MEMBRANESRATFNZDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
93154Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)PENTAZOCINE (+)6.03Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
701155-HT1DCORTICAL MEMBRANESRAT3H-SerotoninONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
72931BZPCORTICAL MEMBRANESRATFNZvicenin-2>10000Moawad A et al 2017Jan 15, 2025Jan 29, 2025
75747BZPCORTICAL MEMBRANESRATFNZ3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
12003H1CORTICAL MEMBRANESHUMAN3H-doxepinNORTRYPTYLINE8.4Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
70116CORTICAL MEMBRANESRAT3H-SPIPERONEONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
12004H1CORTICAL MEMBRANESHUMAN3H-doxepinIMIPRAMINE16Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
70117CORTICAL MEMBRANESRAT3H-SPIPERONEcilansetron7800Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
74725BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
12005H1CORTICAL MEMBRANESHUMAN3H-doxepinTrimipramine1.4Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
14565NMDACORTICAL MEMBRANESRAT3H-5,7-DCKADCUKA>10000Snell LD, et al., 2000Jan 15, 2025Jan 15, 2025
82917A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione51.1Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
701185-HT3CORTICAL MEMBRANESRAT3H-GR-65630cilansetron0.19Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
12006H1CORTICAL MEMBRANESHUMAN3H-doxepinMAPROTILINE0.79Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
14566NMDACORTICAL MEMBRANESRAT3H-5,7-DCKA5,7-DCKA90Snell LD, et al., 2000Jan 15, 2025Jan 15, 2025
83174A1CORTICAL MEMBRANESRAT3H-CCPA8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione170Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
701195-HT4CORTICAL MEMBRANESRAT3H-GR113808cilansetron960Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
12007H1CORTICAL MEMBRANESHUMAN3H-doxepinMIANSERIN0.36Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
14567NMDACORTICAL MEMBRANESRAT3H-BatrachotoxinDCUKA>10000Snell LD, et al., 2000Jan 15, 2025Jan 15, 2025
701205-HT4CORTICAL MEMBRANESRAT3H-GR113808ONDANSETRON1200Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
72680KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2,3-dihydrohinokiflavone>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
12008H1CORTICAL MEMBRANESHUMAN3H-doxepinDESIPRAMINE120Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
14568NMDACORTICAL MEMBRANESRAT3H-BatrachotoxinDCUK-Ome>10000Snell LD, et al., 2000Jan 15, 2025Jan 15, 2025
87528KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
70121CORTICAL MEMBRANESRAT3H-PAROXETINEONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
74473BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
12009H1CORTICAL MEMBRANESHUMAN3H-doxepinIPRINDOLE120Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
14569NMDACORTICAL MEMBRANESRAT3H-BatrachotoxinCARBAMAZEPINE>10000Snell LD, et al., 2000Jan 15, 2025Jan 15, 2025
82921A1CORTICAL MEMBRANESRAT3H-CCPA8-(4-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
84201BZPCORTICAL MEMBRANESRATFNZ(±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide5163PDSP Certified DataJan 15, 2025Jan 29, 2025
70122CORTICAL MEMBRANESRAT3H-PAROXETINEcilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
75498BZPCORTICAL MEMBRANESRATFNZpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
12010H1CORTICAL MEMBRANESHUMAN3H-doxepinNOMIFENSINE2700Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
70123CORTICAL MEMBRANESRAT3H-tryptaminecilansetron>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
72939KORCORTICAL MEMBRANESRAT3H-MUSCIMOLvicenin-2>10000Moawad A et al 2017Jan 15, 2025Jan 27, 2025
12011H1CORTICAL MEMBRANESHUMAN3H-doxepinCHLORPROMAZINE3Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
40427NMDACORTICAL MEMBRANESRAT3H-CGP39653(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid370Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
70124CORTICAL MEMBRANESRAT3H-tryptamineONDANSETRON>10000Van Wijingaarden, I. et, al. 1993Jan 15, 2025Jan 15, 2025
75756KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76524BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
12012H1CORTICAL MEMBRANESHUMAN3H-doxepinHALOPERIDOL1700Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
83180A1CORTICAL MEMBRANESRAT3H-CCPA8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione343Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
30444AMPACORTICAL MEMBRANESRAT3H-AMPAAMPA39Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40428AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
12013H1CORTICAL MEMBRANESHUMAN3H-doxepinTHIOTHIXENE4.4Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
30445AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-ATPA1800Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40429KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
12014H1CORTICAL MEMBRANESHUMAN3H-doxepinMOLINDONE>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
82926A1CORTICAL MEMBRANESRAT3H-CCPA1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione98.8Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
30446AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-Thio-ATPA270Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
12015H1CORTICAL MEMBRANESHUMAN3H-doxepinLevomepromazine0.58Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
30447AMPACORTICAL MEMBRANESRAT3H-AMPA(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid280Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
12016H1CORTICAL MEMBRANESHUMAN3H-doxepinCLOZAPINE1.2Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
83184A1CORTICAL MEMBRANESRAT3H-CCPA8-(3,4,5-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
89328CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide9.3Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
30448AMPACORTICAL MEMBRANESRAT3H-AMPA(R)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid>10000Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40432NMDACORTICAL MEMBRANESRAT3H-CGP39653(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid233Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
12017H1CORTICAL MEMBRANESHUMAN3H-doxepinCIMETIDINE>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
89329CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide245Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
30449KACORTICAL MEMBRANESRAT3H-Kainic acidAMPA>10000Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40433NMDACORTICAL MEMBRANESRAT3H-CGP39653(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
74482KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
12018H1CORTICAL MEMBRANESHUMAN3H-doxepinTiotidine>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
84210BZPCORTICAL MEMBRANESRATFNZ(±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2398PDSP Certified DataJan 15, 2025Jan 29, 2025
30450KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-ATPA>10000Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40434NMDACORTICAL MEMBRANESRAT3H-CGP39653(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
75507KORCORTICAL MEMBRANESRAT3H-MUSCIMOLpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
12019H1CORTICAL MEMBRANESHUMAN3H-doxepinRANITIDINE>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
30451KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-Thio-ATPA>10000Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40435NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid210Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
12020H1CORTICAL MEMBRANESHUMAN3H-doxepinHISTAMINE>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
82932A1CORTICAL MEMBRANESRAT3H-CCPA1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione10.1Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
30452KACORTICAL MEMBRANESRAT3H-Kainic acid(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid1600Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40436NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid1900Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
75253BZPCORTICAL MEMBRANESRAT3H-CGP12177ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76533KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
12021H1CORTICAL MEMBRANESHUMAN3H-doxepinCARBAMAZEPINE>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
30453KACORTICAL MEMBRANESRAT3H-Kainic acid(R)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid>10000Brehm, L et al., 2003Jan 15, 2025Jan 15, 2025
40437NMDACORTICAL MEMBRANESRAT3H-CGP39653(5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid100Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
12022H1CORTICAL MEMBRANESHUMAN3H-doxepinEthosuximide>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
86006KORCORTICAL MEMBRANESRAT3H-MUSCIMOLDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
30454NMDACORTICAL MEMBRANESRAT3H-CGP39653(R)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid28Brehm, L et al., 2003Jan 15, 2025Jan 28, 2025
40438NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid 960Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
12023H1CORTICAL MEMBRANESHUMAN3H-doxepinAlprazolam>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
30455NMDACORTICAL MEMBRANESRAT3H-CGP39653(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid>10000Brehm, L et al., 2003Jan 15, 2025Jan 28, 2025
40439NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid510Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
70648BZPCORTICAL MEMBRANESRATFNZMRP32155.2Porter, MR et. al, 2019Jan 15, 2025Jan 29, 2025
12024H1CORTICAL MEMBRANESHUMAN3H-doxepinNitrazepam>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
26872mGluR2CORTICAL MEMBRANESRAT3H-LY354740(+)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid9Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
30456NMDACORTICAL MEMBRANESRAT3H-CGP39653(S)-Thio-ATPA>10000Brehm, L et al., 2003Jan 15, 2025Jan 28, 2025
40440NMDACORTICAL MEMBRANESRAT3H-CGP39653(5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid2500Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
12025H1CORTICAL MEMBRANESHUMAN3H-doxepinPentobarbital>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
84217Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide1410PDSP Certified DataJan 15, 2025Jan 28, 2025
26873mGluR2CORTICAL MEMBRANESRAT3H-LY354740LY34149510Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
30457NMDACORTICAL MEMBRANESRAT3H-CGP39653(S)-ATPA>10000Brehm, L et al., 2003Jan 15, 2025Jan 28, 2025
40441AMPACORTICAL MEMBRANESRAT3H-AMPA(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
12026H1CORTICAL MEMBRANESHUMAN3H-doxepinATR1600Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
82938A1CORTICAL MEMBRANESRAT3H-CCPA8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione21.4Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
89338CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide94Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
26874mGluR2CORTICAL MEMBRANESRAT3H-LY354740DCG-IV60Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
30458NMDACORTICAL MEMBRANESRAT3H-CGP39653AMPA>10000Brehm, L et al., 2003Jan 15, 2025Jan 28, 2025
40442AMPACORTICAL MEMBRANESRAT3H-AMPA(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
12027H1CORTICAL MEMBRANESHUMAN3H-doxepinBENZTROPINE1.1Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
89339CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide288Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
26875mGluR2CORTICAL MEMBRANESRAT3H-LY354740L-CCG-I70Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40443AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
12028H1CORTICAL MEMBRANESHUMAN3H-doxepinFLUOXETINE1100Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
26876mGluR2CORTICAL MEMBRANESRAT3H-LY354740Glutamate1100Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40444AMPACORTICAL MEMBRANESRAT3H-AMPA(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
12029H1CORTICAL MEMBRANESHUMAN3H-doxepinPROPRANOLOL>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
81149BZPCORTICAL MEMBRANESRATFNZN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 29, 2025
81917BZPCORTICAL MEMBRANESRATFNZ(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 29, 2025
26877mGluR2CORTICAL MEMBRANESRAT3H-LY3547401S, 3R-ACPD2000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40445AMPACORTICAL MEMBRANESRAT3H-AMPA(5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
75262KORCORTICAL MEMBRANESRAT3H-MUSCIMOLethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
12030H1CORTICAL MEMBRANESHUMAN3H-doxepinPHENTOLAMINE4000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
84222BZPCORTICAL MEMBRANESRATFNZ(±)-3-chloro-4-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide2043PDSP Certified DataJan 15, 2025Jan 29, 2025
26878mGluR2CORTICAL MEMBRANESRAT3H-LY354740MCCG>10000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40446AMPACORTICAL MEMBRANESRAT3H-AMPA(5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
70655KORCORTICAL MEMBRANESRAT3H-MUSCIMOLMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 27, 2025
75007BZPCORTICAL MEMBRANESRATFNZ(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
12031H1CORTICAL MEMBRANESHUMAN3H-doxepinBicuculline>10000Kanba S, et al., 1984Jan 15, 2025Jan 15, 2025
26879mGluR2CORTICAL MEMBRANESRAT3H-LY354740Quisqualate>10000Schaffhauser, H et al., 1998Jan 15, 2025Jan 28, 2025
40447AMPACORTICAL MEMBRANESRAT3H-AMPA(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
7685-HT2CChoroid PlexusPIG3H-MESULERGINEIPSAPIRONE>10000SCHLICKER ET AL., 1989Jan 15, 2025Jan 15, 2025
7695-HT2CChoroid PlexusPIG3H-MESULERGINEIPSAPIRONE>10000ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
243215-HT2CChoroid PlexusPORCINE3H-MESULERGINEEscitalopram2531Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
25-HT2CChoroid PlexusPIG3H-MESULERGINE5-Methoxytryptamine23.4HOYER, 1988Jan 15, 2025Jan 15, 2025
7705-HT2CChoroid PlexusPIG3H-MESULERGINEIPSAPIRONE>10000HOYER, 1989 (J.R.R.)Jan 15, 2025Jan 15, 2025
243225-HT2CChoroid PlexusPORCINE3H-MESULERGINER-citalopram1804Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
35-HT2CChoroid PlexusPIG3H-MESULERGINE5-Methoxytryptamine25.1HOYER, 1988 or 9 (book)Jan 15, 2025Jan 15, 2025
7715-HT2CChoroid PlexusPIG3H-MESULERGINEIPSAPIRONE>10000HOYER, 1988 or 9 (book)Jan 15, 2025Jan 15, 2025
243235-HT2CChoroid PlexusPORCINE3H-MESULERGINECITALOPRAM2051Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
45-HT2CChoroid PlexusPIG3H-MESULERGINE5-Methoxytryptamine43.7MARKSTEIN ET AL, 1986Jan 15, 2025Jan 15, 2025
7725-HT2CChoroid PlexusPIG3H-MESULERGINEISAMOLTANE8130HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
243245-HT2CChoroid PlexusPORCINE3H-MESULERGINEFluoxetine-R-(-)64Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
55-HT2CChoroid PlexusPIG3H-MESULERGINE5-Methoxytryptamine43.8ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
7735-HT2CChoroid PlexusPIG3H-MESULERGINEISAMOLTANE8130SCHOEFFTER & HOYER, 1989Jan 15, 2025Jan 15, 2025
243255-HT2CChoroid PlexusPORCINE3H-MESULERGINEFLUOXETINE72Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
65-HT2CChoroid PlexusPIG3H-MESULERGINEDMT,5-Me100HOYER, 1988 or 9 (book)Jan 15, 2025Jan 15, 2025
7745-HT2CChoroid PlexusCANINE3H-SCH23390KETANSERIN13NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
217665-HT2CChoroid PlexusPIG3H-MESULERGINECLOZAPINE11Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
243265-HT2CChoroid PlexusPORCINE3H-MESULERGINEPAROXETINE9034Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
75-HT2CChoroid PlexusPIG3H-MESULERGINE5-Methoxytryptamine7.9HOYER, 1988 or 9 (book)Jan 15, 2025Jan 15, 2025
217675-HT2CChoroid PlexusPIG3H-MESULERGINEHALOPERIDOL>10000Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
243275-HT2CChoroid PlexusPORCINE3H-MESULERGINESERTRALINE2298Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
85-HT2CChoroid PlexusPIG3H-MESULERGINE5-NH2T70.8ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
7765-HT2CChoroid PlexusRAT3H-MIANSERINKETANSERIN30Sanders-Bush E, Breeding M., 1988Jan 15, 2025Jan 15, 2025
217685-HT2CChoroid PlexusPIG3H-MESULERGINEAmisulpride>10000Schoemaker H et al., 1997Jan 15, 2025Jan 15, 2025
243285-HT2CChoroid PlexusPORCINE3H-MESULERGINEFluvoxamine5786Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
95-HT2CChoroid PlexusPIG3H-MESULERGINE5-NH2T79.4HOYER, 1988 or 9 (book)Jan 15, 2025Jan 15, 2025
7775-HT2CChoroid PlexusRAT125I-LSDKETANSERIN30.1YAMAMOTO & KEBABIAN, 1989Jan 15, 2025Jan 15, 2025
105-HT2CChoroid PlexusPIG3H-MESULERGINE6-HT5500ENGEL ET AL, 1986Jan 15, 2025Jan 15, 2025
115-HT2CChoroid PlexusPIG3H-MESULERGINE8-OH-AT7410HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
7795-HT2CChoroid PlexusPIG3H-MESULERGINEKETANSERIN50PAZOS ET AL, 1984Jan 15, 2025Jan 15, 2025
133235-HT2CChoroid PlexusBeef3H-MESULERGINEFLUOXETINE269.15Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
125-HT2CChoroid PlexusPIG3H-MESULERGINE8-OH-DPAT5000PAZOS ET AL, 1984Jan 15, 2025Jan 15, 2025
7805-HT2CChoroid PlexusRAT125I-SCH 23982KETANSERIN60.3YAMAMOTO & KEBABIAN, 1989Jan 15, 2025Jan 15, 2025
133245-HT2CChoroid PlexusBeef3H-MESULERGINEFluoxetine-R-(-)154.88Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
135-HT2CChoroid PlexusPIG3H-5HT8-OH-DPAT5000PAZOS ET AL, 1984Jan 15, 2025Jan 15, 2025
133255-HT2CChoroid PlexusBeef3H-MESULERGINEFluoxetine-S-(+)3630.78Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
7825-HT2CChoroid PlexusPIG3H-MESULERGINEKETANSERIN97.7HOYER ET AL., 1985Jan 15, 2025Jan 15, 2025
133265-HT2CChoroid PlexusBeef3H-MESULERGINECITALOPRAM3311.31Wong DT, et al., 1991Jan 15, 2025Jan 15, 2025
7835-HT2CChoroid PlexusPIG125I-LSDKETANSERIN97.7HOYER ET AL., 1986Jan 15, 2025Jan 15, 2025