The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 1-1,000 of 99,458 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
7745-HT2CChoroid PlexusCANINE3H-SCH23390KETANSERIN13NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
32795D2STRIATUMCANINE3H-SPIPERONEETICLOPRIDE0.09Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32796D2STRIATUMCANINE3H-SPIPERONEFLUPHENAZINE0.5Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32800D2STRIATUMCANINE3H-SPIPERONEKETANSERIN192Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32801D2STRIATUMCANINE3H-SPIPERONEOCTOCLOTHEPIN-S1.5Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32802D2STRIATUMCANINE3H-SPIPERONEOCTOCLOTHEPIN-R13.5Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32806D2STRIATUMCANINE3H-SPIPERONEREMOXIPRIDE300Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32816D2STRIATUMCANINE3H-SPIPERONETRIFLUOPERAZINE1.2Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32817D2STRIATUMCANINE3H-SPIPERONEYM-09151-20.06Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32818D2STRIATUMCANINE3H-SPIPERONEADTN1.7Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32819D2STRIATUMCANINE3H-SPIPERONEAPOMORPHINE2Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32822D2STRIATUMCANINE3H-SPIPERONEDOPAMINE7.5Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32826D2STRIATUMCANINE3H-SPIPERONEErgocryptine, beta0.4Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32827D2STRIATUMCANINE3H-SPIPERONEFENOLDOPAM2.8Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32828D2STRIATUMCANINE3H-SPIPERONEN-04370.7Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32829D2STRIATUMCANINE3H-SPIPERONENOREPINEPHRINE6000Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32830D2STRIATUMCANINE3H-SPIPERONENPA0.4Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32831D2STRIATUMCANINE3H-SPIPERONEPHNO,(+)1.2Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32833D2STRIATUMCANINE3H-SPIPERONEQuinpirole,(-)4.8Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32834D2STRIATUMCANINE3H-SPIPERONE5-Hydroxy Tryptamine>10000Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32835D2STRIATUMCANINE3H-SPIPERONESKF 38393157Van Tol, HH et al., 1991Jan 15, 2025Jan 27, 2025
32838D4STRIATUMCANINE3H-SPIPERONECLOZAPINE9Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32839D4STRIATUMCANINE3H-SPIPERONEETICLOPRIDE2.1Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32840D4STRIATUMCANINE3H-SPIPERONEFLUPHENAZINE46Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32842D4STRIATUMCANINE3H-SPIPERONEKETANSERIN148Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32843D4STRIATUMCANINE3H-SPIPERONEOCTOCLOTHEPIN-S0.6Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32844D4STRIATUMCANINE3H-SPIPERONEOCTOCLOTHEPIN-R1.6Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32847D4STRIATUMCANINE3H-SPIPERONEREMOXIPRIDE3690Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
865-HT2CChoroid PlexusCANINE3H-SCH233905-Hydroxy Tryptamine165NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
32854D4STRIATUMCANINE3H-SPIPERONETRIFLUOPERAZINE3Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32855D4STRIATUMCANINE3H-SPIPERONEYM-09151-20.09Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32856D4STRIATUMCANINE3H-SPIPERONEADTN24Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32857D4STRIATUMCANINE3H-SPIPERONEAPOMORPHINE4.1Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32859D4STRIATUMCANINE3H-SPIPERONEDOPAMINE28Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32861D4STRIATUMCANINE3H-SPIPERONEErgocryptine, beta109Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32862D4STRIATUMCANINE3H-SPIPERONEFENOLDOPAM321Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32863D4STRIATUMCANINE3H-SPIPERONEN-0437122Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32864D4STRIATUMCANINE3H-SPIPERONENOREPINEPHRINE1760Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32865D4STRIATUMCANINE3H-SPIPERONENPA6.5Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32866D4STRIATUMCANINE3H-SPIPERONEPHNO,(+)79Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32867D4STRIATUMCANINE3H-SPIPERONEQuinpirole,(-)46Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32868D4STRIATUMCANINE3H-SPIPERONE5-Hydroxy Tryptamine4180Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
32869D4STRIATUMCANINE3H-SPIPERONESKF 383931800Van Tol, HH et al., 1991Jan 15, 2025Jan 15, 2025
9365-HT2CChoroid PlexusCANINE3H-SCH23390MIANSERIN2.8NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12528D1Choroid PlexusCANINE3H-SCH233905-Hydroxy Tryptamine>10000NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12529D1Choroid PlexusCANINE3H-SCH23390MIANSERIN161NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12530D1Choroid PlexusCANINE3H-SCH23390KETANSERIN166NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12531D1Choroid PlexusCANINE3H-SCH23390DOPAMINE>10000NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12532D1Choroid PlexusCANINE3H-SCH23390FLUPENTHIXOL, Alpha30NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12533D1Choroid PlexusCANINE3H-SCH23390BUTACLAMOL,(+)3.7NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
12534D1Choroid PlexusCANINE3H-SCH23390BUTACLAMOL, (-)>10000NICKLAUS ET AL., 1988Jan 15, 2025Jan 15, 2025
65536GABAACLONEDHUMAN[3H] FlunitrazepamXHE-III-06a37Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65792GABAACLONEDHUMAN[3H] FlunitrazepamDM-1730.78Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66048NETCLONEDHUMAN3H-NisoxetineOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
663045-HT7CLONEDHUMAN3H-LSDFinazine357Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
665605-HT5ACLONEDHUMAN3H-LSD3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride1022Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
668165-HT1DCLONEDHUMAN3H-5-CTN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67328M4CLONEDHUMAN3H-QNB1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67584A1KIDNEYHUMAN3H-N6 -phenylisopropyladenosine(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexane-2,3-diol104Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
67840D2CLONEDHUMAN3H-RACLOPRIDE(R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
25605-HT2ACORTEXHUMAN3H-SPIPERONETHIOTHIXENE,cis-2.32ANDORN ET AL., 1984Jan 15, 2025Jan 15, 2025
68608recombinantHUMAN3H-AdoMet8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline980Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
3328D3CLONEDHUMAN3H-YM 09151-2SKF 81297792TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68864SST2CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH219.9526Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69120H4CLONEDHUMAN3H-HistamineVUF468210Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693765-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL1202Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
69632Alpha1DCLONEDHUMAN3H-PRAZOSIN3-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43525-HT6CLONEDHUMAN3H-LSDMETERGOLINE400KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
4608SLC6A3CLONEDHUMAN3H-DA UPTAKEWIN 35,42813PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48645-HT2BCLONEDHUMAN3H-5HTMESULERGINE3.3WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70400D4CLONEDHUMAN3H-Methylspiperone(+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide>10000Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
51205-HT2ACLONEDHUMAN125I-DOIM-15494.2NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70656H1CLONEDHUMAN3H-PYRILAMINEMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
56325-HT4CLONEDHUMAN3H-GR-113808ZACOPRIDE281.83CLAEYSEN S, ET AL., 1997Jan 15, 2025Jan 27, 2025
71168D3CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE240Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
66565-HT1ECLONEDHUMAN3H-5HTSPIPERONE5051ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72192Beta3CLONEDHUMAN125I-Pindolol2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
6912D4CLONEDHUMAN3H-SPIPERONETRIFLUOPERAZINE44SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
727045-HT5ACLONEDHUMAN3H-LSDnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7424MORCLONEDHUMAN3H-DAMGOMORPHINE-SULFATE14Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
729605-HT2BCLONEDHUMAN3H-LSDcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7680GABAACLONEDHUMAN3H-MUSCIMOLThiomuscimol85.11Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7936GABAACLONEDHUMAN3H-RO-15-1788326000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8192GABAACLONEDHUMAN3H-RO-15-178840 (DMCM)134Huang Q, et al., 1999Jan 15, 2025Jan 27, 2025
8448SST5CLONEDHUMAN125I-CGP23996cycloantagonist SA16.98Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8704SST5CLONEDHUMAN125I-Tyr3-octreotideCGP 239962.08Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8960SST1CLONEDHUMAN125I-SRIF-28BIM 23056100Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
744965-HT1BCLONEDHUMAN3H-5-CT(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74752Alpha1BCLONEDHUMAN3H-PRAZOSIN(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75008D1CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9728MT2CLONEDHUMAN125I-IodomelatoninMelatonin,6-Cl-2-Me2.2Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75264M2CLONEDHUMAN3H-QNBethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
755205-HT1BCLONEDHUMAN3H-5-CTpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10240CLONEDHUMAN125I-HEATSPIPERONE39.81Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
757765-HT5ACLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76032Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
768005-HT1DCLONEDHUMAN3H-5-CT(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
770565-HT2CCLONEDHUMAN3H-MESULERGINE(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide8410Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11776H1FR. CORTEXHUMAN3H-doxepinTHIOTHIXENE,cis-6Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
773125-HT7CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77568Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77824Beta3CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12544NeutrophilHUMAN3H-LTB4LTB42Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78080D2CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78336H1CLONEDHUMAN3H-PYRILAMINE(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78592M2CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78848NETCLONEDHUMAN3H-Nisoxetine(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
791045-HT5ACLONEDHUMAN3H-LSD6-Fluoro-N,N-dimethyltryptamine960.5Ray TS 2010 Jan 15, 2025Jan 15, 2025
79360Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-2,5-Dimethoxy-4-methylamphetamine3219Ray TS 2010 Jan 15, 2025Jan 28, 2025
14080CLONEDHUMAN3H-LTD4LTE4693Heise CE, et al., 2000Jan 15, 2025Jan 15, 2025
79616NETCLONEDHUMAN3H-Nisoxetinecis-2a>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
143365-HT2CCLONEDHUMAN125I-DOINor-d-fenfluramine56FITZGERALD LW, ET AL., 1999Jan 15, 2025Jan 15, 2025
79872M4CLONEDHUMAN3H-QNB5-MeO-TMT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80128CLONEDHUMAN3H-VASOPRESSIN5-Methoxy-N,N-diisopropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14848TPWashed PlateletsHUMAN3H-SQ 29548SQ 2866831.8Hedberg, A, et al., 1988Jan 15, 2025Jan 15, 2025
803845-HT2ACLONEDHUMAN3H-KETANSERIN(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one1413Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15104CLONEDHUMAN3H-PGE2AGN 1909117300Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806405-HT4CLONEDHUMAN3H-GR113808(Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
808965-HT1ACLONEDHUMAN3H-8-OH-DPAT(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
81152D2CLONEDHUMAN3H-N-MethylspiperoneN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
158725-HT7CLONEDHUMAN3H-5HTTRYPTAMINE147.91BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81408D2CLONEDHUMAN3H-Methylspiperone1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine5698Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16128D1CLONEDHUMAN3H-SCH23390BROMOCRIPTINE672Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81920D2CLONEDHUMAN3H-N-Methylspiperone(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16640Y4CLONEDHUMAN125I-hPPDes-AA10-17[Cys7,21, Pro34]-NPY5Mullins D et al., 2001Jan 15, 2025Jan 15, 2025
821765-HT4CLONEDHUMAN3H-GR-1138082-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824325-HT2ACLONEDHUMAN3H-KETANSERIN(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171525-HT2ABRAINHUMAN3H-KETANSERINMELPERONE102Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
82688D4CLONEDHUMAN3H-N-Methylspiperone(S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine3362Besnard J et al 2012Jan 15, 2025Jan 28, 2025
17664CLONEDHUMAN125I-VIPVIP Ala20.43Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832005-HT1ACLONEDHUMAN3H-8-OH-DPATLSD2.78Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83456M2CLONEDHUMAN3H-NMS1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide2137.96Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83712KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide2961PDSP Certified DataJan 15, 2025Jan 28, 2025
83968KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-nitrophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide141PDSP Certified DataJan 15, 2025Jan 28, 2025
18944H1CLONEDHUMAN3H-MEPYRAMINEcis-H2-PAT(+)129Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84480DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19200M2CLONEDHUMAN3H-4-DAMPp-F-HHSiD125.893Eglen RM et al., 1994Jan 15, 2025Jan 15, 2025
84736DORCLONEDHUMAN3H-DADLE(±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19456GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHhAc-MCH(6-16)-NH20.16Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84992KORCLONEDHUMAN3H-U69593±)-(4aS,8R,8aS)-2-benzyl-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
860165-HT5ACLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86272KORCLONEDHUMAN3H-U69593JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86528A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione311Koch P et al 2018Jan 15, 2025Jan 15, 2025
875525-HT3CLONEDHUMAN3H-GR-656302-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
22272A3CLONEDHUMAN125I-Aba4b227Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878085-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine2037Staron J et al 2016Jan 15, 2025Jan 15, 2025
225285-HT7CLONEDHUMAN3H-LSDSL6501553260Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
22784H2CLONEDHUMAN3H-TIOTIDINEL-methionine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88576M1CLONEDHUMAN3H-QNB1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88832A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89088A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893445-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide52Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240645-HT2ACLONEDHUMANUNDEFINEDHALOPERIDOL46Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89600M2CLONEDHUMAN3H-NMS1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
24320NETCLONEDHUMAN3H-NorepinephrineFluvoxamine1119Owens JM et al., 2002Jan 15, 2025Jan 15, 2025
89856nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride190Liu J et al 2010Jan 15, 2025Jan 29, 2025
90112D1CLONEDHUMAN3H-SCH233902-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
250885-HT7CLONEDHUMAN3H-LSDQuetiapine308Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90624A2ACLONEDHUMAN3H-MSX-2(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide118 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25344M5CLONEDHUMAN3H-QNBZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
90880Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane10.9648Franchini S et al 2014Jan 15, 2025Jan 28, 2025
256005-HT7CLONEDHUMAN3H-LSDEphedrine,(+)2300Rothman RB, et al., 2003aJan 15, 2025Jan 15, 2025
91136A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide6500Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
25856nAChRCLONEDHUMAN3H-EpibatidinePseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
91392CB1CLONEDHUMAN3H-SR144528O-621152Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26112nAChRCLONEDHUMAN3H-EpibatidinePseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
91648A3CLONEDHUMAN3H-PSB-11N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26368DORCLONEDHUMAN3H-DADLEAmentoflavone36.5Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91904A1CLONEDHUMAN3H-DPCPX2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (3-trifluoromethylphenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
921605-HT6CLONEDHUMAN3H-LSDN-{1-[2-(Biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}quinoline-2-carboxamide1335Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
92416DORCLONEDHUMAN3H-DADLE9,13-epoxylabd-5-en-7-on-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271365-HT1ACLONEDHUMAN3H-8-OH-DPATCP-132,4848410May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92672M1CLONEDHUMAN3H-QNB15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27392Beta1CLONEDHUMAN3H-CGP-12177Quinelorane>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
92928A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one450Varano F et al 2015Jan 15, 2025Jan 15, 2025
27648Alpha2CCLONEDHUMAN35S-GTPGammaSCLONIDINE501.187Millan MJ, et al., 2000aJan 15, 2025Jan 15, 2025
279045-HT2ACLONEDHUMAN3H-KETANSERINmCPP212Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
281605-HT5ACLONEDHUMAN3H-LSDMETHYSERGIDE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93696A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester14.9Federico S et al 2018Jan 15, 2025Jan 15, 2025
286725-HT2C VGICLONEDHUMAN3H-MESULERGINEARIPIPRAZOLE180Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942085-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine3300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29184SST1CLONEDHUMANUNDEFINEDL-817,8183.3Patel YC, 1999Jan 15, 2025Jan 15, 2025
947205-HT1ECLONEDHUMAN3H-5-HT2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94976D2CLONEDHUMAN3H-N-Methylspiperone4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29952H4CLONEDHUMAN3H-Histamine(5-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone15Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
30208Alpha2ACLONEDHUMANUNDEFINEDDuloxetine1000Bymaster F.P., et. al., 2001Jan 15, 2025Jan 15, 2025
957445-HT6CLONEDHUMAN3H-LSD6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96000DATCLONEDHUMAN3H-WIN 35,4286-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96256Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30976D1CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
965125-HT1ECLONEDHUMAN[3H]5-HT6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
312325-HT6CLONEDHUMAN3H-LSDMDL 1009072388PDSP Certified DataJan 15, 2025Jan 15, 2025
96768D1CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314885-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)5011.87Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97024Alpha1BCLONEDHUMAN[3H]prazosinFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
972805-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamineBUSPIRONE50Perry CK et al 2020Jan 15, 2025Jan 15, 2025
97536A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97792H1Sf9HUMAN3H-MEPYRAMINEUR-AK627000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
98048CB2CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98304H1CLONEDHUMAN[3H]-Pyrilamine5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride553Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985605-HT2BCLONEDHUMAN[3H]-LSD2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride1247Ofon E et al 2016aJan 15, 2025Jan 15, 2025
33280M5CLONEDHUMAN3H-QNBnimesulide>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
988165-HT5ACLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
33536KORCLONEDHUMAN3H-DiprenorphineNaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99072Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99328D2CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol819Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34048P2X3CLONEDHUMAN3H-A-317491AP4A7.7Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99584A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phenyl]xanthine0.796Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99840KORCLONEDHUMAN[3H]U69,593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb9Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
100096SERTCLONEDHUMAN3H-CITALOPRAMCariprazine3597PDSP Certified DataJan 15, 2025Jan 28, 2025
1003525-HT7CLONEDHUMAN3H-LSDARIPIPRAZOLE38PDSP Certified DataJan 15, 2025Jan 15, 2025
100608CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.03Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100864nAChRCLONEDHUMANFunctionalTrimethaphan>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
35584CLONEDHUMAN3H-SQ 29548ZK1108411121Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35840Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole9.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
101376D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one82Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
36096COX-2whole blood assay (WBA)HUMANFunctionalibuprofen7200Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
1016325-HT1ACLONEDHUMAN[3H]-8-OH-DPATPerospirone0.7PDSP Certified DataMar 21, 2025Jul 28, 2026
1018885-HT1ECLONEDHUMAN3H-5HTZiprasidone1.7PDSP Certified DataMar 24, 2025Jul 28, 2026
36608D1CLONEDHUMAN3H-SCH23390MIANSERIN1420Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102144D3CLONEDHUMAN[3H]N-methylspiperoneNEMONAPRIDE1.2PDSP Certified DataMar 25, 2025Jul 28, 2026
37888MPP-2CLONEDHUMANFunctional5-[4-(2-Amino-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione10Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38656UNDEFINEDHUMAN3H-hypoxanthineN-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propyl}-2,4,6-trifluoro-benzamide48Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
38912H1CLONEDHUMAN3H-PYRILAMINEMDL 11,9391604Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
39168D4CLONEDHUMANR-SATCHLORPROMAZINE24Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39424CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396805-HT2BCLONEDHUMAN3H-5HTDOB43.6516Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40704mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopentylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
41216CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-phenylpiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41984GABAACLONEDHUMAN3H-RO-15-1788N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine6.1van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
43008FRKCLONEDHUMAN3H-StaurosporineSB2035804400Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43264CaMKCLONEDHUMAN3H-StaurosporineFlavopiridol320Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
43520EPHB4CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43776STK36CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44032PTK6CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44288PKMYT1CLONEDHUMAN3H-StaurosporineCI-1033>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44544EPHB4CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44800CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45056PAK3CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45568SLC6A4CLONEDHUMAN3H-IMIPRAMINEDesmethylcitalopram3.6Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458245-HT2BCLONEDHUMAN3H-LSD(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46080Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46592SLC6A3CLONEDHUMAN3H-WIN 35,428(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46848M5CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47360GRIA2CLONEDHUMAN3H-AMPALY 525327>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47616ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine1.5Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47872CLONEDHUMAN3H-propionyl-K24-CGRP 8-37[Tic29,D31,p34,F35]-h-alpha-CGRP 27-370.02Lang M, et al., 2006Jan 15, 2025Jan 15, 2025
48128Y1CLONEDHUMAN3H-Propionyl-NPYNPY [hPP(1-17), Ala31,Aib32], human1000Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48640CLONEDHUMANFunctionalN-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.29Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49152DORCLONEDHUMAN3H-DPDPELYS3220.48Lee YS, et al., 2006Jan 15, 2025Jan 15, 2025
49664SST3CLONEDHUMAN125I-LTT-SST-28Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8)6.7Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50176mGluR1CLONEDHUMANFunctionalQuisqualate250Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50432SST2CLONEDHUMAN125I-LTT-SST-28octreotide0.27Yang L, et.al., 1998aJan 15, 2025Jan 15, 2025
50944MORUNDEFINEDHUMANUNDEFINED17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate0.29Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51456Alpha1AUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide1.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51968KORUNDEFINEDHUMANUNDEFINED7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine6.6Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522245-HT1AUNDEFINEDHUMANUNDEFINED(S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol11.2Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52480H3UNDEFINEDHUMANUNDEFINED7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline3.8Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52992CB2UNDEFINEDHUMANUNDEFINEDRimonabant554Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53248D2UNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea183Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53760H1UNDEFINEDHUMANUNDEFINEDQuetiapine8.7Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54272SLC6A4UNDEFINEDHUMANUNDEFINEDPAROXETINE0.42Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54528A2BUNDEFINEDHUMANUNDEFINEDN-(4-cyanophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide1.97Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54784D2UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide5500Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550405-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide19Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55296DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one376Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55808SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline2980Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
56320A1UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione921Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56576DORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol2490Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56832SLC6A2UNDEFINEDHUMANUNDEFINEDBUPROPION6970Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57088D2UNDEFINEDHUMANUNDEFINEDHALOPERIDOL1Pettersson F et al., 2010Jan 15, 2025Jan 15, 2025
57344A1UNDEFINEDHUMANUNDEFINED4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)cyclohexanol1Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57600SST3UNDEFINEDHUMANUNDEFINEDN1-(benzo[d]thiazol-2-yl)-N4-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57856MORUNDEFINEDHUMANUNDEFINED(+)-1-[(1S,2S,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone180Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581125-HT2ACLONEDHUMAN125I-DOIN-(2-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine hydrochloride1.51Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58368H2CLONEDHUMAN3H-CimetidineMRS5755>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58624DORCLONEDHUMAN3H-DADLEMRS56786620Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58880D4CLONEDHUMAN3H-YM 09151-2N-[2-(4-Phenyl-1,2,3,6-tetrahydropyridin-1-yl) ethyl]-3-quinoline Carboxamide34Graulich A, et al., 2010Jan 15, 2025Jan 27, 2025
59392D4CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4'-chloro-4-biphenylcarboxamide5Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
596485-HT2ACLONEDHUMAN3H-KETANSERINSK&F 83959164O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
599045-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide4451Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60160A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiophen-3-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60416GABAACLONEDHUMANFNZCM-A-8714.7Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60672GABAACLONEDHUMANFNZSPH-383000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60928GABAACLONEDHUMANFNZXLi343150.5Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61184GABAACLONEDHUMANFNZCM-A58120Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61440GABAACLONEDHUMANFNZJYI-033.34Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
616965-HT2ACLONEDHUMAN3H-KETANSERIN2-(benzo[d][1,3]dioxol-5-yl)-N-(3,4-dimethoxyphenethyl)-N-phenethylethan-1-amine1472Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
61952CLONEDHUMANUNDEFINEDASTEMIZOLE69Chachin, M et al., 1999Jan 15, 2025Jan 15, 2025
62208NETCLONEDHUMAN[3H] WIN354285-APB2383Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62464M3CLONEDHUMAN3H-QNBDiphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
63232GCCRCLONEDHUMAN125I-Glucagon2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone O-methyloxime>10000Madsen, P et al., 1998Jan 15, 2025Jan 15, 2025
63488D2CLONEDHUMAN3H-N-Methylspiperonebifeprunox0.41Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640005-HT6CLONEDHUMAN3H-LSDN-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]-4-phenylbenzenesulfonamide6.8Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642565-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE4.46684Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64512D2CLONEDHUMAN3H-N-MethylspiperoneLOXAPINE23.9883Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65024H1FR. CORTEXHUMAN3H-MEPYRAMINEBUTACLAMOL,(+)2100Chang, R et., 1978Jan 15, 2025Jan 15, 2025
65280GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-073A (R Enriched)5.9Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65537GABAACLONEDHUMAN[3H] FlunitrazepamRo15-17880.8Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
2575-HT1ACORTEXHUMAN3H-8-OH-DPATDILTIAZEM>10000PEROUTKA, 1988Jan 15, 2025Jan 15, 2025
65793GABAACLONEDHUMAN[3H] FlunitrazepamDM-173118Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66049OTCLONEDHUMAN3H-OxytocinOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
66305Alpha1ACLONEDHUMAN3H-PRAZOSINFinazine771Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
665615-HT6CLONEDHUMAN3H-LSD3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
668175-HT1ECLONEDHUMAN3H-5-HTN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67329M5CLONEDHUMAN3H-QNB1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
20495-HT1DCORTEXHUMAN3H-5HTQUIPAZINE1100PEROUTKA ET AL., 1989Jan 15, 2025Jan 15, 2025
67585A2AKIDNEYHUMAN3H-2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexane-2,3-diol1520Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
678415-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68609recombinantHUMAN3H-AdoMet1-(Aminomethyl)-6-methoxynaphthalene1500Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
3329D3CLONEDHUMAN3H-YM 09151-2SPIPERONE0.2TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68865SST3CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2199.526Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69121H4CLONEDHUMAN3H-HistamineVUF46837.94328Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693775-HT1ACLONEDHUMAN3H-8-OH-DPATFLUPHENAZINE145Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
69633Alpha1DCLONEDHUMAN3H-PRAZOSIN4-MXP>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43535-HT6CLONEDHUMAN3H-LSDTFMPP430KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69889D1CLONEDHUMAN3H-SCH233904-(1-phenylcyclohexyl)morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4609SLC6A3CLONEDHUMAN3H-DA UPTAKEGBR-1290914PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48655-HT2BCLONEDHUMAN3H-5HTMETHYSERGIDE1.51WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70401D3CLONEDHUMAN3H-Methylspiperone(+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide27Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
51215-HT2ACLONEDHUMAN125I-DOID-36788.5NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
706575-HT1DCLONEDHUMAN125I-iodoaminopotentidineMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
53775-HT2BCLONEDHUMAN3H-5HTYOHIMBINE398.1BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
56335-HT4CLONEDHUMAN3H-GR-1138085-Methoxytryptamine154.88CLAEYSEN S, ET AL., 1997Jan 15, 2025Jan 27, 2025
71169D3CLONEDHUMAN3H-N-MethylspiperoneSYA013159Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5889Alpha2BCLONEDHUMAN3H-RAUWOLSCINERAUWOLSCINE0.32WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714255-HT1ACLONEDHUMANWAY1006354-acetoxy-N,N-diallyltryptamine383Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66575-HT1ECLONEDHUMAN3H-5HTTFMPP6293ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72193Beta 2CLONEDHUMAN3H-CGP121772-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 15, 2025
69135-HT2ACLONEDHUMAN3H-KETANSERINCHLORPROMAZINE3.5SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
727055-HT6CLONEDHUMAN3H-LSDnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7425MORCLONEDHUMAN3H-DAMGOSufentanyl0.15Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
729615-HT2CCLONEDHUMAN3H-MESULERGINEcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7681GABAACLONEDHUMAN3H-MUSCIMOLTHIP371.53Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7937GABAACLONEDHUMAN3H-RO-15-1788337000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8193GABAACLONEDHUMAN3H-RO-15-1788413000Huang Q, et al., 1999Jan 15, 2025Jan 27, 2025
8449SST5CLONEDHUMAN125I-Tyr3-octreotideSomatostatin-140.13Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8705SST5CLONEDHUMAN125I-Tyr3-octreotideBIM 230564.78Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8961SST1CLONEDHUMAN125I-SRIF-28SA398.1Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
744975-HT1DCLONEDHUMAN3H-5-CT(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74753Alpha1DCLONEDHUMAN3H-PRAZOSIN(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75009D5CLONEDHUMAN3H-SCH23390(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9729MT2CLONEDHUMAN125I-IodomelatoninGR 1964290.48Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75265M3CLONEDHUMAN3H-QNBethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
755215-HT1DCLONEDHUMAN3H-5-CTpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10241CLONEDHUMAN125I-HEATTerazosin3.98Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
757775-HT6CLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76033Beta 2CLONEDHUMAN3H-CGP-12177Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76289M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765455-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768015-HT1ECLONEDHUMAN3H-5-HT(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
770575-HT3CLONEDHUMAN3H-GR-65630(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11777H1FR. CORTEXHUMAN3H-doxepinPERPHENAZINE8Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77313Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77569Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77825Beta 2CLONEDHUMAN3H-CGP12177(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
12545NeutrophilHUMAN3H-LTB420-OH-LTB413Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78081D3CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
783375-HT1DCLONEDHUMAN3H-Cimetidine(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78593M3CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78849SERTCLONEDHUMAN3H-CITALOPRAM(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791055-HT5ACLONEDHUMAN3H-LSDLISURIDE3.1Ray TS 2010 Jan 15, 2025Jan 15, 2025
79361Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-3,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14081CLONEDHUMAN3H-LTD4BAY u9773597Heise CE, et al., 2000Jan 15, 2025Jan 15, 2025
79617NETCLONEDHUMAN3H-NisoxetineR,R-2b>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
143375-HT2CCLONEDHUMAN125I-DOIl-norfenfluramine99FITZGERALD LW, ET AL., 1999Jan 15, 2025Jan 15, 2025
79873M4CLONEDHUMAN3H-QNBEMDT>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80129CLONEDHUMAN3H-VASOPRESSINN,N-Dipropyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14849TPWashed PlateletsHUMAN3H-SQ 29548SQ 3074128.3Hedberg, A, et al., 1988Jan 15, 2025Jan 15, 2025
803855-HT2BCLONEDHUMAN3H-LSD(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one784Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15105CLONEDHUMAN3H-PGE2AGN 19439434Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806415-HT5ACLONEDHUMAN3H-LSD(Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
808975-HT1BCLONEDHUMAN3H-5-CT(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
81153D3CLONEDHUMAN3H-N-MethylspiperoneN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
158735-HT7CLONEDHUMAN3H-5HT1-NP83.17BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81409H1CLONEDHUMAN3H-PYRILAMINE1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16129D1CLONEDHUMAN3H-SCH23390SKF-76783645Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81921D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16641Y4CLONEDHUMAN125I-hPPDes-AA11-18[Cys7,21,D-Lys9 (Ac)]-NPY53.5Mullins D et al., 2001Jan 15, 2025Jan 15, 2025
821775-HT5ACLONEDHUMAN3H-LSD2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one1982Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824335-HT2BCLONEDHUMAN3H-LSD(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone6416Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171535-HT2ABRAINHUMAN3H-KETANSERINOLANZAPINE1.48Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826895-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82945A2ACHO cellsHUMAN3H-MSX-21,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione569Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
832015-HT2ACLONEDHUMAN125I-DOILSD0.71Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83457M1CLONEDHUMAN3H-NMS1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide549.541Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83713MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide4655PDSP Certified DataJan 15, 2025Jan 28, 2025
83969KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide83PDSP Certified DataJan 15, 2025Jan 28, 2025
18945H1CLONEDHUMAN3H-MEPYRAMINEcis-H2-PAT(+/-)13.6Booth RG et al., 2002Jan 15, 2025Jan 15, 2025
84481MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84737MORCLONEDHUMAN3H-DAMGO(±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19457GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHhMCH0.17Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84993DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85249recombinantHUMAN3H-EstradiolTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
860175-HT6CLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86273MORCLONEDHUMAN3H-DAMGOJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86529A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione210Koch P et al 2018Jan 15, 2025Jan 15, 2025
875535-HT5ACLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
22273A3CLONEDHUMAN125I-Aba4c670Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
87809D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine423Staron J et al 2016Jan 15, 2025Jan 28, 2025
22529SLC6A4CLONEDHUMAN125I-RTI-55 BindingSL650155905Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
22785H4CLONEDHUMAN3H-HistamineDL-homocysteine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88577M1CLONEDHUMAN3H-QNB1-(3-Phenoxypropyl)-4-phenylpiperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88833A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89089A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893455-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide365Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240655-HT2ACLONEDHUMANUNDEFINEDLOXAPINE1.9Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89601M3CLONEDHUMAN3H-NMS1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
90113D1CLONEDHUMAN3H-SCH233902-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine8700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
250895-HT3CLONEDHUMAN3H-ZACOPRIDEQuetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
90625A2ACLONEDHUMAN3H-MSX-2(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide91.8 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25345M4CLONEDHUMAN3H-QNBZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
908815-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane50.1187Franchini S et al 2014Jan 15, 2025Jan 15, 2025
256015-HT7CLONEDHUMAN3H-LSDPseudoephedrine, (-)2000Rothman RB, et al., 2003aJan 15, 2025Jan 15, 2025
91137A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide8600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
25857D4CLONEDHUMAN3H-NMSPPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91393CB1CLONEDHUMAN3H-CP55940O-6211138Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91649A3CLONEDHUMAN3H-PSB-11N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide428Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26369Alpha2ACLONEDHUMAN3H-CLONIDINEHyperoside>10000Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91905A1CLONEDHUMAN3H-DPCPX2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (4-methylphenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
921615-HT6CLONEDHUMAN3H-LSDN-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)thiophene-2-sulfonamide258Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
92417DORCLONEDHUMAN3H-DADLE15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271375-HT1ACLONEDHUMAN3H-8-OH-DPATCP-132,484(4b)287May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92673M2CLONEDHUMAN3H-QNB15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27393Beta1CLONEDHUMAN3H-CGP-12177QUINPIROLE>10000Millan MJ, et al., 2002Jan 15, 2025Jan 15, 2025
92929A3CLONEDHUMAN125I-AB-MECA2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
276495-HT2BCLONEDHUMAN3H-LSDMDMA700PDSP Certified DataJan 15, 2025Jan 15, 2025
279055-HT2ACLONEDHUMAN3H-DOBmCPP74Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
281615-HT6CLONEDHUMAN3H-LSDMETHYSERGIDE52PDSP Certified DataJan 15, 2025Jan 15, 2025
93697A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester34.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
286735-HT2CCLONEDHUMAN3H-MESULERGINEARIPIPRAZOLE75Shapiro DA, et.al., 2003Jan 15, 2025Jan 27, 2025
942095-HT1ACLONEDHUMAN3H-8-OH-DPAT4-benzyloxy-2,5-dimethoxyphenethylamine2700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29185SST2CLONEDHUMANUNDEFINEDL-817,81852Patel YC, 1999Jan 15, 2025Jan 15, 2025
947215-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94977D2CLONEDHUMAN3H-N-Methylspiperone4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29953H4CLONEDHUMAN3H-Histamine(5-Methoxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone3000Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957455-HT7CLONEDHUMAN3H-LSD6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96001DATCLONEDHUMAN3H-WIN 35,428Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96257Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30977D2CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
965135-HT2ACLONEDHUMAN[3H]-ketanserin6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
312335-HT2ACLONEDHUMAN3H-KETANSERINMDL 1009070.81PDSP Certified DataJan 15, 2025Jan 15, 2025
96769D1CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314895-HT2BCLONEDHUMAN3H-5HT(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)2511.89Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97025Alpha2ACLONEDHUMAN[3H]ClonidineFluorolintane (2-F-DPPy)829Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97281MORCLONEDHUMAN[3H]diprenorphineSRI-221387.55Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97537A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98049CB1CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime7Amato G et al 2019Jan 15, 2025Jan 28, 2025
98305D2CLONEDHUMAN[3H]-N-methylspiperone2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 167Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985615-HT2BCLONEDHUMAN[3H]-LSD2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride1713Ofon E et al 2016aJan 15, 2025Jan 15, 2025
988175-HT7CLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
99073Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99329D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)butan-2-ol1210Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34049P2X3CLONEDHUMAN3H-A-317491AP5A10.4Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99585A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthine0.419Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99841KORCLONEDHUMAN[3H]U69,593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide230Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
100097Sigma 1CLONEDHUMAN3H-Pentazocine(+)Cariprazine29PDSP Certified DataJan 15, 2025Jan 28, 2025
1003535-HT7CLONEDHUMAN3H-LSDNEMONAPRIDE81PDSP Certified DataJan 15, 2025Jan 15, 2025
100609CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-4-phenyl-2(2H)-oxoimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.05Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100865nAChRCLONEDHUMANFunctionalHEXAMETHONIUM>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
35585CLONEDHUMAN3H-SQ 29548PGF2Alpha8700Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35841SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole0.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013775-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one22Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36097COX-2whole blood assay (WBA)HUMANFunctionalKetorolac tris salt86Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
1016335-HT1BCLONEDHUMAN[3H]GR127543Perospirone1070PDSP Certified DataMar 21, 2025Jul 28, 2026
101889D1CLONEDHUMAN[3H]SCH23390Ziprasidone41PDSP Certified DataMar 24, 2025Jul 28, 2026
36609D2CLONEDHUMAN3H-SPIPERONE(2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin191Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102145D3CLONEDHUMAN[3H]N-methylspiperoneNEMONAPRIDE1.4PDSP Certified DataMar 25, 2025Jul 28, 2026
37889MPP-9CLONEDHUMANFunctional5-[4-(2-Amino-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione14Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38657UNDEFINEDHUMAN3H-hypoxanthineN-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl]-2,4,6-trifluoro-benzamide55Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
38913H1CLONEDHUMAN3H-PYRILAMINEMDL 10090766.7Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
39169D4CLONEDHUMANR-SATMELPERONE1000Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39425CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396815-HT2BCLONEDHUMAN3H-5HTDOI,(+)28.1838Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40705mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one139Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41217CLONEDHUMAN125I-Chemokine5-(4-(3-Chloro-4-trifluoromethylphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41985GABAACLONEDHUMAN3H-RO-15-17883-(5-Phenylpyridazin-3-yl)benzonitrile666van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
43009FRKCLONEDHUMAN3H-StaurosporineVX-7453300Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43265CDK2CLONEDHUMAN3H-StaurosporineRoscovitine2900Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
43521ERBB2CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43777STK38LCLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44033RPS6KA2CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44289MAPK14CLONEDHUMAN3H-StaurosporineCI-1033>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44545FERCLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44801KDRCLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45057PAK4CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45313CDK2CLONEDHUMANFunctionalpurvalanol A100Bain J, et al., 2003Jan 15, 2025Jan 28, 2025
45569NETCLONEDHUMAN3H-NisoxetineDesmethylcitalopram1820Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458255-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46081Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46593SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46849M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47361CLONEDHUMAN3H-AMPALY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47617ADKrecombinantHUMANFunctional4-N-(4-Methoxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine6Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47873CLONEDHUMAN3H-propionyl-K24-CGRP 8-37[Hyp29,D31,p34,F35]-h-alpha-CGRP 27-370.006Lang M, et al., 2006Jan 15, 2025Jan 15, 2025
48129Y1CLONEDHUMAN3H-Propionyl-NPYPP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human530Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48641GNRHRCLONEDHUMANFunctionalN-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49665SST2CLONEDHUMAN125I-LTT-SST-28Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8)>10000Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50177mGluR1CLONEDHUMANFunctionalL-CCG-I>10000Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50433SST3CLONEDHUMAN125I-LTT-SST-28octreotide45Yang L, et.al., 1998aJan 15, 2025Jan 15, 2025
50945MORUNDEFINEDHUMANUNDEFINED(5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate0.46Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51457Alpha1AUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide4.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51969KORUNDEFINEDHUMANUNDEFINED7alpha-[(4'-chlorocinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine67.9Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522255-HT1AUNDEFINEDHUMANUNDEFINED(S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol3.89Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52481SLC6A2UNDEFINEDHUMANUNDEFINED7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline118Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52993CB2UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N-ethyl-3-methylbenzofuran-2-carboxamide3100Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53249D2UNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea6.5Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53761H1UNDEFINEDHUMANUNDEFINEDOLANZAPINE2.8Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54273SLC6A4UNDEFINEDHUMANUNDEFINEDtrans-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile327Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54529A3UNDEFINEDHUMANUNDEFINEDTheophylline (1,3-dimethylxanthine)>10000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54785D2UNDEFINEDHUMANUNDEFINEDN-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide40Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550415-HT1AUNDEFINEDHUMANUNDEFINED4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide325Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55297DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one867Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55809SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline13.3Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
56321A1UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione346Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56577DORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol2690Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56833SLC6A2UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-4'-methylpropiophenone6840Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57089D2UNDEFINEDHUMANUNDEFINEDOLANZAPINE6.1Pettersson F et al., 2010Jan 15, 2025Jan 15, 2025
57345A1UNDEFINEDHUMANUNDEFINEDTonapofylline7.4Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57601SST3UNDEFINEDHUMANUNDEFINEDN1-(benzo[d]thiazol-2-ylmethyl)-N4-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57857MORUNDEFINEDHUMANUNDEFINED(-)-1-[(1R,2R,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone1150Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581135-HT2ACLONEDHUMAN125I-DOIN-(3-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate1.05Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58369H2CLONEDHUMAN3H-CimetidineMRS5698>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
586255-HT3CLONEDHUMAN3H-GR-65630MRS52023260Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58881NETCLONEDHUMAN3H-NisoxetineN,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine500Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
59137CB2CLONEDHUMAN3H-CP-55940tert-butyl 4-((9-pentyl-9H-carbazole-3-carboxamido)methyl)piperidine-1-carboxylate>10000Bladen C, et al., 2014Jan 15, 2025Jan 15, 2025
59393D2CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-4'-chloro-4-biphenylcarboxamide2600Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59649Alpha1ACLONEDHUMAN3H-PRAZOSINSK&F 83959654O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
599055-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60161A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiophen-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60417GABAACLONEDHUMANFNZCM-A-871000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60673GABAACLONEDHUMANFNZSPH-3818.5Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60929GABAACLONEDHUMANFNZXLi34317.71Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61185GABAACLONEDHUMANFNZCM-A58184Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61441GABAACLONEDHUMANFNZJYI-030.954Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
616975-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-phenylpropan-1-amine165Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
61953CLONEDHUMANUNDEFINEDASTEMIZOLE330Taglialatela, M et al., 1998Jan 15, 2025Jan 15, 2025
62209NETCLONEDHUMAN[3H] WIN354285-APB85Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62465M3CLONEDHUMAN3H-QNB2-methoxy-diphenidine>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
63233GCCRCLONEDHUMAN125I-Glucagon2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone O-benzyloxime>10000Madsen, P et al., 1998Jan 15, 2025Jan 15, 2025
63489D3CLONEDHUMAN3H-N-Methylspiperonebifeprunox0.63Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640015-HT6CLONEDHUMAN3H-LSD2-[5-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxoacetamide1000Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642575-HT2ACLONEDHUMAN3H-KETANSERINPERPHENAZINE5.62341Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64513D2CLONEDHUMAN3H-N-MethylspiperoneMELPERONE114.815Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65281GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-073A (R Enriched)11Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65538GABAACLONEDHUMAN[3H] FlunitrazepamRo15-17880.9Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
2585-HT1ACORTEXHUMAN3H-8-OH-DPATDMT119.51PIERCE & PEROUTKA, 1989Jan 15, 2025Jan 15, 2025
65794GABAACLONEDHUMAN[3H] FlunitrazepamRY-05349Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66306Alpha1BCLONEDHUMAN3H-PRAZOSINFinazine947Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
665625-HT7CLONEDHUMAN3H-LSD3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride720Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
12825-HT1DCAUDATEHUMAN3H-5HTHALOPERIDOL>10000WAEBER ET AL., 1988Jan 15, 2025Jan 15, 2025
668185-HT2ACLONEDHUMAN3H-KETANSERINN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide1572Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67330MORCLONEDHUMAN3H-DAMGO1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride2351.5Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
67586A3KIDNEYHUMANI-125-N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamide(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexane-2,3-diol3450Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
23065-HT3AMYGDALAHUMAN3H-ZACOPRIDEDOPAMINE>10000BARNES ET AL., 1989Jan 15, 2025Jan 15, 2025
678425-HT2ACLONEDHUMAN3H-Ketaserin(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline110Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
25625-HT2ACORTEXHUMAN3H-KETANSERINTHIOTHIXENE,cis-130WANDER ET AL., 1987Jan 15, 2025Jan 15, 2025
28185-HT2AFR. CORTEXHUMAN125I-LSDHISTAMINE>10000ELLIOT & KENT, 1989Jan 15, 2025Jan 15, 2025
68354nAChRKIDNEYHUMAN3H-EpibatidineNicotine303.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68610recombinantHUMAN3H-AdoMet1-(Aminomethyl)-6-hydroxynaphthalene8400Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
3330D3CLONEDHUMAN3H-YM 09151-2SULPIRIDE15TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68866SST4CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH279.4328Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69122H4CLONEDHUMAN3H-HistamineVUF468650.1187Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693785-HT1ACLONEDHUMAN3H-8-OH-DPATCHLORPROMAZINE3115Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
69634Alpha1DCLONEDHUMAN3H-PRAZOSIN2-CI-DPH>10000Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43545-HT6CLONEDHUMAN3H-LSDRU 24969570KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69890D1CLONEDHUMAN3H-SCH233904-[1-(3-methylphenyl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4610SLC6A3CLONEDHUMAN3H-DA UPTAKEMETHYLPHENIDATE42PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48665-HT2BCLONEDHUMAN3H-5HTMIANSERIN8.98WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
70402D2CLONEDHUMAN3H-Methylspiperone(+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide345Omran, A. et, al. 2018Jan 15, 2025Jan 28, 2025
51225-HT2ACLONEDHUMAN125I-DOIQDOB2155NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70658H4CLONEDHUMAN3H-HistamineMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 28, 2025
53785-HT2BCLONEDHUMAN3H-5HTmCPP31.62BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
56345-HT4CLONEDHUMAN3H-GR-1138085-CT>10000CLAEYSEN S, ET AL., 1997Jan 15, 2025Jan 27, 2025
71170D3CLONEDHUMAN3H-N-MethylspiperoneSYA1626386Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5890Alpha2BCLONEDHUMAN3H-RAUWOLSCINEYOHIMBINE1.2WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714265-HT1BCLONEDHUMAN3H-5CT4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66585-HT1ECLONEDHUMAN3H-5HT5-CT7875ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
69145-HT2ACLONEDHUMAN3H-KETANSERINCLOZAPINE11SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
727065-HT7CLONEDHUMAN3H-LSDnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7426MORCLONEDHUMAN3H-DAMGOCTOP0.18Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
729625-HT3CLONEDHUMAN3H-GR-65630catechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7682GABAACLONEDHUMAN3H-MUSCIMOLP4S97.72Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7938GABAACLONEDHUMAN3H-RO-15-1788RY 8028.8He X, et al., 1999Jan 15, 2025Jan 27, 2025
8194GABAACLONEDHUMAN3H-RO-15-178842>10000Huang Q, et al., 1999Jan 15, 2025Jan 27, 2025
8450SST5CLONEDHUMAN125I-Tyr3-octreotidesomatostatin-280.05Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8706SST5CLONEDHUMAN125I-Tyr3-octreotidecycloantagonist SA5.62Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8962SST1CLONEDHUMAN125I-SRIF-28SMS 201-995251.18Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
744985-HT1ECLONEDHUMAN3H-5-HT(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74754Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75010D2CLONEDHUMAN3H-N-Methylspiperone(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9730MT2CLONEDHUMAN125I-IodomelatoninMelatonin,6,7 di-cl-2-Me0.23Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75266M4CLONEDHUMAN3H-QNBethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
755225-HT1ECLONEDHUMAN3H-5-HTpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
10242CLONEDHUMAN125I-HEATWB 410110Schwinn, et al.,1995Jan 15, 2025Jan 15, 2025
757785-HT7CLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76290M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765465-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768025-HT2ACLONEDHUMAN3H-KETANSERIN(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
770585-HT5ACLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11778H1FR. CORTEXHUMAN3H-doxepinCHLORPROMAZINE9Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77314Alpha1BCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77570Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77826D1CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12546NeutrophilHUMAN3H-LTB4DIHETE 12(s), 5(s)454Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78082D4CLONEDHUMAN3H-N-Methylspiperone(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78338H3CLONEDHUMAN3H-Alpha-methylhistamine(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78594M4CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78850Sigma 1CLONEDHUMAN3H-Pentazocine(+)(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791065-HT5ACLONEDHUMAN3H-LSD(±)-2,5-Dimethoxy-4-iodoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79362Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-2,5-Dimethoxy-4-ethylamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14082CLONEDHUMAN3H-LTD4Pranlukast3620Heise CE, et al., 2000Jan 15, 2025Jan 15, 2025
79618NETCLONEDHUMAN3H-NisoxetineS,S-2c>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
143385-HT2BCLONEDHUMAN3H-LSDd-Fenfluramine3920FITZGERALD LW, ET AL., 1999Jan 15, 2025Jan 15, 2025
79874M4CLONEDHUMAN3H-QNBSalvinorin A>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80130CLONEDHUMAN3H-VASOPRESSIN4-Ethylthio-2,5-dimethoxyphenylbutylamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14850TPWashed PlateletsHUMAN3H-SQ 29548BM 131771404Hedberg, A, et al., 1988Jan 15, 2025Jan 15, 2025
803865-HT2CCLONEDHUMAN3H-MESULERGINE(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one2013Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15106CLONEDHUMAN3H-PGE2AGN 191995>10000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806425-HT6CLONEDHUMAN3H-LSD(Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
808985-HT1DCLONEDHUMAN3H-5-CT(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
81154D4CLONEDHUMAN3H-N-MethylspiperoneN-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 28, 2025
158745-HT7CLONEDHUMAN3H-5HT8-OH-DPAT467.73BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
814105-HT2ACLONEDHUMAN3H-KETANSERINmethyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate>10000Weiss DR et al 2018Jan 15, 2025Jan 15, 2025
16130D1CLONEDHUMAN3H-SCH23390SKF-82526, (-)1818Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81922D4CLONEDHUMAN3H-N-Methylspiperone(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16642Y4CLONEDHUMAN125I-hPPDes-AA11-18[Cys7,21,D-Lys9 (Ac), Pro34]-NPY7.3Mullins D et al., 2001Jan 15, 2025Jan 15, 2025
821785-HT6CLONEDHUMAN3H-LSD2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one2192Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824345-HT2CCLONEDHUMAN3H-MESULERGINE(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171545-HT2ABRAINHUMAN3H-KETANSERINORG-52220.77Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826905-HT1BCLONEDHUMAN3H-5-CT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
17666PANC1HUMAN125I-VIPVasoactive intestinal polypeptide1.7Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832025-HT2CCLONEDHUMAN125I-DOILSD2.91Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83458M1CLONEDHUMAN3H-NMS1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide0.301995Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
837145-HT2BCLONEDHUMAN3H-LSD(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide453PDSP Certified DataJan 15, 2025Jan 15, 2025
83970KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide302PDSP Certified DataJan 15, 2025Jan 28, 2025
84226DORCLONEDHUMAN3H-DADLE(±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide1928PDSP Certified DataJan 15, 2025Jan 28, 2025
84482KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84738MORCLONEDHUMAN3H-DAMGO(±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19458GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Nle80.34Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84994DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85250recombinantHUMAN3H-EstradiolTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
860185-HT7CLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86274DORCLONEDHUMAN3H-DADLEJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
875545-HT6CLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
22274A3CLONEDHUMAN125I-Aba4d25.6Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878105-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine137Staron J et al 2016Jan 15, 2025Jan 15, 2025
225305-HT4CLONEDHUMAN3H-GR-113808SL6501550.6Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
22786H2CLONEDHUMAN3H-TIOTIDINEL-cystine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88578H1CLONEDHUMAN3H-PYRILAMINE1-(3-Phenoxypropyl)-4-phenylpiperazine67.9Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88834A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
23554H3BRAIN CORTEXHUMAN3H-NAMHA-317920117.49Esbenshade TA, et al., 2003Jan 15, 2025Jan 15, 2025
89090A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893465-HT6CLONEDHUMAN3H-LSD3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide1039Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
240665-HT2ACLONEDHUMANUNDEFINEDMELPERONE150Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89602M3CLONEDHUMAN3H-NMS3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89858nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride108Liu J et al 2010Jan 15, 2025Jan 29, 2025
90114D1CLONEDHUMAN3H-SCH233902-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
24834Alpha1BCLONEDHUMAN125I-HEATCLOZAPINE7PDSP Certified DataJan 15, 2025Jan 15, 2025
90626A2ACLONEDHUMAN3H-MSX-24-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90882Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane21.3796Franchini S et al 2014Jan 15, 2025Jan 28, 2025
256025-HT7CLONEDHUMAN3H-LSDNorephedrine, (+)7000Rothman RB, et al., 2003aJan 15, 2025Jan 15, 2025
91138A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
25858M1CLONEDHUMAN3H-QNBPseudoephedrine,(+)>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91394CB2CLONEDHUMAN3H-CP55940O-6211>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26114SLC6A4CLONEDHUMAN3H-CITALOPRAMPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91650A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide111Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26370Alpha2ACLONEDHUMAN3H-CLONIDINEMiquelianin716.5Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91906A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (4-chlorophenyl)-methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
921625-HT6CLONEDHUMAN3H-LSDN-{1-[2-(Biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide267Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
92418DORCLONEDHUMAN3H-DADLE9,13-epoxy-15,16-dihydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271385-HT1ACLONEDHUMAN3H-8-OH-DPATN,N-dimethyl derivative562May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92674M3CLONEDHUMAN3H-QNB15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27394Beta2CLONEDHUMAN3H-CGP-12177QUINPIROLE>10000Millan MJ, et al., 2002Jan 15, 2025Jan 28, 2025
92930A3CLONEDHUMAN125I-AB-MECA2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
27650Alpha1ACLONEDHUMAN125I-HEATMDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
279065-HT2ACLONEDHUMAN3H-KETANSERINQUIPAZINE362Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
281625-HT7CLONEDHUMAN3H-LSDMETHYSERGIDE30PDSP Certified DataJan 15, 2025Jan 15, 2025
93698A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester102Federico S et al 2018Jan 15, 2025Jan 15, 2025
286745-HT2C VGICLONEDHUMAN125I-DOIARIPIPRAZOLE97Shapiro DA, et.al., 2003Jan 15, 2025Jan 15, 2025
942105-HT1ACLONEDHUMAN3H-8-OH-DPAT4-allyloxy-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29186SST2CLONEDHUMANUNDEFINEDL-803,0874720Patel YC, 1999Jan 15, 2025Jan 15, 2025
947225-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94978D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29698D2CLONEDHUMAN3H-SPIPERONEHALOPERIDOL4.9Liao Y, et.al., 1999Jan 15, 2025Jan 15, 2025
29954H4CLONEDHUMAN3H-Histamine(7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone19Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957465-HT5ACLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96002DATCLONEDHUMAN3H-WIN 35,428Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96258Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
30978D3CLONEDHUMANUNDEFINEDSR 1477781000Rinaldi-Carmona M et al., 2004Jan 15, 2025Jan 15, 2025
965145-HT2BCLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
312345-HT2CCLONEDHUMAN3H-MESULERGINEMDL 10090763.44PDSP Certified DataJan 15, 2025Jan 15, 2025
96770D1CLONEDHUMAN[3H]SCH233904-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314905-HT4CLONEDHUMANUNDEFINED(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)>10000Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97026Alpha2BCLONEDHUMAN[3H]ClonidineFluorolintane (2-F-DPPy)388Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97282MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol23.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97538A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
98050CB1CHO cellsHUMAN3H-CP-559406-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine47Amato G et al 2019Jan 15, 2025Jan 28, 2025
98306D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985625-HT2BCLONEDHUMAN[3H]-LSD2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride561Ofon E et al 2016aJan 15, 2025Jan 15, 2025
988185-HT6CLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
33538H1CLONEDHUMAN3H-PYRILAMINENaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99074Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99330D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(2-Methoxyphenyl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol1020Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34050P2X3CLONEDHUMAN3H-A-317491AP6A4.8Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99586A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine0.609Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99842Alpha1ACLONEDHUMAN[125I] HEAT(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide6800Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
100098Sigma 2CLONEDHUMAN3H-DTGCariprazine1531PDSP Certified DataJan 15, 2025Jan 28, 2025
1003545-HT7CLONEDHUMAN3H-LSDOLANZAPINE157PDSP Certified DataJan 15, 2025Jan 15, 2025
100866nAChRCLONEDHUMANFunctionald-Tubocurarine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
35586CLONEDHUMAN3H-SQ 29548FLUPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35842Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013785-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one222Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36098COX-2whole blood assay (WBA)HUMANFunctionalNaproxen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
1016345-HT1DCLONEDHUMAN[3H]GR127543Perospirone20PDSP Certified DataMar 21, 2025Jul 28, 2026
101890D2CLONEDHUMAN[3H]N-methylspiperoneZiprasidone81PDSP Certified DataMar 24, 2025Jul 28, 2026
36610D2CLONEDHUMAN3H-SPIPERONEHALOPERIDOL2.5Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102146D5CLONEDHUMAN[3H]SCH23390NEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
37890MPP-2CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-carboxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione85Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38658UNDEFINEDHUMAN3H-hypoxanthineN-{(1S,2S)-1-(4-Benzo[1,3]dioxol-5-yl-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propyl}-2,4,6-trifluoro-benzamide19Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
38914H4CLONEDHUMAN3H-HistamineMDL 100907>10000Pehek EA, et al., 2005Jan 15, 2025Jan 15, 2025
39170D4CLONEDHUMANR-SATOCTOCLOTHEPIN0.4Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39426CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396825-HT2BCLONEDHUMAN3H-5HTDOI,(-)53.7032Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
399385-HT2BCLONEDHUMANUNDEFINEDBW-723C8679.4328Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
40706mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41218CLONEDHUMAN125I-Chemokine5-(4-(4-Bromophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41986M1CLONEDHUMAN3H-QNBAdinazolam>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
43010FRKCLONEDHUMAN3H-StaurosporineBIRB-796360Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43266CDK2CLONEDHUMAN3H-StaurosporineFlavopiridol200Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
43522FERCLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43778STK4CLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44034RPS6KA3CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44290MAPK P38CLONEDHUMAN3H-StaurosporineCI-1033>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44546FGFR1CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44802YES1CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45058PAK6CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45570SLC6A3CLONEDHUMAN3H-WIN 35,428Desmethylcitalopram>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458265-HT2BCLONEDHUMAN3H-LSD(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46082Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46594SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46850M5CLONEDHUMAN3H-QNB(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47362CLONEDHUMAN3H-AMPALY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47618ADKrecombinantHUMANFunctional4-N-(4-Hydroxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine1Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47874CLONEDHUMAN3H-propionyl-K24-CGRP 8-37[Aib29,D31,p34,F35]-h-alpha-CGRP 27-370.002Lang M, et al., 2006Jan 15, 2025Jan 15, 2025
48130Y1CLONEDHUMAN3H-Propionyl-NPYPP, human170Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48642CLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride350Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49666SST1CLONEDHUMAN125I-LTT-SST-28Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8)>10000Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50178mGluR1CLONEDHUMANFunctional1S, 3R-ACPD>10000Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50434SST4CLONEDHUMAN125I-LTT-SST-28octreotide2191Yang L, et.al., 1998aJan 15, 2025Jan 15, 2025
50946MORUNDEFINEDHUMANUNDEFINEDNaloxone(-)0.79Peng X et al., 2007Jan 15, 2025Jan 15, 2025
51458Alpha1AUNDEFINEDHUMANUNDEFINED3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide1.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51970KORUNDEFINEDHUMANUNDEFINED7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine26.4Rennison D et al., 2007Jan 15, 2025Jan 15, 2025
522265-HT1AUNDEFINEDHUMANUNDEFINED(S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol1.33Krushinski JH Jr et al., 2007Jan 15, 2025Jan 15, 2025
52482SLC6A2UNDEFINEDHUMANUNDEFINED(S)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline121Letavic MA et al., 2007Jan 15, 2025Jan 15, 2025
52994CB2UNDEFINEDHUMANUNDEFINEDazepan-1-yl(5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-yl)methanone4900Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53250D2UNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea103Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53762H1UNDEFINEDHUMANUNDEFINEDZiprasidone47Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
54274SLC6A4UNDEFINEDHUMANUNDEFINEDcis-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile6.16Funke U et al., 2008Jan 15, 2025Jan 15, 2025
54530A3UNDEFINEDHUMANUNDEFINEDN-Benzo[1,3]dioxol-5-yl-2-[5-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1-methyl-1H-pyrazol-3-yloxy]-acetamide1000Borrmann T et al., 2009Jan 15, 2025Jan 15, 2025
54786D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine690Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
550425-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide70Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55298DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one379Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55810SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline44.7Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
56322A1UNDEFINEDHUMANUNDEFINED2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione132Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56578DORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol4270Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56834SLC6A2UNDEFINEDHUMANUNDEFINED2-(N-Cyclopentylamino)-3'-chloropropiophenone5700Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
57090D2UNDEFINEDHUMANUNDEFINEDPPP, S(-)-317.4Pettersson F et al., 2010Jan 15, 2025Jan 15, 2025
57346A1UNDEFINEDHUMANUNDEFINED4-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-butyric acid12Scheiff AB et al., 2010Jan 15, 2025Jan 15, 2025
57602SST3UNDEFINEDHUMANUNDEFINEDN-(benzo[d]thiazol-2-yl)-4-(3-ethoxy-4-methoxyphenyl)piperazine-1-carboxamide>10000Martin RE et al., 2009Jan 15, 2025Jan 15, 2025
57858MORUNDEFINEDHUMANUNDEFINED(+)-1-[(1S,2R,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone470Geiger C et al., 2010Jan 15, 2025Jan 15, 2025
581145-HT2ACLONEDHUMAN125I-DOIN-(4-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate10.5Nichols DE, 2014Jan 15, 2025Jan 15, 2025
58370H3CLONEDHUMAN3H-Alpha-Me-histamineMRS5698>10000Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58626hERGCLONEDHUMAN3H-N-Me-DofetilideMRS56767930Jacobson KA, et al., 2014Jan 15, 2025Jan 15, 2025
58882SLC6A3CLONEDHUMAN3H-WIN 35,428N,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine1000Mavel S, et al., 2009Jan 15, 2025Jan 15, 2025
591385-HT2ACLONEDHUMAN3H-KETANSERINCHLORPROMAZINE2.75Gillman P, et al., 2005Jan 15, 2025Jan 15, 2025
59394D4CLONEDHUMAN3H-N-MethylspiporoneN-(1-Benzyl-3-pyrrolidinyl)-2'-formyl-4-biphenylcarboxamide36Egle, I. et. al., 2004Jan 15, 2025Jan 15, 2025
59650Alpha1BCLONEDHUMAN3H-PRAZOSINSK&F 83959688O'sullivan, G. et. al., 2005Jan 15, 2025Jan 15, 2025
599065-HT6CLONEDHUMAN3H-LSD4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide>10000Huang Y, et al, 2005aJan 15, 2025Jan 15, 2025
60162A2ACLONEDHUMAN[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide>10000Tosh DK, et al., 2014Jan 15, 2025Jan 15, 2025
60418GABAACLONEDHUMANFNZCM-A-874.61Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60674GABAACLONEDHUMANFNZSPH-3810.8Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
60930GABAACLONEDHUMANFNZXLi3436.375Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61186GABAACLONEDHUMANFNZCM-A581000Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
61442GABAACLONEDHUMANFNZJYI-03107Clayton, Terry et. al. 2015Jan 15, 2025Jan 27, 2025
616985-HT2ACLONEDHUMAN3H-KETANSERINN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2-methoxyphenyl)propan-1-amine140Ponnala, Shashikanth et. al. 2015Jan 15, 2025Jan 15, 2025
61954CLONEDHUMANUNDEFINEDASTEMIZOLE>10000Suessbrich, H et al., 1996Jan 15, 2025Jan 15, 2025
62210SerotoninCLONEDHUMAN[3H] Citalopram5-APB552Iversen l., et al., 2012Jan 15, 2025Jan 15, 2025
62466M3CLONEDHUMAN3H-QNB3-methoxy-diphenidine2296Wallach, Jason, et. al. 2016Jan 15, 2025Jan 28, 2025
63234GCCRCLONEDHUMAN125I-Glucagon4-[2-(1H-Benzimidazol-2-ylsulfanyl)-1-hydroxyethyl]-2-chlorophenol>10000Madsen, P et al., 1998Jan 15, 2025Jan 15, 2025
634905-HT1ACLONEDHUMAN3H-WAY100635bifeprunox0.73Maeda, K. et, al. 2014Jan 15, 2025Jan 28, 2025
640025-HT6CLONEDHUMAN3H-LSD2-[5-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxoacetamide18.4Holenz J, et al., 2005Jan 15, 2025Jan 15, 2025
642585-HT2ACLONEDHUMAN3H-KETANSERINPIMOZIDE37.1535Silvestre, JS. et, al. 2005Jan 15, 2025Jan 15, 2025
64514D2CLONEDHUMAN3H-N-MethylspiperoneMESORIDAZINE19.0546Silvestre, JS. et, al. 2005Jan 15, 2025Jan 28, 2025
65282GABAACLONEDHUMAN[3H] FlunitrazepamXHE-II-073A (R Enriched)10Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65539GABAACLONEDHUMAN[3H] FlunitrazepamRo15-17881.05Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
65795GABAACLONEDHUMAN[3H] FlunitrazepamRY-05329Clayton, Terry et. al. 2015Jan 15, 2025Jan 28, 2025
66051SERTCLONEDHUMAN3H-CITALOPRAMOndansetron HCl>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
66307Alpha1DCLONEDHUMAN3H-PRAZOSINFinazine707Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
66563Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
12835-HT1DCORTEXHUMAN3H-5HTHALOPERIDOL>10000PEROUTKA ET AL., 1989Jan 15, 2025Jan 15, 2025
668195-HT2BCLONEDHUMAN3H-LSDN-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide913Rennekamp, A, et. al. 2016Jan 15, 2025Jan 15, 2025
67331KORCLONEDHUMAN3H-U695931-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride>10000Rennekamp, A, et. al. 2016Jan 15, 2025Jan 28, 2025
675875-HT2BKIDNEYHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol34Tosh, DK, et. al. 2016Jan 15, 2025Jan 15, 2025
23075-HT3HIPPOCAMPUSHUMAN3H-ZACOPRIDEDOPAMINE>10000BARNES ET AL., 1989Jan 15, 2025Jan 15, 2025
678435-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline2533Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
25635-HT2ACORTEXHUMAN3H-SPIPERONETHIOTHIXENE,trans-140.3ANDORN ET AL., 1984Jan 15, 2025Jan 15, 2025
68355nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid288.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68611recombinantHUMAN3H-AdoMet8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline1400Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
3331D3CLONEDHUMAN3H-YM 09151-2YM-09151-20.2TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
68867SST5CLONEDHUMAN125I-SRIFH-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2100Lewis I, et al., 2003Jan 15, 2025Jan 15, 2025
69123H4CLONEDHUMAN3H-HistamineVUF468763.0957Lim HD, et al., 2005Jan 15, 2025Jan 15, 2025
693795-HT1ACLONEDHUMAN3H-8-OH-DPATRACLOPRIDE>10000Maheux J, et al., 2005Jan 15, 2025Jan 15, 2025
4099KORCLONEDHUMAN3H-U69,593TIPPpsi>10000TOLL L, et. al., 1998Jan 15, 2025Jan 15, 2025
69635Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-CI-DPH2690Wallach, Jason, et. al. 2016Jan 15, 2025Jan 15, 2025
43555-HT6CLONEDHUMAN3H-LSD5-CT720KOHEN R, ET AL., 1996Jan 15, 2025Jan 15, 2025
69891D1CLONEDHUMAN3H-SCH233904-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine>10000Colestock, T. et, al 2018Jan 15, 2025Jan 28, 2025
4611SLC6A3CLONEDHUMAN3H-DA UPTAKENOMIFENSINE53PRISTUPA ZB, ET AL., 1994Jan 15, 2025Jan 15, 2025
48675-HT2BCLONEDHUMAN3H-5HT5-HT,N-ACETYL6800WAINSCOTT DB, ET AL., 1998Jan 15, 2025Jan 15, 2025
704035-HT1ACLONEDHUMAN3H-WAY100635(+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide328Omran, A. et, al. 2018Jan 15, 2025Jan 15, 2025
51235-HT2BCLONEDHUMAN3H-5HTDMA1039NELSON DL, ET AL., 1999Jan 15, 2025Jan 15, 2025
70659M1CLONEDHUMAN3H-QNBMRP3215>10000Porter, MR et. al, 2019Jan 15, 2025Jan 15, 2025
53795-HT2BCLONEDHUMAN3H-5HTMIANSERIN19.95BONHAUS DW, ET AL., 1995Jan 15, 2025Jan 15, 2025
71171D4CLONEDHUMAN3H-N-MethylspiperoneARIPIPRAZOLE510Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
5891Alpha2BCLONEDHUMAN3H-RAUWOLSCINEPHENOXYBENZAMINE3.5WEINSHANK RL, ET AL, 1990Jan 15, 2025Jan 15, 2025
714275-HT1DCLONEDHUMAN3H-5CT4-acetoxy-N,N-diallyltryptamine801Klein LM et al 2018Jan 15, 2025Jan 15, 2025
66595-HT1ECLONEDHUMAN3H-5HTKETANSERIN>10000ZGOMBICK JM, ET AL., 1992Jan 15, 2025Jan 15, 2025
72195D1CLONEDHUMAN3H-SCH233902-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl>10000Magnus CJ et al 2019Jan 15, 2025Jan 28, 2025
69155-HT2ACLONEDHUMAN3H-KETANSERINFLUPHENAZINE80SEEMAN P, ET AL., 1997Jan 15, 2025Jan 15, 2025
72707Alpha1ACLONEDHUMAN3H-PRAZOSINnaringenin>10000Moawad A et al 2017Jan 15, 2025Jan 28, 2025
7427MORCLONEDHUMAN3H-DAMGOb-FNA-HCl0.33Raynor K, et al., 1994Jan 15, 2025Jan 15, 2025
729635-HT5ACLONEDHUMAN3H-LSDcatechin>10000Moawad A et al 2017Jan 15, 2025Jan 15, 2025
7683GABAACLONEDHUMAN3H-MUSCIMOLGamma-Aminobutyric acid50.11Ebert B, et al., 1997Jan 15, 2025Jan 27, 2025
7939GABAACLONEDHUMAN3H-RO-15-1788Beta-CCT5000He X, et al., 1999Jan 15, 2025Jan 27, 2025
8195GABAACLONEDHUMAN3H-RO-15-178843>10000Huang Q, et al., 1999Jan 15, 2025Jan 27, 2025
8451SST5CLONEDHUMAN125I-Tyr3-octreotideLTT-SRIF280.25Siehler S, et al., 1999Jan 15, 2025Jan 15, 2025
8707SST5CLONEDHUMAN125I-Tyr3-octreotideBIM 2303035.48Siehler S, et al., 1998Jan 15, 2025Jan 15, 2025
8963SST1CLONEDHUMAN125I-SRIF-28BIM 23014501.18Bruns C, et al., 1996Jan 15, 2025Jan 15, 2025
744995-HT2ACLONEDHUMAN3H-KETANSERIN(1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
74755Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75011D3CLONEDHUMAN3H-N-Methylspiperone(1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
9731MT2CLONEDHUMAN125I-Iodomelatonin8-M-CADOT0.69Dubocovich M, Masana S, Sauri D, 1997Jan 15, 2025Jan 15, 2025
75267M5CLONEDHUMAN3H-QNBethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
755235-HT2ACLONEDHUMAN3H-KETANSERINpropan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75779Alpha1ACLONEDHUMAN3H-PRAZOSIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76035D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76291M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765475-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
768035-HT2BCLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
770595-HT6CLONEDHUMAN3H-LSD(±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
11779H1FR. CORTEXHUMAN3H-doxepinTHIORIDAZINE16Richelson E, et al., 1984Jan 15, 2025Jan 15, 2025
77315Alpha1DCLONEDHUMAN3H-PRAZOSIN(±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
77571Beta 1CLONEDHUMAN125I-Pindolol(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
77827D5CLONEDHUMAN3H-SCH23390(±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
12547NeutrophilHUMAN3H-LTB420-COOH-LTB4855Jackson RH, et al., 1992Jan 15, 2025Jan 15, 2025
78083DATCLONEDHUMAN3H-WIN 35,428(±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78339H4CLONEDHUMAN3H-Histamine(±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
78595M5CLONEDHUMAN3H-QNB(±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 15, 2025
78851Sigma 2CLONEDHUMAN3H-DTG(±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000Frankowski KJ et al 2010Jan 15, 2025Jan 28, 2025
791075-HT5ACLONEDHUMAN3H-LSD1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
79363Alpha1ACLONEDHUMAN3H-PRAZOSIN(±)-2,4,5-Trimethoxamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 28, 2025
14083CLONEDHUMAN3H-LTD4Zafirlukast7397Heise CE, et al., 2000Jan 15, 2025Jan 15, 2025
79619NETCLONEDHUMAN3H-Nisoxetine5-MeO-TMT6380Ray TS 2010 Jan 15, 2025Jan 15, 2025
143395-HT2BCLONEDHUMAN3H-LSDl-Fenfluramine680FITZGERALD LW, ET AL., 1999Jan 15, 2025Jan 15, 2025
79875M5CLONEDHUMAN3H-QNB(±)-2,5-Dimethoxy-4-bromoamphetamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
80131CLONEDHUMAN3H-VASOPRESSIN6-Fluoro-N,N-dimethyltryptamine>10000Ray TS 2010 Jan 15, 2025Jan 15, 2025
14851TPWashed PlateletsHUMAN3H-SQ 29548BM 135055.43Hedberg, A, et al., 1988Jan 15, 2025Jan 15, 2025
803875-HT3CLONEDHUMAN3H-GR-65630(E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
15107CLONEDHUMAN3H-PGE2AGN 192151>10000Schuster V.L. et.al., 2000Jan 15, 2025Jan 15, 2025
806435-HT7CLONEDHUMAN3H-LSD(Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one3350Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
808995-HT1ECLONEDHUMAN3H-5-HT(Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one>10000Lewellyn K et al 2013Jan 15, 2025Jan 15, 2025
81155DATCLONEDHUMAN3H-WIN 35,428N-Benzyl-2-azatricyclo[3.3.1.13,7]decane>10000Banister SD et al 2011Jan 15, 2025Jan 15, 2025
158755-HT7CLONEDHUMAN3H-5HTCYPROHEPTADINE123.02BOESS FG, ET AL., 1994Jan 15, 2025Jan 15, 2025
81411D2CLONEDHUMAN3H-N-Methylspiperonemethyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate>10000Weiss DR et al 2018Jan 15, 2025Jan 28, 2025
16131D1CLONEDHUMAN3H-SCH23390ADTN, (+)4600Sunahara RK, et al., 1991Jan 15, 2025Jan 15, 2025
81923D5CLONEDHUMAN3H-N-Methylspiperone(2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol>10000Severance AJ et al 2007Jan 15, 2025Jan 28, 2025
16643Y4CLONEDHUMAN125I-hPPDes-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26]-NPY206Mullins D et al., 2001Jan 15, 2025Jan 15, 2025
821795-HT7CLONEDHUMAN3H-LSD2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one181Besnard J et al 2012Jan 15, 2025Jan 15, 2025
824355-HT3CLONEDHUMAN3H-GR65630(S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
171555-HT2ABRAINHUMAN3H-KETANSERINPIMOZIDE14.3Richelson E, Souder T. 2000Jan 15, 2025Jan 15, 2025
826915-HT1DCLONEDHUMAN3H-5-CT(R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine>10000Besnard J et al 2012Jan 15, 2025Jan 15, 2025
82947A2BCHO cellsHUMAN3H-PSB-6031,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2014Jan 15, 2025Jan 15, 2025
17667CLONEDHUMAN125I-VIPVIP [D-His1]0.74Igarashi H et al., 2002Jan 15, 2025Jan 15, 2025
832035-HT2CCLONEDHUMAN125I-DOIDMT166Janowsky A et al 2014Jan 15, 2025Jan 15, 2025
83459M2CLONEDHUMAN3H-NMS1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide6.0256Del Bello F et al 2020Jan 15, 2025Jan 15, 2025
83715DATCLONEDHUMAN3H-WIN 35,428(±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide3596PDSP Certified DataJan 15, 2025Jan 15, 2025
83971KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide297PDSP Certified DataJan 15, 2025Jan 28, 2025
84227KORCLONEDHUMAN3H-U69593(±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide76PDSP Certified DataJan 15, 2025Jan 28, 2025
84483KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84739DORCLONEDHUMAN3H-DADLE(±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
19459GPR24CLONEDHUMAN125I-[Phe13, Tyr19]-hMCHN-Me-Leu962Bednarek MA et al., 2002Jan 15, 2025Jan 15, 2025
84995MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85251recombinantHUMAN125I-QRFP-43Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
86019SERTCLONEDHUMAN3H-CITALOPRAM(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86275Sigma 1CLONEDHUMAN3H-Pentazocine(+)JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
875555-HT7CLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
22275A3CLONEDHUMAN125I-Aba5816Kim, YC, et. al. 2000Jan 15, 2025Jan 15, 2025
878115-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline21Staron J et al 2016Jan 15, 2025Jan 15, 2025
225315-HT3CLONEDHUMAN3H-GR-65630SL650155>10000Moser PC et. al., 2002Jan 15, 2025Jan 15, 2025
22787H2CLONEDHUMAN3H-TIOTIDINED-methionine>10000Shi Q, et.al., 2003Jan 15, 2025Jan 15, 2025
88579H1CLONEDHUMAN3H-PYRILAMINE1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine167Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88835A3HeLaHUMAN3H-NECAN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89091A3HeLaHUMAN3H-NECAN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide10.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89347D2CLONEDHUMAN3H-RACLOPRIDE3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide268Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
240675-HT2ACLONEDHUMANUNDEFINEDMOLINDONE5800Seeman, Philip 2001Jan 15, 2025Jan 15, 2025
89603M2CLONEDHUMAN3H-NMS3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89859nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride124Liu J et al 2010Jan 15, 2025Jan 29, 2025
90115D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
248355-HT5ACLONEDHUMAN3H-LSDCLOZAPINE3857PDSP Certified DataJan 15, 2025Jan 15, 2025
90627A2ACLONEDHUMAN3H-MSX-24-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide58.3 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
25347M1CLONEDHUMAN3H-QNBZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
90883Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane158.489Franchini S et al 2014Jan 15, 2025Jan 28, 2025
256035-HT7CLONEDHUMAN3H-LSDCathinone, (-)2700Rothman RB, et al., 2003aJan 15, 2025Jan 15, 2025
91139A1CHO cellsHUMAN3H-CCPAEthyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91395CB2CLONEDHUMAN3H-CP55940O-6212>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
26115D2CLONEDHUMAN3H-NMSPPseudonorephedrine, (+) [cathine, (+)]>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
91651A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide9.05Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
26371Alpha2CCLONEDHUMAN3H-CLONIDINERutin9637Butterweck V, et. al., 2002Jan 15, 2025Jan 15, 2025
91907A1CLONEDHUMAN3H-DPCPX(2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3-chlorophenyl)methanone>10000Romagnoli R et al 2014Jan 15, 2025Jan 15, 2025
921635-HT6CLONEDHUMAN3H-LSDN-{1-[2-(5,6,7,8-Tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide102Zajdel P et al 2012Jan 15, 2025Jan 15, 2025
92419DORCLONEDHUMAN3H-DADLE9,13-epoxylabd-5-ene-7 β,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
271395-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride>10000May JA, et al., 2003Jan 15, 2025Jan 15, 2025
92675M4CLONEDHUMAN3H-QNB15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 15, 2025
27395Beta2CLONEDHUMAN3H-CGP-12177Ropinirole>10000Millan MJ, et al., 2002Jan 15, 2025Jan 28, 2025
92931A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
27651D5CLONEDHUMAN3H-SCH23390MDMA>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
93187D2CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine76Lober S et al 2012Jan 15, 2025Jan 28, 2025
279075-HT2ACLONEDHUMAN3H-DOBQUIPAZINE59Egan C, et.al., 2000Jan 15, 2025Jan 15, 2025
281635-HT1DCLONEDHUMAN3H-GR-125743METHYSERGIDE69PDSP Certified DataJan 15, 2025Jan 15, 2025
93699A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester194Federico S et al 2018Jan 15, 2025Jan 15, 2025
286755-HT2CCLONEDHUMAN125I-DOIARIPIPRAZOLE22Shapiro DA, et.al., 2003Jan 15, 2025Jan 27, 2025
942115-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
29187SST2CLONEDHUMANUNDEFINEDL-796,778>10000Patel YC, 1999Jan 15, 2025Jan 15, 2025
947235-HT2ACLONEDHUMAN3H-KETANSERIN4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94979D2CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
29699D3CLONEDHUMANUNDEFINEDHALOPERIDOL10Liao Y, et.al., 1999Jan 15, 2025Jan 15, 2025
29955H4CLONEDHUMAN3H-Histamine(7-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone8Jablonowski JA, et al., 2003Jan 15, 2025Jan 15, 2025
957475-HT6CLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96003DATCLONEDHUMAN3H-WIN 35,4286-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96259Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
965155-HT3CLONEDHUMAN[3H]GR656306-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
31235D1CLONEDHUMAN3H-SCH23390MDL 100907628PDSP Certified DataJan 15, 2025Jan 15, 2025
96771D1CLONEDHUMAN[3H]SCH233904-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
314915-HT7CLONEDHUMAN3H-5CT(R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt)3.16228Lovell, P.J., et.al. 2000Jan 15, 2025Jan 15, 2025
97027Alpha2CCLONEDHUMAN[3H]ClonidineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97283MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o138Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97539A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97795H1Sf9HUMAN3H-MEPYRAMINEUR-AK64990Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
98051CB2CHO cellsHUMAN3H-CP-559406-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine830Amato G et al 2019Jan 15, 2025Jan 28, 2025
98307D2CLONEDHUMAN[3H]-N-methylspiperone2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole990Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985635-HT2BCLONEDHUMAN[3H]-LSD2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride204Ofon E et al 2016aJan 15, 2025Jan 15, 2025
98819H1CLONEDHUMAN3H-PYRILAMINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine40Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
33539H2CLONEDHUMAN3H-TIOTIDINENaproxen>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
99075Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99331D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol607Keck TM et al 2015Jan 15, 2025Jan 28, 2025
34051P2X3CLONEDHUMAN3H-A-317491AP3A1670Jarvis, MF et. al., 2004Jan 15, 2025Jan 15, 2025
99587A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine1.25Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99843Alpha1ACLONEDHUMAN[125I] HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide6600Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
100099D1CLONEDHUMAN3H-SCH23390Cariprazine3749PDSP Certified DataJan 15, 2025Jan 28, 2025
1003555-HT7CLONEDHUMAN3H-LSDGMC 1-116200PDSP Certified DataJan 15, 2025Jan 15, 2025
100867nAChRCLONEDHUMANFunctionalSuberyldicholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
35587CLONEDHUMAN3H-SQ 29548CLOPROSTENOL6123Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35843Alpha2CCLONEDHUMAN3H-RAUWOLSCINE5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole4.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
1013795-HT6CLONEDHUMAN3H-LSD1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one999Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
36099COX-2whole blood assay (WBA)HUMANFunctionalPiroxicam7900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
1016355-HT1ECLONEDHUMAN3H-5HTPerospirone>10000PDSP Certified DataMar 21, 2025Jul 28, 2026
101891D3CLONEDHUMAN[3H]-N-methylspiperoneZiprasidone52PDSP Certified DataMar 24, 2025Jul 28, 2026
36611D2CLONEDHUMAN3H-SPIPERONECLOZAPINE144Fernandez J, et al., 2005Jan 15, 2025Jan 15, 2025
102147SERTCLONEDHUMAN[3H]CitalopramNEMONAPRIDE>10000PDSP Certified DataMar 25, 2025Jul 28, 2026
37891MPP-9CLONEDHUMANFunctional5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-carboxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione26Breyholz HJ, et al., 2005Jan 15, 2025Jan 15, 2025
38659UNDEFINEDHUMAN3H-hypoxanthineN-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-2-hydroxy-3-[2-(3-methoxyphenyl)ethylcarbamoyl]propyl}-2,4,6-tri-fluorobenzamide390Johansson P, et al., 2005Jan 15, 2025Jan 15, 2025
39171D4CLONEDHUMANR-SATMESORIDAZINE9.1Burstein ES, et al., 2005Jan 15, 2025Jan 15, 2025
39427CLONEDHUMANUNDEFINED[5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid1000Armer RE, et al., 2005Jan 15, 2025Jan 15, 2025
396835-HT2BCLONEDHUMAN3H-5HTERGOTAMINE1.28825Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
40707mGluR5CLONEDHUMANFunctional3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one19Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
41219CLONEDHUMAN125I-Chemokine5-(4-(4-Methoxyphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41987M1CLONEDHUMAN3H-QNBAMITRIPTYLINE14.7Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
43011FRKCLONEDHUMAN3H-StaurosporineGleevec3500Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43267CDK5CLONEDHUMAN3H-StaurosporineBAY-43-90066200Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43523FGFR1CLONEDHUMAN3H-StaurosporineSB202190>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
43779SykCLONEDHUMAN3H-StaurosporineVX-745>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44035RPS6KA5CLONEDHUMAN3H-StaurosporineIressa>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44291MAPK12CLONEDHUMAN3H-StaurosporineCI-1033>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
44547FGFR2CLONEDHUMAN3H-StaurosporineGW-2016>10000Fabian MA, et al., 2005Jan 15, 2025Jan 28, 2025
44803JAK1CLONEDHUMAN3H-StaurosporineLY-333531>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45059PAK7CLONEDHUMAN3H-StaurosporineFlavopiridol>10000Fabian MA, et al., 2005Jan 15, 2025Jan 15, 2025
45315CDK2CLONEDHUMANFunctionalIndirubin-3monoxime590Bain J, et al., 2003Jan 15, 2025Jan 28, 2025
45571SLC6A4CLONEDHUMAN3H-IMIPRAMINEDesmethylsertraline3Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
458275-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46083Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46595SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid6121Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46851M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47363CLONEDHUMAN3H-AMPALY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47619ADKrecombinantHUMANFunctional4-N-Cyclohexylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine250Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47875CLONEDHUMAN3H-propionyl-K24-CGRP 8-37[A29,D31,p34,F35]-h-alpha-CGRP 27-378.4Lang M, et al., 2006Jan 15, 2025Jan 15, 2025
48131Y1CLONEDHUMAN3H-Propionyl-NPYPYY 3-36760Cabrele C, et al., 2000Jan 15, 2025Jan 15, 2025
48643CLONEDHUMANFunctionalN-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride0.1Becker DP, et al., 2005Jan 15, 2025Jan 15, 2025
49667SST1CLONEDHUMAN125I-LTT-SST-28L-796,778>10000Reubi JC, et.al., 2000Jan 15, 2025Jan 15, 2025
50179mGluR3CLONEDHUMANFunctionalQuisqualate6000Flor PJ, et.al., 1996Jan 15, 2025Jan 28, 2025
50435SST5CLONEDHUMAN125I-LTT-SST-28octreotide137Yang L, et.al., 1998aJan 15, 2025Jan 15, 2025