774 5-HT2C Choroid Plexus CANINE 3H-SCH23390 KETANSERIN 13 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
32795 D2 STRIATUM CANINE 3H-SPIPERONE ETICLOPRIDE 0.09 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32796 D2 STRIATUM CANINE 3H-SPIPERONE FLUPHENAZINE 0.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32800 D2 STRIATUM CANINE 3H-SPIPERONE KETANSERIN 192 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32801 D2 STRIATUM CANINE 3H-SPIPERONE OCTOCLOTHEPIN-S 1.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32802 D2 STRIATUM CANINE 3H-SPIPERONE OCTOCLOTHEPIN-R 13.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32806 D2 STRIATUM CANINE 3H-SPIPERONE REMOXIPRIDE 300 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32816 D2 STRIATUM CANINE 3H-SPIPERONE TRIFLUOPERAZINE 1.2 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32817 D2 STRIATUM CANINE 3H-SPIPERONE YM-09151-2 0.06 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32818 D2 STRIATUM CANINE 3H-SPIPERONE ADTN 1.7 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32819 D2 STRIATUM CANINE 3H-SPIPERONE APOMORPHINE 2 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32822 D2 STRIATUM CANINE 3H-SPIPERONE DOPAMINE 7.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32826 D2 STRIATUM CANINE 3H-SPIPERONE Ergocryptine, beta 0.4 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32827 D2 STRIATUM CANINE 3H-SPIPERONE FENOLDOPAM 2.8 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32828 D2 STRIATUM CANINE 3H-SPIPERONE N-0437 0.7 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32829 D2 STRIATUM CANINE 3H-SPIPERONE NOREPINEPHRINE 6000 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32830 D2 STRIATUM CANINE 3H-SPIPERONE NPA 0.4 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32831 D2 STRIATUM CANINE 3H-SPIPERONE PHNO,(+) 1.2 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32833 D2 STRIATUM CANINE 3H-SPIPERONE Quinpirole,(-) 4.8 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32834 D2 STRIATUM CANINE 3H-SPIPERONE 5-Hydroxy Tryptamine >10000 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32835 D2 STRIATUM CANINE 3H-SPIPERONE SKF 38393 157 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 27, 2025
32838 D4 STRIATUM CANINE 3H-SPIPERONE CLOZAPINE 9 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32839 D4 STRIATUM CANINE 3H-SPIPERONE ETICLOPRIDE 2.1 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32840 D4 STRIATUM CANINE 3H-SPIPERONE FLUPHENAZINE 46 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32842 D4 STRIATUM CANINE 3H-SPIPERONE KETANSERIN 148 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32843 D4 STRIATUM CANINE 3H-SPIPERONE OCTOCLOTHEPIN-S 0.6 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32844 D4 STRIATUM CANINE 3H-SPIPERONE OCTOCLOTHEPIN-R 1.6 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32847 D4 STRIATUM CANINE 3H-SPIPERONE REMOXIPRIDE 3690 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
86 5-HT2C Choroid Plexus CANINE 3H-SCH23390 5-Hydroxy Tryptamine 165 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
32854 D4 STRIATUM CANINE 3H-SPIPERONE TRIFLUOPERAZINE 3 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32855 D4 STRIATUM CANINE 3H-SPIPERONE YM-09151-2 0.09 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32856 D4 STRIATUM CANINE 3H-SPIPERONE ADTN 24 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32857 D4 STRIATUM CANINE 3H-SPIPERONE APOMORPHINE 4.1 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32859 D4 STRIATUM CANINE 3H-SPIPERONE DOPAMINE 28 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32861 D4 STRIATUM CANINE 3H-SPIPERONE Ergocryptine, beta 109 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32862 D4 STRIATUM CANINE 3H-SPIPERONE FENOLDOPAM 321 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32863 D4 STRIATUM CANINE 3H-SPIPERONE N-0437 122 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32864 D4 STRIATUM CANINE 3H-SPIPERONE NOREPINEPHRINE 1760 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32865 D4 STRIATUM CANINE 3H-SPIPERONE NPA 6.5 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32866 D4 STRIATUM CANINE 3H-SPIPERONE PHNO,(+) 79 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32867 D4 STRIATUM CANINE 3H-SPIPERONE Quinpirole,(-) 46 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32868 D4 STRIATUM CANINE 3H-SPIPERONE 5-Hydroxy Tryptamine 4180 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
32869 D4 STRIATUM CANINE 3H-SPIPERONE SKF 38393 1800 Van Tol, HH et al., 1991 Jan 15, 2025 Jan 15, 2025
936 5-HT2C Choroid Plexus CANINE 3H-SCH23390 MIANSERIN 2.8 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12528 D1 Choroid Plexus CANINE 3H-SCH23390 5-Hydroxy Tryptamine >10000 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12529 D1 Choroid Plexus CANINE 3H-SCH23390 MIANSERIN 161 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12530 D1 Choroid Plexus CANINE 3H-SCH23390 KETANSERIN 166 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12531 D1 Choroid Plexus CANINE 3H-SCH23390 DOPAMINE >10000 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12532 D1 Choroid Plexus CANINE 3H-SCH23390 FLUPENTHIXOL, Alpha 30 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12533 D1 Choroid Plexus CANINE 3H-SCH23390 BUTACLAMOL,(+) 3.7 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
12534 D1 Choroid Plexus CANINE 3H-SCH23390 BUTACLAMOL, (-) >10000 NICKLAUS ET AL., 1988 Jan 15, 2025 Jan 15, 2025
65536 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-III-06a 37 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65792 GABAA CLONED HUMAN [3H] Flunitrazepam DM-173 0.78 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66048 NET CLONED HUMAN 3H-Nisoxetine Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
66304 5-HT7 CLONED HUMAN 3H-LSD Finazine 357 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
66560 5-HT5A CLONED HUMAN 3H-LSD 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 1022 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
66816 5-HT1D CLONED HUMAN 3H-5-CT N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67328 M4 CLONED HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67584 A1 KIDNEY HUMAN 3H-N6 -phenylisopropyladenosine (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexane-2,3-diol 104 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67840 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
2560 5-HT2A CORTEX HUMAN 3H-SPIPERONE THIOTHIXENE,cis- 2.32 ANDORN ET AL., 1984 Jan 15, 2025 Jan 15, 2025
68608 recombinant HUMAN 3H-AdoMet 8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 980 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
3328 D3 CLONED HUMAN 3H-YM 09151-2 SKF 81297 792 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68864 SST2 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 19.9526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69120 H4 CLONED HUMAN 3H-Histamine VUF4682 10 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 1202 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
69632 Alpha1D CLONED HUMAN 3H-PRAZOSIN 3-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4352 5-HT6 CLONED HUMAN 3H-LSD METERGOLINE 400 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
4608 SLC6A3 CLONED HUMAN 3H-DA UPTAKE WIN 35,428 13 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4864 5-HT2B CLONED HUMAN 3H-5HT MESULERGINE 3.3 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70400 D4 CLONED HUMAN 3H-Methylspiperone (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide >10000 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
5120 5-HT2A CLONED HUMAN 125I-DOI M-154 94.2 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70656 H1 CLONED HUMAN 3H-PYRILAMINE MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5632 5-HT4 CLONED HUMAN 3H-GR-113808 ZACOPRIDE 281.83 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
71168 D3 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 240 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
6656 5-HT1E CLONED HUMAN 3H-5HT SPIPERONE 5051 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72192 Beta3 CLONED HUMAN 125I-Pindolol 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6912 D4 CLONED HUMAN 3H-SPIPERONE TRIFLUOPERAZINE 44 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72704 5-HT5A CLONED HUMAN 3H-LSD naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7424 MOR CLONED HUMAN 3H-DAMGO MORPHINE-SULFATE 14 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72960 5-HT2B CLONED HUMAN 3H-LSD catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7680 GABAA CLONED HUMAN 3H-MUSCIMOL Thiomuscimol 85.11 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7936 GABAA CLONED HUMAN 3H-RO-15-1788 32 6000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8192 GABAA CLONED HUMAN 3H-RO-15-1788 40 (DMCM) 134 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
8448 SST5 CLONED HUMAN 125I-CGP23996 cycloantagonist SA 16.98 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8704 SST5 CLONED HUMAN 125I-Tyr3-octreotide CGP 23996 2.08 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8960 SST1 CLONED HUMAN 125I-SRIF-28 BIM 23056 100 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74496 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74752 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75008 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9728 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6-Cl-2-Me 2.2 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75264 M2 CLONED HUMAN 3H-QNB ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75520 5-HT1B CLONED HUMAN 3H-5-CT propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10240 CLONED HUMAN 125I-HEAT SPIPERONE 39.81 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75776 5-HT5A CLONED HUMAN 3H-LSD 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76032 Beta3 CLONED HUMAN 125I-Pindolol Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76800 5-HT1D CLONED HUMAN 3H-5-CT (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77056 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 8410 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11776 H1 FR. CORTEX HUMAN 3H-doxepin THIOTHIXENE,cis- 6 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77312 5-HT7 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77568 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77824 Beta3 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12544 Neutrophil HUMAN 3H-LTB4 LTB4 2 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78080 D2 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78336 H1 CLONED HUMAN 3H-PYRILAMINE (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78592 M2 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78848 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
79104 5-HT5A CLONED HUMAN 3H-LSD 6-Fluoro-N,N-dimethyltryptamine 960.5 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79360 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-2,5-Dimethoxy-4-methylamphetamine 3219 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14080 CLONED HUMAN 3H-LTD4 LTE4 693 Heise CE, et al., 2000 Jan 15, 2025 Jan 15, 2025
79616 NET CLONED HUMAN 3H-Nisoxetine cis-2a >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14336 5-HT2C CLONED HUMAN 125I-DOI Nor-d-fenfluramine 56 FITZGERALD LW, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
79872 M4 CLONED HUMAN 3H-QNB 5-MeO-TMT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80128 CLONED HUMAN 3H-VASOPRESSIN 5-Methoxy-N,N-diisopropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14848 TP Washed Platelets HUMAN 3H-SQ 29548 SQ 28668 31.8 Hedberg, A, et al., 1988 Jan 15, 2025 Jan 15, 2025
80384 5-HT2A CLONED HUMAN 3H-KETANSERIN (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 1413 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15104 CLONED HUMAN 3H-PGE2 AGN 190911 7300 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80640 5-HT4 CLONED HUMAN 3H-GR113808 (Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80896 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81152 D2 CLONED HUMAN 3H-N-Methylspiperone N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
15872 5-HT7 CLONED HUMAN 3H-5HT TRYPTAMINE 147.91 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81408 D2 CLONED HUMAN 3H-Methylspiperone 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine 5698 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16128 D1 CLONED HUMAN 3H-SCH23390 BROMOCRIPTINE 672 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81920 D2 CLONED HUMAN 3H-N-Methylspiperone (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16640 Y4 CLONED HUMAN 125I-hPP Des-AA10-17[Cys7,21, Pro34]-NPY 5 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
82176 5-HT4 CLONED HUMAN 3H-GR-113808 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82432 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17152 5-HT2A BRAIN HUMAN 3H-KETANSERIN MELPERONE 102 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82688 D4 CLONED HUMAN 3H-N-Methylspiperone (S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine 3362 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
17664 CLONED HUMAN 125I-VIP VIP Ala2 0.43 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83200 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LSD 2.78 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83456 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2137.96 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83712 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2961 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83968 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-(4-nitrophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 141 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18944 H1 CLONED HUMAN 3H-MEPYRAMINE cis-H2-PAT(+) 129 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84480 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19200 M2 CLONED HUMAN 3H-4-DAMP p-F-HHSiD 125.893 Eglen RM et al., 1994 Jan 15, 2025 Jan 15, 2025
84736 DOR CLONED HUMAN 3H-DADLE (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19456 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH hAc-MCH(6-16)-NH2 0.16 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84992 KOR CLONED HUMAN 3H-U69593 ±)-(4aS,8R,8aS)-2-benzyl-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
86016 5-HT5A CLONED HUMAN 3H-LSD (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
86272 KOR CLONED HUMAN 3H-U69593 JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86528 A2A CLONED HUMAN 3H-MSX-2 1-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 311 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87552 5-HT3 CLONED HUMAN 3H-GR-65630 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
22272 A3 CLONED HUMAN 125I-Aba 4b 227 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87808 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 2037 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22528 5-HT7 CLONED HUMAN 3H-LSD SL650155 3260 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
22784 H2 CLONED HUMAN 3H-TIOTIDINE L-methionine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88576 M1 CLONED HUMAN 3H-QNB 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88832 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89088 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89344 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 52 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24064 5-HT2A CLONED HUMAN UNDEFINED HALOPERIDOL 46 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89600 M2 CLONED HUMAN 3H-NMS 1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
24320 NET CLONED HUMAN 3H-Norepinephrine Fluvoxamine 1119 Owens JM et al., 2002 Jan 15, 2025 Jan 15, 2025
89856 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 190 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90112 D1 CLONED HUMAN 3H-SCH23390 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
25088 5-HT7 CLONED HUMAN 3H-LSD Quetiapine 308 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90624 A2A CLONED HUMAN 3H-MSX-2 (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 118 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25344 M5 CLONED HUMAN 3H-QNB ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90880 Alpha1D CHO cells HUMAN 3H-PRAZOSIN 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane 10.9648 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
25600 5-HT7 CLONED HUMAN 3H-LSD Ephedrine,(+) 2300 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
91136 A1 CHO cells HUMAN 3H-CCPA N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide 6500 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
25856 nAChR CLONED HUMAN 3H-Epibatidine Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
91392 CB1 CLONED HUMAN 3H-SR144528 O-6211 52 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26112 nAChR CLONED HUMAN 3H-Epibatidine Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
91648 A3 CLONED HUMAN 3H-PSB-11 N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide 1000 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26368 DOR CLONED HUMAN 3H-DADLE Amentoflavone 36.5 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91904 A1 CLONED HUMAN 3H-DPCPX 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (3-trifluoromethylphenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92160 5-HT6 CLONED HUMAN 3H-LSD N-{1-[2-(Biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}quinoline-2-carboxamide 1335 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
92416 DOR CLONED HUMAN 3H-DADLE 9,13-epoxylabd-5-en-7-on-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27136 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CP-132,484 8410 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92672 M1 CLONED HUMAN 3H-QNB 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27392 Beta1 CLONED HUMAN 3H-CGP-12177 Quinelorane >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92928 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 450 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27648 Alpha2C CLONED HUMAN 35S-GTPGammaS CLONIDINE 501.187 Millan MJ, et al., 2000a Jan 15, 2025 Jan 15, 2025
27904 5-HT2A CLONED HUMAN 3H-KETANSERIN mCPP 212 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28160 5-HT5A CLONED HUMAN 3H-LSD METHYSERGIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93696 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester 14.9 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28672 5-HT2C VGI CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 180 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94208 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine 3300 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29184 SST1 CLONED HUMAN UNDEFINED L-817,818 3.3 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94720 5-HT1E CLONED HUMAN 3H-5-HT 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94976 D2 CLONED HUMAN 3H-N-Methylspiperone 4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29952 H4 CLONED HUMAN 3H-Histamine (5-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 15 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
30208 Alpha2A CLONED HUMAN UNDEFINED Duloxetine 1000 Bymaster F.P., et. al., 2001 Jan 15, 2025 Jan 15, 2025
95744 5-HT6 CLONED HUMAN 3H-LSD 6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96000 DAT CLONED HUMAN 3H-WIN 35,428 6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96256 Alpha1B CLONED HUMAN 3H-PRAZOSIN 4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30976 D1 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96512 5-HT1E CLONED HUMAN [3H]5-HT 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31232 5-HT6 CLONED HUMAN 3H-LSD MDL 100907 2388 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96768 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31488 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 5011.87 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97024 Alpha1B CLONED HUMAN [3H]prazosin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97280 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine BUSPIRONE 50 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97536 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97792 H1 Sf9 HUMAN 3H-MEPYRAMINE UR-AK62 7000 Xie, S. et. al., 2006 Jan 15, 2025 Jan 15, 2025
98048 CB2 CHO cells HUMAN 3H-CP-55940 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime >10000 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98304 H1 CLONED HUMAN [3H]-Pyrilamine 5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride 553 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98560 5-HT2B CLONED HUMAN [3H]-LSD 2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 1247 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
33280 M5 CLONED HUMAN 3H-QNB nimesulide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
98816 5-HT5A CLONED HUMAN 3H-LSD 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
33536 KOR CLONED HUMAN 3H-Diprenorphine Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99072 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99328 D2 CLONED HUMAN [3H]N-methylspiperone 4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 819 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34048 P2X3 CLONED HUMAN 3H-A-317491 AP4A 7.7 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99584 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phenyl]xanthine 0.796 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99840 KOR CLONED HUMAN [3H]U69,593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 9 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
100096 SERT CLONED HUMAN 3H-CITALOPRAM Cariprazine 3597 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100352 5-HT7 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 38 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100608 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.03 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100864 nAChR CLONED HUMAN Functional Trimethaphan >10000 Kuo YP, et al., 2005 Jan 15, 2025 Jan 29, 2025
35584 CLONED HUMAN 3H-SQ 29548 ZK110841 1121 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35840 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 9.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101376 D2 CLONED HUMAN 3H-RACLOPRIDE 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 82 Zareba P, et al., 2019 Jan 15, 2025 Jan 28, 2025
36096 COX-2 whole blood assay (WBA) HUMAN Functional ibuprofen 7200 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101632 5-HT1A CLONED HUMAN [3H]-8-OH-DPAT Perospirone 0.7 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101888 5-HT1E CLONED HUMAN 3H-5HT Ziprasidone 1.7 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36608 D1 CLONED HUMAN 3H-SCH23390 MIANSERIN 1420 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102144 D3 CLONED HUMAN [3H]N-methylspiperone NEMONAPRIDE 1.2 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37888 MPP-2 CLONED HUMAN Functional 5-[4-(2-Amino-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 10 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38656 UNDEFINED HUMAN 3H-hypoxanthine N-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propyl}-2,4,6-trifluoro-benzamide 48 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
38912 H1 CLONED HUMAN 3H-PYRILAMINE MDL 11,939 1604 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39168 D4 CLONED HUMAN R-SAT CHLORPROMAZINE 24 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39424 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39680 5-HT2B CLONED HUMAN 3H-5HT DOB 43.6516 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40704 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-3-cyclopentylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one >10000 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 28, 2025
41216 CLONED HUMAN 125I-Chemokine 5-(4-Hydroxy-4-phenylpiperidin-1-yl)-2,2-diphenylpentanenitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41984 GABAA CLONED HUMAN 3H-RO-15-1788 N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine 6.1 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
43008 FRK CLONED HUMAN 3H-Staurosporine SB203580 4400 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43264 CaMK CLONED HUMAN 3H-Staurosporine Flavopiridol 320 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
43520 EPHB4 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43776 STK36 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44032 PTK6 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44288 PKMYT1 CLONED HUMAN 3H-Staurosporine CI-1033 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44544 EPHB4 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44800 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45056 PAK3 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45568 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Desmethylcitalopram 3.6 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45824 5-HT2B CLONED HUMAN 3H-LSD (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46080 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46592 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46848 M5 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47360 GRIA2 CLONED HUMAN 3H-AMPA LY 525327 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47616 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47872 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Tic29,D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
48128 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48640 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.29 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49152 DOR CLONED HUMAN 3H-DPDPE LYS322 0.48 Lee YS, et al., 2006 Jan 15, 2025 Jan 15, 2025
49664 SST3 CLONED HUMAN 125I-LTT-SST-28 Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8) 6.7 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50176 mGluR1 CLONED HUMAN Functional Quisqualate 250 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50432 SST2 CLONED HUMAN 125I-LTT-SST-28 octreotide 0.27 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
50944 MOR UNDEFINED HUMAN UNDEFINED 17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate 0.29 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51456 Alpha1A UNDEFINED HUMAN UNDEFINED 2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 1.6 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51968 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 6.6 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52224 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 11.2 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52480 H3 UNDEFINED HUMAN UNDEFINED 7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 3.8 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52992 CB2 UNDEFINED HUMAN UNDEFINED Rimonabant 554 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53248 D2 UNDEFINED HUMAN UNDEFINED 1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 183 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53760 H1 UNDEFINED HUMAN UNDEFINED Quetiapine 8.7 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54272 SLC6A4 UNDEFINED HUMAN UNDEFINED PAROXETINE 0.42 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54528 A2B UNDEFINED HUMAN UNDEFINED N-(4-cyanophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide 1.97 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54784 D2 UNDEFINED HUMAN UNDEFINED N-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide 5500 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55040 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 19 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55296 DOR UNDEFINED HUMAN UNDEFINED 8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 376 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55808 SLC6A4 UNDEFINED HUMAN UNDEFINED [C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline 2980 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
56320 A1 UNDEFINED HUMAN UNDEFINED 2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione 921 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56576 DOR UNDEFINED HUMAN UNDEFINED 4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 2490 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56832 SLC6A2 UNDEFINED HUMAN UNDEFINED BUPROPION 6970 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57088 D2 UNDEFINED HUMAN UNDEFINED HALOPERIDOL 1 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
57344 A1 UNDEFINED HUMAN UNDEFINED 4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)cyclohexanol 1 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57600 SST3 UNDEFINED HUMAN UNDEFINED N1-(benzo[d]thiazol-2-yl)-N4-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57856 MOR UNDEFINED HUMAN UNDEFINED (+)-1-[(1S,2S,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone 180 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58112 5-HT2A CLONED HUMAN 125I-DOI N-(2-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine hydrochloride 1.51 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58368 H2 CLONED HUMAN 3H-Cimetidine MRS5755 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58624 DOR CLONED HUMAN 3H-DADLE MRS5678 6620 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58880 D4 CLONED HUMAN 3H-YM 09151-2 N-[2-(4-Phenyl-1,2,3,6-tetrahydropyridin-1-yl) ethyl]-3-quinoline Carboxamide 34 Graulich A, et al., 2010 Jan 15, 2025 Jan 27, 2025
59392 D4 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4'-chloro-4-biphenylcarboxamide 5 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59648 5-HT2A CLONED HUMAN 3H-KETANSERIN SK&F 83959 164 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
59904 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 4451 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60160 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiophen-3-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60416 GABAA CLONED HUMAN FNZ CM-A-87 14.7 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60672 GABAA CLONED HUMAN FNZ SPH-38 3000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60928 GABAA CLONED HUMAN FNZ XLi343 150.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61184 GABAA CLONED HUMAN FNZ CM-A58 120 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61440 GABAA CLONED HUMAN FNZ JYI-03 3.34 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61696 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(benzo[d][1,3]dioxol-5-yl)-N-(3,4-dimethoxyphenethyl)-N-phenethylethan-1-amine 1472 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
61952 CLONED HUMAN UNDEFINED ASTEMIZOLE 69 Chachin, M et al., 1999 Jan 15, 2025 Jan 15, 2025
62208 NET CLONED HUMAN [3H] WIN35428 5-APB 2383 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62464 M3 CLONED HUMAN 3H-QNB Diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63232 GCCR CLONED HUMAN 125I-Glucagon 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone O-methyloxime >10000 Madsen, P et al., 1998 Jan 15, 2025 Jan 15, 2025
63488 D2 CLONED HUMAN 3H-N-Methylspiperone bifeprunox 0.41 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64000 5-HT6 CLONED HUMAN 3H-LSD N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]-4-phenylbenzenesulfonamide 6.8 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64256 5-HT2A CLONED HUMAN 3H-KETANSERIN OLANZAPINE 4.46684 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64512 D2 CLONED HUMAN 3H-N-Methylspiperone LOXAPINE 23.9883 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65024 H1 FR. CORTEX HUMAN 3H-MEPYRAMINE BUTACLAMOL,(+) 2100 Chang, R et., 1978 Jan 15, 2025 Jan 15, 2025
65280 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073A (R Enriched) 5.9 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65537 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-1788 0.8 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
257 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DILTIAZEM >10000 PEROUTKA, 1988 Jan 15, 2025 Jan 15, 2025
65793 GABAA CLONED HUMAN [3H] Flunitrazepam DM-173 118 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66049 OT CLONED HUMAN 3H-Oxytocin Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
66305 Alpha1A CLONED HUMAN 3H-PRAZOSIN Finazine 771 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66561 5-HT6 CLONED HUMAN 3H-LSD 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
66817 5-HT1E CLONED HUMAN 3H-5-HT N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67329 M5 CLONED HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2049 5-HT1D CORTEX HUMAN 3H-5HT QUIPAZINE 1100 PEROUTKA ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67585 A2A KIDNEY HUMAN 3H-2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexane-2,3-diol 1520 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67841 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68609 recombinant HUMAN 3H-AdoMet 1-(Aminomethyl)-6-methoxynaphthalene 1500 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
3329 D3 CLONED HUMAN 3H-YM 09151-2 SPIPERONE 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68865 SST3 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 199.526 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69121 H4 CLONED HUMAN 3H-Histamine VUF4683 7.94328 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT FLUPHENAZINE 145 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
69633 Alpha1D CLONED HUMAN 3H-PRAZOSIN 4-MXP >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4353 5-HT6 CLONED HUMAN 3H-LSD TFMPP 430 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69889 D1 CLONED HUMAN 3H-SCH23390 4-(1-phenylcyclohexyl)morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4609 SLC6A3 CLONED HUMAN 3H-DA UPTAKE GBR-12909 14 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4865 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 1.51 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70401 D3 CLONED HUMAN 3H-Methylspiperone (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 27 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
5121 5-HT2A CLONED HUMAN 125I-DOI D-367 88.5 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70657 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5377 5-HT2B CLONED HUMAN 3H-5HT YOHIMBINE 398.1 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
5633 5-HT4 CLONED HUMAN 3H-GR-113808 5-Methoxytryptamine 154.88 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
71169 D3 CLONED HUMAN 3H-N-Methylspiperone SYA013 159 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5889 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE RAUWOLSCINE 0.32 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71425 5-HT1A CLONED HUMAN WAY100635 4-acetoxy-N,N-diallyltryptamine 383 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6657 5-HT1E CLONED HUMAN 3H-5HT TFMPP 6293 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72193 Beta 2 CLONED HUMAN 3H-CGP12177 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 15, 2025
6913 5-HT2A CLONED HUMAN 3H-KETANSERIN CHLORPROMAZINE 3.5 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72705 5-HT6 CLONED HUMAN 3H-LSD naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7425 MOR CLONED HUMAN 3H-DAMGO Sufentanyl 0.15 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72961 5-HT2C CLONED HUMAN 3H-MESULERGINE catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7681 GABAA CLONED HUMAN 3H-MUSCIMOL THIP 371.53 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7937 GABAA CLONED HUMAN 3H-RO-15-1788 33 7000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8193 GABAA CLONED HUMAN 3H-RO-15-1788 41 3000 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
8449 SST5 CLONED HUMAN 125I-Tyr3-octreotide Somatostatin-14 0.13 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8705 SST5 CLONED HUMAN 125I-Tyr3-octreotide BIM 23056 4.78 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8961 SST1 CLONED HUMAN 125I-SRIF-28 SA 398.1 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74497 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74753 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75009 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9729 MT2 CLONED HUMAN 125I-Iodomelatonin GR 196429 0.48 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75265 M3 CLONED HUMAN 3H-QNB ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75521 5-HT1D CLONED HUMAN 3H-5-CT propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10241 CLONED HUMAN 125I-HEAT Terazosin 3.98 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75777 5-HT6 CLONED HUMAN 3H-LSD 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76033 Beta 2 CLONED HUMAN 3H-CGP-12177 Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76289 M1 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76545 5-HT1A CLONED HUMAN 3H-WAY100635 (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76801 5-HT1E CLONED HUMAN 3H-5-HT (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77057 5-HT3 CLONED HUMAN 3H-GR-65630 (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11777 H1 FR. CORTEX HUMAN 3H-doxepin PERPHENAZINE 8 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77313 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77569 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77825 Beta 2 CLONED HUMAN 3H-CGP12177 (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
12545 Neutrophil HUMAN 3H-LTB4 20-OH-LTB4 13 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78081 D3 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78337 5-HT1D CLONED HUMAN 3H-Cimetidine (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78593 M3 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78849 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79105 5-HT5A CLONED HUMAN 3H-LSD LISURIDE 3.1 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79361 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-3,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14081 CLONED HUMAN 3H-LTD4 BAY u9773 597 Heise CE, et al., 2000 Jan 15, 2025 Jan 15, 2025
79617 NET CLONED HUMAN 3H-Nisoxetine R,R-2b >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14337 5-HT2C CLONED HUMAN 125I-DOI l-norfenfluramine 99 FITZGERALD LW, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
79873 M4 CLONED HUMAN 3H-QNB EMDT >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80129 CLONED HUMAN 3H-VASOPRESSIN N,N-Dipropyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14849 TP Washed Platelets HUMAN 3H-SQ 29548 SQ 30741 28.3 Hedberg, A, et al., 1988 Jan 15, 2025 Jan 15, 2025
80385 5-HT2B CLONED HUMAN 3H-LSD (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 784 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15105 CLONED HUMAN 3H-PGE2 AGN 194394 34 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80641 5-HT5A CLONED HUMAN 3H-LSD (Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80897 5-HT1B CLONED HUMAN 3H-5-CT (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81153 D3 CLONED HUMAN 3H-N-Methylspiperone N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
15873 5-HT7 CLONED HUMAN 3H-5HT 1-NP 83.17 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81409 H1 CLONED HUMAN 3H-PYRILAMINE 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16129 D1 CLONED HUMAN 3H-SCH23390 SKF-76783 645 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81921 D3 CLONED HUMAN 3H-N-Methylspiperone (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16641 Y4 CLONED HUMAN 125I-hPP Des-AA11-18[Cys7,21,D-Lys9 (Ac)]-NPY 53.5 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
82177 5-HT5A CLONED HUMAN 3H-LSD 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 1982 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82433 5-HT2B CLONED HUMAN 3H-LSD (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone 6416 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17153 5-HT2A BRAIN HUMAN 3H-KETANSERIN OLANZAPINE 1.48 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82689 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82945 A2A CHO cells HUMAN 3H-MSX-2 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 569 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83201 5-HT2A CLONED HUMAN 125I-DOI LSD 0.71 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83457 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 549.541 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83713 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 4655 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83969 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 83 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
18945 H1 CLONED HUMAN 3H-MEPYRAMINE cis-H2-PAT(+/-) 13.6 Booth RG et al., 2002 Jan 15, 2025 Jan 15, 2025
84481 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84737 MOR CLONED HUMAN 3H-DAMGO (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19457 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH hMCH 0.17 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84993 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85249 recombinant HUMAN 3H-Estradiol Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 15, 2025
86017 5-HT6 CLONED HUMAN 3H-LSD (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
86273 MOR CLONED HUMAN 3H-DAMGO JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86529 A1 CLONED HUMAN 3H-CCPA 1-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 210 Koch P et al 2018 Jan 15, 2025 Jan 15, 2025
87553 5-HT5A CLONED HUMAN 3H-LSD 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
22273 A3 CLONED HUMAN 125I-Aba 4c 670 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87809 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 423 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
22529 SLC6A4 CLONED HUMAN 125I-RTI-55 Binding SL650155 905 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
22785 H4 CLONED HUMAN 3H-Histamine DL-homocysteine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88577 M1 CLONED HUMAN 3H-QNB 1-(3-Phenoxypropyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88833 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89089 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 365 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24065 5-HT2A CLONED HUMAN UNDEFINED LOXAPINE 1.9 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89601 M3 CLONED HUMAN 3H-NMS 1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
90113 D1 CLONED HUMAN 3H-SCH23390 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 8700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
25089 5-HT3 CLONED HUMAN 3H-ZACOPRIDE Quetiapine >10000 Jensen NH, et al., 2008 Jan 15, 2025 Jan 15, 2025
90625 A2A CLONED HUMAN 3H-MSX-2 (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 91.8 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25345 M4 CLONED HUMAN 3H-QNB ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90881 5-HT1A HeLa HUMAN 3H-8-OH-DPAT 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane 50.1187 Franchini S et al 2014 Jan 15, 2025 Jan 15, 2025
25601 5-HT7 CLONED HUMAN 3H-LSD Pseudoephedrine, (-) 2000 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
91137 A2A CHO cells HUMAN 3H-NECA N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide 8600 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
25857 D4 CLONED HUMAN 3H-NMSP Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91393 CB1 CLONED HUMAN 3H-CP55940 O-6211 138 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
91649 A3 CLONED HUMAN 3H-PSB-11 N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide 428 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26369 Alpha2A CLONED HUMAN 3H-CLONIDINE Hyperoside >10000 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91905 A1 CLONED HUMAN 3H-DPCPX 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (4-methylphenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92161 5-HT6 CLONED HUMAN 3H-LSD N-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)thiophene-2-sulfonamide 258 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
92417 DOR CLONED HUMAN 3H-DADLE 15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27137 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CP-132,484(4b) 287 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92673 M2 CLONED HUMAN 3H-QNB 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27393 Beta1 CLONED HUMAN 3H-CGP-12177 QUINPIROLE >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 15, 2025
92929 A3 CLONED HUMAN 125I-AB-MECA 2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27649 5-HT2B CLONED HUMAN 3H-LSD MDMA 700 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27905 5-HT2A CLONED HUMAN 3H-DOB mCPP 74 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28161 5-HT6 CLONED HUMAN 3H-LSD METHYSERGIDE 52 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93697 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester 34.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28673 5-HT2C CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 75 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 27, 2025
94209 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-benzyloxy-2,5-dimethoxyphenethylamine 2700 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29185 SST2 CLONED HUMAN UNDEFINED L-817,818 52 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94721 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94977 D2 CLONED HUMAN 3H-N-Methylspiperone 4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29953 H4 CLONED HUMAN 3H-Histamine (5-Methoxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 3000 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95745 5-HT7 CLONED HUMAN 3H-LSD 6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96001 DAT CLONED HUMAN 3H-WIN 35,428 Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96257 Alpha1D CLONED HUMAN 3H-PRAZOSIN 4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30977 D2 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96513 5-HT2A CLONED HUMAN [3H]-ketanserin 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31233 5-HT2A CLONED HUMAN 3H-KETANSERIN MDL 100907 0.81 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96769 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31489 5-HT2B CLONED HUMAN 3H-5HT (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 2511.89 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97025 Alpha2A CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) 829 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97281 MOR CLONED HUMAN [3H]diprenorphine SRI-22138 7.55 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97537 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98049 CB1 CHO cells HUMAN 3H-CP-55940 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime 7 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98305 D2 CLONED HUMAN [3H]-N-methylspiperone 2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 167 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98561 5-HT2B CLONED HUMAN [3H]-LSD 2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride 1713 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98817 5-HT7 CLONED HUMAN 3H-LSD 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
99073 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99329 D2 CLONED HUMAN [3H]N-methylspiperone 1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)butan-2-ol 1210 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34049 P2X3 CLONED HUMAN 3H-A-317491 AP5A 10.4 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99585 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthine 0.419 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99841 KOR CLONED HUMAN [3H]U69,593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 230 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
100097 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) Cariprazine 29 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100353 5-HT7 CLONED HUMAN 3H-LSD NEMONAPRIDE 81 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100609 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-4-phenyl-2(2H)-oxoimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.05 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100865 nAChR CLONED HUMAN Functional HEXAMETHONIUM >10000 Kuo YP, et al., 2005 Jan 15, 2025 Jan 29, 2025
35585 CLONED HUMAN 3H-SQ 29548 PGF2Alpha 8700 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35841 SLC6A4 CLONED HUMAN 3H-PAROXETINE 3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 0.5 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 22 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36097 COX-2 whole blood assay (WBA) HUMAN Functional Ketorolac tris salt 86 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101633 5-HT1B CLONED HUMAN [3H]GR127543 Perospirone 1070 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101889 D1 CLONED HUMAN [3H]SCH23390 Ziprasidone 41 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36609 D2 CLONED HUMAN 3H-SPIPERONE (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin 191 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102145 D3 CLONED HUMAN [3H]N-methylspiperone NEMONAPRIDE 1.4 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37889 MPP-9 CLONED HUMAN Functional 5-[4-(2-Amino-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 14 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38657 UNDEFINED HUMAN 3H-hypoxanthine N-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl]-2,4,6-trifluoro-benzamide 55 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
38913 H1 CLONED HUMAN 3H-PYRILAMINE MDL 100907 66.7 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39169 D4 CLONED HUMAN R-SAT MELPERONE 1000 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39425 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39681 5-HT2B CLONED HUMAN 3H-5HT DOI,(+) 28.1838 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40705 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one 139 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41217 CLONED HUMAN 125I-Chemokine 5-(4-(3-Chloro-4-trifluoromethylphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41985 GABAA CLONED HUMAN 3H-RO-15-1788 3-(5-Phenylpyridazin-3-yl)benzonitrile 666 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
43009 FRK CLONED HUMAN 3H-Staurosporine VX-745 3300 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43265 CDK2 CLONED HUMAN 3H-Staurosporine Roscovitine 2900 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
43521 ERBB2 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43777 STK38L CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44033 RPS6KA2 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44289 MAPK14 CLONED HUMAN 3H-Staurosporine CI-1033 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44545 FER CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44801 KDR CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45057 PAK4 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45313 CDK2 CLONED HUMAN Functional purvalanol A 100 Bain J, et al., 2003 Jan 15, 2025 Jan 28, 2025
45569 NET CLONED HUMAN 3H-Nisoxetine Desmethylcitalopram 1820 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45825 5-HT2B CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46081 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46593 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46849 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47361 CLONED HUMAN 3H-AMPA LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47617 ADK recombinant HUMAN Functional 4-N-(4-Methoxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 6 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47873 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Hyp29,D31,p34,F35]-h-alpha-CGRP 27-37 0.006 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
48129 Y1 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 530 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48641 GNRHR CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49665 SST2 CLONED HUMAN 125I-LTT-SST-28 Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8) >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50177 mGluR1 CLONED HUMAN Functional L-CCG-I >10000 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50433 SST3 CLONED HUMAN 125I-LTT-SST-28 octreotide 45 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
50945 MOR UNDEFINED HUMAN UNDEFINED (5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate 0.46 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51457 Alpha1A UNDEFINED HUMAN UNDEFINED 2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4.5 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51969 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(4'-chlorocinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 67.9 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52225 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 3.89 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52481 SLC6A2 UNDEFINED HUMAN UNDEFINED 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline 118 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52993 CB2 UNDEFINED HUMAN UNDEFINED N-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N-ethyl-3-methylbenzofuran-2-carboxamide 3100 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53249 D2 UNDEFINED HUMAN UNDEFINED 1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea 6.5 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53761 H1 UNDEFINED HUMAN UNDEFINED OLANZAPINE 2.8 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54273 SLC6A4 UNDEFINED HUMAN UNDEFINED trans-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile 327 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54529 A3 UNDEFINED HUMAN UNDEFINED Theophylline (1,3-dimethylxanthine) >10000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54785 D2 UNDEFINED HUMAN UNDEFINED N-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide 40 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55041 5-HT1A UNDEFINED HUMAN UNDEFINED 4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide 325 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55297 DOR UNDEFINED HUMAN UNDEFINED 3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 867 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55809 SLC6A4 UNDEFINED HUMAN UNDEFINED [C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline 13.3 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
56321 A1 UNDEFINED HUMAN UNDEFINED 2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione 346 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56577 DOR UNDEFINED HUMAN UNDEFINED 4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 2690 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56833 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-(N-tert-Butylamino)-4'-methylpropiophenone 6840 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57089 D2 UNDEFINED HUMAN UNDEFINED OLANZAPINE 6.1 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
57345 A1 UNDEFINED HUMAN UNDEFINED Tonapofylline 7.4 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57601 SST3 UNDEFINED HUMAN UNDEFINED N1-(benzo[d]thiazol-2-ylmethyl)-N4-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57857 MOR UNDEFINED HUMAN UNDEFINED (-)-1-[(1R,2R,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone 1150 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58113 5-HT2A CLONED HUMAN 125I-DOI N-(3-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 1.05 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58369 H2 CLONED HUMAN 3H-Cimetidine MRS5698 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58625 5-HT3 CLONED HUMAN 3H-GR-65630 MRS5202 3260 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58881 NET CLONED HUMAN 3H-Nisoxetine N,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine 500 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
59137 CB2 CLONED HUMAN 3H-CP-55940 tert-butyl 4-((9-pentyl-9H-carbazole-3-carboxamido)methyl)piperidine-1-carboxylate >10000 Bladen C, et al., 2014 Jan 15, 2025 Jan 15, 2025
59393 D2 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-4'-chloro-4-biphenylcarboxamide 2600 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59649 Alpha1A CLONED HUMAN 3H-PRAZOSIN SK&F 83959 654 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
59905 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60161 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiophen-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60417 GABAA CLONED HUMAN FNZ CM-A-87 1000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60673 GABAA CLONED HUMAN FNZ SPH-38 18.5 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60929 GABAA CLONED HUMAN FNZ XLi343 17.71 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61185 GABAA CLONED HUMAN FNZ CM-A58 184 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61441 GABAA CLONED HUMAN FNZ JYI-03 0.954 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61697 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-phenylpropan-1-amine 165 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
61953 CLONED HUMAN UNDEFINED ASTEMIZOLE 330 Taglialatela, M et al., 1998 Jan 15, 2025 Jan 15, 2025
62209 NET CLONED HUMAN [3H] WIN35428 5-APB 85 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62465 M3 CLONED HUMAN 3H-QNB 2-methoxy-diphenidine >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63233 GCCR CLONED HUMAN 125I-Glucagon 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone O-benzyloxime >10000 Madsen, P et al., 1998 Jan 15, 2025 Jan 15, 2025
63489 D3 CLONED HUMAN 3H-N-Methylspiperone bifeprunox 0.63 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64001 5-HT6 CLONED HUMAN 3H-LSD 2-[5-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxoacetamide 1000 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64257 5-HT2A CLONED HUMAN 3H-KETANSERIN PERPHENAZINE 5.62341 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64513 D2 CLONED HUMAN 3H-N-Methylspiperone MELPERONE 114.815 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65281 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073A (R Enriched) 11 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65538 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-1788 0.9 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
258 5-HT1A CORTEX HUMAN 3H-8-OH-DPAT DMT 119.51 PIERCE & PEROUTKA, 1989 Jan 15, 2025 Jan 15, 2025
65794 GABAA CLONED HUMAN [3H] Flunitrazepam RY-053 49 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66306 Alpha1B CLONED HUMAN 3H-PRAZOSIN Finazine 947 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66562 5-HT7 CLONED HUMAN 3H-LSD 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 720 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
1282 5-HT1D CAUDATE HUMAN 3H-5HT HALOPERIDOL >10000 WAEBER ET AL., 1988 Jan 15, 2025 Jan 15, 2025
66818 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 1572 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67330 MOR CLONED HUMAN 3H-DAMGO 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 2351.5 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67586 A3 KIDNEY HUMAN I-125-N6 -(4-amino-3-iodobenzyl)adenosine-5′-N-methyluronamide (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexane-2,3-diol 3450 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2306 5-HT3 AMYGDALA HUMAN 3H-ZACOPRIDE DOPAMINE >10000 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67842 5-HT2A CLONED HUMAN 3H-Ketaserin (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 110 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
2562 5-HT2A CORTEX HUMAN 3H-KETANSERIN THIOTHIXENE,cis- 130 WANDER ET AL., 1987 Jan 15, 2025 Jan 15, 2025
2818 5-HT2A FR. CORTEX HUMAN 125I-LSD HISTAMINE >10000 ELLIOT & KENT, 1989 Jan 15, 2025 Jan 15, 2025
68354 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 303.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68610 recombinant HUMAN 3H-AdoMet 1-(Aminomethyl)-6-hydroxynaphthalene 8400 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
3330 D3 CLONED HUMAN 3H-YM 09151-2 SULPIRIDE 15 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68866 SST4 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 79.4328 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69122 H4 CLONED HUMAN 3H-Histamine VUF4686 50.1187 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CHLORPROMAZINE 3115 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
69634 Alpha1D CLONED HUMAN 3H-PRAZOSIN 2-CI-DPH >10000 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4354 5-HT6 CLONED HUMAN 3H-LSD RU 24969 570 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69890 D1 CLONED HUMAN 3H-SCH23390 4-[1-(3-methylphenyl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4610 SLC6A3 CLONED HUMAN 3H-DA UPTAKE METHYLPHENIDATE 42 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4866 5-HT2B CLONED HUMAN 3H-5HT MIANSERIN 8.98 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70402 D2 CLONED HUMAN 3H-Methylspiperone (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 345 Omran, A. et, al. 2018 Jan 15, 2025 Jan 28, 2025
5122 5-HT2A CLONED HUMAN 125I-DOI QDOB 2155 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70658 H4 CLONED HUMAN 3H-Histamine MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 28, 2025
5378 5-HT2B CLONED HUMAN 3H-5HT mCPP 31.62 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
5634 5-HT4 CLONED HUMAN 3H-GR-113808 5-CT >10000 CLAEYSEN S, ET AL., 1997 Jan 15, 2025 Jan 27, 2025
71170 D3 CLONED HUMAN 3H-N-Methylspiperone SYA16263 86 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5890 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE YOHIMBINE 1.2 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71426 5-HT1B CLONED HUMAN 3H-5CT 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6658 5-HT1E CLONED HUMAN 3H-5HT 5-CT 7875 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
6914 5-HT2A CLONED HUMAN 3H-KETANSERIN CLOZAPINE 11 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72706 5-HT7 CLONED HUMAN 3H-LSD naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7426 MOR CLONED HUMAN 3H-DAMGO CTOP 0.18 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72962 5-HT3 CLONED HUMAN 3H-GR-65630 catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7682 GABAA CLONED HUMAN 3H-MUSCIMOL P4S 97.72 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7938 GABAA CLONED HUMAN 3H-RO-15-1788 RY 80 28.8 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8194 GABAA CLONED HUMAN 3H-RO-15-1788 42 >10000 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
8450 SST5 CLONED HUMAN 125I-Tyr3-octreotide somatostatin-28 0.05 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8706 SST5 CLONED HUMAN 125I-Tyr3-octreotide cycloantagonist SA 5.62 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8962 SST1 CLONED HUMAN 125I-SRIF-28 SMS 201-995 251.18 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74498 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74754 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75010 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9730 MT2 CLONED HUMAN 125I-Iodomelatonin Melatonin,6,7 di-cl-2-Me 0.23 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75266 M4 CLONED HUMAN 3H-QNB ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75522 5-HT1E CLONED HUMAN 3H-5-HT propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
10242 CLONED HUMAN 125I-HEAT WB 4101 10 Schwinn, et al.,1995 Jan 15, 2025 Jan 15, 2025
75778 5-HT7 CLONED HUMAN 3H-LSD 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76290 M2 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76546 5-HT1B CLONED HUMAN 3H-5-CT (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76802 5-HT2A CLONED HUMAN 3H-KETANSERIN (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77058 5-HT5A CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11778 H1 FR. CORTEX HUMAN 3H-doxepin CHLORPROMAZINE 9 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77314 Alpha1B CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77570 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77826 D1 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12546 Neutrophil HUMAN 3H-LTB4 DIHETE 12(s), 5(s) 454 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78082 D4 CLONED HUMAN 3H-N-Methylspiperone (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78338 H3 CLONED HUMAN 3H-Alpha-methylhistamine (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78594 M4 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78850 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79106 5-HT5A CLONED HUMAN 3H-LSD (±)-2,5-Dimethoxy-4-iodoamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79362 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-2,5-Dimethoxy-4-ethylamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14082 CLONED HUMAN 3H-LTD4 Pranlukast 3620 Heise CE, et al., 2000 Jan 15, 2025 Jan 15, 2025
79618 NET CLONED HUMAN 3H-Nisoxetine S,S-2c >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14338 5-HT2B CLONED HUMAN 3H-LSD d-Fenfluramine 3920 FITZGERALD LW, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
79874 M4 CLONED HUMAN 3H-QNB Salvinorin A >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80130 CLONED HUMAN 3H-VASOPRESSIN 4-Ethylthio-2,5-dimethoxyphenylbutylamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14850 TP Washed Platelets HUMAN 3H-SQ 29548 BM 13177 1404 Hedberg, A, et al., 1988 Jan 15, 2025 Jan 15, 2025
80386 5-HT2C CLONED HUMAN 3H-MESULERGINE (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one 2013 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15106 CLONED HUMAN 3H-PGE2 AGN 191995 >10000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80642 5-HT6 CLONED HUMAN 3H-LSD (Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80898 5-HT1D CLONED HUMAN 3H-5-CT (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81154 D4 CLONED HUMAN 3H-N-Methylspiperone N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 28, 2025
15874 5-HT7 CLONED HUMAN 3H-5HT 8-OH-DPAT 467.73 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81410 5-HT2A CLONED HUMAN 3H-KETANSERIN methyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 15, 2025
16130 D1 CLONED HUMAN 3H-SCH23390 SKF-82526, (-) 1818 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81922 D4 CLONED HUMAN 3H-N-Methylspiperone (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16642 Y4 CLONED HUMAN 125I-hPP Des-AA11-18[Cys7,21,D-Lys9 (Ac), Pro34]-NPY 7.3 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
82178 5-HT6 CLONED HUMAN 3H-LSD 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 2192 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82434 5-HT2C CLONED HUMAN 3H-MESULERGINE (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17154 5-HT2A BRAIN HUMAN 3H-KETANSERIN ORG-5222 0.77 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82690 5-HT1B CLONED HUMAN 3H-5-CT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17666 PANC1 HUMAN 125I-VIP Vasoactive intestinal polypeptide 1.7 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83202 5-HT2C CLONED HUMAN 125I-DOI LSD 2.91 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83458 M1 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.301995 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83714 5-HT2B CLONED HUMAN 3H-LSD (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 453 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83970 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 302 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84226 DOR CLONED HUMAN 3H-DADLE (±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 1928 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84482 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84738 MOR CLONED HUMAN 3H-DAMGO (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19458 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Nle8 0.34 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84994 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85250 recombinant HUMAN 3H-Estradiol Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 15, 2025
86018 5-HT7 CLONED HUMAN 3H-LSD (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 15, 2025
86274 DOR CLONED HUMAN 3H-DADLE JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
87554 5-HT6 CLONED HUMAN 3H-LSD 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
22274 A3 CLONED HUMAN 125I-Aba 4d 25.6 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87810 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 137 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22530 5-HT4 CLONED HUMAN 3H-GR-113808 SL650155 0.6 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
22786 H2 CLONED HUMAN 3H-TIOTIDINE L-cystine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88578 H1 CLONED HUMAN 3H-PYRILAMINE 1-(3-Phenoxypropyl)-4-phenylpiperazine 67.9 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88834 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
23554 H3 BRAIN CORTEX HUMAN 3H-NAMH A-317920 117.49 Esbenshade TA, et al., 2003 Jan 15, 2025 Jan 15, 2025
89090 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89346 5-HT6 CLONED HUMAN 3H-LSD 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 1039 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
24066 5-HT2A CLONED HUMAN UNDEFINED MELPERONE 150 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89602 M3 CLONED HUMAN 3H-NMS 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89858 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 108 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90114 D1 CLONED HUMAN 3H-SCH23390 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24834 Alpha1B CLONED HUMAN 125I-HEAT CLOZAPINE 7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90626 A2A CLONED HUMAN 3H-MSX-2 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90882 Alpha1A CHO cells HUMAN 3H-PRAZOSIN 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 21.3796 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
25602 5-HT7 CLONED HUMAN 3H-LSD Norephedrine, (+) 7000 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
91138 A3 CHO cells HUMAN 3H-HEMADO N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide >10000 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
25858 M1 CLONED HUMAN 3H-QNB Pseudoephedrine,(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91394 CB2 CLONED HUMAN 3H-CP55940 O-6211 >10000 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26114 SLC6A4 CLONED HUMAN 3H-CITALOPRAM Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91650 A3 CLONED HUMAN 3H-PSB-11 N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 111 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26370 Alpha2A CLONED HUMAN 3H-CLONIDINE Miquelianin 716.5 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91906 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (4-chlorophenyl)-methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92162 5-HT6 CLONED HUMAN 3H-LSD N-{1-[2-(Biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 267 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
92418 DOR CLONED HUMAN 3H-DADLE 9,13-epoxy-15,16-dihydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27138 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N,N-dimethyl derivative 562 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92674 M3 CLONED HUMAN 3H-QNB 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27394 Beta2 CLONED HUMAN 3H-CGP-12177 QUINPIROLE >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 28, 2025
92930 A3 CLONED HUMAN 125I-AB-MECA 2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27650 Alpha1A CLONED HUMAN 125I-HEAT MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
27906 5-HT2A CLONED HUMAN 3H-KETANSERIN QUIPAZINE 362 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28162 5-HT7 CLONED HUMAN 3H-LSD METHYSERGIDE 30 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93698 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 102 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28674 5-HT2C VGI CLONED HUMAN 125I-DOI ARIPIPRAZOLE 97 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 15, 2025
94210 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-allyloxy-2,5-dimethoxyamphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29186 SST2 CLONED HUMAN UNDEFINED L-803,087 4720 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94722 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94978 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29698 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 4.9 Liao Y, et.al., 1999 Jan 15, 2025 Jan 15, 2025
29954 H4 CLONED HUMAN 3H-Histamine (7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 19 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95746 5-HT5A CLONED HUMAN 3H-LSD Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96002 DAT CLONED HUMAN 3H-WIN 35,428 Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96258 Alpha1A CLONED HUMAN 3H-PRAZOSIN 3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
30978 D3 CLONED HUMAN UNDEFINED SR 147778 1000 Rinaldi-Carmona M et al., 2004 Jan 15, 2025 Jan 15, 2025
96514 5-HT2B CLONED HUMAN [3H]-LSD 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31234 5-HT2C CLONED HUMAN 3H-MESULERGINE MDL 100907 63.44 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96770 D1 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31490 5-HT4 CLONED HUMAN UNDEFINED (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) >10000 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97026 Alpha2B CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) 388 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97282 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 23.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97538 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
98050 CB1 CHO cells HUMAN 3H-CP-55940 6-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine 47 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98306 D2 CLONED HUMAN [3H]-N-methylspiperone 2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide >10000 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98562 5-HT2B CLONED HUMAN [3H]-LSD 2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 561 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98818 5-HT6 CLONED HUMAN 3H-LSD 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine >10000 Reilly SW et al 2019 Jan 15, 2025 Jan 15, 2025
33538 H1 CLONED HUMAN 3H-PYRILAMINE Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99074 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99330 D2 CLONED HUMAN [3H]N-methylspiperone 4-(4-(2-Methoxyphenyl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 1020 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34050 P2X3 CLONED HUMAN 3H-A-317491 AP6A 4.8 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99586 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 0.609 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99842 Alpha1A CLONED HUMAN [125I] HEAT (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 6800 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100098 Sigma 2 CLONED HUMAN 3H-DTG Cariprazine 1531 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100354 5-HT7 CLONED HUMAN 3H-LSD OLANZAPINE 157 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100866 nAChR CLONED HUMAN Functional d-Tubocurarine >10000 Kuo YP, et al., 2005 Jan 15, 2025 Jan 29, 2025
35586 CLONED HUMAN 3H-SQ 29548 FLUPROSTENOL >10000 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35842 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 1.6 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101378 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 222 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36098 COX-2 whole blood assay (WBA) HUMAN Functional Naproxen >10000 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101634 5-HT1D CLONED HUMAN [3H]GR127543 Perospirone 20 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101890 D2 CLONED HUMAN [3H]N-methylspiperone Ziprasidone 81 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36610 D2 CLONED HUMAN 3H-SPIPERONE HALOPERIDOL 2.5 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102146 D5 CLONED HUMAN [3H]SCH23390 NEMONAPRIDE >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37890 MPP-2 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-carboxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 85 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38658 UNDEFINED HUMAN 3H-hypoxanthine N-{(1S,2S)-1-(4-Benzo[1,3]dioxol-5-yl-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propyl}-2,4,6-trifluoro-benzamide 19 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
38914 H4 CLONED HUMAN 3H-Histamine MDL 100907 >10000 Pehek EA, et al., 2005 Jan 15, 2025 Jan 15, 2025
39170 D4 CLONED HUMAN R-SAT OCTOCLOTHEPIN 0.4 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39426 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39682 5-HT2B CLONED HUMAN 3H-5HT DOI,(-) 53.7032 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39938 5-HT2B CLONED HUMAN UNDEFINED BW-723C86 79.4328 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
40706 mGluR5 CLONED HUMAN Functional 9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one >10000 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41218 CLONED HUMAN 125I-Chemokine 5-(4-(4-Bromophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41986 M1 CLONED HUMAN 3H-QNB Adinazolam >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
43010 FRK CLONED HUMAN 3H-Staurosporine BIRB-796 360 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43266 CDK2 CLONED HUMAN 3H-Staurosporine Flavopiridol 200 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
43522 FER CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43778 STK4 CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44034 RPS6KA3 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44290 MAPK P38 CLONED HUMAN 3H-Staurosporine CI-1033 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44546 FGFR1 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44802 YES1 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45058 PAK6 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45570 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Desmethylcitalopram >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45826 5-HT2B CLONED HUMAN 3H-LSD (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46082 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46594 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46850 M5 CLONED HUMAN 3H-QNB (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47362 CLONED HUMAN 3H-AMPA LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47618 ADK recombinant HUMAN Functional 4-N-(4-Hydroxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47874 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Aib29,D31,p34,F35]-h-alpha-CGRP 27-37 0.002 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
48130 Y1 CLONED HUMAN 3H-Propionyl-NPY PP, human 170 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48642 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 350 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49666 SST1 CLONED HUMAN 125I-LTT-SST-28 Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8) >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50178 mGluR1 CLONED HUMAN Functional 1S, 3R-ACPD >10000 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50434 SST4 CLONED HUMAN 125I-LTT-SST-28 octreotide 2191 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025
50946 MOR UNDEFINED HUMAN UNDEFINED Naloxone(-) 0.79 Peng X et al., 2007 Jan 15, 2025 Jan 15, 2025
51458 Alpha1A UNDEFINED HUMAN UNDEFINED 3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 1.5 Chiu G et al., 2007 Jan 15, 2025 Jan 15, 2025
51970 KOR UNDEFINED HUMAN UNDEFINED 7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 26.4 Rennison D et al., 2007 Jan 15, 2025 Jan 15, 2025
52226 5-HT1A UNDEFINED HUMAN UNDEFINED (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 1.33 Krushinski JH Jr et al., 2007 Jan 15, 2025 Jan 15, 2025
52482 SLC6A2 UNDEFINED HUMAN UNDEFINED (S)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline 121 Letavic MA et al., 2007 Jan 15, 2025 Jan 15, 2025
52994 CB2 UNDEFINED HUMAN UNDEFINED azepan-1-yl(5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-yl)methanone 4900 Foloppe N et al., 2008 Jan 15, 2025 Jan 15, 2025
53250 D2 UNDEFINED HUMAN UNDEFINED 1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea 103 Chiu G et al., 2008 Jan 15, 2025 Jan 15, 2025
53762 H1 UNDEFINED HUMAN UNDEFINED Ziprasidone 47 Ablordeppey SY et al., 2008 Jan 15, 2025 Jan 15, 2025
54274 SLC6A4 UNDEFINED HUMAN UNDEFINED cis-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile 6.16 Funke U et al., 2008 Jan 15, 2025 Jan 15, 2025
54530 A3 UNDEFINED HUMAN UNDEFINED N-Benzo[1,3]dioxol-5-yl-2-[5-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1-methyl-1H-pyrazol-3-yloxy]-acetamide 1000 Borrmann T et al., 2009 Jan 15, 2025 Jan 15, 2025
54786 D2 UNDEFINED HUMAN UNDEFINED N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine 690 Dörfler M et al., 2008 Jan 15, 2025 Jan 15, 2025
55042 5-HT1A UNDEFINED HUMAN UNDEFINED 4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 70 Leopoldo M et al., 2008 Jan 15, 2025 Jan 15, 2025
55298 DOR UNDEFINED HUMAN UNDEFINED 8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 379 Caldwell JP et al., 2009 Jan 15, 2025 Jan 15, 2025
55810 SLC6A4 UNDEFINED HUMAN UNDEFINED [C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline 44.7 Ben-Daniel R et al., 2008 Jan 15, 2025 Jan 15, 2025
56322 A1 UNDEFINED HUMAN UNDEFINED 2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione 132 Ishiyama H et al., 2009 Jan 15, 2025 Jan 15, 2025
56578 DOR UNDEFINED HUMAN UNDEFINED 4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4270 Zhang Y et al., 2009 Jan 15, 2025 Jan 15, 2025
56834 SLC6A2 UNDEFINED HUMAN UNDEFINED 2-(N-Cyclopentylamino)-3'-chloropropiophenone 5700 Carroll FI et al., 2009 Jan 15, 2025 Jan 15, 2025
57090 D2 UNDEFINED HUMAN UNDEFINED PPP, S(-)-3 17.4 Pettersson F et al., 2010 Jan 15, 2025 Jan 15, 2025
57346 A1 UNDEFINED HUMAN UNDEFINED 4-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-butyric acid 12 Scheiff AB et al., 2010 Jan 15, 2025 Jan 15, 2025
57602 SST3 UNDEFINED HUMAN UNDEFINED N-(benzo[d]thiazol-2-yl)-4-(3-ethoxy-4-methoxyphenyl)piperazine-1-carboxamide >10000 Martin RE et al., 2009 Jan 15, 2025 Jan 15, 2025
57858 MOR UNDEFINED HUMAN UNDEFINED (+)-1-[(1S,2R,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone 470 Geiger C et al., 2010 Jan 15, 2025 Jan 15, 2025
58114 5-HT2A CLONED HUMAN 125I-DOI N-(4-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate 10.5 Nichols DE, 2014 Jan 15, 2025 Jan 15, 2025
58370 H3 CLONED HUMAN 3H-Alpha-Me-histamine MRS5698 >10000 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58626 hERG CLONED HUMAN 3H-N-Me-Dofetilide MRS5676 7930 Jacobson KA, et al., 2014 Jan 15, 2025 Jan 15, 2025
58882 SLC6A3 CLONED HUMAN 3H-WIN 35,428 N,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine 1000 Mavel S, et al., 2009 Jan 15, 2025 Jan 15, 2025
59138 5-HT2A CLONED HUMAN 3H-KETANSERIN CHLORPROMAZINE 2.75 Gillman P, et al., 2005 Jan 15, 2025 Jan 15, 2025
59394 D4 CLONED HUMAN 3H-N-Methylspiporone N-(1-Benzyl-3-pyrrolidinyl)-2'-formyl-4-biphenylcarboxamide 36 Egle, I. et. al., 2004 Jan 15, 2025 Jan 15, 2025
59650 Alpha1B CLONED HUMAN 3H-PRAZOSIN SK&F 83959 688 O'sullivan, G. et. al., 2005 Jan 15, 2025 Jan 15, 2025
59906 5-HT6 CLONED HUMAN 3H-LSD 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide >10000 Huang Y, et al, 2005a Jan 15, 2025 Jan 15, 2025
60162 A2A CLONED HUMAN [3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- hexane-1-carboxamide >10000 Tosh DK, et al., 2014 Jan 15, 2025 Jan 15, 2025
60418 GABAA CLONED HUMAN FNZ CM-A-87 4.61 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60674 GABAA CLONED HUMAN FNZ SPH-38 10.8 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
60930 GABAA CLONED HUMAN FNZ XLi343 6.375 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61186 GABAA CLONED HUMAN FNZ CM-A58 1000 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61442 GABAA CLONED HUMAN FNZ JYI-03 107 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 27, 2025
61698 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2-methoxyphenyl)propan-1-amine 140 Ponnala, Shashikanth et. al. 2015 Jan 15, 2025 Jan 15, 2025
61954 CLONED HUMAN UNDEFINED ASTEMIZOLE >10000 Suessbrich, H et al., 1996 Jan 15, 2025 Jan 15, 2025
62210 Serotonin CLONED HUMAN [3H] Citalopram 5-APB 552 Iversen l., et al., 2012 Jan 15, 2025 Jan 15, 2025
62466 M3 CLONED HUMAN 3H-QNB 3-methoxy-diphenidine 2296 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 28, 2025
63234 GCCR CLONED HUMAN 125I-Glucagon 4-[2-(1H-Benzimidazol-2-ylsulfanyl)-1-hydroxyethyl]-2-chlorophenol >10000 Madsen, P et al., 1998 Jan 15, 2025 Jan 15, 2025
63490 5-HT1A CLONED HUMAN 3H-WAY100635 bifeprunox 0.73 Maeda, K. et, al. 2014 Jan 15, 2025 Jan 28, 2025
64002 5-HT6 CLONED HUMAN 3H-LSD 2-[5-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxoacetamide 18.4 Holenz J, et al., 2005 Jan 15, 2025 Jan 15, 2025
64258 5-HT2A CLONED HUMAN 3H-KETANSERIN PIMOZIDE 37.1535 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 15, 2025
64514 D2 CLONED HUMAN 3H-N-Methylspiperone MESORIDAZINE 19.0546 Silvestre, JS. et, al. 2005 Jan 15, 2025 Jan 28, 2025
65282 GABAA CLONED HUMAN [3H] Flunitrazepam XHE-II-073A (R Enriched) 10 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65539 GABAA CLONED HUMAN [3H] Flunitrazepam Ro15-1788 1.05 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
65795 GABAA CLONED HUMAN [3H] Flunitrazepam RY-053 29 Clayton, Terry et. al. 2015 Jan 15, 2025 Jan 28, 2025
66051 SERT CLONED HUMAN 3H-CITALOPRAM Ondansetron HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
66307 Alpha1D CLONED HUMAN 3H-PRAZOSIN Finazine 707 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
66563 Alpha1A CLONED HUMAN 3H-PRAZOSIN 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
1283 5-HT1D CORTEX HUMAN 3H-5HT HALOPERIDOL >10000 PEROUTKA ET AL., 1989 Jan 15, 2025 Jan 15, 2025
66819 5-HT2B CLONED HUMAN 3H-LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 913 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 15, 2025
67331 KOR CLONED HUMAN 3H-U69593 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp, A, et. al. 2016 Jan 15, 2025 Jan 28, 2025
67587 5-HT2B KIDNEY HUMAN 3H-LSD (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- hexane-2,3-diol 34 Tosh, DK, et. al. 2016 Jan 15, 2025 Jan 15, 2025
2307 5-HT3 HIPPOCAMPUS HUMAN 3H-ZACOPRIDE DOPAMINE >10000 BARNES ET AL., 1989 Jan 15, 2025 Jan 15, 2025
67843 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 2533 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
2563 5-HT2A CORTEX HUMAN 3H-SPIPERONE THIOTHIXENE,trans- 140.3 ANDORN ET AL., 1984 Jan 15, 2025 Jan 15, 2025
68355 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 288.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68611 recombinant HUMAN 3H-AdoMet 8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 1400 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
3331 D3 CLONED HUMAN 3H-YM 09151-2 YM-09151-2 0.2 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
68867 SST5 CLONED HUMAN 125I-SRIF H-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 100 Lewis I, et al., 2003 Jan 15, 2025 Jan 15, 2025
69123 H4 CLONED HUMAN 3H-Histamine VUF4687 63.0957 Lim HD, et al., 2005 Jan 15, 2025 Jan 15, 2025
69379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RACLOPRIDE >10000 Maheux J, et al., 2005 Jan 15, 2025 Jan 15, 2025
4099 KOR CLONED HUMAN 3H-U69,593 TIPPpsi >10000 TOLL L, et. al., 1998 Jan 15, 2025 Jan 15, 2025
69635 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-CI-DPH 2690 Wallach, Jason, et. al. 2016 Jan 15, 2025 Jan 15, 2025
4355 5-HT6 CLONED HUMAN 3H-LSD 5-CT 720 KOHEN R, ET AL., 1996 Jan 15, 2025 Jan 15, 2025
69891 D1 CLONED HUMAN 3H-SCH23390 4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine >10000 Colestock, T. et, al 2018 Jan 15, 2025 Jan 28, 2025
4611 SLC6A3 CLONED HUMAN 3H-DA UPTAKE NOMIFENSINE 53 PRISTUPA ZB, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
4867 5-HT2B CLONED HUMAN 3H-5HT 5-HT,N-ACETYL 6800 WAINSCOTT DB, ET AL., 1998 Jan 15, 2025 Jan 15, 2025
70403 5-HT1A CLONED HUMAN 3H-WAY100635 (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide 328 Omran, A. et, al. 2018 Jan 15, 2025 Jan 15, 2025
5123 5-HT2B CLONED HUMAN 3H-5HT DMA 1039 NELSON DL, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
70659 M1 CLONED HUMAN 3H-QNB MRP3215 >10000 Porter, MR et. al, 2019 Jan 15, 2025 Jan 15, 2025
5379 5-HT2B CLONED HUMAN 3H-5HT MIANSERIN 19.95 BONHAUS DW, ET AL., 1995 Jan 15, 2025 Jan 15, 2025
71171 D4 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 510 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
5891 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE PHENOXYBENZAMINE 3.5 WEINSHANK RL, ET AL, 1990 Jan 15, 2025 Jan 15, 2025
71427 5-HT1D CLONED HUMAN 3H-5CT 4-acetoxy-N,N-diallyltryptamine 801 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
6659 5-HT1E CLONED HUMAN 3H-5HT KETANSERIN >10000 ZGOMBICK JM, ET AL., 1992 Jan 15, 2025 Jan 15, 2025
72195 D1 CLONED HUMAN 3H-SCH23390 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl >10000 Magnus CJ et al 2019 Jan 15, 2025 Jan 28, 2025
6915 5-HT2A CLONED HUMAN 3H-KETANSERIN FLUPHENAZINE 80 SEEMAN P, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
72707 Alpha1A CLONED HUMAN 3H-PRAZOSIN naringenin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 28, 2025
7427 MOR CLONED HUMAN 3H-DAMGO b-FNA-HCl 0.33 Raynor K, et al., 1994 Jan 15, 2025 Jan 15, 2025
72963 5-HT5A CLONED HUMAN 3H-LSD catechin >10000 Moawad A et al 2017 Jan 15, 2025 Jan 15, 2025
7683 GABAA CLONED HUMAN 3H-MUSCIMOL Gamma-Aminobutyric acid 50.11 Ebert B, et al., 1997 Jan 15, 2025 Jan 27, 2025
7939 GABAA CLONED HUMAN 3H-RO-15-1788 Beta-CCT 5000 He X, et al., 1999 Jan 15, 2025 Jan 27, 2025
8195 GABAA CLONED HUMAN 3H-RO-15-1788 43 >10000 Huang Q, et al., 1999 Jan 15, 2025 Jan 27, 2025
8451 SST5 CLONED HUMAN 125I-Tyr3-octreotide LTT-SRIF28 0.25 Siehler S, et al., 1999 Jan 15, 2025 Jan 15, 2025
8707 SST5 CLONED HUMAN 125I-Tyr3-octreotide BIM 23030 35.48 Siehler S, et al., 1998 Jan 15, 2025 Jan 15, 2025
8963 SST1 CLONED HUMAN 125I-SRIF-28 BIM 23014 501.18 Bruns C, et al., 1996 Jan 15, 2025 Jan 15, 2025
74499 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74755 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
75011 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]-hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
9731 MT2 CLONED HUMAN 125I-Iodomelatonin 8-M-CADOT 0.69 Dubocovich M, Masana S, Sauri D, 1997 Jan 15, 2025 Jan 15, 2025
75267 M5 CLONED HUMAN 3H-QNB ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75523 5-HT2A CLONED HUMAN 3H-KETANSERIN propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
75779 Alpha1A CLONED HUMAN 3H-PRAZOSIN 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76035 D1 CLONED HUMAN 3H-SCH23390 Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
76291 M3 CLONED HUMAN 3H-QNB (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76547 5-HT1D CLONED HUMAN 3H-5-CT (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
76803 5-HT2B CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77059 5-HT6 CLONED HUMAN 3H-LSD (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
11779 H1 FR. CORTEX HUMAN 3H-doxepin THIORIDAZINE 16 Richelson E, et al., 1984 Jan 15, 2025 Jan 15, 2025
77315 Alpha1D CLONED HUMAN 3H-PRAZOSIN (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
77571 Beta 1 CLONED HUMAN 125I-Pindolol (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
77827 D5 CLONED HUMAN 3H-SCH23390 (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
12547 Neutrophil HUMAN 3H-LTB4 20-COOH-LTB4 855 Jackson RH, et al., 1992 Jan 15, 2025 Jan 15, 2025
78083 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78339 H4 CLONED HUMAN 3H-Histamine (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
78595 M5 CLONED HUMAN 3H-QNB (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 15, 2025
78851 Sigma 2 CLONED HUMAN 3H-DTG (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 Frankowski KJ et al 2010 Jan 15, 2025 Jan 28, 2025
79107 5-HT5A CLONED HUMAN 3H-LSD 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
79363 Alpha1A CLONED HUMAN 3H-PRAZOSIN (±)-2,4,5-Trimethoxamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 28, 2025
14083 CLONED HUMAN 3H-LTD4 Zafirlukast 7397 Heise CE, et al., 2000 Jan 15, 2025 Jan 15, 2025
79619 NET CLONED HUMAN 3H-Nisoxetine 5-MeO-TMT 6380 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14339 5-HT2B CLONED HUMAN 3H-LSD l-Fenfluramine 680 FITZGERALD LW, ET AL., 1999 Jan 15, 2025 Jan 15, 2025
79875 M5 CLONED HUMAN 3H-QNB (±)-2,5-Dimethoxy-4-bromoamphetamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
80131 CLONED HUMAN 3H-VASOPRESSIN 6-Fluoro-N,N-dimethyltryptamine >10000 Ray TS 2010 Jan 15, 2025 Jan 15, 2025
14851 TP Washed Platelets HUMAN 3H-SQ 29548 BM 13505 5.43 Hedberg, A, et al., 1988 Jan 15, 2025 Jan 15, 2025
80387 5-HT3 CLONED HUMAN 3H-GR-65630 (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
15107 CLONED HUMAN 3H-PGE2 AGN 192151 >10000 Schuster V.L. et.al., 2000 Jan 15, 2025 Jan 15, 2025
80643 5-HT7 CLONED HUMAN 3H-LSD (Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one 3350 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
80899 5-HT1E CLONED HUMAN 3H-5-HT (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one >10000 Lewellyn K et al 2013 Jan 15, 2025 Jan 15, 2025
81155 DAT CLONED HUMAN 3H-WIN 35,428 N-Benzyl-2-azatricyclo[3.3.1.13,7]decane >10000 Banister SD et al 2011 Jan 15, 2025 Jan 15, 2025
15875 5-HT7 CLONED HUMAN 3H-5HT CYPROHEPTADINE 123.02 BOESS FG, ET AL., 1994 Jan 15, 2025 Jan 15, 2025
81411 D2 CLONED HUMAN 3H-N-Methylspiperone methyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate >10000 Weiss DR et al 2018 Jan 15, 2025 Jan 28, 2025
16131 D1 CLONED HUMAN 3H-SCH23390 ADTN, (+) 4600 Sunahara RK, et al., 1991 Jan 15, 2025 Jan 15, 2025
81923 D5 CLONED HUMAN 3H-N-Methylspiperone (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol >10000 Severance AJ et al 2007 Jan 15, 2025 Jan 28, 2025
16643 Y4 CLONED HUMAN 125I-hPP Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26]-NPY 206 Mullins D et al., 2001 Jan 15, 2025 Jan 15, 2025
82179 5-HT7 CLONED HUMAN 3H-LSD 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 181 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82435 5-HT3 CLONED HUMAN 3H-GR65630 (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
17155 5-HT2A BRAIN HUMAN 3H-KETANSERIN PIMOZIDE 14.3 Richelson E, Souder T. 2000 Jan 15, 2025 Jan 15, 2025
82691 5-HT1D CLONED HUMAN 3H-5-CT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82947 A2B CHO cells HUMAN 3H-PSB-603 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
17667 CLONED HUMAN 125I-VIP VIP [D-His1] 0.74 Igarashi H et al., 2002 Jan 15, 2025 Jan 15, 2025
83203 5-HT2C CLONED HUMAN 125I-DOI DMT 166 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83459 M2 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 6.0256 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83715 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3596 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83971 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 297 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84227 KOR CLONED HUMAN 3H-U69593 (±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide 76 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84483 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
84739 DOR CLONED HUMAN 3H-DADLE (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
19459 GPR24 CLONED HUMAN 125I-[Phe13, Tyr19]-hMCH N-Me-Leu9 62 Bednarek MA et al., 2002 Jan 15, 2025 Jan 15, 2025
84995 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
85251 recombinant HUMAN 125I-QRFP-43 Tasimelteon >10000 Lavedan C et al 2015 Jan 15, 2025 Jan 15, 2025
86019 SERT CLONED HUMAN 3H-CITALOPRAM (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
86275 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) JWH-391 >10000 Wiley JL et al 2016 Jan 15, 2025 Jan 28, 2025
87555 5-HT7 CLONED HUMAN 3H-LSD 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine >10000 Singh P et al 2018 Jan 15, 2025 Jan 15, 2025
22275 A3 CLONED HUMAN 125I-Aba 5 816 Kim, YC, et. al. 2000 Jan 15, 2025 Jan 15, 2025
87811 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€3,4â€difluoroâ€Nâ€(2â€phenylethyl)aniline 21 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
22531 5-HT3 CLONED HUMAN 3H-GR-65630 SL650155 >10000 Moser PC et. al., 2002 Jan 15, 2025 Jan 15, 2025
22787 H2 CLONED HUMAN 3H-TIOTIDINE D-methionine >10000 Shi Q, et.al., 2003 Jan 15, 2025 Jan 15, 2025
88579 H1 CLONED HUMAN 3H-PYRILAMINE 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 167 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88835 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89091 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 10.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89347 D2 CLONED HUMAN 3H-RACLOPRIDE 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 268 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
24067 5-HT2A CLONED HUMAN UNDEFINED MOLINDONE 5800 Seeman, Philip 2001 Jan 15, 2025 Jan 15, 2025
89603 M2 CLONED HUMAN 3H-NMS 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89859 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 124 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
90115 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
24835 5-HT5A CLONED HUMAN 3H-LSD CLOZAPINE 3857 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90627 A2A CLONED HUMAN 3H-MSX-2 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 58.3 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
25347 M1 CLONED HUMAN 3H-QNB ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
90883 Alpha1B CHO cells HUMAN 3H-PRAZOSIN 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 158.489 Franchini S et al 2014 Jan 15, 2025 Jan 28, 2025
25603 5-HT7 CLONED HUMAN 3H-LSD Cathinone, (-) 2700 Rothman RB, et al., 2003a Jan 15, 2025 Jan 15, 2025
91139 A1 CHO cells HUMAN 3H-CCPA Ethyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2014 Jan 15, 2025 Jan 15, 2025
91395 CB2 CLONED HUMAN 3H-CP55940 O-6212 >10000 Wiley JL et al 2012 Jan 15, 2025 Jan 28, 2025
26115 D2 CLONED HUMAN 3H-NMSP Pseudonorephedrine, (+) [cathine, (+)] >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
91651 A3 CLONED HUMAN 3H-PSB-11 N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 9.05 Abdelrahman A et al 2020 Jan 15, 2025 Jan 15, 2025
26371 Alpha2C CLONED HUMAN 3H-CLONIDINE Rutin 9637 Butterweck V, et. al., 2002 Jan 15, 2025 Jan 15, 2025
91907 A1 CLONED HUMAN 3H-DPCPX (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3-chlorophenyl)methanone >10000 Romagnoli R et al 2014 Jan 15, 2025 Jan 15, 2025
92163 5-HT6 CLONED HUMAN 3H-LSD N-{1-[2-(5,6,7,8-Tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 102 Zajdel P et al 2012 Jan 15, 2025 Jan 15, 2025
92419 DOR CLONED HUMAN 3H-DADLE 9,13-epoxylabd-5-ene-7 β,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
27139 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride >10000 May JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
92675 M4 CLONED HUMAN 3H-QNB 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 15, 2025
27395 Beta2 CLONED HUMAN 3H-CGP-12177 Ropinirole >10000 Millan MJ, et al., 2002 Jan 15, 2025 Jan 28, 2025
92931 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
27651 D5 CLONED HUMAN 3H-SCH23390 MDMA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93187 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 76 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
27907 5-HT2A CLONED HUMAN 3H-DOB QUIPAZINE 59 Egan C, et.al., 2000 Jan 15, 2025 Jan 15, 2025
28163 5-HT1D CLONED HUMAN 3H-GR-125743 METHYSERGIDE 69 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
93699 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 194 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
28675 5-HT2C CLONED HUMAN 125I-DOI ARIPIPRAZOLE 22 Shapiro DA, et.al., 2003 Jan 15, 2025 Jan 27, 2025
94211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine 5600 Kolaczynska KE et al 2019 Jan 15, 2025 Jan 15, 2025
29187 SST2 CLONED HUMAN UNDEFINED L-796,778 >10000 Patel YC, 1999 Jan 15, 2025 Jan 15, 2025
94723 5-HT2A CLONED HUMAN 3H-KETANSERIN 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
94979 D2 CLONED HUMAN 3H-N-Methylspiperone 2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate >10000 Jung et al 2021 Jan 15, 2025 Jan 28, 2025
29699 D3 CLONED HUMAN UNDEFINED HALOPERIDOL 10 Liao Y, et.al., 1999 Jan 15, 2025 Jan 15, 2025
29955 H4 CLONED HUMAN 3H-Histamine (7-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 8 Jablonowski JA, et al., 2003 Jan 15, 2025 Jan 15, 2025
95747 5-HT6 CLONED HUMAN 3H-LSD Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96003 DAT CLONED HUMAN 3H-WIN 35,428 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene >10000 Jung et al 2021 Jan 15, 2025 Jan 15, 2025
96259 Alpha1B CLONED HUMAN 3H-PRAZOSIN 3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid >10000 Jung et al 2020 Jan 15, 2025 Jan 28, 2025
96515 5-HT3 CLONED HUMAN [3H]GR65630 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione >10000 Martini ML et al 2019a Jan 15, 2025 Jan 15, 2025
31235 D1 CLONED HUMAN 3H-SCH23390 MDL 100907 628 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
96771 D1 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
31491 5-HT7 CLONED HUMAN 3H-5CT (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) 3.16228 Lovell, P.J., et.al. 2000 Jan 15, 2025 Jan 15, 2025
97027 Alpha2C CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97283 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 138 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97539 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97795 H1 Sf9 HUMAN 3H-MEPYRAMINE UR-AK64 990 Xie, S. et. al., 2006 Jan 15, 2025 Jan 15, 2025
98051 CB2 CHO cells HUMAN 3H-CP-55940 6-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine 830 Amato G et al 2019 Jan 15, 2025 Jan 28, 2025
98307 D2 CLONED HUMAN [3H]-N-methylspiperone 2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole 990 Ofon E et al 2016 Jan 15, 2025 Jan 28, 2025
98563 5-HT2B CLONED HUMAN [3H]-LSD 2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 204 Ofon E et al 2016a Jan 15, 2025 Jan 15, 2025
98819 H1 CLONED HUMAN 3H-PYRILAMINE 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine 40 Reilly SW et al 2019 Jan 15, 2025 Jan 28, 2025
33539 H2 CLONED HUMAN 3H-TIOTIDINE Naproxen >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
99075 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide >10000 Tosh DK et al 2020 Jan 15, 2025 Jan 28, 2025
99331 D2 CLONED HUMAN [3H]N-methylspiperone 4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 607 Keck TM et al 2015 Jan 15, 2025 Jan 28, 2025
34051 P2X3 CLONED HUMAN 3H-A-317491 AP3A 1670 Jarvis, MF et. al., 2004 Jan 15, 2025 Jan 15, 2025
99587 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine 1.25 Yasdav R et al 2016 Jan 15, 2025 Jan 15, 2025
99843 Alpha1A CLONED HUMAN [125I] HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 6600 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
100099 D1 CLONED HUMAN 3H-SCH23390 Cariprazine 3749 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100355 5-HT7 CLONED HUMAN 3H-LSD GMC 1-116 200 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100867 nAChR CLONED HUMAN Functional Suberyldicholine >10000 Kuo YP, et al., 2005 Jan 15, 2025 Jan 29, 2025
35587 CLONED HUMAN 3H-SQ 29548 CLOPROSTENOL 6123 Abramovitz M, et al., 2000 Jan 15, 2025 Jan 15, 2025
35843 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 4.5 Andres JI, et al., 2005 Jan 15, 2025 Jan 15, 2025
101379 5-HT6 CLONED HUMAN 3H-LSD 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 999 Zareba P, et al., 2019 Jan 15, 2025 Jan 15, 2025
36099 COX-2 whole blood assay (WBA) HUMAN Functional Piroxicam 7900 Warner TD, et al., 1999 Jan 15, 2025 Jan 15, 2025
101635 5-HT1E CLONED HUMAN 3H-5HT Perospirone >10000 PDSP Certified Data Mar 21, 2025 Jul 28, 2026
101891 D3 CLONED HUMAN [3H]-N-methylspiperone Ziprasidone 52 PDSP Certified Data Mar 24, 2025 Jul 28, 2026
36611 D2 CLONED HUMAN 3H-SPIPERONE CLOZAPINE 144 Fernandez J, et al., 2005 Jan 15, 2025 Jan 15, 2025
102147 SERT CLONED HUMAN [3H]Citalopram NEMONAPRIDE >10000 PDSP Certified Data Mar 25, 2025 Jul 28, 2026
37891 MPP-9 CLONED HUMAN Functional 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-carboxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 26 Breyholz HJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
38659 UNDEFINED HUMAN 3H-hypoxanthine N-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-2-hydroxy-3-[2-(3-methoxyphenyl)ethylcarbamoyl]propyl}-2,4,6-tri-fluorobenzamide 390 Johansson P, et al., 2005 Jan 15, 2025 Jan 15, 2025
39171 D4 CLONED HUMAN R-SAT MESORIDAZINE 9.1 Burstein ES, et al., 2005 Jan 15, 2025 Jan 15, 2025
39427 CLONED HUMAN UNDEFINED [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid 1000 Armer RE, et al., 2005 Jan 15, 2025 Jan 15, 2025
39683 5-HT2B CLONED HUMAN 3H-5HT ERGOTAMINE 1.28825 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
40707 mGluR5 CLONED HUMAN Functional 3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one 19 Zheng GZ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41219 CLONED HUMAN 125I-Chemokine 5-(4-(4-Methoxyphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile >10000 Hulshof JW, et al., 2005 Jan 15, 2025 Jan 15, 2025
41987 M1 CLONED HUMAN 3H-QNB AMITRIPTYLINE 14.7 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
43011 FRK CLONED HUMAN 3H-Staurosporine Gleevec 3500 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43267 CDK5 CLONED HUMAN 3H-Staurosporine BAY-43-9006 6200 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43523 FGFR1 CLONED HUMAN 3H-Staurosporine SB202190 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
43779 Syk CLONED HUMAN 3H-Staurosporine VX-745 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44035 RPS6KA5 CLONED HUMAN 3H-Staurosporine Iressa >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44291 MAPK12 CLONED HUMAN 3H-Staurosporine CI-1033 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
44547 FGFR2 CLONED HUMAN 3H-Staurosporine GW-2016 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 28, 2025
44803 JAK1 CLONED HUMAN 3H-Staurosporine LY-333531 >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45059 PAK7 CLONED HUMAN 3H-Staurosporine Flavopiridol >10000 Fabian MA, et al., 2005 Jan 15, 2025 Jan 15, 2025
45315 CDK2 CLONED HUMAN Functional Indirubin-3monoxime 590 Bain J, et al., 2003 Jan 15, 2025 Jan 28, 2025
45571 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Desmethylsertraline 3 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45827 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46083 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46595 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid 6121 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46851 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47363 CLONED HUMAN 3H-AMPA LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47619 ADK recombinant HUMAN Functional 4-N-Cyclohexylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 250 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47875 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [A29,D31,p34,F35]-h-alpha-CGRP 27-37 8.4 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
48131 Y1 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 760 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48643 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
49667 SST1 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Reubi JC, et.al., 2000 Jan 15, 2025 Jan 15, 2025
50179 mGluR3 CLONED HUMAN Functional Quisqualate 6000 Flor PJ, et.al., 1996 Jan 15, 2025 Jan 28, 2025
50435 SST5 CLONED HUMAN 125I-LTT-SST-28 octreotide 137 Yang L, et.al., 1998a Jan 15, 2025 Jan 15, 2025